Assignee profile:

OTSUKA PHARMACEUTICAL CO., LTD.

City:

Tokyo

Country:

Japan

Published Applications:

640

Last publication date:

2026-04-30

Patent Grants:

429

Last grant date:

2025-07-29

Quarterly OTSUKA PHARMACEUTICAL CO., LTD. Patent Applications

Top Inventors for applications by OTSUKA PHARMACEUTICAL CO., LTD.

These are the the leading inventors for applications assigned to OTSUKA PHARMACEUTICAL CO., LTD.:

Recent patent applications by OTSUKA PHARMACEUTICAL CO., LTD.

OTSUKA PHARMACEUTICAL CO., LTD. based in Tokyo, JP has been assigned the rights to these inventions. The list includes both Pending Applications and Patent Grants:

#1 | 2026-04-30
US20260118357A1
Physics

TETRA-FUNCTIONAL CHEMICAL PROBE AND METHOD FOR IDENTIFYING TARGET MEMBRANE PROTEIN FROM LIVING CELL OR LIVING TISSUE BY USING SAID PROBE

#2 | 2026-04-30
US20260115131A1
Human necessities

METHODS OF ADMINISTERING AN ARIPIPRAZOLE INJECTABLE PREPARATION

#3 | 2026-04-16
US20260102394A1
Human necessities

PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS

#4 | 2026-01-29
US20260027103A1
Human necessities

PHARMACEUTICAL COMPOSITIONS COMPRISING A QUINOLONE COMPOUND FOR IRRITABLE BOWEL SYNDROME

#5 | 2025-11-27
US20250361224A1
Chemistry; metallurgy

PYRIMIDINE COMPOUND

#6 | 2025-10-23
US20250325541A1
Human necessities

METHODS OF DISPERSING ARIPIPRAZOLE INJECTABLE PREPARATIONS

#7 | 2025-10-16
US20250320453A1
Chemistry; metallurgy

MICROORGANISM BELONGING TO GENUS AKKERMANSIA

#8 | 2025-10-02
US20250304558A1
Chemistry; metallurgy

HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF EPILEPSY

#9 | 2025-08-07
US20250250243A1
Chemistry; metallurgy

OXAZOLE COMPOUND CRYSTAL

#10 | 2025-07-31
US20250241909A1
Human necessities

INJECTABLE FORMULATION

#11 | 2025-06-12
US20250191730A1
Physics

COMPUTER PROGRAM, AND INFORMATION PROCESSING DEVICE AND METHOD

#12 | 2025-06-05
US20250177385A1
Human necessities

COMBINATIONS COMPRISING BREXPIPRAZOLE OR A SALT THEREOF AND A SECOND DRUG FOR USE IN THE TREATMENT OF A CNS DISORDER

#13 | 2025-05-08
US20250144112A1
Human necessities

SUSPENSION FOR ORAL ADMINISTRATION COMPRISING AMORPHOUS TOLVAPTAN

#14 | 2025-05-01
US20250134872A1
Human necessities

ANTITUMOR COMPOSITION

#15 | 2025-04-24
US20250129029A1
Chemistry; metallurgy

ACRIDINE COMPOUND

#16 | 2025-04-24
US20250127813A1
Human necessities

COMBINATION DRUG

#17 | 2025-04-24
US20250127776A1
Human necessities

ORAL PHARMACEUTICAL COMPOSITION

#18 | 2025-04-17
US20250121065A1
Human necessities

INJECTABLE PREPARATION

#19 | 2025-03-27
US20250099459A1
Human necessities

PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF

#20 | 2025-03-13
US20250082631A1
Human necessities

SLEEP IMPROVING AGENT

#21 | 2025-02-27
US20250064745A1
Human necessities

FREEZE-DRIED ARIPIRAZOLE FORMULATION

#22 | 2025-02-20
US20250057835A1
Human necessities

ORAL PHARMACEUTICAL COMPOSITION CONTAINING HETEROCYCLIC COMPOUND

#23 | 2025-02-13
US20250051310A1
Chemistry; metallurgy

BENZAZEPINE DERIVATIVES

#24 | 2025-02-13
US20250049749A1
Human necessities

COMPOSITION FOR IMPROVING SLEEP QUALITY OR CONTROLLING AUTONOMIC NERVOUS SYSTEM

#25 | 2025-02-06
US20250042924A1
Chemistry; metallurgy

WATER-SOLUBLE PHYTIN

#26 | 2025-02-06 ✅ Patent 12,370,144 granted on 2025-07-29
US20250041225A1
Human necessities

CENTANAFADINE PHARMACEUTICAL FORMULATIONS, AND METHODS OF MAKING AND USING SAME

#27 | 2025-01-30
US20250031716A1
Human necessities

FROZEN DESSERT COMPOSITION

#28 | 2025-01-02
US20250002481A1
Chemistry; metallurgy

6-PYRIMIDIN-ISOINDOLE DERIVATIVE AS ERK1/2 INHIBITOR

#29 | 2024-12-19
US20240417376A1
Chemistry; metallurgy

4-(METHYLAMINOPHENOXY)PYRDIN-3-YL-BENZAMIDE DERIVATIVES FOR TREATING CANCER

#30 | 2024-12-19
US20240415774A1
Human necessities

DELAMANID-CONTAINING COMPOSITION

#31 | 2024-12-12
US20240409519A1
Chemistry; metallurgy

HYDROGENATED QUINOXALINES

#32 | 2024-12-05
US20240400520A1
Chemistry; metallurgy

5-METHYL-6-PHENYL-4,5-DIHYDRO-2H-PYRIDAZIN-3-ONE DERIVATIVE

#33 | 2024-11-14
US20240379241A1
Physics

INFORMATION PROVISION METHOD FOR PREDICTING HEALTH CONDITION OF CONSUMER AND SUPPORTING HEALTH MAINTENANCE AND IMPROVEMENT

#34 | 2024-11-14
US20240376435A1
Chemistry; metallurgy

KIDNEY ORGANOID AND METHOD FOR PRODUCING SAME

#35 | 2024-11-14
US20240376109A1
Chemistry; metallurgy

PYRAZOLO[1,5-A]PYRIMIDINE COMPOUND FOR THE TREATMENT OF DERMAL DISORDERS

#36 | 2024-11-07 ✅ Patent 12,655,137 granted on 2026-06-16
US20240368136A1
Chemistry; metallurgy

BENZOLACTAM COMPOUNDS AS PROTEIN KINASE INHIBITORS

#37 | 2024-11-07
US20240366573A1
Human necessities

OINTMENT CONTAINING AN OXAZOLE COMPOUND

#38 | 2024-10-03
US20240325348A1
Human necessities

KAEMPFEROL ANALOG-CONTAINING COMPOSITION

#39 | 2024-09-12
US20240299339A1
Human necessities

COMPOSITION FOR SUPPRESSING MUSCLE DAMAGE

#40 | 2024-09-05
US20240293364A1
Human necessities

BIOMARKERS FOR CANCER THERAPY USING MDM2 ANTAGONISTS

#41 | 2024-08-29
US20240286999A1
Chemistry; metallurgy

AZABICYCLO[3.1.0]HEXANE COMPOUND

#42 | 2024-08-22
US20240277703A1
Human necessities

TABLET COMPRISING 7-[4-(4-BENZO[B]THIOPHEN-4-YL-PIPERAZIN-1-YL)BUTOXY]-1H-QUINOLIN-2-ONE OR A SALT THEREOF

#43 | 2024-08-22
US20240277702A1
Human necessities

INJECTABLE FORMULATION

#44 | 2024-07-04
US20240216389A1
Human necessities

DRUG FOR PREVENTING AND/OR TREATING POLYCYSTIC KIDNEY DISEASE

#45 | 2024-07-04 ✅ Patent 12,564,335 granted on 2026-03-03
US20240215867A1
Human necessities

LOW POWER RECEIVER FOR IN VIVO CHANNEL SENSING AND INGESTIBLE SENSOR DETECTION WITH WANDERING FREQUENCY

#46 | 2024-06-27
US20240208999A1
Chemistry; metallurgy

HETEROCYCLIC COMPOUND

#47 | 2024-05-23 ✅ Patent 12,156,941 granted on 2024-12-03
US20240165030A1
Human necessities

Centanafadine pharmaceutical formulations, and methods of making and using same

#48 | 2024-05-16
US20240158380A1
Chemistry; metallurgy

AMORPHOUS FORM AND COMPOSITION CONTAINING SAID AMORPHOUS FORM

#49 | 2024-05-16
US20240156811A1
Human necessities

COMBINATIONS COMPRISING BREXPIPRAZOLE OR A SALT THEREOF AND A SECOND DRUG FOR USE IN THE TREATMENT OF A CNS DISORDER

#50 | 2024-05-09
US20240148699A1
Human necessities

OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION

#51 | 2024-05-02 ✅ Patent 12,528,771 granted on 2026-01-20
US20240140910A1
Chemistry; metallurgy

METHOD FOR PRODUCING CENTANAFADINE

#52 | 2024-04-25
US20240131169A1
Human necessities

CLIPTAC COMPOSITION

#53 | 2024-04-04
US20240109842A1
Chemistry; metallurgy

ACRYLAMIDE COMPOUNDS

#54 | 2024-03-07
US20240076275A1
Chemistry; metallurgy

OXAZOLE COMPOUND CRYSTAL

#55 | 2024-02-08
US20240041774A1
Human necessities

FREEZE-DRIED ARIPIPRAZOLE FORMULATION

#56 | 2023-12-07 ✅ Patent 12,016,927 granted on 2024-06-25
US20230390399A1
Human necessities

Injectable preparation

#57 | 2023-11-30
US20230381194A1
Human necessities

SUSPENSION FOR ORAL ADMINISTRATION COMPRISING AMORPHOUS TOLVAPTAN

#58 | 2023-10-26
US20230338337A1
Human necessities

BIOMARKERS FOR CANCER THERAPY USING MDM2 ANTAGONISTS

#59 | 2023-10-26 ✅ Patent 11,980,690 granted on 2024-05-14
US20230338293A1
Human necessities

Centanafadine pharmaceutical formulations, and methods of making and using same

#60 | 2023-10-26 ✅ Patent 11,957,642 granted on 2024-04-16
US20230338238A1
Human necessities

Internal substance supplier and method of producing molded product

#61 | 2023-10-12
US20230322812A1
Chemistry; metallurgy

CRYSTALLINE FORM OF HETEROBICYCLIC COMPOUND

#62 | 2023-10-12
US20230321113A1
Human necessities

PHARMACEUTICAL SOLID PREPARATION COMPRISING BENZAZEPINES AND PRODUCTION METHOD THEREOF

#63 | 2023-10-12
US20230321030A1
Human necessities

KAEMPFEROL AGLYCONE-CONTAINING EXTRACT

#64 | 2023-10-05
US20230313313A1
Chemistry; metallurgy

BIOMARKERS FOR CANCER THERAPY USING MDM2 ANTAGONISTS

#65 | 2023-09-28
US20230303981A1
Chemistry; metallurgy

BLADDER ORGANOID AND METHOD FOR PRODUCING SAME

#66 | 2023-09-28 ✅ Patent 12,195,496 granted on 2025-01-14
US20230303609A1
Chemistry; metallurgy

2′-deoxy-2′,2′-difluorotetrahydrouridines with high purity and methods of making the same

#67 | 2023-08-31
US20230270142A1
Human necessities

COMPOSITION CONTAINING EQUOL AND ORNITHINE

#68 | 2023-08-24
US20230265073A1
Chemistry; metallurgy

BENZAZEPINE DERIVATIVES

#69 | 2023-08-24 ✅ Patent 11,963,971 granted on 2024-04-23
US20230263818A1
Human necessities

Combination decitabine and cedazuridine solid oral dosage forms

#70 | 2023-07-06
US20230216595A1
Electricity

PHARMA-INFORMATICS SYSTEM

#71 | 2023-06-29
US20230203450A1
Chemistry; metallurgy

METHOD OF PRODUCING ORGANOID DERIVED FROM LUNG EPITHELIAL CELL OR LUNG CANCER CELL

#72 | 2023-06-15 ✅ Patent 12,196,674 granted on 2025-01-14
US20230184676A1
Physics

Detection device and detection method

#73 | 2023-05-25
US20230163864A1
Electricity

COMMUNICATION SYSTEM WITH PARTIAL POWER SOURCE

#74 | 2023-05-25
US20230157570A1
Human necessities

IN-BODY POWER SOURCE HAVING HIGH SURFACE AREA ELECTRODE

#75 | 2023-05-18 ✅ Patent 12,306,106 granted on 2025-05-20
US20230152234A1
Physics

Detection device

#76 | 2023-05-11
US20230146795A1
Human necessities

ENHANCEMENT OF ANTI-TUMOR ACTIVITY OF SHP2 INHIBITOR PYRIMIDINONE IN COMBINATION WITH NOVEL CANCER MEDICINES IN CANCERS

#77 | 2023-05-04
US20230139808A1
Chemistry; metallurgy

4-(METHYLAMINOPHENOXY)PYRDIN-3-YL-BENZAMIDE DERIVATIVES FOR TREATING CANCER

#78 | 2023-04-06 ✅ Patent 11,759,426 granted on 2023-09-19
US20230104529A1
Human necessities

Centanafadine pharmaceutical formulations, and methods of making and using same

#79 | 2023-03-09 ✅ Patent 11,793,419 granted on 2023-10-24
US20230076111A1
Human necessities

Methods for manufacturing capsules with ingestible event markers

#80 | 2023-03-02
US20230062476A1
Human necessities

GENETICALLY MODIFIED MEGAKARYOCYTE, MODIFIED PLATELET, AND METHODS RESPECTIVELY FOR PRODUCING SAID GENETICALLY MODIFIED MEGAKARYOCYTE AND SAID MODIFIED PLATELET

#81 | 2023-02-16 ✅ Patent 12,458,640 granted on 2025-11-04
US20230049719A1
Human necessities

PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS

#82 | 2023-02-16
US20230049327A1
Chemistry; metallurgy

DIHYDRATE OF BENZOTHIOPHENE COMPOUND OR OF A SALT THEREOF, AND PROCESS FOR PRODUCING THE SAME

#83 | 2023-02-16 ✅ Patent 11,703,519 granted on 2023-07-18
US20230048882A1
Physics

Temperature control system

#84 | 2023-02-02 ✅ Patent 12,643,943 granted on 2026-06-02
US20230036655A1
Chemistry; metallurgy

ANTI-GDF15 ANTIBODY

#85 | 2023-02-02
US20230034761A1
Human necessities

INGESTIBLE DEVICE WITH PHARMACEUTICAL PRODUCT

#86 | 2023-01-26
US20230027710A1
Physics

METHOD FOR PROVIDING SUPPORT TO MAINTAIN AND IMPROVE HEALTH OF CONSUMERS BY USING HEALTH PREDICTION MODEL THROUGH RECOGNITION OF THEIR HEALTH CONDITION, AND METHOD FOR PROVIDING INFORMATION

#87 | 2023-01-26
US20230021481A1
Physics

STANDARD SUBSTANCE FOR PSA QUANTIFICATION, PREPARATION METHOD THEREFOR, STANDARD SOLUTION FOR PSA QUANTIFICATION, AND PSA QUANTIFICATION METHOD

#88 | 2023-01-19 ✅ Patent 11,939,321 granted on 2024-03-26
US20230019032A1
Chemistry; metallurgy

Benzolactam compounds as protein kinase inhibitors

#89 | 2023-01-19 ✅ Patent 12,186,312 granted on 2025-01-07
US20230017155A1
Human necessities

Sleep improving agent

#90 | 2022-12-29 ✅ Patent 12,187,757 granted on 2025-01-07
US20220411457A1
Chemistry; metallurgy

2′-deoxy-2′,2′-difluorotetrahydrouridines with high purity and methods of making the same

#91 | 2022-12-29 ✅ Patent 11,840,512 granted on 2023-12-12
US20220411386A1
Chemistry; metallurgy

Oxazole compound crystal

#92 | 2022-12-08
US20220387464A1
Human necessities

INOSITOL PHOSPHATE-CONTAINING COMPOSITION

#93 | 2022-11-24
US20220370442A1
Human necessities

PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF

#94 | 2022-11-17 ✅ Patent 12,037,345 granted on 2024-07-16
US20220363693A1
Chemistry; metallurgy

Heterobicyclic compounds for inhibiting the activity of SHP2

#95 | 2022-11-03
US20220346664A1
Human necessities

INGESTION-RELATED BIOFEEDBACK AND PERSONALIZED MEDICAL THERAPY METHOD AND SYSTEM

#96 | 2022-10-20
US20220331311A1
Human necessities

TABLET COMPRISING 7-[4-(4-BENZO[B]THIOPHEN-4-YL-PIPERAZIN-1-YL)BUTOXY]-1H-QUINOLIN-2-ONE OR A SALT THEREOF

#97 | 2022-10-13
US20220326234A1
Physics

DETECTION METHOD AND DETECTION DEVICE

#98 | 2022-10-13
US20220323364A1
Human necessities

CONTROLLED ACTIVATION INGESTIBLE IDENTIFIER

#99 | 2022-10-06
US20220313602A1
Human necessities

MEDICAL TABLET, AND MANUFACTURING METHOD AND MANUFACTURING APPARATUS FOR MEDICAL TABLET

#100 | 2022-09-29 ✅ Patent 11,870,508 granted on 2024-01-09
US20220311474A1
Electricity

System for supply chain management

Also check out OTSUKA PHARMACEUTICAL CO., LTD.'s (Tokyo, Japan) applicant profile with 254 patent applications submitted.

AssigneeID:

1905 ⎘