Tokyo
Japan
640
2026-04-30
429
2025-07-29
These are the the leading inventors for applications assigned to OTSUKA PHARMACEUTICAL CO., LTD.:
OTSUKA PHARMACEUTICAL CO., LTD. based in Tokyo, JP has been assigned the rights to these inventions. The list includes both Pending Applications and Patent Grants:
TETRA-FUNCTIONAL CHEMICAL PROBE AND METHOD FOR IDENTIFYING TARGET MEMBRANE PROTEIN FROM LIVING CELL OR LIVING TISSUE BY USING SAID PROBE
#2 | 2026-04-30METHODS OF ADMINISTERING AN ARIPIPRAZOLE INJECTABLE PREPARATION
#3 | 2026-04-16PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS
#4 | 2026-01-29PHARMACEUTICAL COMPOSITIONS COMPRISING A QUINOLONE COMPOUND FOR IRRITABLE BOWEL SYNDROME
#5 | 2025-11-27PYRIMIDINE COMPOUND
#6 | 2025-10-23METHODS OF DISPERSING ARIPIPRAZOLE INJECTABLE PREPARATIONS
#7 | 2025-10-16MICROORGANISM BELONGING TO GENUS AKKERMANSIA
#8 | 2025-10-02HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF EPILEPSY
#9 | 2025-08-07OXAZOLE COMPOUND CRYSTAL
#10 | 2025-07-31INJECTABLE FORMULATION
#11 | 2025-06-12COMPUTER PROGRAM, AND INFORMATION PROCESSING DEVICE AND METHOD
#12 | 2025-06-05COMBINATIONS COMPRISING BREXPIPRAZOLE OR A SALT THEREOF AND A SECOND DRUG FOR USE IN THE TREATMENT OF A CNS DISORDER
#13 | 2025-05-08SUSPENSION FOR ORAL ADMINISTRATION COMPRISING AMORPHOUS TOLVAPTAN
#14 | 2025-05-01ANTITUMOR COMPOSITION
#15 | 2025-04-24ACRIDINE COMPOUND
#16 | 2025-04-24COMBINATION DRUG
#17 | 2025-04-24ORAL PHARMACEUTICAL COMPOSITION
#18 | 2025-04-17INJECTABLE PREPARATION
#19 | 2025-03-27PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF
#20 | 2025-03-13SLEEP IMPROVING AGENT
#21 | 2025-02-27FREEZE-DRIED ARIPIRAZOLE FORMULATION
#22 | 2025-02-20ORAL PHARMACEUTICAL COMPOSITION CONTAINING HETEROCYCLIC COMPOUND
#23 | 2025-02-13BENZAZEPINE DERIVATIVES
#24 | 2025-02-13COMPOSITION FOR IMPROVING SLEEP QUALITY OR CONTROLLING AUTONOMIC NERVOUS SYSTEM
#25 | 2025-02-06WATER-SOLUBLE PHYTIN
#26 | 2025-02-06 ✅ Patent 12,370,144 granted on 2025-07-29CENTANAFADINE PHARMACEUTICAL FORMULATIONS, AND METHODS OF MAKING AND USING SAME
#27 | 2025-01-30FROZEN DESSERT COMPOSITION
#28 | 2025-01-026-PYRIMIDIN-ISOINDOLE DERIVATIVE AS ERK1/2 INHIBITOR
#29 | 2024-12-194-(METHYLAMINOPHENOXY)PYRDIN-3-YL-BENZAMIDE DERIVATIVES FOR TREATING CANCER
#30 | 2024-12-19DELAMANID-CONTAINING COMPOSITION
#31 | 2024-12-12HYDROGENATED QUINOXALINES
#32 | 2024-12-055-METHYL-6-PHENYL-4,5-DIHYDRO-2H-PYRIDAZIN-3-ONE DERIVATIVE
#33 | 2024-11-14INFORMATION PROVISION METHOD FOR PREDICTING HEALTH CONDITION OF CONSUMER AND SUPPORTING HEALTH MAINTENANCE AND IMPROVEMENT
#34 | 2024-11-14KIDNEY ORGANOID AND METHOD FOR PRODUCING SAME
#35 | 2024-11-14PYRAZOLO[1,5-A]PYRIMIDINE COMPOUND FOR THE TREATMENT OF DERMAL DISORDERS
#36 | 2024-11-07 ✅ Patent 12,655,137 granted on 2026-06-16BENZOLACTAM COMPOUNDS AS PROTEIN KINASE INHIBITORS
#37 | 2024-11-07OINTMENT CONTAINING AN OXAZOLE COMPOUND
#38 | 2024-10-03KAEMPFEROL ANALOG-CONTAINING COMPOSITION
#39 | 2024-09-12COMPOSITION FOR SUPPRESSING MUSCLE DAMAGE
#40 | 2024-09-05BIOMARKERS FOR CANCER THERAPY USING MDM2 ANTAGONISTS
#41 | 2024-08-29AZABICYCLO[3.1.0]HEXANE COMPOUND
#42 | 2024-08-22TABLET COMPRISING 7-[4-(4-BENZO[B]THIOPHEN-4-YL-PIPERAZIN-1-YL)BUTOXY]-1H-QUINOLIN-2-ONE OR A SALT THEREOF
#43 | 2024-08-22INJECTABLE FORMULATION
#44 | 2024-07-04DRUG FOR PREVENTING AND/OR TREATING POLYCYSTIC KIDNEY DISEASE
#45 | 2024-07-04 ✅ Patent 12,564,335 granted on 2026-03-03LOW POWER RECEIVER FOR IN VIVO CHANNEL SENSING AND INGESTIBLE SENSOR DETECTION WITH WANDERING FREQUENCY
#46 | 2024-06-27HETEROCYCLIC COMPOUND
#47 | 2024-05-23 ✅ Patent 12,156,941 granted on 2024-12-03Centanafadine pharmaceutical formulations, and methods of making and using same
#48 | 2024-05-16AMORPHOUS FORM AND COMPOSITION CONTAINING SAID AMORPHOUS FORM
#49 | 2024-05-16COMBINATIONS COMPRISING BREXPIPRAZOLE OR A SALT THEREOF AND A SECOND DRUG FOR USE IN THE TREATMENT OF A CNS DISORDER
#50 | 2024-05-09OXAZOLE COMPOUND AND PHARMACEUTICAL COMPOSITION
#51 | 2024-05-02 ✅ Patent 12,528,771 granted on 2026-01-20METHOD FOR PRODUCING CENTANAFADINE
#52 | 2024-04-25CLIPTAC COMPOSITION
#53 | 2024-04-04ACRYLAMIDE COMPOUNDS
#54 | 2024-03-07OXAZOLE COMPOUND CRYSTAL
#55 | 2024-02-08FREEZE-DRIED ARIPIPRAZOLE FORMULATION
#56 | 2023-12-07 ✅ Patent 12,016,927 granted on 2024-06-25Injectable preparation
#57 | 2023-11-30SUSPENSION FOR ORAL ADMINISTRATION COMPRISING AMORPHOUS TOLVAPTAN
#58 | 2023-10-26BIOMARKERS FOR CANCER THERAPY USING MDM2 ANTAGONISTS
#59 | 2023-10-26 ✅ Patent 11,980,690 granted on 2024-05-14Centanafadine pharmaceutical formulations, and methods of making and using same
#60 | 2023-10-26 ✅ Patent 11,957,642 granted on 2024-04-16Internal substance supplier and method of producing molded product
#61 | 2023-10-12CRYSTALLINE FORM OF HETEROBICYCLIC COMPOUND
#62 | 2023-10-12PHARMACEUTICAL SOLID PREPARATION COMPRISING BENZAZEPINES AND PRODUCTION METHOD THEREOF
#63 | 2023-10-12KAEMPFEROL AGLYCONE-CONTAINING EXTRACT
#64 | 2023-10-05BIOMARKERS FOR CANCER THERAPY USING MDM2 ANTAGONISTS
#65 | 2023-09-28BLADDER ORGANOID AND METHOD FOR PRODUCING SAME
#66 | 2023-09-28 ✅ Patent 12,195,496 granted on 2025-01-142′-deoxy-2′,2′-difluorotetrahydrouridines with high purity and methods of making the same
#67 | 2023-08-31COMPOSITION CONTAINING EQUOL AND ORNITHINE
#68 | 2023-08-24BENZAZEPINE DERIVATIVES
#69 | 2023-08-24 ✅ Patent 11,963,971 granted on 2024-04-23Combination decitabine and cedazuridine solid oral dosage forms
#70 | 2023-07-06PHARMA-INFORMATICS SYSTEM
#71 | 2023-06-29METHOD OF PRODUCING ORGANOID DERIVED FROM LUNG EPITHELIAL CELL OR LUNG CANCER CELL
#72 | 2023-06-15 ✅ Patent 12,196,674 granted on 2025-01-14Detection device and detection method
#73 | 2023-05-25COMMUNICATION SYSTEM WITH PARTIAL POWER SOURCE
#74 | 2023-05-25IN-BODY POWER SOURCE HAVING HIGH SURFACE AREA ELECTRODE
#75 | 2023-05-18 ✅ Patent 12,306,106 granted on 2025-05-20Detection device
#76 | 2023-05-11ENHANCEMENT OF ANTI-TUMOR ACTIVITY OF SHP2 INHIBITOR PYRIMIDINONE IN COMBINATION WITH NOVEL CANCER MEDICINES IN CANCERS
#77 | 2023-05-044-(METHYLAMINOPHENOXY)PYRDIN-3-YL-BENZAMIDE DERIVATIVES FOR TREATING CANCER
#78 | 2023-04-06 ✅ Patent 11,759,426 granted on 2023-09-19Centanafadine pharmaceutical formulations, and methods of making and using same
#79 | 2023-03-09 ✅ Patent 11,793,419 granted on 2023-10-24Methods for manufacturing capsules with ingestible event markers
#80 | 2023-03-02GENETICALLY MODIFIED MEGAKARYOCYTE, MODIFIED PLATELET, AND METHODS RESPECTIVELY FOR PRODUCING SAID GENETICALLY MODIFIED MEGAKARYOCYTE AND SAID MODIFIED PLATELET
#81 | 2023-02-16 ✅ Patent 12,458,640 granted on 2025-11-04PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS
#82 | 2023-02-16DIHYDRATE OF BENZOTHIOPHENE COMPOUND OR OF A SALT THEREOF, AND PROCESS FOR PRODUCING THE SAME
#83 | 2023-02-16 ✅ Patent 11,703,519 granted on 2023-07-18Temperature control system
#84 | 2023-02-02 ✅ Patent 12,643,943 granted on 2026-06-02ANTI-GDF15 ANTIBODY
#85 | 2023-02-02INGESTIBLE DEVICE WITH PHARMACEUTICAL PRODUCT
#86 | 2023-01-26METHOD FOR PROVIDING SUPPORT TO MAINTAIN AND IMPROVE HEALTH OF CONSUMERS BY USING HEALTH PREDICTION MODEL THROUGH RECOGNITION OF THEIR HEALTH CONDITION, AND METHOD FOR PROVIDING INFORMATION
#87 | 2023-01-26STANDARD SUBSTANCE FOR PSA QUANTIFICATION, PREPARATION METHOD THEREFOR, STANDARD SOLUTION FOR PSA QUANTIFICATION, AND PSA QUANTIFICATION METHOD
#88 | 2023-01-19 ✅ Patent 11,939,321 granted on 2024-03-26Benzolactam compounds as protein kinase inhibitors
#89 | 2023-01-19 ✅ Patent 12,186,312 granted on 2025-01-07Sleep improving agent
#90 | 2022-12-29 ✅ Patent 12,187,757 granted on 2025-01-072′-deoxy-2′,2′-difluorotetrahydrouridines with high purity and methods of making the same
#91 | 2022-12-29 ✅ Patent 11,840,512 granted on 2023-12-12Oxazole compound crystal
#92 | 2022-12-08INOSITOL PHOSPHATE-CONTAINING COMPOSITION
#93 | 2022-11-24PROPHYLACTIC AND/OR THERAPEUTIC AGENT FOR BEHAVIORAL AND PSYCHOLOGICAL SYMPTOMS ASSOCIATED WITH NEURODEGENERATIVE DISEASE OR IMPULSIVE SYMPTOMS ASSOCIATED WITH MENTAL DISEASE CONTAINING BREXPIPRAZOLE OR SALT THEREOF
#94 | 2022-11-17 ✅ Patent 12,037,345 granted on 2024-07-16Heterobicyclic compounds for inhibiting the activity of SHP2
#95 | 2022-11-03INGESTION-RELATED BIOFEEDBACK AND PERSONALIZED MEDICAL THERAPY METHOD AND SYSTEM
#96 | 2022-10-20TABLET COMPRISING 7-[4-(4-BENZO[B]THIOPHEN-4-YL-PIPERAZIN-1-YL)BUTOXY]-1H-QUINOLIN-2-ONE OR A SALT THEREOF
#97 | 2022-10-13DETECTION METHOD AND DETECTION DEVICE
#98 | 2022-10-13CONTROLLED ACTIVATION INGESTIBLE IDENTIFIER
#99 | 2022-10-06MEDICAL TABLET, AND MANUFACTURING METHOD AND MANUFACTURING APPARATUS FOR MEDICAL TABLET
#100 | 2022-09-29 ✅ Patent 11,870,508 granted on 2024-01-09System for supply chain management
Also check out OTSUKA PHARMACEUTICAL CO., LTD.'s (Tokyo, Japan) applicant profile with 254 patent applications submitted.
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