Berlin
Germany
545
2026-01-15
377
2025-11-25
These are the the leading inventors for applications assigned to Bayer Pharma Aktiengesellschaft:
Bayer Pharma Aktiengesellschaft based in Berlin, DE has been assigned the rights to these inventions. The list includes both Pending Applications and Patent Grants:
METHOD FOR THE PREPARATION OF (4S)-4-(4-CYANO-2-METHOXYPHENYL)-5-ETHOXY-2,8-DIMETHYL-1,4-DIHYDRO-1-6-NAPHTHYRIDINE-3-CARBOX-AMIDE BY RACEMATE SEPARATION BY MEANS OF DIASTEREOMERIC TARTARIC ACID ESTERS
#2 | 2025-11-06METHOD FOR THE PREPARATION OF (4S)-4-(4-CYANO-2-METHOXYPHENYL)-5-ETHOXY-2,8-DIMETHYL-1,4-DIHYDRO-1-6-NAPHTHYRIDINE-3-CARBOX-AMIDE BY RACEMATE SEPARATION BY MEANS OF DIASTEREOMERIC TARTARIC ACID ESTERS
#3 | 2025-05-15DIAZABICYCLIC SUBSTITUTED IMIDAZOPYRIMIDINES AND THEIR USE FOR THE TREATMENT OF BREATHING DISORDERS
#4 | 2025-04-10 ✅ Patent 12,478,696 granted on 2025-11-25GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING
#5 | 2025-01-30 ✅ Patent 12,559,473 granted on 2026-02-24SUBSTITUTED INDAZOLES, METHODS FOR THE PRODUCTION THEREOF, PHARMACEUTICAL PREPARATIONS THAT CONTAIN SAID NEW SUBSTITUTED INDAZOLES, AND USE OF SAID NEW SUBSTITUTED INDAZOLES TO PRODUCE DRUGS
#6 | 2024-11-21COMBINATIONS OF COPANLISIB WITH ANTI-PD-1 ANTIBODY
#7 | 2024-11-14METHOD FOR THE PREPARATION OF (4S)-4-(4-CYANO-2-METHOXYPHENYL)-5-ETHOXY-2,8-DIMETHYL-1,4-DIHYDRO-1-6-NAPHTHYRIDINE-3-CARBOX-AMIDE BY RACEMATE SEPARATION BY MEANS OF DIASTEREOMERIC TARTARIC ACID ESTERS
#8 | 2024-11-07COMPOUNDS, COMPOSITIONS AND METHODS FOR CANCER PATIENT STRATIFICATION AND CANCER TREATMENT
#9 | 2024-09-05 ✅ Patent 12,522,594 granted on 2026-01-132-HETEROARYL-3-OXO-2,3-DIHYDROPYRIDAZINE-4-CARBOXAMIDES FOR THE TREATMENT OF CANCER
#10 | 2024-08-01 ✅ Patent 12,303,573 granted on 2025-05-20Formulation of contrast media and process of preparation thereof
#11 | 2024-06-066-PHENYL-4,5-DIHYDROPYRIDAZIN-3(2H)-ONE DERIVATIVES AS PDE3A AND PDE3B INHIBITORS FOR TREATING CANCER
#12 | 2024-05-09 ✅ Patent 12,138,256 granted on 2024-11-12Treatment of cardiopulmonary disorders
#13 | 2024-04-18 ✅ Patent 12,503,491 granted on 2025-12-23MASP INHIBITORY COMPOUNDS AND USES THEREOF
#14 | 2024-04-11 ✅ Patent 12,202,805 granted on 2025-01-21Process for preparing (5S)-{[2-(4-carboxyphenyl)ethyl] |2-(2-{|3-chloro-4'-(trifluoromethyl)biphenyl-4-yl]methoxy}phenyl)ethyl]aminol-5,6,7,8-tetrahydroquinoline-2-carboxylic acid and its crystalline forms for use as pharmaceutically active compound
#15 | 2023-12-28N-[2-({4-[3-(ANILINO)-4-OXO-4,5,6,7-TETRAHYDRO-1H-PYRROLO[3,2-C]PYRIDIN-2-YL]PYRIDIN-3-YL)OXY)ETHYL]PROP-2-ENAMIDE DERIVATIVES AND SIMILAR COMPOUNDS AS EGFR INHIBITORS FOR THE TREATMENT OF CANCER
#16 | 2023-11-16 ✅ Patent 12,486,248 granted on 2025-12-022,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH
#17 | 2023-11-02COMBINATION of ATR KINASE INHIBITORS and PD-1/PD-L1 INHIBITORS
#18 | 2023-08-31 ✅ Patent 12,239,630 granted on 2025-03-04Carboxylic acid aromatic amides as antagonists of bradykinin B1 receptor
#19 | 2023-06-29 ✅ Patent 11,998,539 granted on 2024-06-04Substituted aminoquinolones as DGKalpha inhibitors for immune activation
#20 | 2023-06-08 ✅ Patent 12,006,303 granted on 2024-06-11Substituted indazoles, methods for the production thereof, pharmaceutical preparations that contain said substituted indazoles, and use of said substituted indazoles to produce drugs
#21 | 2023-05-11 ✅ Patent 12,478,621 granted on 2025-11-25SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION
#22 | 2023-04-20 ✅ Patent 11,795,164 granted on 2023-10-242-heteroaryl-3-oxo-2,3-dihydropyridazine-4-carboxamides for the treatment of cancer
#23 | 2023-04-13[1,2,4]TRIAZOLO[1,5-C]QUINAZOLIN-5-AMINES
#24 | 2023-04-13 ✅ Patent 11,891,404 granted on 2024-02-06Substituted macrocyclic indole derivatives
#25 | 2023-03-23 ✅ Patent 11,905,270 granted on 2024-02-20Carboxylic acid aromatic amides as antagonists of bradykinin B1 receptor
#26 | 2023-03-02SUBSTITUTED 6-(1H-PYRAZOL-1-YL)PYRIMIDIN-4-AMINE DERIVATIVES AND USES THEREOF
#27 | 2023-03-02SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION
#28 | 2023-03-02SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION
#29 | 2023-02-09 ✅ Patent 12,023,319 granted on 2024-07-02Carboxylic acid aromatic amides
#30 | 2023-02-09 ✅ Patent 12,144,865 granted on 2024-11-19Antibody drug conjugates with enzymatically cleavable groups
#31 | 2023-01-19 ✅ Patent 12,258,323 granted on 2025-03-25Dihydrooxadiazinones
#32 | 2023-01-19ANALOGUES OF 3-(5-METHYL-1,3-THIAZOL-2-YL)-N-{(1R)-1-[2-(TRIFLUORO-METHYL)PYRIMIDIN-5-YL]ETHYL}BENZAMIDE
#33 | 2022-12-15 ✅ Patent 11,773,070 granted on 2023-10-03Dihydrooxadiazinones
#34 | 2022-12-08 ✅ Patent 12,006,304 granted on 2024-06-11Substituted indazoles, methods for the production thereof, pharmaceutical preparations that contain said substituted indazoles, and use of said substituted indazoles to produce drugs
#35 | 2022-11-10PROCESS FOR PREPARING BENZOTHIOPHEN-2YL BORONATE
#36 | 2022-11-08 ✅ Patent 11,492,358 granted on 2022-11-08Macrocyclic indole derivatives
#37 | 2022-10-25 ✅ Patent 11,478,451 granted on 2022-10-25Macrocyclic chlorine substituted indole derivatives
#38 | 2022-10-13 ✅ Patent 11,524,938 granted on 2022-12-13Aromatic sulfonamide derivatives
#39 | 2022-09-08 ✅ Patent 12,152,041 granted on 2024-11-26Macrocyclic fluorine substituted indole derivatives
#40 | 2022-09-012-METHYL-AZA-QUINAZOLINES
#41 | 2022-08-25 ✅ Patent 11,643,469 granted on 2023-05-09Specific antibody-drug-conjugates (ADCs) with KSP inhibitors and anti-CD123-antibodies
#42 | 2022-08-25 ✅ Patent 11,691,986 granted on 2023-07-04PTEFB inhibiting macrocyclic compounds
#43 | 2022-08-18SUBSTITUTED DIAZAHETERO-BICYCLIC COMPOUNDS AND THEIR USE
#44 | 2022-08-18ORALLY ADMINISTRABLE MODIFIED-RELEASE PHARMACEUTICAL DOSAGE FORM
#45 | 2022-08-11 ✅ Patent 11,992,481 granted on 2024-05-28Use of 2-substituted indazoles for the treatment and prophylaxis of autoimmune diseases
#46 | 2022-08-04COMBINATIONS OF INHIBITORS OF IRAK4 WITH INHIBITORS OF BTK
#47 | 2022-08-04COMBINATION CONTAINING SGC ACTIVATORS AND MINERALOCORTICOID RECEPTOR ANTAGONISTS
#48 | 2022-07-282-METHYL-QUINAZOLINES
#49 | 2022-07-28Method for Producing (3S)-3-(4-chloro-3-{[(2S,3R)-2-(4-chlorophenyl)-4,4,4-trifluoro-3-methylbutanoyl]amino}phenyl)-3-cyclo-propylpropanoic Acid and the Crystalline Form Thereof for Use as a Pharmaceutical Ingredient
#50 | 2022-06-30 ✅ Patent 12,459,916 granted on 2025-11-04SUBSTITUTED INDAZOLES USEFUL FOR TREATMENT AND PREVENTION OF ALLERGIC AND/OR INFLAMMATORY DISEASES IN ANIMALS
#51 | 2022-05-24 ✅ Patent 11,339,157 granted on 2022-05-244H-pyrrolo[3,2-c]pyridin-4-one derivatives
#52 | 2022-05-19 ✅ Patent 12,152,006 granted on 2024-11-26Process for preparing 4-amino-5-methylpyridone
#53 | 2022-05-19 ✅ Patent 12,358,877 granted on 2025-07-15SYNTHESIS OF 4-AMINO-5-METHYL-1H-PYRIDIN-2(1H)-ON (INTERMEDIATE COMPOUND FOR THE SYNTHESIS OF THE MR ANTAGONIST FINERENONE) FROM 2-CHLORO-5-METHYL-4-NITRO-PYRIDINE-1-OXIDE USING THE INTERMEDIATE COMPOUND 2-CHLORO-5-METHYL-4-PYRIDINAMINE
#54 | 2022-05-12RADIO-PHARMACEUTICAL COMPLEXES
#55 | 2022-05-05 ✅ Patent 11,713,304 granted on 2023-08-012,4,5-trisubstituted 1,2,4-triazolones useful as inhibitors of DHODH
#56 | 2022-03-31THE MONOHYDRATE OF ROGARATINIB HYDROCHLORIDE AND SOLID STATES THEREOF
#57 | 2022-03-247-SUBSTITUTED 1-ARYL-NAPHTHYRIDINE-3-CARBOXYLIC ACID AMIDES AND USE THEREOF
#58 | 2022-03-10COMPOSITIONS AND METHODS FOR CANCER EXPRESSING PDE3A OR SLFN12
#59 | 2022-01-27 ✅ Patent 12,427,131 granted on 2025-09-30STIMULATORS AND/OR ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE (SGC) IN COMBINATION WITH AN INHIBITOR OF NEUTRAL ENDOPEPTIDASE (NEP INHIBITOR) AND/OR AN ANGIOTENSIN AII ANTAGONIST AND THE USE THEREOF
#60 | 2022-01-20 ✅ Patent 12,180,227 granted on 2024-12-31Diazabicyclic substituted imidazopyrimidines and their use for the treatment of breathing disorders
#61 | 2022-01-20 ✅ Patent 11,478,554 granted on 2022-10-25Antibody drug conjugates (ADCS) having enzymatically cleavable groups
#62 | 2022-01-20COMPOUNDS AND METHODS USEFUL FOR TREATING OR PREVENTING HEMATOLOGICAL CANCERS
#63 | 2021-12-30 ✅ Patent 11,976,334 granted on 2024-05-07Inhibitor of ATR kinase for use in a method of treating a hyper-proliferative disease
#64 | 2021-12-30INHIBITORS AND ANTAGONISTS OF GPR84 FOR THE TREATMENT OF ENDOMETRIOSIS
#65 | 2021-12-23REVERSAL AGENTS FOR NEUTRALIZING THE THERAPEUTIC ACTIVITY OF ANTI-FXIA ANTIBODIES
#66 | 2021-12-23PROCESS FOR PRODUCING PHARMACEUTICAL DOSAGE FORMS CONTAINING TASK-1 AND TASK-3 CHANNEL INHIBITORS, AND THE USE OF SAME IN BREATHING DISORDER THERAPY
#67 | 2021-10-14 ✅ Patent 11,319,324 granted on 2022-05-03Pyrazolo-pyrrolo-pyrimidine-dione derivatives as P2X3 inhibitors
#68 | 2021-09-23 ✅ Patent 11,401,278 granted on 2022-08-02Macrocyclic indole derivatives
#69 | 2021-09-16PHARMACEUTICAL DOSAGE FORM WHICH CAN BE ADMINISTERED ORALLY AND HAS MODIFIED RELEASE
#70 | 2021-09-09 ✅ Patent 11,447,504 granted on 2022-09-20Macrocyclic chlorine substituted indole derivatives
#71 | 2021-08-26 ✅ Patent 11,472,803 granted on 2022-10-187-substituted 1-aryl-naphthyridine-3-carboxylic acid amides and use thereof
#72 | 2021-08-19 ✅ Patent 12,258,343 granted on 2025-03-25Method for preparing 2-[(3R)-3-methylmorpholin-4-yl]-4-[1-methyl-1H-pyrazol-5-yl)-8-(1H-pyrazol-5-yl)-1,7-naphthyridine
#73 | 2021-08-19 ✅ Patent 11,806,404 granted on 2023-11-07Site specific homogeneous with KSP inhibitors
#74 | 2021-08-12 ✅ Patent 11,667,675 granted on 2023-06-06MASP inhibitory compounds and uses thereof
#75 | 2021-08-05 ✅ Patent 12,053,476 granted on 2024-08-06Compounds, compositions and methods for cancer patient stratification and cancer treatment
#76 | 2021-07-29SPECIFIC ANTIBODY-DRUG-CONJUGATES (ADCS) WITH KSP INHIBITORS AND ANTI-CD123-ANTIBODIES
#77 | 2021-07-22 ✅ Patent 11,814,369 granted on 2023-11-14HIGH RELAXIVITY GADOLINIUM CHELATE COMPOUNDS FOR USE IN MAGNETIC RESONANCE IMAGING
#78 | 2021-07-221,3-THIAZOL-2-YL SUBSTITUTED BENZAMIDES FOR THE TREATMENT OF DISEASES ASSOCIATED WITH NERVE FIBER SENSITIZATION
#79 | 2021-07-221,3-THIAZOL-2-YL SUBSTITUTED BENZAMIDES FOR THE TREATMENT OF DISEASES ASSOCIATED WITH NERVE FIBER SENSITIZATION
#80 | 2021-06-24 ✅ Patent 11,787,797 granted on 2023-10-174,5-annulated 1,2,4-triazolones
#81 | 2021-06-17 ✅ Patent 11,230,540 granted on 2022-01-25Substituted triazole derivatives and uses thereof
#82 | 2021-06-17 ✅ Patent 11,332,435 granted on 2022-05-17Method for producing (3S)-3-(4-chloro-3-{[(2S,3R)-2-(4- chlorophenyl)-4,4,4-trifluoro-3-methylbutanoyl]amino}phenyl)-3-cyclo-propylpropanoic acid and the crystalline form thereof for use as a pharmaceutical ingredient
#83 | 2021-06-03 ✅ Patent 12,054,481 granted on 2024-08-06Method for the preparation of (4S)-4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1-6-naphthyridine-3-carbox-amide by racemate separation by means of diastereomeric tartaric acid esters
#84 | 2021-05-20 ✅ Patent 11,884,660 granted on 2024-01-30Substituted oxopyridine derivative
#85 | 2021-05-06PROLACTIN RECEPTOR ANTIBODY FOR MALE AND FEMALE PATTERN HAIR LOSS
#86 | 2021-05-06 ✅ Patent 11,690,911 granted on 2023-07-04Combination of ATR kinase inhibitors and PD-1/PD-L1 inhibitors
#87 | 2021-05-06 ✅ Patent 11,660,301 granted on 2023-05-30Combination of ATR kinase inhibitors with PARP inhibitors
#88 | 2021-04-29 ✅ Patent 11,684,621 granted on 2023-06-27Combination containing sGC stimulators and mineralocorticoid receptor antagonists
#89 | 2021-04-22 ✅ Patent 11,344,519 granted on 2022-05-31Orally administrable modified-release pharmaceutical dosage form
#90 | 2021-03-25USE OF 2-SUBSTITUTED INDAZOLES FOR THE TREATMENT AND PROPHYLAXIS OF AUTOIMMUNE DISEASES
#91 | 2021-03-25 ✅ Patent 11,311,520 granted on 2022-04-26Substituted dihydroimidazopyridinediones as MKNK1 and MKNK2 inhibitors
#92 | 2021-03-18 ✅ Patent 11,286,263 granted on 2022-03-29Macrocyclic fluorine substituted indole derivatives
#93 | 2021-02-25SUBSTITUTED INDAZOLES, METHODS FOR THE PRODUCTION THEREOF, PHARMACEUTICAL PREPARATIONS THAT CONTAIN SAID NEW SUBSTITUTED INDAZOLES, AND USE OF SAID NEW SUBSTITUTED INDAZOLES TO PRODUCE DRUGS
#94 | 2021-02-184-(3-AMINO-6-FLUORO-1H-INDAZOL-5-YL)-1,2,6-TRIMETHYL-1,4-DIHYDROPYRIDINE-3,5-DIC ARBONITRILE COMPOUNDS FOR TREATING HYPERPROLIFERATIVE DISORDERS
#95 | 2021-02-04 ✅ Patent 11,365,179 granted on 2022-06-21Method for the preparation of a 2,4,5-trisubstituted 1,2,4-triazolone
#96 | 2021-01-28SUBSTITUTED DIAZAHETERO-BICYCLIC COMPOUNDS AND THEIR USE
#97 | 2021-01-28METHOD FOR THE PREPARATION OF THE METABOLITES OF (4S)- AND (4R)-4-(4-CYANO-2-METHOXYPHENYL)-5-ETHOXY-2,8-DIMETHYL-1,4-DIHYDRO-1,6-NAPHTHYRIDINE-3-CARBOXAMIDE AND THE USE THEREOF
#98 | 2021-01-28REDUCING THE RISK OF CARDIOVASCULAR EVENTS
#99 | 2021-01-21 ✅ Patent 11,701,347 granted on 2023-07-18Use of 5-fluoro-4-(4-fluoro-2-methoxyphenyl)-N-{4-[(S-methylsulfonimidoyl)methyl]pyridin-2-yl}pyridin-2-amine for treating diffuse large B-cell lymphoma
#100 | 2021-01-14 ✅ Patent 11,390,592 granted on 2022-07-19Method for producing the crystalline form of modification a of calcobutrol
Also check out Bayer Pharma Aktiengesellschaft's (Berlin, Germany) applicant profile with 339 patent applications submitted.
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