Assignee profile:

Exelixis, Inc.

City:

Alameda, California

Country:

United States

Published Applications:

65

Last publication date:

2026-06-04

Patent Grants:

55

Last grant date:

2025-04-15

Top Inventors for applications by Exelixis, Inc.

These are the the leading inventors for applications assigned to Exelixis, Inc.:

Recent patent applications by Exelixis, Inc.

Exelixis, Inc. based in Alameda, US has been assigned the rights to these inventions. The list includes both Pending Applications and Patent Grants:

#1 | 2026-06-04
US20260152498A1
Chemistry; metallurgy

4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[4,3-c]PYRIDINE COMPOUNDS AND DERIVATIVES AS USP1 INHIBITORS

#2 | 2025-10-23
US20250326858A1
Chemistry; metallurgy

5T4 BINDING AGENTS AND USES THEREOF

#3 | 2025-09-25
US20250295803A1
Human necessities

5T4 ANTIBODY-DRUG CONJUGATES AND USES THEREOF

#4 | 2025-06-19
US20250197502A1
Chemistry; metallurgy

MULTISPECIFIC BINDING AGENTS AND USES THEREOF

#5 | 2025-03-27
US20250099604A1
Human necessities

PHARMACEUTICAL COMPOSITIONS COMPRISING ANTI-TISSUE FACTOR ANTIBODY-DRUG CONJUGATES

#6 | 2025-03-13 βœ… Patent 12,275,706 granted on 2025-04-15
US20250084037A1
Chemistry; metallurgy

Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-Nβ€²-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer

#7 | 2024-11-28
US20240392002A1
Chemistry; metallurgy

ANTI-ROR ANTIBODY CONSTRUCTS

#8 | 2024-06-13 βœ… Patent 12,128,039 granted on 2024-10-29
US20240189298A1
Human necessities

Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds

#9 | 2024-01-11
US20240010751A1
Chemistry; metallurgy

MULTISPECIFIC BINDING AGENTS AND USES THEREOF

#10 | 2024-01-11 βœ… Patent 12,227,481 granted on 2025-02-18
US20240010621A1
Chemistry; metallurgy

Crystalline solid forms of salts of N-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}-N'-(4-fluorophenyl) cyclopropane-1,1-dicarboxamide, processes for making, and methods of use

#11 | 2023-11-30 βœ… Patent 12,264,161 granted on 2025-04-01
US20230382917A1
Chemistry; metallurgy

Heterocyclic adenosine receptor antagonists

#12 | 2023-11-30 βœ… Patent 12,486,233 granted on 2025-12-02
US20230382867A1
Chemistry; metallurgy

CRYSTALLINE SOLID FORMS OF N-{4-[(6,7-DIMETHOXYQUINOLIN-4-YL)OXY]PHENYL}-N'-(4-FLUOROPHENYL) CYCLOPROPANE-1,1-DICARBOXAMIDE, PROCESSES FOR MAKING, AND METHODS OF USE

#13 | 2023-11-23 βœ… Patent 12,195,475 granted on 2025-01-14
US20230374024A1
Chemistry; metallurgy

Compounds for the treatment of kinase-dependent disorders

#14 | 2023-11-09
US20230357391A1
Chemistry; metallurgy

CD47 BINDING AGENTS AND USES THEREOF

#15 | 2023-09-28
US20230303699A1
Chemistry; metallurgy

PD-L1 BINDING AGENTS AND USES THEREOF

#16 | 2023-09-28 βœ… Patent 11,969,419 granted on 2024-04-30
US20230301980A1
Human necessities

Method of treating cancer

#17 | 2023-09-28 βœ… Patent 12,016,854 granted on 2024-06-25
US20230301978A1
Human necessities

Liquid dosage forms to treat cancer

#18 | 2023-06-22 βœ… Patent 12,497,367 granted on 2025-12-16
US20230192619A1
Chemistry; metallurgy

Processes for the Preparation of a Kinase Inhibitor

#19 | 2023-02-09 βœ… Patent 12,503,438 granted on 2025-12-23
US20230043835A1
Chemistry; metallurgy

Compounds for the Treatment of Kinase-Dependent Disorders

#20 | 2023-01-26 βœ… Patent 12,017,995 granted on 2024-06-25
US20230029213A1
Chemistry; metallurgy

Crystalline forms and salt forms of a kinase inhibitor

#21 | 2022-10-06 βœ… Patent 12,371,428 granted on 2025-07-29
US20220315579A1
Chemistry; metallurgy

PYRIDONE COMPOUNDS AND METHODS OF USE

#22 | 2021-09-23 βœ… Patent 11,718,622 granted on 2023-08-08
US20210292332A1
Chemistry; metallurgy

Heterocyclic adenosine receptor antagonists

#23 | 2021-08-26 βœ… Patent 11,279,675 granted on 2022-03-22
US20210261509A1
Chemistry; metallurgy

Crystalline solid forms of salts of N-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}-Nβ€²-(4-fluorophenyl) cyclopropane-1, 1-dicarboxamide, processes for making, and methods of use

#24 | 2021-08-19 βœ… Patent 11,124,482 granted on 2021-09-21
US20210253530A9
Chemistry; metallurgy

C-met modulators and methods of use

#25 | 2021-07-08 βœ… Patent 11,760,726 granted on 2023-09-19
US20210206722A1
Chemistry; metallurgy

Crystalline solid forms of N-{4-[(6,7-Dimethoxyquinolin-4-yl)oxy]phenyl} -n'-(4-fluorophenyl) cyclopropane-1,1-dicarboxamide, processes for making, and methods of use

#26 | 2021-06-03 βœ… Patent 11,098,015 granted on 2021-08-24
US20210163416A1
Chemistry; metallurgy

Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-Nβ€²-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms thereof for the treatment of cancer

#27 | 2021-06-03 βœ… Patent 11,298,349 granted on 2022-04-12
US20210161885A1
Human necessities

Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds

#28 | 2021-05-27 βœ… Patent 12,084,496 granted on 2024-09-10
US20210155692A1
Chemistry; metallurgy

Anti-ROR antibody constructs

#29 | 2021-05-13 βœ… Patent 11,091,440 granted on 2021-08-17
US20210139430A1
Chemistry; metallurgy

Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)- Nβ€²-(4-fluorophenyl)cyclopropane-1,1 -dicarboxamide, and crystalline forms thereof for the treatment of cancer

#30 | 2021-02-11 βœ… Patent 11,708,367 granted on 2023-07-25
US20210040099A1
Chemistry; metallurgy

Compounds for the treatment of kinase-dependent disorders

#31 | 2021-02-11 βœ… Patent 11,542,259 granted on 2023-01-03
US20210040076A1
Chemistry; metallurgy

Compounds for the treatment of kinase-dependent disorders

#32 | 2021-02-04 βœ… Patent 11,673,897 granted on 2023-06-13
US20210032263A1
Chemistry; metallurgy

Compounds for the treatment of kinase-dependent disorders

#33 | 2021-02-04
US20210030737A1
Human necessities

Triple Negative Breast Cancer Treatment Method

#34 | 2021-01-28 βœ… Patent 11,091,439 granted on 2021-08-17
US20210024467A1
Chemistry; metallurgy

Malate salt of N-(4-{[6,7-bis(methyloxy) quinolin-4-yl]oxy}phenyl)-Nβ€²-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, and crystalline forms therof for the treatment of cancer

#35 | 2020-12-17 βœ… Patent 11,414,396 granted on 2022-08-16
US20200392104A1
Chemistry; metallurgy

Process for making compounds for use in the treatment of cancer

#36 | 2020-10-22 βœ… Patent 11,433,064 granted on 2022-09-06
US20200330451A1
Human necessities

Methods of using c-Met modulators

#37 | 2020-10-22 βœ… Patent 11,612,597 granted on 2023-03-28
US20200330450A1
Human necessities

Method of treating cancer

#38 | 2020-09-10 βœ… Patent 11,597,699 granted on 2023-03-07
US20200283383A1
Chemistry; metallurgy

MEK inhibitors and methods of their use

#39 | 2020-08-27 βœ… Patent 11,504,362 granted on 2022-11-22
US20200268737A1
Human necessities

Liquid dosage forms to treat cancer

#40 | 2020-08-13 βœ… Patent 11,254,649 granted on 2022-02-22
US20200255398A1
Chemistry; metallurgy

Crystalline fumarate salt of (S)-[3,4-difluoro-2-(2-fluoro-4-iodophenylamino)phenyl] [3-hydroxy-3-(piperidin-2-yl) azetidin-1-yl]-methanone

#41 | 2020-08-13 βœ… Patent 11,504,363 granted on 2022-11-22
US20200255382A1
Chemistry; metallurgy

Method of treating cancer and bone cancer pain

#42 | 2020-06-18 βœ… Patent 10,851,061 granted on 2020-12-01
US20200190033A1
Chemistry; metallurgy

Crystalline solid forms of N-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}-Nβ€²-(4-fluorophenyl) cyclopropane-1,1-dicarboxamide, processes for making, and methods of use

#43 | 2020-04-23 βœ… Patent 11,123,338 granted on 2021-09-21
US20200121671A1
Human necessities

C-met modulator pharmaceutical compositions

#44 | 2019-11-21 βœ… Patent 11,198,731 granted on 2021-12-14
US20190352403A1
Chemistry; metallurgy

Combinations of cabozantinib and atezolizumab to treat cancer

#45 | 2019-07-11 βœ… Patent 11,141,413 granted on 2021-10-12
US20190209547A1
Human necessities

Method of treating renal cell carcinoma using N-(4-(6,7-dimethoxyquinolin-4-yloxy)phenyl)-Nβ€²-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide, (2S)-hydroxybutanedioate

#46 | 2019-06-20 βœ… Patent 10,793,541 granted on 2020-10-06
US20190185447A1
Chemistry; metallurgy

Process for making compounds for use in the treatment of cancer

#47 | 2019-05-23 βœ… Patent 10,736,886 granted on 2020-08-11
US20190151302A1
Human necessities

Methods of using c-Met modulators

#48 | 2019-03-28 βœ… Patent 11,116,759 granted on 2021-09-14
US20190091215A1
Human necessities

Method of treating cancer

#49 | 2019-01-31 βœ… Patent 10,543,206 granted on 2020-01-28
US20190030021A1
Human necessities

Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds

#50 | 2018-12-06 βœ… Patent 10,590,102 granted on 2020-03-17
US20180346442A1
Chemistry; metallurgy

Crystalline fumarate salt of (S)-[3,4-difluoro-2-(2-fluoro-4-iodophenylamino)phenyl] [3-hydroxy-3-(piperidin-2-yl) azetidin-1-yl]methanone

#51 | 2017-12-14 βœ… Patent 11,124,482 granted on 2021-09-21
US20170355678A1
Chemistry; metallurgy

C-met modulators and methods of use

#52 | 2017-12-07 βœ… Patent 10,239,858 granted on 2019-03-26
US20170349569A1
Chemistry; metallurgy

Process for making compounds for use in the treatment of cancer

#53 | 2017-10-19 βœ… Patent 10,328,069 granted on 2019-06-25
US20170296529A1
Human necessities

Phosphatidylinositol 3-kinase inhibitors for the treatment of lymphoproliferative malignancies

#54 | 2017-09-21 βœ… Patent 10,034,873 granted on 2018-07-31
US20170266178A1
Human necessities

C-met modulator pharmaceutical compositions

#55 | 2017-08-10 βœ… Patent 10,053,470 granted on 2018-08-21
US20170226131A1
Chemistry; metallurgy

Inhibitors of PI3K-delta and methods of their use and manufacture

#56 | 2017-08-10 βœ… Patent 11,065,240 granted on 2021-07-20
US20170224672A1
Human necessities

Drug combinations to treat multiple myeloma

#57 | 2017-08-03 βœ… Patent 11,124,481 granted on 2021-09-21
US20170217896A1
Chemistry; metallurgy

Method of preparing fluorine-18 labeled Cabozantinib and its analogs

#58 | 2017-05-25 βœ… Patent 10,039,757 granted on 2018-08-07
US20170143689A1
Human necessities

C-Met modulator pharmaceutical compositions

#59 | 2017-03-30 βœ… Patent 10,159,666 granted on 2018-12-25
US20170087143A1
Human necessities

Dosing of cabozantinib formulations

#60 | 2017-03-02 βœ… Patent 10,123,999 granted on 2018-11-13
US20170057921A1
Chemistry; metallurgy

Processes for preparing quinoline compounds and pharmaceutical compositions containing such compounds

#61 | 2017-02-16 βœ… Patent 10,501,418 granted on 2019-12-10
US20170044106A1
Chemistry; metallurgy

Crystalline solid forms of N-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}-Nβ€²-(4-fluorophenyl) cyclopropane-1,1-dicarboxamide, processes for making, and methods of use

#62 | 2016-02-04 βœ… Patent 10,273,211 granted on 2019-04-30
US20160031818A1
Chemistry; metallurgy

Metabolites of N-{4-([6,7-bis(methyloxy)quinolin-4-yl]oxy}phenyl)-Nβ€²-(4-fluorophenyl)cyclopropane-1,1-dicarboxamide

#63 | 2016-01-28 βœ… Patent 11,564,915 granted on 2023-01-31
US20160022662A1
Human necessities

Cabozantinib dosage form and use in the treatment of cancer

#64 | 2015-09-24 βœ… Patent 10,035,790 granted on 2018-07-31
US20150266856A1
Chemistry; metallurgy

RORΞ³ modulators

#65 | 2014-08-14 βœ… Patent 10,166,225 granted on 2019-01-01
US20140228401A1
Human necessities

Method for treating osteoporosis

Also check out Exelixis, Inc.'s (Alameda, United States) applicant profile with 74 patent applications submitted.

AssigneeID:

307005 ⎘