ClassID:

90494

C07B2200/13 - page 9 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#2401
20210179817
2021-06-17

Purification of sugammadex

#2402
20210179647
2021-06-17

Phosphonamide ester compound, salt thereof, related crystal form thereof, preparation method therefor and use thereof

#2403
20210179637
2021-06-17

Methods for treating Crohn's disease using 3-((1R,3s,5S)-3-((7-((5-methyl-1H-pyrazol-3-yl)amino)-1,6-naphthyridin-5-yl)amino)-8-azabicyclo[3.2.1]octan-8-yl)propanenitrile

#2404
20210179587
2021-06-17

Modulators of alpha-1 antitrypsin

#2405
20210179586
2021-06-17

SOLID STATE FORMS OF BRANAPLAM AND THEIR PREPARATION

#2406
20210179585
2021-06-17

CRYSTAL FORM OF ABEMACICLIB MESYLATE, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL COMPOSITION THEREOF

#2407
20210179566
2021-06-17

Compositions and methods for delivering pharmaceutical agents

#2408
20210179561
2021-06-17

ACID ADDITION SALTS OF APOMORPHINE, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME

#2409
20210179558
2021-06-17

Crystalline form of EB-1020, processes for preparation and use thereof

#2410
20210179549
2021-06-17

Co-crystal of sorafenib derivatives and process for preparation thereof

#2411
20210179541
2021-06-17

Method for producing (3S)-3-(4-chloro-3-{[(2S,3R)-2-(4- chlorophenyl)-4,4,4-trifluoro-3-methylbutanoyl]amino}phenyl)-3-cyclo-propylpropanoic acid and the crystalline form thereof for use as a pharmaceutical ingredient

#2412
20210177758
2021-06-17

Platform drug delivery system utilizing crystal engineering and theanine dissolution

#2413
20210171568
2021-06-10

CRYSTALLINE FORMS OF SELECTIVE PROGESTERONE RECEPTOR MODULATOR, PROCESSES FOR PREPARATION THEREOF

#2414
20210171560
2021-06-10

D-allose crystal and production method thereof

#2415
20210171541
2021-06-10

Pyridine and pyrimidine derivatives

#2416
20210171536
2021-06-10

COMPOUND OF EOC315 MOD.I CRYSTAL FORM AND PREPARATION METHOD THEREOF

#2417
20210171525
2021-06-10

Purinone compounds and their use in treating cancer

#2418
20210171506
2021-06-10

Process for Manufacturing Pibrentasvir Active Drug Substance

#2419
20210171496
2021-06-10

Solid forms of a plasma kallikrein inhibitor and salts thereof

#2420
20210171494
2021-06-10

Crystalline and salt forms of PPAR agonist compounds

#2421
20210171493
2021-06-10

Processes for preparing 2-(4-chlorophenyl)-N-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)methyl)-2,2-difluoroacetamide

#2422
20210171464
2021-06-10

AMORPHOUS FORM OF PIMAVANSERIN HEMITARTRATE

#2423
20210171460
2021-06-10

Crystalline form of sofpironium bromide and preparation method thereof

#2424
20210170301
2021-06-10

Diamond pressure apparatus for crystallizing cannabinoids

#2425
20210163586
2021-06-03

Gremlin-1 crystal structure and inhibitory antibody

#2426
20210163523
2021-06-03

Crystalline forms of (S)-2-ethylbutyl 2-(((S)-(((2R,3S,4R,5R)-5-(4-aminopyrrolo[2,1-f] [1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxytetrahydrofuran-2-yl)methoxy) (phenoxy) phosphoryl)amino)propanoate

#2427
20210163522
2021-06-03

Salts and polymorphs of cethromycin for the treatment of disease

#2428
20210163507
2021-06-03

Borate of azetidine derivative

#2429
20210163498
2021-06-03

SOLID STATE FORMS OF LORLATINIB AND THEIR PREPARATION

#2430
20210163488
2021-06-03

Ion channel modulators

#2431
20210163463
2021-06-03

Process for preparing modulators of p300 and/or CBP

#2432
20210163457
2021-06-03

CANAGLIFLOZIN MONOHYDRATE AND ITS CRYSTALLINE FORMS, PREPARATION METHODS AND USES THEREOF

#2433
20210163455
2021-06-03

GLP-1 Receptor Agonists and Uses Thereof

#2434
20210163442
2021-06-03

Crystalline forms of lenalidomide

#2435
20210163398
2021-06-03

Crystalline form of triethylenetetramine tetrahydrochloride and its pharmaceutical use

#2436
20210161904
2021-06-03

Methods of synthesizing thyroid hormone analogs and polymorphs thereof

#2437
20210155642
2021-05-27

Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use

#2438
20210155630
2021-05-27

Crystal of benzoxazole derivative

#2439
20210155613
2021-05-27

Fruquintinib eutectic crystal, preparation method therefor, composition, and uses thereof

#2440
20210155605
2021-05-27

Salts of a Pim kinase inhibitor

#2441
20210155603
2021-05-27

THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE

#2442
20210155589
2021-05-27

Method of preparing (3R,4S)-3-acetamido-4-allyl-n-(tert-butyl)pyrrolidine-3-carboxamide

#2443
20210155587
2021-05-27

Method for preparing novel crystalline forms of 1-(4-benzyloxy-benzyl)-3-methyl-thiourea

#2444
20210155586
2021-05-27

Polymorphs of 1-(4-benzyloxy-benzyl)-3-methyl-thiourea

#2445
20210155577
2021-05-27

Crystalline tranilast salts and their pharmaceutical use

#2446
20210147472
2021-05-20

SOLID FORMS AND FORMULATIONS COMPRISING A GLUCOCORTICOID RECEPTOR ANTAGONIST AND USES THEREOF

#2447
20210147471
2021-05-20

Crystalline forms of a fatty acid bile acid conjugate, preparation method thereof and use thereof

#2448
20210147466
2021-05-20

IMPROVED PROCESSES FOR THE PREPARATION OF GUADECITABINE AND INTERMEDIATES THEREOF

#2449
20210147440
2021-05-20

Methods for the preparation of 1,3-benzodioxole heterocyclic compounds

#2450
20210147433
2021-05-20

Crystalline forms of (S)-1-(4-fluorophenyl)-1-(2-(4-(6-(1-methyl-1H-pyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl)piperazinyl)-pyrimidin-5-yl)ethan-1-amine and methods of making

#2451
20210147423
2021-05-20

Crystal form of Baricitinib and preparation method thereof

#2452
20210147417
2021-05-20

Processes for preparing an FGFR inhibitor

#2453
20210147413
2021-05-20

ISOTHERMAL REACTIVE CRYSTALLISATION PROCESS FOR THE PREPARATION OF A CRYSTALLINE FORM OF PIMODIVIR HYDROCHLORIDE HEMIHYDRATE

#2454
20210147402
2021-05-20

Compounds and methods of preparing compounds S1P1 modulators

#2455
20210147401
2021-05-20

Process for the production of 5-(4-((2S,5S)-5-(4-chlorobenzyl)-2-methyl-morpholino)piperidin-1-yl)-1H-1,2,4-triazol-3-amine

#2456
20210147394
2021-05-20

Polymorph of HDAC6-selective inhibitor and application thereof

#2457
20210147384
2021-05-20

Densely charged catenanes

#2458
20210147370
2021-05-20

Oxazole compound crystal

#2459
20210147367
2021-05-20

CRYSTALLINE FORMS OF A MAGL INHIBITOR

#2460
20210147363
2021-05-20

Solid state crystalline forms of a selective potassium channel modulator

#2461
20210147353
2021-05-20

Method for extracting and isolating lutein crystal from vegetable oil resin containing lutein diester

#2462
20210147342
2021-05-20

Crystalline solids of 3-palmitoyl-amido-1,2-propanediol and 3-palmitoyl-amido-2-hydroxy-1-dimethoxytriphenylmethylether-propane and methods of making and using the same

#2463
20210147341
2021-05-20

Crystal form and amorphous form of dezocine analogue hydrochloride

#2464
20210147338
2021-05-20

Zuclomiphene salts and crystalline forms thereof

#2465
20210147335
2021-05-20

Fenfluramine compositions and methods of preparing the same

#2466
20210147329
2021-05-20

Process for the preparation of iloprost

#2467
20210145831
2021-05-20

Crystalline forms of 5-bromo-2,6-di(1H-pyrazol-1- yl)pyrimidin-4-amine and new salts

#2468
20210139528
2021-05-13

CRYSTALLINE FORMS OF OBETICHOLIC ACID

#2469
20210139518
2021-05-13

NOVEL POLYMORPHIC FORM OF FERRIC MALTOL

#2470
20210139511
2021-05-13

Salts and crystalline forms of a PD-1/PD-L1 inhibitor

#2471
20210139502
2021-05-13

Solid forms of an S1P-receptor modulator

#2472
20210139498
2021-05-13

Crystal forms of thiophene derivatives

#2473
20210139489
2021-05-13

Methods of treating painful diabetic peripheral neuropathy

#2474
20210139487
2021-05-13

Crystalline forms of C-C chemokine receptor type 4 antagonist and uses thereof

#2475
20210139474
2021-05-13

Tartrate of selective CDK9 inhibitor and crystal form thereof

#2476
20210139461
2021-05-13

Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same

#2477
20210139437
2021-05-13

Methods and processes for the preparation of KDM1A inhibitors

#2478
20210139433
2021-05-13

Crystal form of 3-(4-methyl-1h-imidazol-1-yl)-5-trifluoromethylaniline monohydrochloride and use thereof

#2479
20210139431
2021-05-13

Crystalline form of lenvatinib mesylate and methods thereof

#2480
20210139427
2021-05-13

Salt forms of a complement component C5A receptor

#2481
20210139424
2021-05-13

Crystalline form of 1-(5-(2,4-difluorophenyl)-1-((3-fluorophenyl)sulfonyl)-4-methoxy-1H-pyrrol-3-yl)-N-methylmethanamine salt

#2482
20210139420
2021-05-13

Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof

#2483
20210139416
2021-05-13

2,2,2-trifluoroacetic acid 1-(2,4-dimethylphenyl)-2-[(3-methoxyphenyl)methylene] method of making the same

#2484
20210139413
2021-05-13

Production method for 1-amino cyclopropane carboxylic acid nonhydrate

#2485
20210139411
2021-05-13

Crystal forms and methods of synthesis of (2R, 6R)-hydroxynorketamine and (2S, 6S)-hydroxynorketamine

#2486
20210139405
2021-05-13

METHODS OF MAKING BEMPEDOIC ACID AND COMPOSITIONS OF THE SAME

#2487
20210139401
2021-05-13

Methods of making bempedoic acid and compositions of the same

#2488
20210137907
2021-05-13

Free base crystalline form of a complement component C5a receptor

#2489
20210137112
2021-05-13

Crystalline forms of ethyl[3-[2-chloro-4-fluoro-5-(1-methyl-6-trifluoromethyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-3-yl)phenoxy]-2-pyridyloxy]acetate

#2490
20210130363
2021-05-06

CRYSTALLINE FORM OF (S)-7-(1-ACRYLOYLPIPERIDIN-4-YL)-2-(4-PHENOXYPHENYL)-4,5,6,7-TETRA-HYDROPYRAZOLO[1,5-a]PYRIMIDINE-3-CARBOXAMIDE, PREPARATION, AND USES THEREOF

#2491
20210130362
2021-05-06

MEDICAL USE OF COMPOUND III

#2492
20210130360
2021-05-06

Crystalline forms of Acalabrutinib

#2493
20210130350
2021-05-06

Solid state forms of Venetoclax and its process for the preparation there of

#2494
20210130332
2021-05-06

OPIOID RECEPTOR (MOR) AGONIST SALT, FUMARATE SALT CRYSTAL FORM I THEREOF AND PREPARATION METHOD THEREOF

#2495
20210130330
2021-05-06

Solid forms of Cerdulatinib

#2496
20210122766
2021-04-29

Salt forms of amino pyrazine purine based selective kinase inhibitor

#2497
20210122756
2021-04-29

Long-acting injectable formulations and crystalline forms of buprenorphine derivatives

#2498
20210122754
2021-04-29

Process for the preparation of ribociclib succinate and its novel crystalline forms thereof

#2499
20210122753
2021-04-29

Tebipenem pivoxil crystalline forms, compositions including the same, methods of manufacture, and methods of use

#2500
20210122740
2021-04-29

SOLID FORMS OF 2-(3,5-DICHLORO-4-((5-ISOPROPYL-6-OXO-1,6-DIHYDROPYRIDAZIN-3-YL)OXY)PHENYL)-3,5-DIOXO-2,3,4,5-TETRAHYDRO-1,2,4-TRIAZINE-6-CARBONITRILE

#2501
20210122738
2021-04-29

Salts and solid state forms of plinabulin

#2502
20210122737
2021-04-29

Polymorph of flibanserin and preparation method thereof and use of same

#2503
20210122726
2021-04-29

Crystalline solid compound of 3-phenyl-4-propyl-1-(pyridin-2-yl)-1H-pyrazol-5-ol hydrochloride

#2504
20210122718
2021-04-29

Forms of fedratinib dihydrochloride

#2505
20210122717
2021-04-29

Process for synthesis of a phenoxy diaminopyrimidine compound

#2506
20210122714
2021-04-29

Crystal forms of oxypyridine amide derivative and preparation method therefor

#2507
20210122708
2021-04-29

Trisodium sacubitril valsartan and process for its preparation

#2508
20210121422
2021-04-29

Glucagon receptor antagonists

#2509
20210115050
2021-04-22

Crystalline forms of 8-(2-fluorobenzyl)-6-(3-(trifluoromethyl)-1H-1,2,4-triazol-5-yl)imidazo[1,2-a]pyrazine as sGC stimulators

#2510
20210115039
2021-04-22

Cocrystal

#2511
20210115033
2021-04-22

Crystalline forms of the CXCR7 receptor antagonist (3S,4S)-1-Cyclopropylmethyl-4-{[5-(2,4-difluoro-phenyl)-isoxazole-3-carbonyl]-amino}-piperidine-3-carboxylic acid (1-pyrimidin-2-yl-cyclopropyl)-amide

#2512
20210115032
2021-04-22

Processes for the preparation of furazanobenzimidazoles and crystalline forms thereof

#2513
20210115019
2021-04-22

Solid forms comprising (S)-2-(2,6-dioxopiperidin-3-yl)-4-((2-fluoro-4-((3-morpholinoazetidin-1-yl)methyl)benzyl)amino)isoindoline-1,3-dione and salts thereof, and compositions comprising and methods of using the same

#2514
20210115004
2021-04-22

A2-73 crystalline polymorph compositions of matter and methods of use thereof

#2515
20210114997
2021-04-22

Preparation of 2-([1,2,3]triazol-2-yl)-benzoic acid derivatives

#2516
20210114995
2021-04-22

Crystalline substituted pyrazines as PGI2 receptor agonists

#2517
20210113572
2021-04-22

Crystalline form of (S)-[2-chloro-4-fluoro-5-(7-morpholin-4-yl-quinazolin-4-yl)phenyl]-(6-methoxy-pyridazin-3-yl)-methanol

#2518
20210113470
2021-04-22

Amorphous dispersion of cyclopropanecarboxylic acid (5-{5-[N′-(2-chloro-6-methylbenzoyl) hydrazinocarbonyl]-2-methyl-phenylethynyl}-pyridin-2-yl) amide

#2519
20210107911
2021-04-15

Monohydrate and crystalline forms of 6-[(3S,4S)-4-methyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl]-3-tetrahydropyran-4-yl-7H-imidazo[1,5-a]pyrazin-8-one

#2520
20210107907
2021-04-15

Hydrochloride salt of 2-((3R,4S)-1-(5-(4-chloro-3,5-difluorophenyl)-7-((2-fluoro-6-methylphenyl)(methyl)amino)pyrazolo[1,5-a]pyrimidine-2-carbonyl)-3-methoxypiperidin-4-yl) acetic acid and crystals thereof

#2521
20210107905
2021-04-15

[1,2,4]triazolo[4,3-b]pyridazines for use in the treatment of proliferative diseases

#2522
20210107902
2021-04-15

Crystalline sodium salt of 5-methyl-(6S)-tetrahydrofolic acid

#2523
20210107897
2021-04-15

Process for the preparation of 6-(cyclopropaneamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyl- D3)pyridazine-3-carboxamide

#2524
20210107892
2021-04-15

Compounds, compositions and methods

#2525
20210107888
2021-04-15

Crystalline 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione dihydrate, compositions and methods of use thereof

#2526
20210107884
2021-04-15

Method for purifying crystals using solvent vapors

#2527
20210107856
2021-04-15

Co-crystals of lithium benzoate and uses thereof

#2528
20210106577
2021-04-15

Methods and compositions for treating retina-associated disease using CCR3-inhibitors

#2529
20210105998
2021-04-15

Crystalline solid forms of a BET inhibitor

#2530
20210101889
2021-04-08

6-pyrimidin-isoindole derivative as ERK1/2 inhibitor

#2531
20210101887
2021-04-08

Isoindolinone inhibitors of the MDM2-P53 interaction and process for making them

#2532
20210101863
2021-04-08

Substituted Phenethylamines with Serotoninergic and/or Norepinephrinergic Activity

#2533
20210100785
2021-04-08

Solid forms comprising 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione and a coformer, compositions and methods of use thereof

#2534
20210094979
2021-04-01

Pharmaceutical co-crystal composition and use thereof

#2535
20210094974
2021-04-01

DIARYL MACROCYCLE POLYMORPH

#2536
20210094970
2021-04-01

Polymorphs and solid forms of (s)-2-((2-((s)-4-(difluoromethyl)-2-oxooxazolidin-3-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)amino)propanamide, and methods of production

#2537
20210094962
2021-04-01

Solid state forms of rucaparib and of rucaparib salts

#2538
20210094961
2021-04-01

Form of ponatinib

#2539
20210094957
2021-04-01

Crystal form a of (5-amino-8-(2-methyl-6-(trifluoromethyl)pyridin-4-yl)-7-phenyl-[1,2,4]triazolo[1,5-c]pyrimidin-2-yl)methanol (compound 1)

#2540
20210094955
2021-04-01

SALT AND CRYSTAL OF TRIAZOLOPYRAZINE DERIVATIVE

#2541
20210094936
2021-04-01

Crystalline forms of nicotinamide riboside chloride

#2542
20210094930
2021-04-01

COFORMER SALTS OF (2S,3S)-METHYL 7-FLUORO-2-(4-FLUOROPHENYL)-3-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-4-OXO-1,2,3,4-TETRAHYDROQUINOLINE-5-CARBOXYLATE AND METHODS OF PREPARING THEM

#2543
20210094918
2021-04-01

Process for the preparation of (S)-Netarsudil,its salts and polymorphs

#2544
20210094901
2021-04-01

Crystalline particles of bis-choline tetrathiomolybdate

#2545
20210092957
2021-04-01

Crystalline forms of deltamethrin and methods of use thereof

#2546
20210087217
2021-03-25

NUCLEOTIDE HEMI-SULFATE SALT FOR THE TREATMENT OF HEPATITIS C VIRUS

#2547
20210087212
2021-03-25

Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use

#2548
20210087205
2021-03-25

Salt serving as AKT inhibitor and crystal thereof

#2549
20210087204
2021-03-25

BCKDK inhibitors

#2550
20210087197
2021-03-25

3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyrazine as an ion channel modulator

#2551
20210087196
2021-03-25

Triazolopyrimidine compounds and their use in treating cancer

#2552
20210087195
2021-03-25

NEW CRYSTAL FORM OF ACALBRUTINIB, PREPARATION METHOD THEREFOR AND USE THEREOF

#2553
20210087194
2021-03-25

Chemical Process for Preparing Imidazopyrrolidinone Derivatives and Intermediates Thereof

#2554
20210087181
2021-03-25

Salt form and crystal form of compound as FGFR4 inhibitor and preparation method thereof

#2555
20210087176
2021-03-25

Polymorphs and solid forms of a pyrimidinylamino-pyrazole compound, and methods of production

#2556
20210087175
2021-03-25

Crystalline Form II of Darolutamide

#2557
20210087165
2021-03-25

PROCESS OF MAKING SOMATOSTATIN MODULATORS

#2558
20210087156
2021-03-25

PHARMACEUTICALLY ACCEPTABLE SALTS OF BENZODICYCLOALKANE DERIVATIVE, POLYMORPHIC SUBSTANCE THEREOF, AND APPLICATION THEREOF

#2559
20210087155
2021-03-25

AN IMPROVED PROCESS FOR THE PREPARATION OF VORTIOXETINE AND SALTS THEREOF

#2560
20210087152
2021-03-25

Tebuconazole polymorph and preparation method therefor

#2561
20210087150
2021-03-25

Crystalline polymorphs of Pracinostat and Pracinostat salts

#2562
20210087140
2021-03-25

Crystalline siponimod fumaric acid and polymorphs thereof

#2563
20210085677
2021-03-25

SHP2 phosphatase inhibitors and methods of making and using the same

#2564
20210079021
2021-03-18

Crystal form and salt form of TGF-βRI inhibitor and preparation method therefor

#2565
20210078993
2021-03-18

Crystalline form of valbenazine ditosylate, processes for preparation thereof and use thereof

#2566
20210078984
2021-03-18

Solid forms of (E)-3-[2-(2-thienyl)vinyl]-1H-pyrazole

#2567
20210078968
2021-03-18

Purification of cannabinoids from crude cannabis oil

#2568
20210078960
2021-03-18

Crystal and salt of 4-(naphthalen-1-yl)-4H-1,2,4-triazole compound and preparation method therefor

#2569
20210078939
2021-03-18

Type-B fenolamine crystal form, preparation method, composition and use thereof

#2570
20210077518
2021-03-18

Polymorphic compounds and uses thereof

#2571
20210070759
2021-03-11

Crystalline forms of a Bruton's tyrosine kinase inhibitor

#2572
20210070755
2021-03-11

Method for the production of lumateperone and its salts

#2573
20210070738
2021-03-11

Polycrystalline form of dehydrophenylahistin-like compound, and manufacturing and purification method and application thereof

#2574
20210070733
2021-03-11

Cyclopentane compounds

#2575
20210070724
2021-03-11

METHOD FOR PRODUCING 2-ACETYL-4H,9H-NAPHTHO[2,3-B]FURAN-4,9-DIONE

#2576
20210070723
2021-03-11

CRYSTAL FORM OF SESQUITERPENE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF

#2577
20210070722
2021-03-11

Method for purifying and removing color of FDCA

#2578
20210070714
2021-03-11

Crystalline forms of [3-(4- {2-butyl-1-[4-(4-chloro-phenoxy)-phenyl]-1H-imidazol-4-yl} -phenoxy)-propyl]-diethyl-amine

#2579
20210069219
2021-03-11

Substituted 1,2-oxaborolan-2-ols as PDE4 inhibitors

#2580
20210061853
2021-03-04

Crystalline bis- and tris-hydrochloride salt of elamipretide

#2581
20210061796
2021-03-04

IL-17 and IFN-gamma inhibition for the treatment of autoimmune diseases and chronic inflammation

#2582
20210061792
2021-03-04

Process and crystalline forms of Lumacaftor

#2583
20210061776
2021-03-04

Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2-methylpentanoic acid and uses thereof

#2584
20210061772
2021-03-04

Method for preparing tolimidone on large scale

#2585
20210061759
2021-03-04

Crystal forms and production methods thereof

#2586
20210054014
2021-02-25

Polymorphic forms of deoxycytidine, compositions comprising the same and uses

#2587
20210053996
2021-02-25

4-substituted benzoxaborole compounds and uses thereof

#2588
20210053983
2021-02-25

Salts, crystal forms, and production methods thereof

#2589
20210053974
2021-02-25

Inhibitors of the menin-MLL interaction

#2590
20210053971
2021-02-25

Crystal form of monomethanesulfonate of deuterated 3-(4,5-substituted aminopyrimidine)phenyl compound and preparation method therefor

#2591
20210053963
2021-02-25

Crystalline forms of Actinomycin D for treatment of cancer

#2592
20210053962
2021-02-25

Processes and intermediates for the preparation of soluble guanylate cyclase stimulators

#2593
20210053951
2021-02-25

Salt Forms Of 4-Cyano-N-(4,4-Dimethylcyclohex-1-EN-1-YL)-6-(2,2,6,6-Tetramethyltetrahydro-2H-Pyran-4-YL)Pyridin-3-YL)-1H-Imidazole-2-Carboximide

#2594
20210053949
2021-02-25

Process and crystalline forms of lumacaftor

#2595
20210053945
2021-02-25

Acryloyl-containing nuclear transport regulators and uses thereof

#2596
20210053944
2021-02-25

Salt of a quinazoline derivative-like tyrosine kinase inhibitor and crystal form thereof

#2597
20210053939
2021-02-25

POLYMORPHIC FORMS OF (R)-4-(1-((3-(DIFLUOROMETHYL)-1-METHYL-1H-PYRAZOL-4-YL)SULFONYL)-1-FLUOROETHYL)-N-(ISOXAZOL-3-YL)PIPERIDINE-1-CARBOXAMIDE

#2598
20210053923
2021-02-25

CRYSTAL FORM OF QUINOLINE COMPOUND AND PROCESS FOR ITS PRODUCTION

#2599
20210053914
2021-02-25

Crystalline form of 3-((L-valyl)amino))-3,3-dideuterium-1-propanesulfonic acid, preparation method and uses thereof

#2600
20210053912
2021-02-25

Compositions comprising (R)-2-amino-3-phenylpropyl carbamate and uses thereof

#2601
20210053901
2021-02-25

Process for the preparation of polymorph form B of treprostinil diethanolamine salt

#2602
20210053900
2021-02-25

Aqueous Leaching Method to Produce Microcrystalline Powder

#2603
20210047368
2021-02-18

Crystalline salt forms

#2604
20210047362
2021-02-18

Crystal forms of an antitumor agent and their preparation methods

#2605
20210047339
2021-02-18

Method for preparation of Asenapine

#2606
20210047323
2021-02-18

Crystalline forms of CFTR modulators

#2607
20210047317
2021-02-18

Process for preparation of Deutetrabenazine

#2608
20210047295
2021-02-18

Modulator of the cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator

#2609
20210047292
2021-02-18

Crystal form targeting CDKkinase inhibitor

#2610
20210047288
2021-02-18

Fasoracetam crystalline forms

#2611
20210047272
2021-02-18

Crystalline of compound as c-Met kinase inhibitor and preparation method therefor and use thereof

#2612
20210046092
2021-02-18

LOW DOSE COMPOSITIONS OF ARAMCHOL SALTS

#2613
20210046082
2021-02-18

CRYSTALLINE FORMS OF QUINOLINE ANALOGS AND SALTS THEREOF, COMPOSITIONS, AND THEIR METHODS FOR USE

#2614
20210046066
2021-02-18

ACETATE SALT OF BUPRENORPHINE AND METHODS FOR PREPARING BUPRENORPHINE

#2615
20210046050
2021-02-18

Stable amorphous form of sacubitril valsartan trisodium complex and processes for preparation thereof

#2616
20210045384
2021-02-18

Crystalline form of oxamyl process for its preparation and use of the same

#2617
20210040521
2021-02-11

Solid form of (-)-Ambrox formed by a bioconversion of homofarnesol in the presence of a biocatalyst

#2618
20210040116
2021-02-11

New Polymorphs of Dolutegravir Sodium

#2619
20210040103
2021-02-11

Crystalline salts or co-crystals of 2′,6-difluoro-5′-[3-(1-hydroxy-1-methylethyl)-imidazo[1,2-b] [1,2,4]triazin-7-yl]biphenyl-2-carbonitrile with phosphoric acid as GABAA positive allosteric modulators

#2620
20210040090
2021-02-11

Salts of a PD-1/PD-L1 inhibitor

#2621
20210040071
2021-02-11

Solid forms of an HPK1 inhibitor

#2622
20210040068
2021-02-11

EGFR inhibitors

#2623
20210040064
2021-02-11

Solid forms of 2-(4-chlorophenyl)-N-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)methyl)-2,2-difluoroacetamide, and their pharmaceutical compositions and uses

#2624
20210040051
2021-02-11

Salt of delmopinol

#2625
20210040045
2021-02-11

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#2626
20210040042
2021-02-11

Method for preparing mesaconine and related intermediaries thereof

#2627
20210040040
2021-02-11

Process for the preparation of a PDE4 inhibitor

#2628
20210040035
2021-02-11

Process for the preparation of metformin

#2629
20210039061
2021-02-11

Constant shear continuous reactor device

#2630
20210038590
2021-02-11

Memantine paroxetine cocrystal salt and its preparation method, pharmaceutical composition and application

#2631
20210032258
2021-02-04

CRYSTALLINE FORMS OF A BRUTONS TYROSINE KINASE INHIBITOR

#2632
20210032257
2021-02-04

(E)-1-(4-(DIMETHYLAMINO)BUT-2-ENOYL)PYRROLIDIN-3-YL 4-((3-ISOPROPYL-5-METHYLPYRAZOLO[1,5-A]PYRIMIDIN-7-YL)AMINO)PIPERIDINE-1-CARBOXYLATE FOR INHIBITING CDK7

#2633
20210032255
2021-02-04

Compounds useful as inhibitors of ATR kinase

#2634
20210032235
2021-02-04

Crystalline forms of dasatinib

#2635
20210032232
2021-02-04

Crystalline salts of peptide epoxyketone immunoproteasome inhibitor

#2636
20210032226
2021-02-04

Process for the preparation of lifitegrast

#2637
20210032223
2021-02-04

Crystal form of small molecule immune compound, preparation method thereof and pharmaceutical composition containing the same

#2638
20210032218
2021-02-04

Succinate forms and compositions of Bruton's tyrosine kinase inhibitors

#2639
20210032212
2021-02-04

Method for the preparation of a 2,4,5-trisubstituted 1,2,4-triazolone

#2640
20210032210
2021-02-04

Resveratrol-piperazine co-crystals

#2641
20210032209
2021-02-04

Certain chemical entities, compositions, and methods

#2642
20210032204
2021-02-04

Salt forms of URAT-1 inhibitors

#2643
20210024554
2021-01-28

Crystalline forms and methods of producing crystalline forms of a compound

#2644
20210024541
2021-01-28

Salt of pentacyclic compound and crystal thereof

#2645
20210024538
2021-01-28

Crystal form of 3,4-dihydrothieno[3,2-d]pyrimidine compound and preparation method thereof

#2646
20210024537
2021-01-28

Processes for preparing ACC inhibitors and solid forms thereof

#2647
20210024536
2021-01-28

BCKDK inhibitors

#2648
20210024527
2021-01-28

Crystalline forms of 3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-n-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide and its mono hydrochloride salt

#2649
20210024514
2021-01-28

Solid form of dihydropyrimidine compound and preparation method therefor and use thereof

#2650
20210024506
2021-01-28

Polymorphic forms of Afatinib free base and Afatinib dimaleate

#2651
20210024488
2021-01-28

Crystalline 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione hemihydrate, compositions and methods of use thereof

#2652
20210024475
2021-01-28

Crystal modifications of odevixibat

#2653
20210024461
2021-01-28

(S)-CSA Salt Of S-Ketamine, (R)-CSA Salt Of S-Ketamine And Processes For The Preparation Of S-Ketamine

#2654
20210017191
2021-01-21

Crystal of compound having JAK-inhibiting activity

#2655
20210017188
2021-01-21

Solid state forms of Relugolix

#2656
20210017185
2021-01-21

Morphic forms of marizomib and uses thereof

#2657
20210017181
2021-01-21

Pyridine or N,N-dimethyl acetamide solvated solid state forms of solvated idelalisib, their use and preparation

#2658
20210017163
2021-01-21

HYDROCHLORIDE SALT FORM FOR EZH2 INHIBITION

#2659
20210017151
2021-01-21

Crystalline forms of niraparib tosylate

#2660
20210017148
2021-01-21

Crystalline forms of ARN-509, preparation method and use thereof

#2661
20210017137
2021-01-21

Salts of an epidermal growth factor receptor kinase inhibitor

#2662
20210017125
2021-01-21

Calcium salt polymorphs as anti-inflammatory, immunomodulatory and anti-proliferative agents

#2663
20210015817
2021-01-21

Solid-state forms of Abemaciclib, their use and preparation

#2664
20210015765
2021-01-21

Polymorphic and amorphous forms of (R)-2-hydroxy-2-methyl-4-(2,4,5-trimethyl-3,6-dioxocyclohexa-1,4-dienyl)butanamide

#2665
20210009626
2021-01-14

Solid-state forms of Regadenoson, their use and preparation

#2666
20210009620
2021-01-14

PURE HEPTASULFATED DISACCHARIDES HAVING IMPROVED ORAL BIOAVAILABILITY

#2667
20210009619
2021-01-14

Method for producing allulose crystals

#2668
20210009614
2021-01-14

Crystalline forms

#2669
20210009601
2021-01-14

Manufacturing process and intermediates for a pyrrolo[2,3-d]pyrimidine compound and use thereof

#2670
20210009593
2021-01-14

Purinone derivative hydrochloride

#2671
20210009587
2021-01-14

ERBB receptor inhibitors

#2672
20210009560
2021-01-14

CRYSTALLINE FORMS OF MODULATORS OF CFTR

#2673
20210009534
2021-01-14

Method for producing the crystalline form of modification a of calcobutrol

#2674
20210009525
2021-01-14

Crystalline forms of plasma kallikrein inhibitors

#2675
20210009494
2021-01-14

Menaquinol compositions and methods of treatment

#2676
20210002307
2021-01-07

Crystal forms of crisaborole in free form and preparation method and use thereof

#2677
20210002283
2021-01-07

Crystal form of ethyl (S)-3-(8-bromo-1-methyl-6-(pyridin-2-yl)-4H-benzo[f]imidazo[1,2-a][1,4]diazepin-4-yl)propanoate hydrochloride

#2678
20210002282
2021-01-07

SOLID FORMS OF IBRUTINIB

#2679
20210002275
2021-01-07

PROCESS FOR PREPARATION OF PALBOCICLIB

#2680
20210002273
2021-01-07

Process for preparing N-(5-(3-(7-(3-fluorophenyl)-3H-imidazo[4,5-c]pyridin-2-yl)-1H-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide

#2681
20210002259
2021-01-07

Polycrystalline form of dehydrophenylahistin-like compound, and manufacturing and purification method and application thereof

#2682
20210002235
2021-01-07

Crystal of a caspase inhibitor

#2683
20210002227
2021-01-07

CRYSTALLINE FORMS OF PITAVASTATIN CALCIUM

#2684
20210002209
2021-01-07

NOVEL CRYSTALLINE FORMS OF TAMIBAROTENE FOR TREATMENT OF CANCER

#2685
20210000809
2021-01-07

PROCESS FOR THE PREPARATION OF ABAMETAPIR AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS

#2686
20200407389
2020-12-31

Method for producing functional crystalline sweetener

#2687
20200407382
2020-12-31

POLYMORPHIC FORMS OF (9-[(R)-2-[[(S)-[[(S)-1-(ISOPROPOXYCARBONYL)ETHYL]AMINO]PHENOXY PHOSPHINYL]METHOXY]PROPYL] ADENINE AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF

#2688
20200407377
2020-12-31

Process for the preparation of Crisaborole in a stable crystal form

#2689
20200407368
2020-12-31

Solid forms of stemospironine and its salts

#2690
20200407355
2020-12-31

CRYSTALLINE FORMS OF VENETOCLAX

#2691
20200407354
2020-12-31

Crystal form and salt form of pyridoimidazole compound and preparation method therefor

#2692
20200407334
2020-12-31

Process of preparing a peptide epoxyketone immunoproteasome inhibitor, and precursors thereof

#2693
20200407313
2020-12-31

Method for preparing natural L-cysteine hydrochloride hydrate crystals by continuous chromatography

#2694
20200399286
2020-12-24

Polymorphs and solid forms of (s)-2-((2-((s)-4-(difluoromethyl)-2-oxooxazolidin-3-yl)-5,6-dihydrobenzo[f]imidazo[1,2-d][1,4]oxazepin-9-yl)amino)propanamide, and methods of production

#2695
20200399272
2020-12-24

Crystal form of 2-(6-methyl-pyridin-2-yl)-3-yl-[6-amido-quinolin-4-yl]-5,6-dihydro-4H-pyrrolo[1,2-B]pyrazole, preparation method therefor and pharmaceutical composition thereof

#2696
20200399258
2020-12-24

Benzisoxazole sulfonamide derivatives

#2697
20200399234
2020-12-24

Polymorphs and new path to synthesize Tafamidis

#2698
20200399213
2020-12-24

Solid forms comprising an oxime ether compound, compositions and methods of use thereof

#2699
20200399205
2020-12-24

2,2,2-trifluoroacetic acid 1-(2,4-Dimethylphenyl)-2-[(3-methoxyphenyl)methylene] hydrazide polymorphs and method of making the same

#2700
20200397774
2020-12-24

Piperidin-4-yl azetidine derivatives as JAK1 inhibitors