94044 ⎘
Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
Sub-classes:LACTAM-MODIFIED ADENO-ASSOCIATED VIRUS VECTORS
#2SYNTHETIC CANNABINOID ANALOGS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF TREATING BACTERIAL INFECTIONS AND OTHER DISORDERS
#3COMPOUNDS FOR THE REDUCING LIPOTOXIC DAMAGE
#4Organic Compound And Organic Light-Emitting Element Comprising Same
#5THERAPEUTIC COMPOUNDS AND COMPOSITIONS
#6COMPOUNDS FOR THE REDUCING LIPOTOXIC DAMAGE
#7Antagonists of human integrin α4β7
#8TEAD INHIBITORS
#9THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE
#10MODIFIED EZETIMIBE DRUG FOR CANCER TREATMENT
#11Compounds for the reducing lipotoxic damage
#12BETA-LACTAMS AND THEIR USE AS HERBICIDES
#13Cytotoxic actin-targeting compounds
#14LACTAM-MODIFIED ADENO-ASSOCIATED VIRUS VECTORS
#15ANTAGONISTS OF HUMAN INTEGRIN (ALPHA4)(BETA7)
#16Compounds for the reducing lipotoxic damage
#17SMALL MOLECULE INHIBITORS OF A PROTEIN COMPLEX
#18Therapeutic compounds and compositions
#19Diaryl-B-Lactam Compound and Preparation Method and Pharmaceutical Use Thereof
#20Chiral-substituted poly-N-vinylpyrrolidinones and complexes with bimetallic nanoclusters and uses thereof in asymmetric oxidation reactions
#21Spiro-lactam NMDA receptor modulators and uses thereof
#22Compounds for the reducing lipotoxic damage
#23Therapeutically active compounds and their methods of use
#24Diaryl-B-Lactam Compound and Preparation Method and Pharmaceutical Use Thereof
#25Antagonists of human integrin (α4)(β7)
#26Cytotoxic actin-targeting compounds
#27Necrosis inhibitors
#28Compositions and methods for selective carbonylation of heterocyclic compounds
#29Substituted dihydroindene-4-carboxamides and analogs thereof, and methods using same
#30Therapeutic compounds and compositions
#31Therapeutically active compounds and their methods of use
#32Antagonists of human integrin α4β7
#33Inhibitors of creatine transport and uses thereof
#34Method of preparing ezetimibe and intermediate thereof
#35Spiro-lactam NMDA receptor modulators and uses thereof
#36Beta lactams as modulators of glutamate uptake and methods for use thereof
#37Synthesis of lactams
#38Necrosis inhibitors
#39Therapeutic compounds and compositions
#40Therapeutically active compositions and their methods of use
#41Tricyclic sulfones as ROR gamma modulators
#42Method for preparing azetidinone compound and intermediate of azetidinone compound
#43Peripherally substituted monocyclic beta-lactams
#44Necrosis inhibitors
#45Poly-β-peptides from functionalized β-lactam monomers and antibacterial compositions containing same
#46Method for preparing azetidinone compound and intermediate of azetidinone compound
#47Crystal forms of azetidinone compounds and preparing methods thereof
#48Crystal forms of azetidinone compounds and preparing methods thereof
#49B-LACTAM COMPOUNDS
#50Inhibitors of creatine transport and uses thereof
#51Therapeutic compounds and compositions
#52Therapeutically active compositions and their methods of use
#53METHOD FOR PRODUCING OPTICALLY ACTIVE AZETIDINONE COMPOUND
#54Strain of marine oil-degrading bacteria, compounds obtained by fermentation and their applications
#55Enzymatic process for the preparation of (S)-5-(4-fluoro-phenyl)-5-hydroxy-1morpholin-4-yl-pentan-1-one, an intermediate of ezetimibe and further conversion to ezetimibe
#56Beta lactams as modulators of glutamate uptake and methods for use thereof
#57Compounds useful as immunomodulators
#58N-alkylthio beta-lactams, alkyl-coenzyme A asymmetric disulfides, and aryl-alkyl disulfides as anti-bacterial agents
#59Poly-beta-peptides from functionalized beta-lactam monomers and antibacterial compositions containing same
#60Crystal forms of azetidinone compounds and preparing methods thereof
#61Process for synthesis of ezetimibe and intermediates used in said process
#62Synthetic route for the preparation of β-aminobutyryl substituted 5,6,7,8-tetrahydro[1,4]diazolo[4,3-alpha ]pyrazin-7-yl compounds
#63Synthesis of lactams
#64Taxane compounds, compositions and methods
#65Processes for preparing peptide conjugates and linkers
#66METHOD OF PREPARING EZETIMIBE
#67Taxane compounds, compositions and methods
#68-alkylthio beta-lactams, alkyl-coenzyme A asymmetric disulfides, and aryl-alkyl disulfides as anti-bacterial agents
#69Thio derivatives bearing lactams as potent HDAC inhibitors and their uses as medicaments
#70MULTICOMPONENT CRYSTALLINE SYSTEM OF EZETIMIBE AND PROLINE
#71Chemically Programmed Vaccination
#72N-acyl-β-lactam derivative, macromolecular compound, and photoresist composition
#73Compounds, monomers, and polymers containing a carbonate linkage
#74Securing element, particularly suitable for use with tablet-arm chairs
#75Monobactams
#76Substituted [1,2,4]triazolo[4,3-A]pyrazines for medicaments and pharmaceutical compositions
#77PROCESS FOR THE PREPARATION OF EZETIMIBE AND DERIVATIVES THEREOF
#78Therapeutically active compositions and their methods of use
#79Amide derivative and use thereof as medicine
#80Heterocyclic CETP inhibitors
#81COMBRETASTATIN DERIVATIVES AND USES THEREFOR
#82MONOBACTAMS
#83Taxane compounds, compositions and methods
#84Compounds, pharmaceutical compositions and uses thereof
#85Azetidinone compounds and medical use thereof
#86Method for synthesizing beta lactam compounds by decomposition of an alpha-diazo-beta-ketoamide using a fluorescent light source
#87N-acyl-β-lactam derivative, macromolecular compound, and photoresist composition
#88Process for the synthesis of azetidinones
#89Intermediates in the preparation of 1,4-diphenyl azetidinone
#90Enzymatic process for the preparation of (S)-5-(4-fluoro-phenyl)-5-hydroxy-1morpholin-4-yl-pentan-1-one, an intermediate of Ezetimibe and further conversion to Ezetimibe
#91β-lactam compounds
#92Taxane compounds, compositions and methods
#93Chemically programmed vaccination
#94Poly-β-peptides from functionalized β-lactam monomers and antibacterial compositions containing same
#95PROCESS FOR THE SYNTHESIS OF EZETIMIBE AND INTERMEDIATES USEFUL THEREFOR
#96PROCESS FOR THE SYNTHESIS OF AZETIDINONES
#97EZETIMIBE PROCESS AND COMPOSITION
#98NEW METHODS FOR THE PREPARATION OF TAXANES USING CHIRAL AUXILIARIES
#99NEW METHODS FOR THE PREPARATION OF TAXANES USING CHIRAL AUXILIARIES
#100INTERMEDIATES FOR THE PREPARATION OF (3R, 4S)-1-(4-FLUOROPHENYL)-3-[(3S)-3-(4-FLUOROPHENYL)-3-HYDROXYPROPYL)]-4-(4-HYDROXYPHENYL)-2-AZETIDINONE
#101Ruthenium Catalysts and Uses Thereof
#102Aryl potassium channel blockers and uses thereof
#103Heterocyclic CETP inhibitors
#104Poly-beta-peptides from functionalized beta-lactam monomers and antibacterial compositions containing same
#105NOVEL AZETIDINONES USEFUL AS INHIBITORS OF ELASTASE
#1062-azetidinone derivatives and their use as cholesterol absorption inhibitors for the treatment of hyperlipidaemia
#107PROCESSES FOR PREPARING EZETIMIBE AND INTERMEDIATE COMPOUNDS USEFUL FOR THE PREPARATION THEREOF
#108Novel 2-Azetidinone Derivatives As Cholesterol Absorption Inhibitors For The Treatment Of Hyperlipidaemic Conditions
#109NOVEL DIPHENYLAZETIDINONES, PROCESS FOR THEIR PREPARATION, MEDICAMENTS COMPRISING THESE COMPOUNDS AND THEIR USE
#1102-Azetidinone Derivatives For The Treatment Of Hyperlipidaemic Diseases
#111PHARMACEUTICAL COMPOSITIONS OF POORLY SOLUBLE DRUGS
#112SUBSTITUTED AZETIDINONES
#1132-azetidinone derivatives as cholesterol absorption inhibitors for the treatment of hyperlipidaemic conditions
#114Diphenylazetidinone derivatives possessing cholesterol absorption inhibitory activity
#1151-adamantyl azetidin-2-one derivatives and drugs containing same
#116ANTI-HYPERCHOLESTEROLEMIC COMPOUNDS
#117Processes for the preparation of (3R,4S)-4-((4-benzyloxy)phenyl)-1-(4-fluorophenyl)-3-((S)-3-(4-fluorophenyl)-3-hydroxypropyl)-2-azetidinone, an intermediate for the synthesis of ezetimibe
#118Anti-hypercholesterolemic compounds
#119Substituted beta-lactams
#120NOVEL HYPOCHOLESTEROLEMIC COMPOUNDS
#121NOVEL DIPHENYLAZETIDINONE SUBSTITUTED BY PIPERAZINE-1-SULFONIC ACID AND HAVING IMPROVED PHARMACOLOGICAL PROPERTIES
#122PREPARATION OF BETA-AMINO ACIDS HAVING AFFINITY FOR THE ALPHA-2-DELTA PROTEIN
#123PROCESSES FOR PREPARING INTERMEDIATE COMPOUNDS USEFUL FOR THE PREPARATION OF EZETIMIBE
#124Process for the production of ezetimibe and intermediates used in this process
#125Therapeutic substituted beta-lactams
#126Certain crystalline diphenylazetidinone hydrates, pharmaceutical compositions thereof and methods for their use
#127Therapeutic beta-lactams
#128DIPHENYLHETEROCYCLE CHOLESTEROL ABSORPTION INHIBITORS
#129SUBSTITUTED AZETIDINONES
#130Methods for the preparation of taxanes using chiral auxiliaries
#131Anti-Hypercholesterolemic Compounds
#132BIPHENYLAZETIDINONE CHOLESTEROL ABSORPTION INHIBITORS
#133Processes for Production of 4-(Biphenylyl)Azetidin-2-One Phosphonic Acids
#134Usage of poly-3-hydroxybutyrates in preparation of β-lactam compounds
#135Diphenylazetidinone derivatives possessing cholesterol absorption inhibitor activity
#136Process for preparing optically active alcohols
#137Process for the preparation of ezetimibe
#138Compounds comprising a lactam or a lactam derivative moiety, processes for making them, and their uses
#139DEUTERIUM-ENRICHED EZETIMIBE
#140Process For Production Of 4-Biphenylyazetidin-2-Ones
#141Diphenylazetidinones, process for their preparation, medicaments comprising these compounds and their use
#142Anti-hypercholesterolemic biaryl azetidinone compounds
#143Hydroxy-Substituted Diphenylazetidinones for the Treatment of Hyperlipidemia
#144Novel Substituted Azetidinones
#145Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
#146Processes For Production of Phenolic 4-Biphenylylazetidin-2-Ones
#1474-Biarylyl-1-Phenylazetidin-2-One Glucuronide Derivatives for Hypercholesterolemia
#148Asymmetric disulfides and aryl-alkyl disulfides as anti-bacterial agents
#1494-BIARYLYL-1-PHENYLAZETIDIN-2-ONES
#1504-alkenyl-2-azetidinone derivatives, process for preparing 4-alkenyl-2-azetidinone derivatives and multicyclic compounds prepared using 4-alkenyl-2-azetidinone derivatives
#151Therapeutic β-lactams
#152Diphenylazetidinone derivatives possessing cholesterol absorption inhibitory activity
#153Processes for the purification of (3R,4S)-4-(4-hydroxy-protected-phenyl)-1-(4-fluorophenyl)-3-[3-(4-fluorophenyl)-3-oxopropyl]azetidin-2-one
#154Hypocholesterolemic compounds
#155Processes for the preparation of (3R,4S)-4-((4-benzyloxy)phenyl)-1-(4-fluorophenyl)-3-((S)-3-(4-fluorophenyl)-3-hydroxypropyl)-2-azetidinone, an intermediate for the synthesis of ezetimibe
#156Diphenylazetidinones, process for their preparation, medicaments comprising these compounds and their use
#157Lactams of alkylated acyclic diamine derivatives as modulators of chemokine receptor activity
#158Diphenylazetidinone with improved physiological properties, process for its preparation, medicaments comprising this compound, and its use
#159Tethered dimers and trimers of 1,4-diphenylazetidin-2-ones
#160Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
#161Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
#162Method for producing 1,4-diphenyl azetidinone derivatives
#163Process for the preparation of diphenyl azetidinone derivatives
#164Diphenylazetidinone derivatives possessing chloesterol absorption inhibitory activity
#165Heterocyclic CETP inhibitors
#166Anti-hypercholesterolemic compounds
#167Process for the preparation of chiral azetidinones
#168Acid-group-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use
#169Substituted azetidinones
#170Treatment of diseases associated with the egr-1 enhancer element
#171Poly-β-peptides from functionalized β-lactam monomers and antibacterial compositions containing same
#172Anti-hypercholesterolemic compounds
#173Quaternary salt derivatives of 1,4-diphenylazetidin-2-ones
#174PREPARATION OF EZETIMIBE
#175Novel compounds and compositions as cathepsin inhibitors
#176Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use
#177PROCESS FOR DESILYLATION OF CARBAPENEM INTERMEDIATES
#178Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use
#179Novel dipeptidyl peptidase IV inhibitors used for functionally influencing different cells and treating immunological, infammatory, neuronal, and other diseases
#180Novel taxanes and methods related to use and preparation thereof
#181Resolution of enantiomeric mixtures of beta-lactams
#182β-lactam synthesis
#183Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use
#184Copper-catalyzed formation of carbon-heteroatom and carbon—carbon bonds
#185Intermediate for carbapenem compound for oral administration and process for producing the same
#186Therapeutic substituted β-lactams
#187Novel crystalline form of ezetimibe and processes for the preparation thereof
#188Methods for preventing and treating cancer using -thiolated β-lactam compounds and analogs thereof
#189Ezetimibe polymorphs
#190Process for the synthesis of azetidinones
#191Novel compounds and compositions as cathepsin inhibitors
#192Process for ezetimibe intermediate
#193Bisphenyl compounds useful as vitamin D3 receptor agonists
#194Methods for carbon isotope labeling synthesis by transition metal-promoted carbonylation via isocyanate using azides and carbon-isotope monoxide
#195Anti-hypercholesterolemic compounds
#196Diphenylazetidinones, process for their preparation, medicaments comprising these compounds and their use
#197Process for preparing N-hydroxyformamido-propyl pyrrolidin compounds and intermediates
#198Diphenylazetidinone derivatives for treating disorders of the lipid metabolism
#199Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
#2004-Biarylyl-1-phenylazetidin-2-ones
#201Highly enantiomerically pure lactam-substituted propanoic acid derivatives and methods of making and using same
#202Polymorphs of ezetimibe and process for preparation thereof
#203β-Lactams, methods for the preparation of taxanes, and sidechain-bearing taxanes
#204Cyclisation process for the preparation of c-2 beta-lactam compounds
#205Lactams of alkylated acyclic diamine derivatives as modulators of chemokine receptor activity
#206Diphenylazetidinone with improved physiological properties, process for its preparation, medicaments comprising this compound, and its use