ClassID:

94271

C07D215/227 - CPC Classification

Classification description:

Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms; Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2

Recent Application in this class:
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20260078130
2026-03-19

NAMPT MODULATORS, PREPARATIONS, AND USES THEREOF

#2
20260021085
2026-01-22

CYCLOALKYL CARBOXYLIC ACID DERIVATIVES AS INHIBITORS OF GLYCOGEN SYNTHASE 1 (GYS1) AND METHODS OF USE THEREOF

#3
20260015337
2026-01-15

COMPOUNDS FOR TREATMENT A CORONAVIRUS INFECTION

#4
20250359552
2025-11-27

MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO

#5
20250333371
2025-10-30

COMPOUNDS

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20250313535
2025-10-09

ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF

#7
20250312459
2025-10-09

Pharmaceutical Compositions Having Improved Storage Stability

#8
20250296915
2025-09-25

NOVEL AMINO ACID DERIVATIVES

#9
20250283008
2025-09-11

FLUORINE-CONTAINING ETHER COMPOUND, LUBRICANT FOR MAGNETIC RECORDING MEDIUM, AND MAGNETIC RECORDING MEDIUM

#10
20250214940
2025-07-03

HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHOLOGICAL DISORDERS

#11
20250154106
2025-05-15

ABIETANES AND METHODS OF MAKING AND USING THE SAME

#12
20250154105
2025-05-15

POLYCYCLIC COMPOUND AND USE THEREOF

#13
20250134105
2025-05-01

MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO

#14
20250129045
2025-04-24

SMALL MOLECULE PIM AND MTOR KINASE INHIBITOR AND METHODS OF USE THEREOF

#15
20250122194
2025-04-17

NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS

#16
20250008960
2025-01-09

MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO

#17
20240417377
2024-12-19

COMPOUNDS, COMPOSITIONS, AND METHODS FOR SELECTIVELY INHIBITING ß-GLUCURONIDASES AND ALLEVIATING SIDE EFFECTS ASSOCIATED WITH DRUG TREATMENT INDUCED DIARRHEA

#18
20240400517
2024-12-05

CHIRAL BIMETALLIC COOPERATIVE CATALYSIS SYSTEM AND USE THEREOF IN ASYMMETRIC SYNTHESIS OF BEDAQUILINE

#19
20240360081
2024-10-31

SULFONAMIDE OREXIN RECEPTOR AGONISTS AND USES THEREOF

#20
20240308963
2024-09-19

Low-temperature continuous-flow preparation method of bedaquiline

#21
20240307542
2024-09-19

Pharmaceutical compositions having improved storage stability

#22
20240287022
2024-08-29

IL4I1 INHIBITORS AND METHODS OF USE

#23
20240174665
2024-05-30

CDK2 INHIBITORS AND USES THEREOF

#24
20240174634
2024-05-30

Aldehyde Dehydrogenase Inhibitors and Their Therapeutic Use

#25
20240158339
2024-05-16

TYRAMINE CONTAINING HYDROXYCINNAMIC ACID AMIDE DERIVATIVES AND METHODS OF USE THEREOF

#26
20240140912
2024-05-02

Abietanes and methods of making and using the same

#27
20240010622
2024-01-11

MITOCHONDRIAL ATP INHIBITORS TARGETING THE GAMMA SUBUNIT PREVENT METASTASIS

#28
20240002380
2024-01-04

REV-ERB AGONISTS

#29
20230414625
2023-12-28

Combination Antibacterial Composition and Short-Course Antibacterial Regimen

#30
20230365540
2023-11-16

SMALL MOLECULE INHIBITORS OF ENPP1

#31
20230365488
2023-11-16

TRUXILLIC ACID MONOESTER-DERIVATIVES AS SELECTIVE FABP5 INHIBITORS AND PHARMACEUTICAL COMPOSITIONS AND USES THEREOF

#32
20230322692
2023-10-12

COMPOUND AS PPAR AGONIST AND APPLICATION THEREOF

#33
20230295095
2023-09-21

NOVEL FUSED-HETEROCYCLYL-CARBONOHYDRAZONOYL DICYANIDE COMPOUNDS AND USE THEREOF

#34
20230278962
2023-09-07

Tetrahydrobenzoazepinones and Related Analogs for Inhibiting YAP/TAZ-TEAD

#35
20230242496
2023-08-03

SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA

#36
20230227409
2023-07-20

QUINOLINONE DERIVATIVES AS METHIONINE ADENOSYLTRANSFERASE 2A INHIBITORS

#37
20230180761
2023-06-15

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#38
20230167064
2023-06-01

TREATMENTS OF INFLAMMATORY BOWEL DISEASE

#39
20230150941
2023-05-18

Heterocyclic compounds for the treatment of neurological and psychological disorders

#40
20230113085
2023-04-13

Small molecule inhibitors of TEAD transcription factors

#41
20230040299
2023-02-09

2,3-DISUBSTITUTED 1-ACYL-4-AMINO-1,2,3,4-TETRAHYDROQUINOLINE DERIVATIVES AND THEIR USE AS BROMODOMAIN INHIBITORS

#42
20220315534
2022-10-06

BETA ADRENERGIC AGONIST AND METHODS OF USING THE SAME

#43
20220220075
2022-07-14

SOLID FORM OF AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR

#44
20220204485
2022-06-30

Stabilization of amyloidogenic immunoglobulin light chains

#45
20220125778
2022-04-28

COMPOUNDS, COMPOSITIONS, AND METHODS FOR SELECTIVELY INHIBITING BETA-GLUCURONIDASES AND ALLEVIATING SIDE EFFECTS ASSOCIATED WITH DRUG TREATMENT INDUCED DIARRHEA

#46
20220072133
2022-03-10

Pharmaceutical compositions having improved storage stability

#47
20210395204
2021-12-23

LOW HYGROSCOPIC ARIPIPRAZOLE DRUG SUBSTANCE AND PROCESSES FOR THE PREPARATION THEREOF

#48
20210340106
2021-11-04

Modulators of mas-related g-protein receptor X4 and related products and methods

#49
20210338847
2021-11-04

RADIOLABELLED COMPOUND OF A QUATERNARY AMMONIUM SALT OF A POLYCYCLIC AROMATIC AMINE AND METHODS OF MANUFACTURING AND DIAGNOSTIC USE THEREOF

#50
20210299115
2021-09-30

HETEROARYL INHIBITORS OF PAD4

#51
20210155612
2021-05-27

α,β-unsaturated amide compound

#52
20210147364
2021-05-20

Catalyst bound alpha radical and synthesis of OXO compounds using the same

#53
20210107876
2021-04-15

Histone methyltransferase inhibitors

#54
20210094917
2021-04-01

Compounds, compositions, and methods for selectively inhibiting β-glucuronidases and alleviating side effects associated with drug treatment induced diarrhea

#55
20210070747
2021-03-11

2(1H)-QUINOLINONE DERIVATIVE

#56
20210053967
2021-02-25

Compounds for inhibition of α4 β7 integrin

#57
20210046073
2021-02-18

2,3-disubstituted 1-acyl-4-amino-1,2,3,4-tetrahydroquinoline derivatives and their use as bromodomain inhibitors

#58
20210017100
2021-01-21

Organic reactions carried out in aqueous solution in the presence of a hydroxyalkyl(alkyl)cellulose or an alkylcellulose

#59
20210002229
2021-01-07

Compounds for treatment of PD-L1 diseases

#60
20200407320
2020-12-31

Heterocyclic compounds for the treatment of neurological and psychological disorders

#61
20200377461
2020-12-03

Amine compound for inhibiting SSAO/VAP-1 and use thereof

#62
20200331871
2020-10-22

Method for producing lactam compound, and lactam compound produced thereby

#63
20200331868
2020-10-22

Compound as PPAR agonist and application thereof

#64
20200277277
2020-09-03

Aromatic compound, pharmaceutical composition and use thereof

#65
20200268891
2020-08-27

Pharmaceutical compositions having improved storage stability

#66
20200262805
2020-08-20

Hydrophilic compounds for optically active devices

#67
20200239429
2020-07-30

Aromatic compound, pharmaceutical composition and use thereof

#68
20200237770
2020-07-30

COMBINATION ANTIBACTERIAL COMPOSITION AND SHORT-COURSE ANTIBACTERIAL REGIMEN

#69
20200216430
2020-07-09

Catalyst-free and redox-neutral innate trifluoromethylation and alkylation of (hetero)aromatics enabled by light

#70
20200196607
2020-06-25

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#71
20200172523
2020-06-04

Process and intermediates for the preparation of benzo[b]thiophene compounds

#72
20200148610
2020-05-14

Organic reactions carried out in aqueous solution in the presence of a hydroxyalkyl(alkyl)cellulose or an alkylcellulose

#73
20200138827
2020-05-07

SMALL MOLECULE MODULATORS OF HUMAN STING

#74
20200123110
2020-04-23

LOW HYGROSCOPIC ARIPIPRAZOLE DRUG SUBSTANCE AND PROCESSES FOR THE PREPARATION THEREOF

#75
20200115343
2020-04-16

FUSED-BICYCLIC ARYL QUINOLINONE DERIVATIVES AS MUTANT-ISOCITRATE DEHYDROGENASE INHIBITORS

#76
20200017463
2020-01-16

Process for the preparation of aripiprazole lauroxil

#77
20190375705
2019-12-12

TYRAMINE CONTAINING HYDROXYCINNAMIC ACID AMIDE DERIVATIVES AND METHODS OF USE THEREOF

#78
20190365768
2019-12-05

N-{[2-(piperidin-1-yl)phenyl](phenyl)methyl}-2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-7-yl)acetamide derivatives and related compounds as ROR-gamma modulators for treating autoimmune diseases

#79
20190358216
2019-11-28

Heteroaryl inhibitors of PAD4

#80
20190345162
2019-11-14

Methods and compositions for inhibition of bromodomain-containing proteins

#81
20190331663
2019-10-31

Antibodies to aripiprazole haptens and use thereof

#82
20190276406
2019-09-12

Heterocyclic compounds for the treatment of neurological and psychological disorders

#83
20190275155
2019-09-12

Pharmaceutical compositions having improved storage stability

#84
20190225584
2019-07-25

LOW HYGROSCOPIC ARIPIPRAZOLE DRUG SUBSTANCE AND PROCESSES FOR THE PREPARATION THEREOF

#85
20190210970
2019-07-11

PHENYL QUINOLINONE DERIVATIVES AS MUTANT-ISOCITRATE DEHYDROGENASE INHIBITORS

#86
20190209592
2019-07-11

BICYCLIC ARYL SPHINGOSINE 1-PHOSPHATE ANALOGS

#87
20190202790
2019-07-04

Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#88
20190176134
2019-06-13

Methods of hydrofluorination

#89
20190144450
2019-05-16

Modulators of ATP-binding cassette transporters

#90
20190090488
2019-03-28

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#91
20190084937
2019-03-21

Heterocyclic compounds for the treatment of neurological and psychological disorders

#92
20190071434
2019-03-07

Mutant IDH1 inhibitors useful for treating cancer

#93
20190046511
2019-02-14

Endoparasite control agent

#94
20190040048
2019-02-07

Process and intermediates for the preparation of benzo[b]thiophene compounds

#95
20190000084
2019-01-03

High stress resistant plant growth regulator and preparation method and use thereof

#96
20180344725
2018-12-06

QUINOLONE CHALCONE COMPOUNDS AND USES THEREOF

#97
20180327361
2018-11-15

Phenyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#98
20180312530
2018-11-01

PROCESSES FOR MAKING ALKYLATED ARYLPIPERAZINE AND ALKYLATED ARYLPIPERIDINE COMPOUNDS INCLUDING NOVEL INTERMEDIATES

#99
20180312488
2018-11-01

Heterobicyclic compounds and their use for the treatment of tuberculosis

#100
20180303831
2018-10-25

2,3-disubstituted 1-acyl-4-amino-1,2,3,4-tetrahydroquinoline derivatives and their use as bromodomain inhibitors

#101
20180265473
2018-09-20

Crystal forms of bedaquiline fumarate and preparation methods therefor

#102
20180237410
2018-08-23

Hydrophilic compounds for optically active devices

#103
20180230101
2018-08-16

PROCESS FOR THE PREPARATION OF 5-AMINO-QUINOLIN-2(1H)-ONES AND THEIR TAUTOMER FORMS 5-AMINO-QUINOLIN-2-OLS

#104
20180194732
2018-07-12

Multi-API loading prodrugs

#105
20180186745
2018-07-05

Histone methyltransferase inhibitors

#106
20180162817
2018-06-14

Compounds for optically active devices

#107
20180162816
2018-06-14

Heterocyclic compounds for the treatment of neurological and psychological disorders

#108
20180155359
2018-06-07

SHIP1 MODULATORS AND METHODS RELATED THERETO

#109
20180155290
2018-06-07

Improved Process for the Preparation of Aripiprazole with Reduced Particle Size

#110
20180149637
2018-05-31

Antibodies to aripiprazole haptens and use thereof

#111
20180141921
2018-05-24

Therapeutic compounds

#112
20180141910
2018-05-24

Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#113
20180134715
2018-05-17

Methods and compositions for inhibition of bromodomain-containing proteins

#114
20180133233
2018-05-17

Bicyclic aryl sphingosine 1-phosphate analogs

#115
20180117169
2018-05-03

Haptens of aripiprazole

#116
20180099982
2018-04-12

Processes for making alkylated arylpiperazine and alkylated arylpiperidine compounds including novel intermediates

#117
20180051033
2018-02-22

Inhibitors of Late SV40 Factor (LSF) as cancer chemotherapeutics

#118
20180044297
2018-02-15

2-oxo-3,4-dihydroquinoline compounds as plant growth regulators

#119
20180020662
2018-01-25

Substituted 1-cycloalkyl-2-oxotetrahydroquinolin-6-ylsulfonamides or salts thereof and use thereof to increase stress tolerance in plants

#120
20180016242
2018-01-18

2,4-dioxo-quinazoline-6-sulfonamide derivatives as inhibitors of PARG

#121
20180007911
2018-01-11

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#122
20180007907
2018-01-11

Pesticidally active semi-carbazones and thiosemicarbazones derivatives

#123
20180000944
2018-01-04

Pharmaceutical compositions having improved storage stability

#124
20180000087
2018-01-04

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#125
20170362250
2017-12-21

SHIP1 modulators and methods related thereto

#126
20170349607
2017-12-07

Compounds active towards bromodomains

#127
20170339961
2017-11-30

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#128
20170267639
2017-09-21

Process for synthesizing oxidized lactam compounds

#129
20170253576
2017-09-07

Heterobicyclic compounds and their use for the treatment of tuberculosis

#130
20170247389
2017-08-31

SHIP1 MODULATORS AND METHODS RELATED THERETO

#131
20170239280
2017-08-24

Bicyclic aryl sphingosine 1-phosphate analogs

#132
20170217895
2017-08-03

2-oxo-3,4-dihydroquinolin-6-yl sulphonamide CPDS and their use as plant growth regulators

#133
20170217850
2017-08-03

ORGANIC REACTIONS CARRIED OUT IN AQUEOUS SOLUTION IN THE PRESENCE OF A HYDROXYALKYL(ALKYL)CELLULOSE OR AN ALKYLCELLULOSE

#134
20170204198
2017-07-20

Antibodies to aripiprazole haptens and use thereof

#135
20170166558
2017-06-15

O-GLCNAC TRANSFERASE (OGT) INHIBITORS AND USES THEREOF

#136
20170119753
2017-05-04

Compounds having muscarinic receptor antagonist and BETA2 adrenergic receptor agonist activity

#137
20170088515
2017-03-30

IDENTIFICATION OF COMPOUNDS THAT DISPERSE TDP-43 INCLUSIONS

#138
20170072061
2017-03-16

Haptens of aripiprazole

#139
20170044175
2017-02-16

Inhibitors of late SV40 factor (LSF) as cancer chemotherapeutics

#140
20170035739
2017-02-09

Substituted oxopyridine derivatives and use thereof as factor XIa/plasma

#141
20170015628
2017-01-19

Methods for the preparation of indacaterol and pharmaceutically acceptable salts thereof

#142
20170008859
2017-01-12

Therapeutic compounds

#143
20170001998
2017-01-05

Substituted heterocyclic acetamides as kappa opioid receptor (KOR) agonists

#144
20160318869
2016-11-03

Heterocyclic compounds for the treatment of neurological and psychological disorders

#145
20160311774
2016-10-27

Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#146
20160304522
2016-10-20

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#147
20160302418
2016-10-20

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#148
20160302417
2016-10-20

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#149
20160297767
2016-10-13

Estrogen receptor modulators and uses thereof

#150
20160280671
2016-09-29

Compositions for the treatment of hypertension and/or fibrosis

#151
20160280652
2016-09-29

Arylquinoline and analog compounds and use thereof to treat cancer

#152
20160280651
2016-09-29

COMPOUNDS THAT INDUCE ABA RESPONSES

#153
20160257651
2016-09-08

NOVEL COMPOUND WITH ANTIBACTERIAL ACTIVITY

#154
20160251315
2016-09-01

LOW HYGROSCOPIC ARIPIPRAZOLE DRUG SUBSTANCE AND PROCE3SSES FOR THE PREPARATION THEREOF

#155
20160235734
2016-08-18

Compounds having muscarinic receptor antagonist and BETA2 adrenergic receptor agonist activity

#156
20160214973
2016-07-28

Store overload-induced calcium release inhibitors and methods for producing and using the same

#157
20160194690
2016-07-07

Fluorophore chelated lanthanide luminescent probes with improved quantum efficiency

#158
20160152613
2016-06-02

Substituted oxopyridine derivatives and use thereof as factor xia/plasma

#159
20160137636
2016-05-19

Bicyclic sulfonamide compounds as sodium channel inhibitors

#160
20160136279
2016-05-19

Pharmaceutical compositions having improved storage stability

#161
20160130231
2016-05-12

ROR MODULATORS AND THEIR USES

#162
20160129023
2016-05-12

Bicyclic aryl sphingosine 1-phosphate analogs

#163
20160083349
2016-03-24

Pyridin-2(1H)-one quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#164
20160075708
2016-03-17

Anti-angiogenesis compound, intermediate and use thereof

#165
20160060270
2016-03-03

Aryl-quinoline derivatives

#166
20160052935
2016-02-25

COMPOUNDS FOR USE IN SCREENING METHODS FOR SPINAL MUSCULAR ATROPHY

#167
20160046626
2016-02-18

Bicyclic sulfonamide compounds as sodium channel inhibitors

#168
20160031899
2016-02-04

SHIP1 modulators and methods related thereto

#169
20160024096
2016-01-28

Methods and compositions for inhibition of bromodomain-containing proteins

#170
20160024045
2016-01-28

Chiral compounds, compositions, products and methods employing same

#171
20160024012
2016-01-28

Process for synthesizing oxidized lactam compounds

#172
20160024011
2016-01-28

Multi-API Loading Prodrugs

#173
20160016908
2016-01-21

2,3-disubstituted 1-acyl-4-amino-1,2,3,4-tetrahydroquinoline derivatives and their use as bromodomain inhibitors

#174
20150361099
2015-12-17

Processes for making alkylated arylpiperazine and alkylated arylpiperidine compounds including novel intermediates

#175
20150320875
2015-11-12

Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives

#176
20150316558
2015-11-05

Fluorescent chemical compounds having high selectivity for double stranded DNA, and methods for their use

#177
20150299189
2015-10-22

Amine derivative or salt thereof

#178
20150291531
2015-10-15

Therapeutic hydroxyquinolones

#179
20150274670
2015-10-01

Heterocyclic Compounds for the Treatment of Neurological and Psychological Disorders

#180
20150225347
2015-08-13

Low hygroscopic aripiprazole drug substance and processes for the preparation thereof

#181
20150225346
2015-08-13

Methods for the preparation of indacaterol and pharmaceutically acceptable salts thereof

#182
20150210643
2015-07-30

DERIVATIVES OF 4-(2-AMINO-1-HYDROXYETHYL)PHENOL AS AGONISTS OF THE BETA2 ADRENERGIC RECEPTOR

#183
20150191430
2015-07-09

CONJUGATES OF HUPERZINE AND ANALOGS THEREOF

#184
20150183807
2015-07-02

Compound and asymmetric synthesis reaction

#185
20150183744
2015-07-02

Activators of human pyruvate kinase

#186
20150141409
2015-05-21

Rebamipide prodrugs, preparation method and use thereof

#187
20150105372
2015-04-16

Secondary alcohol quinolinyl modulators of RORγt

#188
20150065480
2015-03-05

MIF inhibitors and their uses

#189
20150057256
2015-02-26

Polymorphic crystal forms of 5-(2-{[6-(2,2-difluoro-2-phenylethoxy)hexyl]amino}-1-(R)-hydroxyethyl)-8-hydroxyquinolin-2(1H)-one, heminapadisytlate as agonist of the β2 adrenergic receptor

#190
20150051205
2015-02-19

Selective β-glucuronidase inhibitors as a treatment for side effects of camptothecin antineoplastic agents

#191
20150047073
2015-02-12

Synthetic compounds for vegetative ABA responses

#192
20150045374
2015-02-12

2-(tert-butoxy)-2-(7-methylquinolin-6-yl) acetic acid derivatives for treating AIDS

#193
20150031685
2015-01-29

Substituted heterocyclic acetamides as kappa opioid receptor (KOR) agonists

#194
20150004597
2015-01-01

Fluorescent chemical compounds having high selectivity for double stranded DNA, and methods for their use

#195
20140371201
2014-12-18

Bicyclic sulfonamide compounds as sodium channel inhibitors

#196
20140343315
2014-11-20

Modulators of ATP-binding cassette transporters

#197
20140343278
2014-11-20

Nitrogen-containing compounds and pharmaceutical compositions thereof for the treatment of atrial fibrillation

#198
20140343277
2014-11-20

NITROGEN-CONTAINING COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS THEREOF FOR THE TREATMENT OF ATRIAL FIBRILLATION

#199
20140343091
2014-11-20

BETA2-adrenoceptor agonists

#200
20140329830
2014-11-06

2-carboxamide-4-piperazinyl-benzofuran derivative

#201
20140323303
2014-10-30

2-(substituted-phenyl)-cyclopentane-1,3-dione compounds, and derivatives thereof

#202
20140322334
2014-10-30

Oral solid preparation comprising aripiprazole and method for producing oral solid preparation comprising aripiprazole

#203
20140309236
2014-10-16

Low hygroscopic aripiprazole drug substance and processes for the preparation thereof

#204
20140309190
2014-10-16

Bicyclic aryl sphingosine 1-phosphate analogs

#205
20140275060
2014-09-18

COMPOUNDS FOR THE TREATMENT OF NEUROLOGIC DISORDERS

#206
20140249306
2014-09-04

HIV replication inhibitor

#207
20140228572
2014-08-14

Method for producing optically active tetrahydroquinolines

#208
20140228310
2014-08-14

Method of modulating stress-activated protein kinase system

#209
20140221423
2014-08-07

Agents and methods for treating ischemic and other diseases

#210
20140193906
2014-07-10

Screening methods for spinal muscular atrophy

#211
20140163206
2014-06-12

Haptens of aripiprazole

#212
20140135344
2014-05-15

Aripiprazole type I microcrystal, aripiprazole solid preparations, and preparation method

#213
20140114071
2014-04-24

Process for the preparation of anhydrous aripiprazole crystal form II

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20140100195
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Fused heterocyclic compounds as ion channel modulators

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Pharmaceutical compositions having improved storage stability

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Identification of compounds that disperse TDP-43 inclusions

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Rebamipide complexes and cocrystals

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NMDA receptor antagonists for neuroprotection

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Viral polymerase inhibitors

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Kappa opioid receptor agonists

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Estrogen receptor modulators and uses thereof

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SKIN LIGHTENING COMPOSITIONS

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Chiral compounds, compositions, products and methods employing same

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2-quinolinyl-acetic acid derivatives as HIV antiviral compounds

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Fluorophore chelated lanthanide luminescent probes with improved quantum efficiency

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TRPV1 antagonists

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Process for making sterile aripiprazole of desired mean particle size

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Aryl-quinoline derivatives

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ACTIVATORS OF HUMAN PYRUVATE KINASE

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Fused heterocyclic compounds as ion channel modulators

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Modulators of ATP-binding cassette transporters

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QUINOLINE DERIVATIVES AS ANTIBACTERIAL AGENTS

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QUINOLINE DERIVATIVES AS ANTIBACTERIAL AGENTS

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Selective beta-glucuronidase inhibitors as a treatment for side effects of camptothecin antineoplastic agents

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Compounds which have activity at Mreceptor and their uses in medicine

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Method of modulating stress-activated protein kinase system

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Nitrogen-containing compounds and pharmaceutical compositions thereof for the treatment of atrial fibrillation

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Quinolinones and quinoxalinones as antibacterial composition

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Viral polymerase inhibitors

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METHODS FOR IDENTIFYING AND USING MarR FAMILY POLYPEPTIDE BINDING COMPOUNDS

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Multi-API Loading Prodrugs

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Bicyclic aryl sphingosine 1-phosphate analogs

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Quinolines and their therapeutic use

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Quinoline derivatives as anti-cancer agents

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Selective inhibitors of CB2 receptor expression and/or activity for the treatment of obesity and obesity-related disorders

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Quinolinone PDE2 inhibitors

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Herbicidal quinoline and 1,8-naphthyridine compounds

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Beta-2-adrenoreceptor agonists

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Herbicides

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Prodrugs of NH-acidic compounds: ester, carbonate, carbamate and phosphonate derivatives

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Ring-fused 2-pyridone derivatives and herbicides

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DI-SUBSTITUTED PHENYL COMPOUNDS

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Glucagon receptor antagonist compounds, compositions containing such compounds and methods of use

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PROCESS FOR MAKING STERILE ARIPIPRAZOLE OF DESIRED MEAN PARTICLE SIZE

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Caspase inhibitors and uses thereof

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NOVEL MYCOBACTERIAL INHIBITORS

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6-alkenyl and 6-phenylalkyl substituted 2-quinolinones and 2-quinoxalinones as poly(ADP-ribose) polymerase inhibitors

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6-pyridin-3-yl-3,4-dihydro-1h-quinolin-2-one derivatives and related compounds as inhibitors of the human aldosterone synthase CYP11B2

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Beta-2-adrenoreceptor agonists

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Oxo-heterocyclic substituted carboxylic acid derivatives and the use thereof

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Viral polymerase inhibitors

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Methods for identifying and using MarR family polypeptide binding compounds

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Heterocyclic compounds for the treatment of neurological and psychological disorders

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Process for preparing anhydrous Aripirazole type I

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TETRAHYDRONAPHTHALENE DERIVATES, PROCESS FOR PREPARING THEM AND THEIR USE AS ANTIINFLAMMATORY AGENTS

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METHOD OF MODULATING STRESS-ACTIVATED PROTEIN KINASE SYSTEM

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Quinolinone derivatives as PARP inhibitors

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New Heterocyclic Derivatives Useful For The Treatment of CNS Disorders

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Amine salt of carbostyril derivative

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METHOD FOR SALT PREPARATION

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Compounds which have activity at Mreceptor and their uses in medicine

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