94371 ⎘
Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms One oxygen or sulfur atom
Sub-classes:NLRP3 INHIBITORS
#2INHIBITORS OF MsbA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
#3INHIBITORS OF MsbA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
#4MODULATORS OF THE INTEGRATED STRESS PATHWAY
#5SULFONIMIDAMIDE COMPOUNDS AS INHIBITORS OF INTERLEUKIN-1 ACTIVITY
#6COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES
#7RXFP1 AGONISTS
#8SULFINYLAMINOBENZAMIDE AND SULFONYLAMINOBENZAMIDE DERIVATIVES
#9HETEROBIFUNCTIONAL COMPOUNDS AND THEIR USE IN TREATING DISEASE
#10SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME
#11COMPOUNDS AND USES THEREOF IN THE TREATMENT AND PREVENTION OF DISEASES AND CONDITIONS ASSOCIATE WITH OR AGGRAVATED BY IMPAIRED MITOPHAGY OR OXIDATIVE STRESS
#12COMPOUND SERVING AS NLRP3 INHIBITOR
#13Small molecule compounds having naphthylamine structure and application thereof
#14PERFLUORINATED AMIDE SALTS AND THEIR USES AS IONIC CONDUCTING MATERIALS
#15Compounds and compositions for treating conditions associated with NLRP activity
#16COMPOUND AS A UBR BOX DOMAIN LIGAND
#17COMPOUND AS A UBR BOX DOMAIN LIGAND
#18[(1,4,5-TRISUBSTITUTED-1H-PYRAZOL-3-YL)SULFANYL]ACETIC ACID DERIVATIVES, SALTS THEREOF, AND USE THEREOF AS ACTIVE HERBICIDAL INGREDIENTS
#192-amino-N-(amino-oxo-aryl-lambda-sulfanylidene)acetamide compounds and their therapeutic use
#20Compounds and compositions for treating conditions associated with NLRP activity
#21COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY
#22Aromatic sulfonamide derivatives
#23AGONISTS OF ROR GAMMAt
#24Sulfonylureas and related compounds and use of same
#25NLRP3 INHIBITORS
#26Alpha-cinnamide compounds and compositions as HDAC8 inhibitors
#27Sulfinylaminobenzamide and sulfonylaminobenzamide derivatives
#28Arylazole compound and pest control agent
#29Compounds
#30TETRALIN AND INDANE DERIVATIVES AND USES THEREOF
#31Sulfonimidamide compounds as inhibitors of interleukin-1 activity
#32DISUBSTITUTED 5(3)-PYRAZOLE CARBOXYLATES AND A PROCESS FOR THEIR PREPARATION FROM ENOLATES AND FLUOROALKYLAMINOREAGENTS (FAR) REAGENTS
#33Method for producing a polymorphic form of 3-[5-amino-4-(3-cyanobenzoyl)-pyrazol-1-yl]-N-cyclopropyl-4-methylbenzamide
#34Compounds and compositions for treating conditions associated with NLRP activity
#35Neprilysin inhibitors
#36Sulfonylureas and sulfonylthioureas as NLRPinhibitors
#37NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS
#38DISUBSTITUTED 3-PYRAZOLE CARBOXYLATES AND A PROCESS FOR THEIR PREPARATION VIA ACYLATION OF ENOLATES
#39Pyrazole compounds and preparation thereof
#40N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#41Compounds
#42HALOGEN SUBSTITUTED DIKETONES, PYRAZOLE COMPOUNDS AND PROCESSES FOR THE MANUFACTURE OF PYRAZOLE COMPOUNDS
#43Sulfonyl acetamides as NLRP3 inhibitors
#44Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto
#45Substituted heterocycles as c-MYC targeting agents
#46NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS
#47Compounds
#48Methods and compositions for treatment of muscle wasting, muscle weakness, and/or cachexia
#49Alpha-cinnamide compounds and compositions as HDAC8 inhibitors
#50Sulfonamide carboxamide compounds
#51Pyrazole compound
#52GLYCOLATE OXIDASE INHIBITORS AND METHODS OF USE FOR THE TREATMENT OF KIDNEY STONES
#53SULFONAMIDE OR AMIDE COMPOUNDS, COMPOSITIONS AND METHODS FOR THE PROPHYLAXIS AND/OR TREATMENT OF AUTOIMMUNE, INFLAMMATION OR INFECTION RELATED DISORDERS
#54High solubility thioether quinones
#55Spiroheptane salicylamides and related compounds as inhibitors of ROCK
#56TETRALIN AND INDANE DERIVATIVES AND USES THEREOF
#57N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#58HALOALLYLAMINE PYRAZOLE DERIVATIVE INHIBITORS OF LYSYL OXIDASES AND USES THEREOF
#59Neprilysin inhibitors
#60Sulfinylaminobenzamide and sulfonylaminobenzamide derivatives
#61Sulfonylureas and related compounds and use of same
#62Method for producing a polymorphic form of 3-[5-amino-4-(3- cyanobenzoyl)-pyrazol-1-yl]-N-cyclopropyl-4-methylbenzamide
#63Amide compounds and use thereof
#64Electrophotographic photosensitive member, process cartridge, and image forming apparatus
#65Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto
#66N-methyl-N-(1-phenyl-2-(1-pyrrolidinyl)ethyl)-2-aminophenylacetamide derivatives agonists for the κ opioid receptor
#67Alpha-cinnamide compounds and compositions as HDAC8 inhibitors
#68Pyridyl reverse sulfonamides for HBV treatment
#69N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#70Compounds and compositions for treating conditions associated with NLRP activity
#71Aromatic sulfonamide derivatives
#72Pyrazole compound
#73Substituted heterocycles as c-MYC targeting agents
#74High-solubility thioether quinones
#75Halogen substituted diketones, pyrazole compounds and processes for the manufacture of pyrazole compounds
#76Selective androgen receptor degrader (SARD) ligands and methods of use thereof
#77Arylazole compound and pest control agent
#78Neprilysin inhibitors
#79TETRALIN AND INDANE DERIVATIVES AND USES THEREOF
#80Alpha-cinnamide compounds and compositions as HDAC8 inhibitors
#81Pyrazole compound
#82N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#83Penflufen polymer particles
#84Tricyclic sulfones as ROR gamma modulators
#85Pyrazole compounds or salts thereof, preparation method therefor, herbicidal composition and use thereof
#86Pyridyl reverse sulfonamides for HBV treatment
#87Neprilysin inhibitors
#88Sulfonylureas and related compounds and use of same
#89ALPHA-CINNAMIDE COMPOUNDS AND COMPOSITIONS AS HDAC8 INHIBITORS
#90FUNGICIDAL PYRAZOLES
#91Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto
#92N-methyl-N-(1-phenyl-2-(1-pyrrolidinyl)ethyl)-2-aminophenylacetamide derivatives agonists for the kappa opioid receptor
#93Neprilysin inhibitors
#94Substituted pyrazolone compounds for use in treatment of amyotrophic lateral sclerosis
#95TETRACYCLINE COMPOUNDS
#96N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#97SUBSTITUTED HETEROCYCLES AS c-MYC TARGETING AGENTS
#98TETRALIN AND INDANE DERIVATIVES AND USES THEREOF
#99Pyridinyloxy- and phenyloxy-pyrazolyl compounds
#100Halogen-substituted compounds
#101Pyrazole compound
#102DERIVATIVES OF N-(ARYLAMINO) SULFONAMIDES AS INHIBITORS OF MEK
#103Small molecule inhibitors of G protein coupled receptor 6 kinases polypeptides
#104N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#105Neprilysin inhibitors
#106Endoparasite control agent and method for using the same
#107Heteroaryl disulfide compounds as allosteric effectors for increasing the oxygen-binding affinity of hemoglobin
#108Fluorophenyl pyrazol compounds
#109Alpha-cinnamide compounds and compositions as HDAC8 inhibitors
#1101,2- bis-sulfonamide derivatives as chemokine receptor modulators
#111Fungicidal pyrazoles
#112Pyridyl reverse sulfonamides for HBV treatment
#113Treatment of amyotrophic lateral sclerosis
#114Apoptosis-inducing agent for the treatment of cancer and immune and autoimmune diseases
#115Neprilysin inhibitors
#116Compounds that modulate intracellular calcium
#117Halogen-substituted pyrazole derivatives as pest-control agents
#118Glucagon receptor modulators
#119Tetralin and indane derivatives and uses thereof
#120Endoparasite control agent and method for using the same
#121Potassium channel blockers
#122Neprilysin inhibitors
#123Compound having ability to inhibit 11Beta-HSD1 enzyme or pharmaceutically acceptable salt thereof, method for producing same, and pharmaceutical composition containing same as active ingredient
#124Substituted sulfonamide compounds
#125Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto
#1261-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof
#127Bicyclic sulfone compounds for inhibition of RORgamma activity and the treatment of disease
#128Processes for the preparation of 1-aryl-5-alkyl pyrazole compounds
#129Methods and compositions for treatment of fibrosis
#130Methods and compositions for treatment of muscle wasting, muscle weakness, and/or cachexia
#131CFO-containing enaminoketones and their utilization for the preparation of CFO-containing pyrazoles
#132DERIVATIVES OF N-(ARYLAMINO) SULFONAMIDES AS INHIBITORS OF MEK
#133Glucagon receptor modulators
#134Neprilysin inhibitors
#135Process for the preparation of N-substituted pyrazole compounds
#136Pyrazole compound
#137Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
#138Sulfonyl semicarbazides, semicarbazides and ureas, pharmaceutical compositions thereof, and methods for treating hemorrhagic fever viruses, including infections associated with arenaviruses
#139Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
#140Compounds that modulate intracellular calcium
#141Fungicidal pyrazoles
#142Potassium channel blockers
#143ATGListatin and pharmaceutical composition comprising the same
#144Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto
#145Acylamino-substituted cyclic carboxylic acid derivatives and their use as pharmaceuticals
#146N-(3-carbamoylphenly)-1H-pyrazole-5-carboxamide derivatives and the use thereof for controlling animal pests
#147O-cyclopropylcyclohexyl-carboxanilides and their use as fungicides
#148Thienopyrazole derivative having PDE7 inhibitory activity
#149HETEROCYCLIC COMPOUNDS AND THROMBOPOIETIN RECEPTOR ACTIVATORS
#150Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy
#151Neprilysin inhibitors
#1521-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof
#153Glucagon receptor modulators
#154Processes for the preparation of 1-aryl-5-alkyl pyrazole compounds
#155Neprilysin inhibitors
#156Substituted N-(2-arylamino)aryl sulfonamide-containing combinations
#157LIPASE INHIBITORS
#158Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
#159Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy
#160Fungicidal pyrazoles
#161Pyrazole compounds that modulate HSP90 activity
#162HETEROCYCLIC COMPOUNDS AND THROMBOPOIETIN RECEPTOR ACTIVATORS
#163Acylamino-substituted cyclic carboxylic acid derivatives and their use as pharmaceuticals
#164Compounds that interact with glucokinase regulatory protein for the treatment of diabetes
#165Neprilysin inhibitors
#166Fused heterocyclic compounds and thrombopoietin receptor activators
#167Tetracycline compounds
#168Glucagon receptor modulators
#169Pyrazole-based thyroid receptor compounds
#170Indane derivatives
#171UREA SUBSTITUTED SULPHONAMIDE DERIVATIVES
#1721,2-bis-sulfonamide derivatives as chemokine receptor modulators
#173SORTASE A INHIBITORS
#174Compounds, Compositions and Methods for Modulating Uric Acid Levels
#175Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
#176Tetralin and indane derivatives and uses thereof
#177Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
#178Derivatives of N-acyl-N′-phenylpiperazine useful (inter alia) for the prophylaxis or treatment of diabetes
#179Sulfonamide compounds for the treatment of respiratory disorders
#180Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
#181Pyrazole Derivatives
#182Derivatives of N-(arylamino)sulfonamides as inhibitors of MEK
#183Fungicidal N-(Phenylcycloalkyl)carboxamide, N-(Benzylcycloalkyl)carboxamide and thiocarboxamide derivatives
#184N-Hydroxylsulfonamide Derivatives as New Physiologically Useful Nitroxyl Donors
#185Dimeric 1-arylpyrazole derivatives for use against ectoparasites, agricultural pests, and household pests
#186Pyrazole derivatives as 11-beta-HSD1 inhibitors
#187PYRAZOLYL SUBSTITUTED CARBONIC ACID DERIVATIVES AS MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO
#188Insecticidal 4-phenyl-1H-pyrazoles
#189THIENOPYRAZOLE DERIVATIVE HAVING PDE7 INHIBITORY ACTIVITY
#190Pyrazole compounds that modulate HSP90 activity
#191PYRAZOLE DERIVATIVES USEFUL AS INHIBITORS OF FAAH
#192Indane derivatives as AMPA receptor modulators
#193Heterocyclic compounds and thrombopoietin receptor activators
#194SUBSTITUTED PHENYLAMINO-BENZENE DERIVATIVES USEFUL FOR TREATING HYPER-PROLIFERATIVE DISORDERS AND DISEASES ASSOCIATED WITH MITOGEN EXTRACELLULAR KINASE ACTIVITY
#195Heterocyclic compounds as factor IXA inhibitors
#196SUBSTITUTED PHENOXYBENZAMIDES
#197Aminotetraline derivatives, pharmaceutical compositions containing them, and their use in therapy
#198N-HETEROCYCLYLPHENYL-SUBSTITUTED CYCLIC KETOENOLS
#1991-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof
#200Nitrogen-containing heterocyclic derivative having 11β-hydroxysteroid dehydrogenase type I inhibitory activity
#201Substituted piperazines
#2025-Membered heterocyclic compound
#203INHIBITORS FOR DISRUPTING THE INTERACTION OF UBIQUITINATION RELATED ENZYMES AND USES THEREOF
#204Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
#205Thyroid like compounds
#206HETEROCYCLE-SUBSTITUTED, N-PHENYL-PHTHALAMIDE DERIVATIVES, RELATED COMPOUNDS AND THEIR USE AS INSECTICIDES
#207Potassium channel blockers
#208Potassium channel blockers
#209Potassium channel blockers
#210PYRAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY
#211Cyclohexanesulfonyl derivatives as GLYT1 inhibitors to treat schizophrenia
#212BIARYL SULFONAMIDE DERIVATIVES
#213PYRAZOLE COMPOUND
#214Fluoro- and trifluoroalkyl-containing heterocyclic sulfonamide inhibitors of beta amyloid production and derivatives thereof
#215Chemical compounds
#216Pyrazole derivatives
#217Sulfonyl semicarbazides, semicarbazides and ureas, pharmaceutical compositions thereof, and methods for treating hemorrhagic fever viruses, including infections associated with arena viruses
#218Substituted arylpyrazoles
#219Heterocyclic compounds having type I 11β hydroxysteroid dehydrogenase inhibitory activity
#2205-Membered heterocyclic compound
#221TRICYCLIC STEROID HORMONE NUCLEAR RECEPTOR MODULATORS
#222Non-nucleoside reverse transcriptase inhibitors
#223Amide compound and thrombopoietin receptor activator
#224Histamine-3 receptor antagonists
#225Thienopyrazole derivative having PDE7 inhibitory activity
#226Compounds Useful in Therapy
#227Novel Sulphonamide Derivatives as Glucocorticoid Receptor Modulators for the Treatment of Inflammatory Diseases
#228Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK
#229Substituted phenylamino-benzene derivatives useful for treating hyper-proliferative disorders and diseases associated with mitogen extracellular kinase activity
#230Pyrazole compounds having cannabinoid receptor (CB1) antagonizing activity
#231Tetralin and indane derivatives and uses thereof
#232Substituted piperazines
#233Cannabinoid Receptor Modulators
#234Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
#2353-(2-Hydroxyphenyl) Pyrazoles and Thier Use as Hsp90 Modulators
#236Thione derivative, method for the preparation thereof, and pharmaceutical composition containing the same
#2371H-pyrazoles useful in therapy
#238Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK
#239Viral polymerase inhibitors
#2401-aryl-5-alkyl pyrazole derivative compounds, processes of making and methods of using thereof
#241Heterocyclic compounds and thrombopoietin receptor activators
#242N-hydroxylsulfonamide derivatives as new physiologically useful nitroxyl donors
#243Heterocycle-substituted n-phenyl-phthalamide derivatives, related compounds and their use as insecticides
#244Process for Preparing Bicyclic Pyrazolyl
#245Fluoro- and trifluoroalkyl-containing heterocyclic sulfonamide inhibitors of beta amyloid production and derivatives thereof
#246ABCA1 elevating compounds
#247SMALL-MOLECULES FOR TREATING CANCER AND ABNORMAL CELL PROLIFERATION DISORDERS
#248Pyrazole compounds that modulate HSP90 activity
#249Method for the production of tetrahydrogeranylacetone
#2501H-pyrazoles useful in therapy
#251Substituted arylpyrazoles
#252Cyclohexanesulfonyl derivatives as GlyT1 inhibitors to treat schizophrenia
#253Aryl and heteroaryl compounds and methods to modulate coagulation
#254Compounds useful in therapy
#255Hydroxysteroid dehydrogenase inhibitors
#256Sulfonamide derivatives as PPAR modulators
#257Pyrazole compounds useful in the treatment of inflammation
#258Tetralin and indane derivatives and uses thereof
#259N-heterocyclyl phenyl-substituted cyclic ketoenols
#260Cinnamide and hydrocinnamide derivatives with kinase inhibitory activity
#261PARP inhibitors
#262Hexafluoroisopropanol substituted cyclohexane derivatives
#2633-cyclopropyl-4-(3-amino-2-methylbenzoyl)pyrazoles and their use as herbicides
#264Substituted piperazines
#265Heterocyclic compounds and thrombopoietin receptor activators
#266Tricyclic steroid hormone nuclear receptor modulators
#267Pyrazole derivatives
#268Non nucleoside reverse transcriptase inhibitors
#269Novel piperidine and piperazine derivatives
#270Sulphones for inhibition of gamma secretase
#271Substituted piperazines
#2723-Heterocyclyl substituted benzoic acid derivatives
#273Novel benzohydrazide derivatives as herbicides and desiccant compositions contaning them
#274Inhibitors of HCV NS5B polymerase
#275Tetrahydropyridazine derivatives and their use as pesticides
#276Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials
#2774-Sulfide/sulfoxide/sulfonyl-1h-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
#2781H-pyrazolyl derivative compounds, for use in diseases associated with the 5-ht2c receptor
#279Perfluorinated amide salts and their uses as ionic conducting materials
#280Pyrazole derivatives