ClassID:

94565

C07D243/24 - CPC Classification

Classification description:

Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems 1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms Oxygen atoms

Recent Application in this class:
#1
20260152473
2026-06-04

POLYMORPHS OF BIS(FLUOROALKYL)-1,4-BENZODIAZEPINONE COMPOUNDS AND USES THEREOF

#2
20260070912
2026-03-12

BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM

#3
20250388586
2025-12-25

NEW BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM

#4
20250346565
2025-11-13

METHODS OF PREPARING CHIRAL BENZODIAZEPINONE DERIVATIVES

#5
20250313537
2025-10-09

BENZODIAZEPINE ANALOGS AND METHODS OF USE IN TREATING CANCER

#6
20250236597
2025-07-24

DEUTERATED BENZODIAZEPINE ANALOGS AND METHODS OF USE IN TREATING CANCER

#7
20250197360
2025-06-19

NOVEL DIAZEPINES THAT TARGET YELLOW FEVER VIRUS NON-STRUCTURAL 4B (NS4B) PROTEIN AND THEIR METHOD OF USE

#8
20250019351
2025-01-16

COMPOSITIONS AND METHODS FOR REDUCING TACTILE DYSFUNCTION, ANXIETY, AND SOCIAL IMPAIRMENT

#9
20230357167
2023-11-09

POLYMORPHS OF BIS(FLUOROALKYL)-1,4-BENZODIAZEPINONE COMPOUNDS AND USES THEREOF

#10
20230142171
2023-05-11

NEW BENZODIAZEPINE DERIVATIVES AS GABA A GAMMA1 PAM

#11
20230108536
2023-04-06

METHODS OF PREPARING CHIRAL BENZODIAZEPINONE DERIVATIVES

#12
20220323460
2022-10-13

Combination pharmaceutical agents as RSV inhibitors

#13
20220162173
2022-05-26

Compositions and methods for reducing tactile dysfunction, anxiety, and social impairment

#14
20220073474
2022-03-10

Crystalline form of propoxazepam, the method of its making and use as medicinal agent

#15
20220040198
2022-02-10

COMPOSITIONS COMPRISING SHORT-ACTING BENZODIAZEPINES

#16
20210309617
2021-10-07

Inhibition of respiratory complex III by ligands that interact with a regulatory switch

#17
20210163490
2021-06-03

PERIPHERALLY RESTRICTED GABA POSITIVE ALLOSTERIC MODULATORS FOR THE TREATMENT OF IRRITABLE BOWEL SYNDROME AND OTHER AILMENTS OF THE PERIPHERAL NERVOUS SYSTEM

#18
20210017138
2021-01-21

Antiviral benzodiazepine compounds

#19
20200361878
2020-11-19

1,4-benzodiazepin-2-one derivatives and use thereof

#20
20200181155
2020-06-11

Peripherally restricted GABA positive allosteric modulators for the treatment of irritable bowel syndrome and other ailments of the peripheral nervous system

#21
20200062759
2020-02-27

Peripherally restricted GABA positive allosteric modulators for the treatment of irritable bowel syndrome and other ailments of the peripheral nervous system

#22
20190256478
2019-08-22

1,3-dihydro-1,4-benzodiazepine-2-thiones for the treatment of CNS related diseases

#23
20190192535
2019-06-27

Combination pharmaceutical agents as RSV inhibitors

#24
20170312292
2017-11-02

Therapeutic compounds and uses thereof

#25
20170233386
2017-08-17

Compounds Which Have a Protective Activity with Respect to the Action of Toxins and of Viruses with an Intracellular Mode of Action

#26
20170197967
2017-07-13

Peripherally restricted GABA positive allosteric modulators for the treatment of irritable bowel syndrome and other ailments of the peripheral nervous system

#27
20160347744
2016-12-01

Fused heterocyclic compounds as ion channel modulators

#28
20160311783
2016-10-27

Benzodiazepine derivatives for use in the treatment of Chlamydiales infections

#29
20160096846
2016-04-07

Fused heterocyclic compounds as ion channel modulators

#30
20160060232
2016-03-03

BIS(FLUOROALKYL)-1,4-BENZODIAZEPINONE COMPOUNDS

#31
20150284342
2015-10-08

BIS(FLUOROALKYL)-1,4-BENZODIAZEPINONE COMPOUNDS

#32
20150239851
2015-08-27

Alkyl, fluoroalkyl-1,4-benzodiazepinone compounds

#33
20150232491
2015-08-20

Prodrugs of 1,4-benzodiazepinone compounds

#34
20150231152
2015-08-20

Fluoroalkyl and fluorocycloalkyl 1,4-benzodiazepinone compounds

#35
20150218111
2015-08-06

Fluoroalkyl-1,4-benzodiazepinone compounds

#36
20150166489
2015-06-18

Bis(fluoroalkyl)-1,4-benzodiazepinone compounds and prodrugs thereof

#37
20150011537
2015-01-08

Benzodiazepine compounds with anti-flavivirus activity

#38
20140357605
2014-12-04

BIS(FLUOROALKYL)-1,4-BENZODIAZEPINONE COMPOUNDS

#39
20140135317
2014-05-15

Fused heterocyclic compounds as ion channel modulators

#40
20140100365
2014-04-10

Bisfluoroalkyl-1,4-benzodiazepinone compounds

#41
20140087992
2014-03-27

Bis(fluoroalkyl)-1,4-benzodiazepinone compounds and prodrugs thereof

#42
20140073633
2014-03-13

Inhibitors of the shiga toxins trafficking through the retrograde pathway

#43
20140038947
2014-02-06

Therapeutic applications of pro-apoptotic benzodiazepines

#44
20140011988
2014-01-09

Dibenzo[b,f][1,4]oxazepin-11-yl-N-hydroxybenzamides as HDAC inhibitors

#45
20130274197
2013-10-17

Benzodiazepinone compounds useful in the treatment of skin conditions

#46
20130190300
2013-07-25

Compositions and methods for inhibiting the proliferation of cells

#47
20130172550
2013-07-04

P2Xreceptor antagonist

#48
20130012492
2013-01-10

Fused heterocyclic compounds as ion channel modulators

#49
20120289498
2012-11-15

Compositions And Methods Relating To Novel Compounds And Targets Thereof

#50
20120283249
2012-11-08

Novel compounds which have a protective activity with respect to the action of toxins and of viruses with an intracellular mode of action

#51
20120245151
2012-09-27

Bisfluoroalkyl-1,4-benzodiazepinone compounds

#52
20120232067
2012-09-13

Benzodiazepinone compounds and methods of treatment using same

#53
20120214801
2012-08-23

COMPOSITIONS AND METHODS RELATING TO NOVEL COMPOUNDS AND TARGETS THEREOF

#54
20120116073
2012-05-10

P2X4 RECEPTOR ANTAGONIST

#55
20120077805
2012-03-29

UNSOLVATED BENZODIAZEPINE COMPOSITIONS AND METHODS

#56
20120040971
2012-02-16

Benzodiazepinone compounds useful in the treatment of skin conditions

#57
20120015938
2012-01-19

1,4-BENZODIAZEPIN-2-ON DERIVATIVES

#58
20110245238
2011-10-06

Novel Soluble 1,4 Benzodiazepine Compounds and Stable Salts Thereof

#59
20110201601
2011-08-18

Inhibitors of the Shiga toxins trafficking through the retrograde pathway

#60
20110196147
2011-08-11

INHIBITORS OF HISTONE DEACETYLASE

#61
20110195959
2011-08-11

Compositions and methods relating to novel compounds and targets thereof

#62
20110059043
2011-03-10

CHEMICAL COMPOUNDS

#63
20110009393
2011-01-13

Novel Soluble 1,4 Benzodiazepine Compounds and Stable Salts Thereof

#64
20100331316
2010-12-30

5-phenyl-1H-benzo [E] [1,4] diazepine compounds substituted with an hydroxamic acid group as histone deacetylase inhibitors

#65
20100317619
2010-12-16

Selective agents for pain suppression

#66
20100256123
2010-10-07

P2X4 RECEPTOR ANTAGONIST

#67
20100130481
2010-05-27

ANTICONVULSANT AND ANXIOLYTIC METHODS OF USING RECEPTOR SUBTYPE SELECTIVE AGENTS

#68
20100069373
2010-03-18

SUBSTITUTED LACTAMS AS INHIBITORS OF A BETA PROTEIN PRODUCTION

#69
20100056501
2010-03-04

SUBSTITUTED LACTAMS AS INHIBITORS OF ABETA PROTEIN PRODUCTION

#70
20100048541
2010-02-25

SUBSTITUTED LACTAMS AS INHIBITORS OF ABETA PROTEIN PRODUCTION

#71
20100041639
2010-02-18

CYCLIC MALONAMIDES AS INHIBITORS OF A BETA PROTEIN PRODUCTION

#72
20100015063
2010-01-21

Benzodiazepine derivatives and pharmaceutical compositions containing them

#73
20100009966
2010-01-14

SUBSTITUTED LACTAMS AS INHIBITORS OF ABETA PROTEIN PRODUCTION

#74
20100009965
2010-01-14

CYCLIC MALONAMIDES AS INHIBITORS OF ABETA PROTEIN PRODUCTION

#75
20100004227
2010-01-07

Compositions and methods relating to novel compounds and targets thereof

#76
20100004226
2010-01-07

STEREOSPECIFIC ANXIOLYTIC AND ANTICONVULSANT AGENTS WITH REDUCED MUSCLE-RELAXANT, SEDATIVE-HYPNOTIC AND ATAXIC EFFECTS

#77
20090318427
2009-12-24

Benzodiazepine derivatives for treating hepatitis C infection

#78
20090264419
2009-10-22

CYCLIC MALONAMIDES AS INHIBITORS OF Abeta PROTEIN PRODUCTION

#79
20090253686
2009-10-08

Unsolvated benzodiazepine compositions and methods

#80
20090215752
2009-08-27

Compounds, preparation and therapeutic use thereof

#81
20090208413
2009-08-20

Registry method and control system for DEA schedule II-V medicines

#82
20090203901
2009-08-13

Process for preparing pyrazole functionalized benzodiazepinones

#83
20090170831
2009-07-02

Substituted lactams as inhibitors of Aβ protein production

#84
20090163478
2009-06-25

Salts and crystal modifications thereof

#85
20090137562
2009-05-28

SUBSTITUTED BENZYL AMINE COMPOUNDS

#86
20090118244
2009-05-07

Benzodiazepinone compounds useful in the treatment of skin conditions

#87
20090111793
2009-04-30

HYDROXYALKANOYLAMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF A BETA PROTEIN PRODUCTION

#88
20090069293
2009-03-12

SUCCINOYLAMINO BENZODIAZEPINES AS INHIBITORS OF AB PROTEIN PRODUCTION

#89
20090062256
2009-03-05

LACTAMS SUBSTITUTED BY CYCLIC SUCCINATES AS INHIBITORS OF Abeta PROTEIN PRODUCTION

#90
20090012065
2009-01-08

Therapeutic applications of pro-apoptotic benzodiazepines

#91
20080293700
2008-11-27

Compositions and Methods Relating to Novel Compounds and Targets Thereof

#92
20080293692
2008-11-27

Succinoylamino lactams as inhibitors of a-β protein production

#93
20080275024
2008-11-06

Cyclic malonamides as inhibitors of aβ protein production

#94
20080269194
2008-10-30

Compositions and methods relating to novel compounds and targets thereof

#95
20080261957
2008-10-23

Dihydro-benzo[B][1,4]diazepin-2-one sulfonamide derivatives

#96
20080221087
2008-09-11

Substituted lactams as inhibitors of Aβ protein production

#97
20080207602
2008-08-28

Succinoylamino benzodiazepines as inhibitors of aβ protein production

#98
20080207590
2008-08-28

Dibenzo[b,f][1,4]oxazepin-11-yl-N-hydroxybenzamides as HDAC inhibitors

#99
20080171735
2008-07-17

SUCCINOYLAMINO BENZODIAZEPINES AS INHIBITORS OF Abeta PROTEIN PRODUCTION

#100
20080139536
2008-06-12

Benzodiazepines for Treating or Preventing Rsv Infection

#101
20080132482
2008-06-05

Hydroxyalkanoylaminolactams and related structures as inhibitors of aβ protein production

#102
20080108605
2008-05-08

ANXIOLYTIC AGENTS WITH REDUCED SEDATIVE AND ATAXIC EFFECTS

#103
20080103128
2008-05-01

Lactams substituted by cyclic succinates as inhibitors of Aβ protein production

#104
20080085891
2008-04-10

Asthma and allergic inflammation modulators

#105
20080064686
2008-03-13

Soluble 1,4 benzodiazepine compounds and stable salts thereof

#106
20080045509
2008-02-21

Substituted benzyl amine compounds

#107
20080021014
2008-01-24

Cyclic malonamides as inhibitors of Aβ protein production

#108
20070299059
2007-12-27

Compostions and methods relating to novel compounds and targets thereof

#109
20070299058
2007-12-27

Anxiolytic Agents With Reduced Sedative And Ataxic Effects

#110
20070293482
2007-12-20

Process for Preparing Benzodiazepines

#111
20070265193
2007-11-15

Tetraazabenzo[e]azulene derivatives and analogs thereof

#112
20070185094
2007-08-09

Novel 3-substitued-1,4-benzodiazepines

#113
20070173491
2007-07-26

Substituted lactams as inhibitors of Aβ protein production

#114
20070155730
2007-07-05

Benzodiazepine And Benzopiperazine Analog Inhibitors Of Histone Deacetylase

#115
20070135418
2007-06-14

Compositions and methods for inhibiting the proliferation of cells

#116
20070123519
2007-05-31

Benzo-1,4-diazepin-2-one derivatives as phosphodiesterase PDE2 inhibitors, preparation and therapeutic use thereof

#117
20070093485
2007-04-26

Substituted n-phenyl sulfonamide bradykinin antagonists

#118
20070054881
2007-03-08

Anxiolytic agents with reduced sedative and ataxic effects

#119
20070049580
2007-03-01

ANXIOLYTIC AGENTS WITH REDUCED SEDATIVE AND ATAXIC EFFECTS

#120
20070043033
2007-02-22

Unsolvated benzodiazepine compositions and methods

#121
20070036854
2007-02-15

Therapeutic applications of pro-apoptotic benzodiazepines

#122
20070027132
2007-02-01

Hydroxyalkanoylaminolactams and related structures as inhibitors of Aβ protein production

#123
20060264417
2006-11-23

Succinoylamino lactams as inhibitors of Aβ protein production

#124
20060258638
2006-11-16

Succinoylamino lactams as inhibitors of Aβ protein production

#125
20060217362
2006-09-28

Novel compounds useful for bradykinin B1 receptor antagonism

#126
20060211679
2006-09-21

Substituted lactams as inhibitors of Abeta protein production

#127
20060135762
2006-06-22

Cyclic malonamides as inhibitors of Aβ protein protection

#128
20060128695
2006-06-15

Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses

#129
20060122169
2006-06-08

Succinoylamino benzodiazepines as inhibitors of Aβ protein production

#130
20060040923
2006-02-23

Benzodiazepine derivatives and pharmaceutical compositions containing them

#131
20060030553
2006-02-09

Cell adhesion inhibitors

#132
20060025407
2006-02-02

Succinoylaminobenzodiazepines as inhibitors of Aβ protein production

#133
20060024832
2006-02-02

Water-soluble derivatives of lipophilic drugs

#134
20060003995
2006-01-05

Stereospecific anxiolytic and anticonvulsant agents with reduced muscle-relaxant, sedative-hypnotic and ataxic effects

#135
20050267100
2005-12-01

Tetraazabenzo[e]azulene derivatives and analogs thereof

#136
20050261318
2005-11-24

Protein kinase inhibitors

#137
20050261274
2005-11-24

Lactams substituted by cyclic succinates as inhibitors of Aβ protein production

#138
20050261176
2005-11-24

Compositions and methods relating to novel compounds and targets thereof

#139
20050245501
2005-11-03

Succinoylamino lactams as inhibitors of A-β protein production

#140
20050234039
2005-10-20

Substituted lactams as inhibitors of Aβ protein production

#141
20050176699
2005-08-11

Benzodiazepine derivatives, preparation thereof and use thereof

#142
20050124605
2005-06-09

Benzo-fused heterocycles as endothelin antagonists

#143
20050113460
2005-05-26

Compositions and methods relating to novel compounds and targets thereof

#144
20050113363
2005-05-26

Hydroxyalkanoylaminolactams and related structures as inhibitors of Aβ protein production

#145
20050075327
2005-04-07

Carbamic acid alkyl ester derivatives

#146
20050054633
2005-03-10

Malonamide derivatives

#147
20050009807
2005-01-13

Cyclic malonamides as inhibitors of A-β protein production