ClassID:

94769

C07D277/54 - CPC Classification

Classification description:

Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms Nitrogen and either oxygen or sulfur atoms

Recent Application in this class:
#1
20250115565
2025-04-10

SOLID CRYSTALLINE FORMS OF HELICASE-PRIMASE INHIBITORS AND PROCESS OF PREPARATION THEREOF

#2
20250100982
2025-03-27

PLEUROMUTILIN DERIVATIVE WITH THIAZOLE SIDE CHAIN AND PREPARATION AND APPLICATION

#3
20250091997
2025-03-20

COMPOSITIONS AND METHODS FOR MAKING AND USING SMALL MOLECULES FOR TUBULIN-TARGETED THERAPY IN THE TREATMENT OF CANCERS AND RELATED CONDITIONS

#4
20250034126
2025-01-30

CHROMOBOX PROTEIN INHIBITORS AND USES THEREOF

#5
20250002467
2025-01-02

DESIGN, SYNTHESIS AND MECHANISMS OF ANTICANCER ACTIVITY OF NEW ACETYLATED 5-AMINOSALICYLATE-THIAZOLINONE HYBRID DERIVATIVES

#6
20240368094
2024-11-07

POLYMORPHS OF PONESIMOD

#7
20240360089
2024-10-31

Metabolically Stable HDAC Inhibitors with Trifluoromethylpyruvamide as Metal-Binding Group

#8
20240199560
2024-06-20

PROCESS FOR PREPARING (2Z)-2-(PHENYLIMINO)-1,3-THIAZOLIDINE-4-ONE-SULFOXIDE DERIVATIVES IN AN ENANTIOMERICALLY ENRICHED FORM

#9
20230391738
2023-12-07

DEUTERATED AMINOTHIAZOLE COMPOUNDS AS ANTIVIRAL COMPOUNDS

#10
20230219910
2023-07-13

CRYSTALLINE FORMS OF {2-[3-CYCLOHEXYL-3-(TRANS-4-PROPOXY-CYCLOHEXYL)-UREIDO]-THIAZOL-5-YLSULFANYL}-ACETIC ACID AND USES THEREOF

#11
20230219909
2023-07-13

SALTS OR CO-CRYSTALS OF {2-[3-CYCLOHEXYL-3-(TRANS-4-PROPOXY-CYCLOHEXYL)-UREIDO]-THIAZOL-5-YLSULFANYL}-ACETIC ACID AND USES THEREOF

#12
20230106983
2023-04-06

SULFOXIDE AND SULFONE GLUCOKINASE ACTIVATORS AND METHODS OF USE THEREOF

#13
20230105595
2023-04-06

PROCESS OF PREPARING 2-(PHENYLIMINO)-3-ALKYL-1,3-THIAZOLIDIN-4-ONES

#14
20230090414
2023-03-23

Physics-driven discovery of novel small therapeutic compounds for use as a BCL-2 inhibitor

#15
20230022304
2023-01-26

WDR5-MYC INHIBITORS

#16
20230020663
2023-01-19

SULFONAMIDE INHIBITORS AS CTPS1 INHIBITORS

#17
20220315545
2022-10-06

PROCESS OF PREPARING 2-(PHENYLIMINO)-1,3-THIAZOLIDIN-4-ONES

#18
20210276963
2021-09-09

Pesticidal compositions and methods

#19
20210085679
2021-03-25

Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria

#20
20200216405
2020-07-09

Crystalline polymorph of Ponesimod

#21
20200148652
2020-05-14

Aminothiazole Derivatives Useful As Antiviral Agents

#22
20200131142
2020-04-30

FARNESOID X RECEPTOR AGONISTS AND USES THEREOF

#23
20200087250
2020-03-19

Pharmaceutical composition for ANO1 antagonist with anticancer activity

#24
20200024267
2020-01-23

Chromobox protein inhibitors and uses thereof

#25
20190382397
2019-12-19

Substituted 2-imino-1,3-thiazolidin-4-ones as N-arachidonoylethanolamine cellular uptake inhibitors

#26
20190375744
2019-12-12

Thiazole derivative and applications thereof

#27
20190183889
2019-06-20

Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria

#28
20190171099
2019-06-06

POLYMERIZABLE COMPOSITION COMPRISING AN OXIME SULFONATE AS THERMAL CURING AGENT

#29
20190119265
2019-04-25

Substituted 2-imino-1,3-thiazolidin-4-ones as N-arachidonoylethanolamine cellular uptake inhibitors

#30
20190112285
2019-04-18

Aminothiazole derivatives useful as antiviral agents

#31
20180370928
2018-12-27

4-oxo-4,5-dihydrothiazole derivative, preparation method and use thereof

#32
20180344706
2018-12-06

Compositions comprising metformin and a glucokinase activator

#33
20180319741
2018-11-08

Sulfonylaminobenzamide compounds as anthelmintics

#34
20180170863
2018-06-21

ROR gamma (RORγ) modulators

#35
20180111924
2018-04-26

Molecules having certain pesticidal utilities, and intermediates, compositions, and processes related thereto

#36
20180086700
2018-03-29

Inhibitors of the Notch transcriptional activation complex and methods for use of the same

#37
20180044332
2018-02-15

MOLECULES HAVING CERTAIN PESTICIDAL UTILITIES, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES RELATED THERETO

#38
20180015086
2018-01-18

Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria

#39
20170354647
2017-12-14

Use of metformin in combination with a glucokinase activator and compositions comprising metformin and a glucokinase activator

#40
20170253569
2017-09-07

Thiazolidinone compounds and use thereof

#41
20170226053
2017-08-10

Sulfonylaminobenzamide compounds as anthelmintics

#42
20170197952
2017-07-13

Substituted 2-imino-1,3-thiazolidin-4-ones as N-arachidonoylethanolamine cellular uptake inhibitors

#43
20170183333
2017-06-29

DERIVATIVES OF N-(ARYLAMINO) SULFONAMIDES AS INHIBITORS OF MEK

#44
20170166569
2017-06-15

Asparagine endopeptidase (AEP) inhibitors for managing cancer and compositions related thereto

#45
20170057914
2017-03-02

N-arylamidine-substituted trifluoroethyl sulfide derivatives as acaricides and insecticides

#46
20170036969
2017-02-09

NITRIFICATION INHIBITORS

#47
20160193207
2016-07-07

Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria

#48
20160184277
2016-06-30

Use of metformin in combination with a glucokinase activator and compositions comprising metformin and a glucokinase activator

#49
20160130240
2016-05-12

Aryl sulfide derivatives and aryl sulfoxide derivatives as acaricides and insecticides

#50
20160096831
2016-04-07

Molecules having certain pesticidal utilities, and intermediates, compositions, and processes related thereto

#51
20160060214
2016-03-03

Polymerizable composition comprising an oxime sulfonate as thermal curing agent

#52
20160002187
2016-01-07

Apoptosis-inducing agent for the treatment of cancer and immune and autoimmune diseases

#53
20150336912
2015-11-26

(4E)-4-(4-substituted benzylideneamino)-2,3-dihydro-3-substituted-2-thioxothiazole-5-carbonitriles as A2AR antagonist and process for preparation thereof

#54
20150225391
2015-08-13

Molecules having certain pesticidal utilities, and intermediates, compositions, and processes related thereto

#55
20150203459
2015-07-23

Process for the preparation of (2Z,5Z)-5-(3-chloro-4-(()-2,3-dihydroxypropdxy)benzylidene)-2-(propylimino)-3-(-tolyl)thiazolidin-4-one and intermediate used in said process

#56
20150051249
2015-02-19

Inhibition of MCL-1 and/or BFL-1/A1

#57
20150025094
2015-01-22

Compounds and compositions for use in augmentation of glucose

#58
20150018371
2015-01-15

Positive allosteric modulators for melanocortin receptors

#59
20150018330
2015-01-15

Broad spectrum benzothiophene-nitrothiazolide and other antimicrobials

#60
20140303026
2014-10-09

Compounds for modulating integrin CD11B/CD18

#61
20140275524
2014-09-18

Molecules having certain pesticidal utilities, and intermediates, compositions, and processes related thereto

#62
20140275047
2014-09-18

Molecules having certain pesticidal utilities, and intermediates, compositions, and processes related thereto

#63
20140256745
2014-09-11

Compounds that modulate intracellular calcium

#64
20140128397
2014-05-08

Synthetic lethal targeting of glucose transport

#65
20140080825
2014-03-20

Modulators of ATP-binding cassette transporters

#66
20140079736
2014-03-20

Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria

#67
20140066466
2014-03-06

Necroptosis inhibitors and methods of use therefor

#68
20130345432
2013-12-26

ASYMMETRIC PROCESS FOR MAKING SUBSTITUTED 2-AMINO-THIAZOLONES

#69
20130310432
2013-11-21

Thiazolidin-4-one-derivatives

#70
20130308219
2013-11-21

Polymerizable composition comprising an oxime sulfonate as thermal curing agent

#71
20130143927
2013-06-06

COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM

#72
20130109019
2013-05-02

HAPTEN CONJUGATES FOR TARGET DETECTION

#73
20130053402
2013-02-28

Substituted 3-thiazoloamino-propionic acid derivatives and their use as pharmaceuticals

#74
20130045967
2013-02-21

Compounds for modulating integrin CD11b/CD18

#75
20130040951
2013-02-14

PROPHYLACTIC OR THERAPEUTIC AGENT FOR CANCER

#76
20120302758
2012-11-29

Process for the preparation of 2-imino-thiazolidin-4-one derivatives

#77
20120302612
2012-11-29

Thiazolidin-4-one derivatives

#78
20120214735
2012-08-23

Acetamide derivatives as glucokinase activators, their process and medicinal applications

#79
20120196864
2012-08-02

PROPHYLACTIC OR THERAPEUTIC AGENT FOR CANCER

#80
20120108591
2012-05-03

Alkylsulfinyl-substituted thiazolide compounds

#81
20120108573
2012-05-03

Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them

#82
20120022076
2012-01-26

Derivatives of N-(arylamino)sulfonamides as inhibitors of MEK

#83
20120010256
2012-01-12

Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1

#84
20120010187
2012-01-12

Broad spectrum benzothiophene-nitrothiazolide and other antimicrobials

#85
20110313007
2011-12-22

Use of metformin in combination with a glucokinase activator and compositions comprising metformin and a glucokinase activator

#86
20110306637
2011-12-15

Modulators of ATP-binding cassette transporters

#87
20110301158
2011-12-08

ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS

#88
20110288083
2011-11-24

Method of treating cancer by inhibition of protein kinase-like endoplasmic reticulum protein kinase

#89
20110230529
2011-09-22

BENZAMIDE GLUCOKINASE ACTIVATORS

#90
20110201821
2011-08-18

Process for the preparation of 2-imino-thiazolidin-4-one derivatives

#91
20110196004
2011-08-11

Crystalline forms of (R)-5-[3-chloro-4-(2,3-dihydroxy-propoxy)-benz[Z]ylidene]-2-([Z]-propylimino)-3-0-tolyl-thiazolidin-4-one

#92
20110190299
2011-08-04

Thiazolidinone derivative

#93
20110178307
2011-07-21

Asymmetric process for making substituted 2-amino-thiazolones

#94
20110160463
2011-06-30

Process for making substituted 2-amino-thiazolones

#95
20110130402
2011-06-02

HETEROAROMATIC GLUCOKINASE ACTIVATORS

#96
20110082107
2011-04-07

INHIBITORS OF 11-BETA-HYDROXY STEROID DEHYDROGENASE TYPE 1

#97
20110039849
2011-02-17

5-substituted-2-imino-thiazolidinone compounds and their use as inhibitors of bacterial infection

#98
20100317867
2010-12-16

NEW PROCESS FOR THE PREPARATION OF 2-IMINO-THIAZOLIDIN-4-ONE DERIVATIVES

#99
20100310493
2010-12-09

Acetamide derivatives as glucokinase activators, their process and medicinal application

#100
20100286171
2010-11-11

Substituted pyrazine compounds

#101
20100280034
2010-11-04

Modulation of pathogenicity

#102
20100184766
2010-07-22

Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases

#103
20100087442
2010-04-08

Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient

#104
20100056503
2010-03-04

Compounds for modulating integrin CD11b/CD18

#105
20090306133
2009-12-10

New Acetyl Coenzyme A Carboxylase (ACC) Inhibitors And Uses In Treatments Of Obesity And Diabetes Mellitus - 087

#106
20090275625
2009-11-05

Thiazolidin 4-one derivatives

#107
20090275538
2009-11-05

ARYLMETHYLIDENE HETEROCYCLES AS NOVEL ANALGESICS

#108
20090215758
2009-08-27

Use of 2,5-Disubstituted Thiazol-4-One Derivatives in Drugs

#109
20090176991
2009-07-09

Benzamide glucokinase activators

#110
20090176773
2009-07-09

Non-Peptidic Inhibitors of AKAP/PKA Interaction

#111
20090118501
2009-05-07

Dicycloalkyl urea glucokinase activators

#112
20090082457
2009-03-26

Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK

#113
20080280962
2008-11-13

Thiazolidin-4-one derivatives

#114
20080269283
2008-10-30

Arylsulfones and uses related thereto

#115
20080269219
2008-10-30

Neurotrophin production/secretion promoting agent

#116
20080176899
2008-07-24

Modulators of ATP-binding cassette transporters

#117
20080146629
2008-06-19

Thiazolidin-4-one derivatives

#118
20080146594
2008-06-19

Thrombopoietin activity modulating compounds and methods

#119
20080139562
2008-06-12

Heteroaromatic glucokinase activators

#120
20080132519
2008-06-05

Heterocyclic compounds as pharmaceutical agents

#121
20080119455
2008-05-22

Aryl carbonyl derivatives as therapeutic agents

#122
20080119454
2008-05-22

Aryl carbonyl derivatives as therapeutic agents

#123
20080103190
2008-05-01

THROMBOPOIETIN ACTIVITY MODULATING COMPOUNDS AND METHODS

#124
20080096936
2008-04-24

Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them

#125
20080090782
2008-04-17

Materials and methods to potentiate cancer treatment

#126
20080058340
2008-03-06

Derivatives of N-(arylamino) sulfonamides as inhibitors of MEK

#127
20080045503
2008-02-21

Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1

#128
20070281979
2007-12-06

FBPase inhibitors for diabetes

#129
20070281938
2007-12-06

Inhibitors of 11-Beta-Hydroxy Steroid Dehydrogenase Type 1

#130
20070248594
2007-10-25

CXCR1 AND CXCR2 CHEMOKINE ANTAGONISTS

#131
20070197598
2007-08-23

Inhibitors of 11-beta-hydroxysteroid dehydrogenase type 1

#132
20070197523
2007-08-23

CALCIUM CHANNEL ANTAGONISTS

#133
20070173504
2007-07-26

Calcium channel antagonists

#134
20070155750
2007-07-05

Integrin-binding small molecules

#135
20070155671
2007-07-05

Diaminopropionic acid derivatives

#136
20070117985
2007-05-24

Catalyzed process of making C-5-substituted heterocyclic inhibitors of 11β-hydroxy steroid dehydrogenase type 1

#137
20070082933
2007-04-12

Thiazolidin-4-one derivatives

#138
20070027147
2007-02-01

Biarylurea derivatives

#139
20060270720
2006-11-30

Iminothiazolidinone derivatives as SFRP-1 antagonists

#140
20060183783
2006-08-17

Aryl carbonyl derivatives as therapeutic agents

#141
20060166990
2006-07-27

Aminobenzophenone compounds

#142
20060142357
2006-06-29

Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1

#143
20060116417
2006-06-01

Thrombopoietin activity modulating compounds and methods

#144
20060111303
2006-05-25

Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient

#145
20060069037
2006-03-30

Peptide-containing alpha-ketoamide cysteine and serine protease inhibitors

#146
20060052358
2006-03-09

Modulators of ATP-binding cassette transporters

#147
20060030598
2006-02-09

Thiazolyl inhibitors of Tec family tyrosine kinases

#148
20060014794
2006-01-19

CXCR1 and CXCR2 chemokine antagonists

#149
20050277665
2005-12-15

Arylsulfones and uses related thereto

#150
20050267173
2005-12-01

Serine protease inhibitors

#151
20050239853
2005-10-27

New compounds

#152
20050215642
2005-09-29

Selective inhibitors of the urokinase plasminogen activator

#153
20050080119
2005-04-14

Diaminopropionic acid derivatives

#154
18443136
2024-11-19

4-thiazolidinone derivatives as EGFR inhibitors for anti-tumor activity

#155
16653629
2021-11-30

Salts of a thiazolidinone compound, solid forms, compositions and methods of use thereof