ClassID:

94883

C07D295/185 - page 3 - CPC Classification

Classification description:

Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof; Radicals derived from carboxylic acids from aliphatic carboxylic acids

Recent Application in this class:
#601
20070032664
2007-02-08

Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1-pyrrole-3-carboxylic acid phenylamide

#602
20070032663
2007-02-08

Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1-pyrrole-3-carboxylic acid phenylamide

#603
20070032662
2007-02-08

Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1-pyrrole-3-carboxylic acid and phenylamide

#604
20070032532
2007-02-08

Hsp90 family protein inhibitors

#605
20070032488
2007-02-08

6-Membered aryl and heteroaryl derivatives for treating viruses

#606
20070027141
2007-02-01

Derivatives of alkylpiperazine and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors

#607
20070015807
2007-01-18

Heteroatom-linked substituted piperidines and derivatives thereof useful as histamine Hantagonists

#608
20070015787
2007-01-18

Apoptosis promoters

#609
20070004750
2007-01-04

N-substituted piperazines

#610
20070004725
2007-01-04

Derivatives of amino acids for treatment of obesity and related disorders

#611
20070004718
2007-01-04

Ion channel modulating compounds and uses thereof

#612
20060293310
2006-12-28

Derivatives of 1-piperazine-and 1-homopiperazine-carboxylates, preparation method thereof and use of same as inhibitors of the FAAH enzyme

#613
20060287306
2006-12-21

Compounds to treat alzheimer's disease

#614
20060287244
2006-12-21

L-Threonine derivatives of high therapeutic index

#615
20060281920
2006-12-14

Derivatives of hydroxamic acid as metalloproteinase inhibitors

#616
20060276642
2006-12-07

Compounds to treat Alzheimer's disease

#617
20060276465
2006-12-07

1,2-di(cyclic) substituted benzene compounds

#618
20060276409
2006-12-07

Antibacterial agents

#619
20060264415
2006-11-23

Inhibitors of histone deacetylase

#620
20060258866
2006-11-16

Carboxylic derivates

#621
20060258657
2006-11-16

Apoptosis promoters

#622
20060252832
2006-11-09

Interleukin-1 and tumor necrosis factor-α modulators, synthesis of said modulators and their enantiomers and methods of using said modulators

#623
20060252778
2006-11-09

Compounds for the treatment of inflammatory disorders

#624
20060247264
2006-11-02

Modulators of the glucocorticoid receptor

#625
20060247223
2006-11-02

Non-imidazole alkylamines as histamine H- receptor ligands and their therapeutic applications

#626
20060241119
2006-10-26

Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives

#627
20060241017
2006-10-26

Compounds with high therapeutic index

#628
20060235073
2006-10-19

Diamino-functional chalcones

#629
20060229254
2006-10-12

Compounds having prolyl oligopeptidase inhibitory activity

#630
20060217422
2006-09-28

Exo-selective synthesis of himbacine analogs

#631
20060199853
2006-09-07

Analogs of 4-hydroxyisoleucine and uses thereof

#632
20060199848
2006-09-07

Ion channel modulating activity II

#633
20060189689
2006-08-24

Arginine mimetics as factor Xa inhibitors

#634
20060183741
2006-08-17

Substituted diamine derivatives useful as motilin antagonists

#635
20060178366
2006-08-10

Compounds for the treatment of inflammatory disorders

#636
20060178360
2006-08-10

Benzenesulphonamide derivatives, method for production and use thereof for treatment of pain

#637
20060173044
2006-08-03

Substituted propargylamines

#638
20060173004
2006-08-03

1-(4-Benzyl-piperazin-1-yl)-3-phenyl-propenone derivatives

#639
20060171882
2006-08-03

Method for the use of [11C] carbon monoxide in labeling synthesis of 11C-labelled compounds by thermally induced free radical carbonylation

#640
20060161020
2006-07-20

N-alkyl phenylcarboxamide beta-secretase inhibitors for the treatment of Alzheimer's disease

#641
20060142305
2006-06-29

Hydroxyamidine and hydroxyguanidine compounds as urokinase inhibitors

#642
20060141597
2006-06-29

Valency platform molecules comprising aminooxy groups

#643
20060135487
2006-06-22

Piperazine derivatives and their use as anti-inflammatory agents

#644
20060128706
2006-06-15

Apoptosis promoters

#645
20060116410
2006-06-01

4-Aminomethyl benzamidine derivatives

#646
20060111406
2006-05-25

Amide linker peroxisome proliferator activated receptor modulators

#647
20060111336
2006-05-25

Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes

#648
20060106016
2006-05-18

Dicarboxamide derivatives

#649
20060094874
2006-05-04

Substituted aryl alkenoic acid heterocyclic amides

#650
20060094718
2006-05-04

O-substituted hydroxyaryl derivatives

#651
20060089357
2006-04-27

Novel compounds and compositions as cathepsin inhibitors

#652
20060089336
2006-04-27

4-Dedimethylamino tetracycline compounds

#653
20060084658
2006-04-20

Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound

#654
20060079527
2006-04-13

Piperazine derivatives having SST1 antagonistic activity

#655
20060079506
2006-04-13

Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors

#656
20060074086
2006-04-06

Phenyl derivatives and methods of use

#657
20060069103
2006-03-30

17β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases

#658
20060063930
2006-03-23

Compositions and methods comprising proteinase activated receptor antagonists

#659
20060063778
2006-03-23

Hydroxamic acid derivatives

#660
20060052600
2006-03-09

Amino-functional chalcones

#661
20060052396
2006-03-09

Arylamines for the treatment of conditions associated with gsk-3

#662
20060052375
2006-03-09

Bis-alkylbenzylamines

#663
20060049061
2006-03-09

Organic salts and their use as reagents in electrochemical reactions

#664
20060047123
2006-03-02

Mercaptoamides as histone deacetylase inhibitors

#665
20060041169
2006-02-23

Preparation of N-substituted 2,7-dialkyl-4-hydroxy-5-amino-8-aryl-octanoyl amides

#666
20060041020
2006-02-23

Cyclohexyl sulphones

#667
20060025404
2006-02-02

Substituted piperazines,(1,4) diazepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine H1 and/or H3 antagonists or histamine H3 reverse antagonists

#668
20060020131
2006-01-26

Inhibitors of histone deacetylase

#669
20060020009
2006-01-26

Succinoylamino hydroxyethylamino sulfonyl urea derivatives useful as retroviral protease inhibitors

#670
20060014755
2006-01-19

17 β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases

#671
20060009491
2006-01-12

Amido compounds and their use as pharmaceuticals

#672
20060009484
2006-01-12

Polycyclic compounds which modulate PPARγ type receptors and cosmetic/pharmaceutical compositions comprised thereof

#673
20060009471
2006-01-12

Amido compounds and their use as pharmaceuticals

#674
20060004062
2006-01-05

Compounds for inhibiting insulin secretion and methods related thereto

#675
20060004048
2006-01-05

Biaromatic compounds which activate PPARgamma type receptors and cosmetic/pharmaceutical compositions comprised thereof

#676
20050282882
2005-12-22

Diamines as modulators of chemokine receptor activity

#677
20050282872
2005-12-22

Thyroid receptor ligands and method II

#678
20050282858
2005-12-22

Amido compounds and their use as pharmaceuticals

#679
20050282822
2005-12-22

Therapeutic agents

#680
20050282821
2005-12-22

Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives

#681
20050277627
2005-12-15

Colchinol derivatives as vascular damaging agents

#682
20050272667
2005-12-08

Analogs and derivatives of (S,S,R)-(-)-actinonin and uses therefor

#683
20050267173
2005-12-01

Serine protease inhibitors

#684
20050267168
2005-12-01

Pentanoic acid derivatives

#685
20050267167
2005-12-01

Pentanoic acid derivatives

#686
20050261501
2005-11-24

Pyrrolidine and thiazolidine compounds

#687
20050261371
2005-11-24

Pentanoic acid derivatives

#688
20050256133
2005-11-17

Thio-substituted arylmethanesulfinyl derivatives

#689
20050256116
2005-11-17

Biaromatic compounds which activate PPARγ type receptors and cosmetic/pharmaceutical compositions comprised thereof

#690
20050250790
2005-11-10

Novel sulfonic acid derivatives

#691
20050250768
2005-11-10

Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds

#692
20050245747
2005-11-03

Thio-substituted biaryl-methanesulfinyl derivatives

#693
20050245616
2005-11-03

Compounds and related methods for mutant p53 reactivation

#694
20050245534
2005-11-03

Inhibitors of the 11-beta-hydroxysteroid dehydrogenase Type 1 enzyme

#695
20050245522
2005-11-03

Novel compounds

#696
20050239870
2005-10-27

Hemiasterlin derivatives and uses thereof

#697
20050239869
2005-10-27

Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1-pyrrole-3-carboxylic acid phenylamide

#698
20050239839
2005-10-27

Adamantylglycine-based inhibitors of dipeptidyl peptidase IV and methods

#699
20050234106
2005-10-20

Cycloalkyl inhibitors of potassium channel function

#700
20050234065
2005-10-20

Dipeptidyl peptidase-IV inhibitors

#701
20050233943
2005-10-20

Polyamine analog conjugates and quinone conjugates as therapies for cancers and prostate diseases

#702
20050228040
2005-10-13

Bicyclic aromatic sulfinyl derivatives

#703
20050228021
2005-10-13

Adamantylglycine-based inhibitors of dipeptidyl peptidase IV and methods

#704
20050227991
2005-10-13

Heterocyclic or benzenic derivatives of lipoic acid, their preparation and their use as medicaments

#705
20050227990
2005-10-13

Aminoalkoxy-functional chalcones

#706
20050227973
2005-10-13

Human ADAM-10 inhibitors

#707
20050222244
2005-10-06

Synthesis of UDP-glucose: -acylsphingosine glucosyltransferase inhibitors

#708
20050222146
2005-10-06

N-substituted-n-sulfonylaminocyclopropane compounds and pharmaceutical use thereof

#709
20050222140
2005-10-06

Phenylalanine derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes

#710
20050215637
2005-09-29

Tuberculosis treatment

#711
20050215587
2005-09-29

Serine protease inhibitors

#712
20050215563
2005-09-29

Proteomimetic compounds and methods

#713
20050215548
2005-09-29

Bisarylsulfonamide compounds and their use in cancer therapy

#714
20050203030
2005-09-15

Novel effectors of dipeptidyl peptidase IV

#715
20050192289
2005-09-01

Novel cinnamic amides

#716
20050192286
2005-09-01

Ligands of melanocortin receptors and compositions and methods related thereto

#717
20050192208
2005-09-01

ION CHANNEL MODULATING COMPOUNDS AND USES THEREOF

#718
20050187198
2005-08-25

Methods of preparing substituted tetracyclines with transition metal-based chemistries

#719
20050176987
2005-08-11

Method for producing vinyl, aryl and heteroaryl acetic acids and derivatives thereof

#720
20050171120
2005-08-04

Stereoselective alkylation of chiral 2-methyl-4-protected piperazines

#721
20050153366
2005-07-14

Protein-protein interaction antagonist screening libraries based upon 1,4-disubstituted naphthalenes and related scaffolds

#722
20050148656
2005-07-07

Carboxylic derivates

#723
20050148584
2005-07-07

Substituted diamine derivatives useful as motilin antagonists

#724
20050143426
2005-06-30

Calcium receptor modulating agents

#725
20050143393
2005-06-30

Pleuromutilin derivatives with antimicrobial activity

#726
20050143385
2005-06-30

Carbamic acid compounds comprising a piperazine linkage as HDAC inhibitors

#727
20050143372
2005-06-30

Compounds, pharmaceutical compositions and methods of use therefor

#728
20050119315
2005-06-02

Ion channel modulating activity method

#729
20050119306
2005-06-02

Alkaloid that inhibits biosynthesis of mycotoxins and method for screening for mycotoxin inhibitors

#730
20050119275
2005-06-02

Salt and crystal forms of (5-chloro-2-{2-[4-(4-fluoro-benzyl)-(2R,5S)-2,5-dimethyl-piperazin-1-yl]-2-oxo-ethoxy}-phenyl)-methanesulfonic acid

#731
20050119252
2005-06-02

Ligands of melanocortin receptors and compositions and methods related thereto

#732
20050113580
2005-05-26

Compounds and methods

#733
20050113344
2005-05-26

Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases

#734
20050107444
2005-05-19

Amide compounds and methods of using the same

#735
20050107354
2005-05-19

Agents for the prevention or treatment of renal diseases

#736
20050106712
2005-05-19

Yellow low fluorescence dye for coated optical bead random array DNA analysis

#737
20050096357
2005-05-05

Pleuromutilin derivatives

#738
20050080271
2005-04-14

Peptidomimetic ligands for cellular receptors and ion channels

#739
20050075392
2005-04-07

Pharmaceuticals

#740
20050075381
2005-04-07

Diastereoselective synthesis of UDP-glucose: N-acylsphingosine glucosyltransferase inhibitors

#741
20050075368
2005-04-07

Conjugated dienamides, methods of production thereof, compositions containing same and uses thereof

#742
20050074533
2005-04-07

Conjugated dienamides, methods of production thereof, compositions containing same and uses thereof

#743
20050070719
2005-03-31

Inhibitors of dipeptidyl peptidase iv

#744
20050070559
2005-03-31

Use of oxindole derivatives in the treatment of dementia related diseases, alzheimer's disease and conditions associated with glycogen synthase kinase-3

#745
20050070485
2005-03-31

Phenylalanine derivatives

#746
20050065346
2005-03-24

Carboxylic acid amides, the preparation thereof and their use as pharmaceutical compositions

#747
20050065210
2005-03-24

Aminoalkylamide substituted cyclohexyl derivatives

#748
20050065095
2005-03-24

Antibacterial agents

#749
20050059668
2005-03-17

Substituted acylpiperazine derivatives

#750
20050043299
2005-02-24

Inhibitors of dipeptidyl peptidase IV

#751
20050038020
2005-02-17

Adamantylglycine-based inhibitors of dipeptidyl peptidase IV and methods

#752
20050032794
2005-02-10

Diamine derivatives of quinone and uses thereof

#753
20050032790
2005-02-10

Compounds

#754
20050026953
2005-02-03

Alkaloid that inhibits biosynthesis of mycotoxins and method for screening for mycotoxin inhibitors

#755
20050020857
2005-01-27

Method for the separation of acids from chemical reaction mixtures by means of ionic fluids

#756
20050020684
2005-01-27

Modulators of peroxisome proliferator activated receptors

#757
20050020504
2005-01-27

C-terminal modified oxamyl dipeptides as inhibitors of the ICE/ced-3 family of cysteine proteases

#758
20050020481
2005-01-27

Ion channel modulating compounds and uses thereof

#759
20050014787
2005-01-20

5-amidino-2-hydroxybenzenesulfonamide derivatives medicinal compoistions containing the same medicinal use thereof and intermediates in the production thereof

#760
20050014702
2005-01-20

Antibacterial agents

#761
20050010060
2005-01-13

Quinones as disease therapies

#762
20050009872
2005-01-13

Synthesis of UDP-glucose: -acylsphingosine glucosyltransferase inhibitors

#763
20050009706
2005-01-13

α-Cyanoacrylates

#764
20050004351
2005-01-06

Therapeutic and diagnostic domain 1 beta2GP1 polypeptides and methods of using same

#765
14839993
2017-01-03

Fumarate compounds, pharmaceutical compositions thereof, and methods of use