95252 ⎘
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
Thrombopoietin mimetics
#6602PROCESSES FOR PREPARING ZAFIRLUKAST
#6603Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
#6604Cinnamic acid amides
#6605Imidazole derivatives having a positive allosteric GABAreceptor modulator effect and methods of use
#6606Monocyclic Heteroaryl compounds
#6607Aminopyridine derivatives having aurora a selective inhibitory action
#6608Tyrosine Kinase Inhibitors
#6609Use of 1,4-bis (3-aminoalkyl) piperazine derivatives in the treatment of neurodegenerative diseases
#6610P38 inhibitors and methods of use thereof
#6611Mmuscarinic acetylcholine receptor antagonists
#6612P38 inhibitors and methods of use thereof
#6613Pyrimidines as PLK inhibitors
#6614RATE-CONTROLLED PARTICLES
#6615Scalable synthesis of imidazole derivatives
#6616Vanilloid receptor ligands and their use in treatments
#6617Acid secretion inhibitor
#6618P38 inhibitors and methods of use thereof
#6619Phenylpiperazine
#6620Melanin concentrating hormone receptor antagonist
#6621Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
#6622Non-nucleoside reverse transcriptase inhibitors
#6623Heteroaryl urea derivatives useful for inhibiting CHK1
#6624Substituted aryl-amine derivatives and methods of use
#6625NOVEL M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS
#6626Compounds and compositions as protein kinase inhibitors
#6627A2B ADENOSINE RECEPTOR ANTAGONISTS
#6628Chemical compounds
#6629Fungicide N-cyclopropyl-sulfonylamide derivatives
#6630Heterocyclic amide compound and use thereof
#66314,6-disubstitued pyrimidines useful as kinase inhibitors
#66322-aminoquinazoline derivatives
#66331,3-disubstituted 4-methyl-1H-pyrrole-2-carboxamides and their use in medicaments
#6634Substituted arylpyrazoles
#6635Organic compounds and their uses
#6636Anti-inflammatory medicaments
#6637P38 inhibitors and methods of use thereof
#6638Indoline-substituted pyrazoline derivatives, their preparation and use as medicaments
#6639Non-Nucleoside Reverse Transcriptase Inhibitors
#6640Indole derivatives as CFTR modulators
#6641Quinoline and quinoxaline derivatives as inhibitors of kinase enzymatic activity
#6642Triazole derivative
#6643DISUBSTITUTED UREAS AS KINASE INHIBITORS
#6644Pyrimidine Derivatives
#6645Substituted tetrazole compounds and uses thereof
#6646Cyclic derivatives as modulators of chemokine receptor activity
#6647Fused heterocyclic derivatives and methods of use
#6648Novel Bicyclic Sulfonamides for Use as Glucocorticoid Receptor Modulators in the Treatment of Inflammatory Diseases
#6649Soft protease inhibitors and pro-soft forms thereof
#6650HYDROXYAMIC ANALOGS AS HEPATITIS C VIRUS SERINE PROTEASE INHIBITOR
#6651Development of molecular imaging probes for carbonic anhydrase-IX using click chemistry
#6652Quaternary polymers
#66535,6-trimethylenepyrimidin-4-one compounds
#6654Compounds that are ERK inhibitors
#6655Compounds which potentiate AMPA receptor and uses thereof in medicine
#6656Compositions useful as inhibitors of GSK-3
#6657QUINAZOLINONE DERIVATIVES AND THEIR USE AS B-RAF INHIBITORS
#6658Pharmaceutical use of substituted amides
#6659Histamine H3 receptor agents, preparation and therapeutic uses
#6660Proline bis-amide orexin receptor antagonists
#6661HETEROCYCLIC COMPOUNDS AND METHODS OF USE
#6662Sulfonylpyrroles as Histone Deacetylase Inhibitors
#6663Histone deacetylase inhibitors
#66641,2,4-TRIAZOLE ETHER DERIVATIVES AS MODULATORS OF MGLUR5
#6665Imidazolidinone compounds useful as β-secretase inhibitors for the treatment of Alzheimer's disease
#6666Substituted isoindolones and their use as metabotropic glutamate receptor potentiators
#66677-membered ring compound and method of production and pharmaceutical application thereof
#6668HISTONE DEACETYLASE INHIBITORS
#6669Substituted pyrazolecarboxylic acid anilide derivative or salt thereof, intermediate thereof, agent for agricultural and horticultural use, and use thereof
#6670Indoline amide derivatives as EP4 receptor ligands
#6671Amidoethylthioether Orexin Receptor Antagonists
#6672Benzoheterocylethylcarboxamide derivatives
#6673Therapeutic Agents - 550
#6674Macrocyclic inhibitors of hepatitis C virus
#6675c-Met modulators and methods of use
#6676Diacylglycerol acyltransferase inhibitors
#6677Triazole derivative and use thereof
#6678Anti-inflammatory medicaments
#6679Benzazepine derivatives for the treatment of neurological disorders
#66803-(aminomethyliden) 2-indolinone derivates and their use as cell proliferation inhibitors
#6681Heteroaryl benzamide derivatives for use as GLK activators in the treatment of diabetes
#6682Inhibitors of hedgehog pathway
#6683Substituted piperazines as CB1 antagonists
#6684PREPARATION OF 7-ALKENYL-3 QUINOLINECARBONITRILES VIA A PALLADIUM MEDIATED COUPLING REACTION
#6685ORGANIC COMPOUNDS
#6686CXCR4 antagonists including diazine and triazine structures for the treatment of medical disorders
#6687PYRIMIDINES AND USES THEREOF
#6688INDAZOLE COMPOUNDS AND METHODS OF USE THEREOF
#6689Sirtuin modulating compounds
#66906-substituted 2,3,4,5-tetrahydro-1H-benzo[d]azepines as 5-HTreceptor agonists
#6691TETRAHYDRO-INDAZOLE CANNABINOID MODULATORS
#6692Compounds and methods for modulating FXR
#6693Diacylglycerol acyltransferase inhibitors
#6694ANTI-CANCER AGENTS AND USES THEREOF
#6695N-AROYL CYCLIC AMINES
#6696Dual-acting antihypertensive agents
#6697miRNA PROCESSING INHIBITOR EFFICACY ASSAYS AND SUBSTANCES
#6698Solid forms of (S)-ethyl 2-amino-3-(4-(2-amino-6-((R)-1- (4-chloro-2-(3-methyl-1H-pyrazol-1-YL)phenyl)2,2,2-trifluoroethoxy)-pyrimidin-4-YL)phenyl)propanoate and methods of their use
#6699Compounds with HIV-1 integrase inhibitory activity and use thereof as anti-HIV/AIDS therapeutics
#6700N,N-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitors
#6701Intermediates for making 2,4-pyrimidinediamine compounds
#6702Pharmaceutical for prevention or treatment of bone metabolic disease
#6703BENZIMIDAZOLES
#67045-aryl-4,5-dihydro-(1H)-pyrazolines as cannabinoid CB1 receptor agonists
#6705DEUTERIUM-ENRICHED TELAPREVIR
#6706Pyrazine compounds and uses as PI3K inhibitors
#6707Pyrimidine compound having dibenzylamine structure and medicament comprising the same
#67083-substituted-5- and 6-aminoalkyl indole-2-carboxylic acid amides and related analogs as inhibitors of casein kinase I
#6709Substituted phenylamino-benzene derivatives useful for treating hyper-proliferative disorders and diseases associated with mitogen extracellular kinase activity
#6710Fluorinated 4-azasteroid derivatives as androgen receptor modulators
#6711Prodrugs of thyroid hormone analogs
#6712DIACYLGLYCEROL ACYLTRANSFERASE INHIBITORS
#6713VEGFR INHIBITORS CONTAINING A ZINC BINDING MOIETY
#6714Tartrate salts of quinazoline based EGFR inhibitors containing a zinc binding moiety
#6715Modulation of pathogenicity
#6716Anti-inflammatory medicaments
#6717Colorants based N-halamines compositions and method of making and using
#6718NEW INDOLE DERIVATIVES AS FACTOR XA INHIBITORS
#6719CLICK CHEMISTRY ROUTE TO TRIAZOLE DENDRIMERS
#6720ALPHA-ALKYL SUBSTITUTED N-ACYLTRYPTOPHANOLS
#6721Anti-inflammatory medicaments
#6722ISOQUINOLINYL AND ISOINDOLINYL DERIVATIVES AS HISTAMINE-3 ANTAGONISTS
#6723Novel therapeutic compounds
#6724Linear and cyclic melanocortin receptor-specific peptidomimetics
#6725Isatin analogues and uses therefor
#6726METHODS OF PREPARING 4-PHENYL-6-(2,2,2-TRIFLUORO-1-PHENYLETHOXY)PYRIMIDINE-BASED COMPOUNDS
#6727N-Formyl Hydrozyamine Compounds
#6728Substituted arylalkanoic acid derivatives and use thereof
#6729Pyrrolidine derivative or salt thereof
#6730Amide derivative or salt thereof
#6731Substituted pyrimidine compounds and their utility as CETP inhibitors
#6732HETEROARYL-SUBSTITUTED UREA MODULATORS OF FATTY ACID AMIDE HYDROLASE
#6733Small molecule PI 3-kinase inhibitors and methods of their use
#6734Octahydropentalene-Substituted Pyrazoline Derivatives, Their Prepartion and Use as Medicaments
#6735Heterocyclylethylcarboxamide derivatives
#6736Pyrazinyl hydroxyacrylamide compounds having an inhibitory effect on the activity of histone deacetylase
#6737HDAC inhibitor
#6738Piperazine derivatives and methods of use
#6739Substituted indoles
#6740COMPOSITIONS AND METHODS OF USE FOR TREATING OR PREVENTING LIPID RELATED DISORDERS
#6741Substituted N-heterocyclic compounds and their use as dopamine Dreceptor ligands
#6742Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors
#67432,3-disubstituted pyrazinesulfonamides as CRTH2 inhibitors
#6744TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS
#6745Substituted bicyclic derivatives and use thereof
#6746Sulfonyl amide derivatives for the treatment of abnormal cell growth
#6747Heteroaroyl-substituted Alanines
#6748Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
#6749Hybridization and mismatch discrimination using oligonucleotides conjugated to minor groove binders
#6750Azabicycloheptyl compounds suitable for treating disorders that respond to modulation of the dopamine D3 receptor
#6751Amino-5-[4-(difluoromethoxy)phenyl]-5-phenylimidazolone compounds for the inhibition of beta-secretase
#6752Piperazine amide derivatives
#6753Pyrazole compounds having cannabinoid receptor (CB1) antagonizing activity
#67544-(1H-indazol-5-yl-amino)-quinazoline compounds as erbB receptor tyrosine kinase inhibitors for the treatment of cancer
#6755Phenylalanine derivatives
#6756Substituted prolinamides, the preparation thereof and the use thereof as pharmaceutical compositions
#6757Compounds and compositions useful as cathepsin S inhibitors
#6758Heterocycle derivatives as histone deacetylase (HDAC) inhibitors
#6759Antiviral compounds
#6760NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION
#6761Indoles Useful in the Treatment of Inflammation
#6762Carbonylamino-derivatives as novel inhibitors of histone deacetylase
#6763SUBSTITUTED ACETAMIDES AS MODULATORS OF THE EP2 RECEPTOR
#6764Sulfonamide derivatives, preparation thereof and use thereof as antagonists of orexin 2 receptors
#6765Tubulin Binding Anti Cancer Agents And Prodrugs Thereof
#6766Compositions and methods for inhibition of the JAK pathway
#67675-pyrrolidinylsulfonyl isatin derivatives
#6768Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them
#6769Cannabinoid receptor antagonists/inverse agonists useful for treating metabolic disorders, including obesity and diabetes
#6770Quinazoline derivatives for use against cancer
#6771Pyridine and pyrimidine derivatives as inhibitors of histone deacetylase
#6772PYRAZOLE COMPOUNDS AND USE THEREOF
#6773Indazolesquaric Acid Derivatives as Chk1, Chk2 and Sgk Inhibitors
#6774PYRIMIDINE DERIVATIVES AND METHODS OF TREATMENT RELATED TO THE USE THEREOF
#6775Indole derivatives as histamine 3 receptor inhibitors for the treatment of cognitive and sleep disorders, obesity and other CNS disorders
#6776Five-membered heterocycles useful as serine protease inhibitors
#6777Compounds useful as Raf kinase inhibitors
#6778Modified carbocyanine dyes and their conjugates
#6779Modified carbocyanine dyes and their conjugates
#6780Bicyclic compound, production and use thereof
#6781Heterobicyclic carboxamides as inhibitors for kinases
#6782Trisubstituted amine compound
#6783SUBSTITUTED PYRAZOLE COMPOUNDS
#6784BENZAMIDE DERIVATIVES USEFUL AS HISTONE DEACETYLASE INHIBITORS
#6785N-aroyl cyclic amines
#6786Pyridazine compounds and methods
#6787Pesticides and uses thereof
#6788Tetrazine-based bio-orthogonal coupling reagents and methods
#6789Anti-cancer cyclopenta[g]quinazoline compounds
#6790ARYL/HETARYLAMIDES AS MODULATORS OF THE EP2 RECEPTOR
#6791DIAMINOPYRIMIDINES AS MODULATORS OF THE EP2 RECEPTOR
#6792PHTHALAZINONE DERIVATIVES
#6793Fused Heteroaryl Derivatives for Use as P38 Kinase Inhibitors
#6794INHIBITORS OF SERINE PROTEASE, PARTICULARLY HCV NS3-NS4A PROTEASE
#6795Radiolabelling via fluorination of aziridines
#6796CAPPED PYRAZINOYLGUANIDINE SODIUM CHANNEL BLOCKERS
#6797Kinase inhibitors, compositions thereof, and methods of use therewith
#6798Inhibitors of glutaminyl cyclase
#6799Compounds for Inhibiting Beta-Amyloid Production
#6800Cyanoguanidines and cyanoamidines as ErbB2 and EGFR inhibitors
#6801Bicyclic derivatives as modulators of ion channels
#6802Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors
#6803New Aza-Bicyclohexane Compounds Useful As Inhibitors Of Thrombin
#6804N-aroyl cyclic amines
#6805Therapeutic applications of pro-apoptotic benzodiazepines
#6806Substituted pyrazinone derivatives for use in MCH-1 mediated diseases
#6807Dipeptidyl peptidase inhibitors
#6808Nitro-imidazole hypoxia imaging agents
#6809Gas generant compositions
#6810Alkinyl-Oxypyrimidines Used in the Form of Pesticides
#6811QUINOXALINYL MACROCYCLIC HEPATITIS C VIRUS SERINE PROTEASE INHIBITORS
#6812Thyroid hormone analogs
#6813Cyclohexyl derivatives
#6814AMINO-SUBSTITUTED QUINAZOLINE DERIVATIVES AS INHIBITORS OF BETA-CATENIN/TCF-4 PATHWAY AND CANCER TREATMENT AGENTS
#6815FLUID STORAGE AND DISPENSING METHODS AND APPARATUS
#6816Pyridine derivatives and pyrimidine derivatives (3)
#6817Phenylacetamides suitable as protein kinase inhibitors
#6818Pyrimidine Kinase Inhibitors
#6819METHODS FOR MODULATING BONE FORMATION AND MINERALIZATION
#6820Urotensin II receptor antagonists
#6821Heteroaryl benzamide derivatives
#68221-[6,7-substituted alkoxyquinoxalinyl)aminocarbonyl]-4-(hetero)arylpiperazine derivatives
#6823Dual-acting benzoimidazole antihypertensive agents
#68244' SUBSTITUTED COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY
#6825Phenoxypyridine derivative salts and crystals thereof, and process for preparing the same
#68261,3-dihydro-2H-indole-2-one compound and pyrrolidine-2-one compound fused with aromatic heterocycle
#6827Pyridazine compounds, compositions and methods
#6828Labels, their production process and their uses
#6829Indole and benzimidazole derivatives
#6830Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
#6831Substituted Piperazines as Metabotropic Glutamate Receptor Antagonists
#6832Substituted amide derivatives and methods of use
#6833Substituted pyrazines for use in the treatment of inflammatory or allergic conditions
#6834Inhibitors of the 11-beta-hydroxysteroid dehydrogenase Type 1 enzyme
#6835Organic Compounds
#6836Compounds
#6837Diaryl Urea Derivatives in the Treatment of Protein Kinase Dependent Diseases
#6838Sulfonylpyrazole and sulfonylpyrazoline carboxamidine derivatives as 5-HTantagonists
#6839Inhibitors of serine proteases, particularly HCV NS3-NS4A protease
#6840Benzimidazoles useful as modulators of ion channels
#6841Compositions and methods for inhibition of the JAK pathway
#6842Quinazoline Derivatives, Process for Their Preparation and Their Use as Anti-Cancer Agents
#6843Prolinamide-tetrazole derivatives as NK3 receptor antagonists
#6844Metalloproteinase inhibitors
#6845Chemical process for the preparation of an amido-phenoxybenzoic acid compound
#6846Prodrugs of pyrazoline compounds, their preparation and use as medicaments
#6847Derivatives of 3-Azabicyclo[3.1.0] Hexane as Dipeptidyl Peptidase-IV Inhibitors
#6848Pharmaceutically Active Diazepanes
#6849Pyrimidine derivatives for the treatment of abnormal cell growth
#6850Methods of treating emesis using growth hormone secretagogues
#6851Anti-inflammatory medicaments
#6852Fluid Storage and Purification Method and System
#6853Cycloalkane-substituted pyrazoline derivatives, their preparation and use as medicaments
#6854Diaryl triazolmethylamine derivatives, preparation and therapeutic use thereof
#6855AZACYCLYLBENZAMIDE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS
#6856Nitrogen-containing heteroaryl compounds and methods of use thereof
#6857Complexes Comprising alpha2-Adrenergic Receptor Agonists and Compositions
#6858Novel sulfonamide inhibitors of aspartyl protease
#6859Therapeutic Pyrazolo[3,4-b]Pyridines and Indazoles
#6860Chemokine receptor modulators
#6861Pyrimidine derivatives
#6862Fused compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor
#6863Inhibitors of Factor XA and Other Serine Proteases Involved in the Coagulation Cascade
#6864CB1 modulator compounds
#6865Carbamoylbenzotriazole derivatives as inhibitors of lipases and phospholipases
#6866CXCR4 antagonists
#6867HETEROARYL/ARYL PYRIMIDINE ANALOGS AND THEIR USE AS AGONISTS OF THE WNT-BETA-CATENIN CELLULAR MESSAGING SYSTEM
#6868Pyrazole compounds useful as protein kinase inhibitors
#6869Agent for preventing or treating neuropathy
#6870Bicyclic amides as kinase inhibitors
#6871AZOLYLACYLGUANIDINES AS beta-SECRETASE INHIBITORS
#6872PYRIMIDINE DERIVATIVES USEFUL AS INHIBITORS OF PKC-THETA
#6873Methods and compounds for preparing CC-1065 analogs
#6874Amines as small molecule inhibitors
#6875Pyridazine derivatives and their use as therapeutic agents
#6876Cinnoline Compounds as Inhibitors of Phosphodiesterase Type IV (Pde4)
#6877Phenylalanine derivatives
#68785-amino 4-hydroxy-7-(1H-indolmethyl)-8-methylnonamide derivatives as renin inhibitors for the treatment of hypertension
#6879Anti-cancer agents and uses thereof
#6880Selected Cgrp-Antagonists, Processes for Preparing Them and Their Use as Pharmaceutical Compositions
#6881Azetidines
#6882Phenoxy Benzamide Compounds with Utility in the Treatment of Type 2 Diabetes and Obesity
#6883Benzamide Derivatives and Their Use as Glucokinase Activating Agents
#6884Aryl ether compounds and their preparation and use thereof
#6885Pyrazole-isoquinoline urea derivatives as p38 kinase inhibitors
#6886Cycloalkyl lactam derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1
#6887Inhibitors of C-FMS kinase
#6888Compounds for Treating Protein-Kinase Mediated Disorders
#6889Piperazinone Derivatives Useful as Histamine H3 Receptor Antagonists and/or Inverse Agonists
#6890Cyclic malonamides as inhibitors of aβ protein production
#6891Substituted Quinazolones as Anti-Cancer Agents
#6892N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase
#6893Hydroxy-Substituted Diphenylazetidinones for the Treatment of Hyperlipidemia
#6894Process for the preparation of macrocyclic compounds
#68954-ANILINO QUINAZOLINE DERIVATIVES AS ANTIPROLIFERATIVE AGENTS
#6896PYRAZOLE DERIVATIVES AS ANTI-PLATELET AND ANTI-THROMBOTIC AGENTS
#6897Compounds and Methods for Treating Dyslipidemia
#6898Therameutin modulators
#6899Inhibitors of poly(ADP-ribose)polymerase
#6900Prokineticin 1 receptor antagonists