95301 ⎘
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
Tetra- and penta-o-benzyl-protected, C-4 activated-epicatechin and -catechin monomers and processes for their preparation and use
#6602Piperazinyl and piperidinyl ureas as modulators of fatty acid amide hydrolase
#6603Multicyclic bis-amide MMP inhibitors
#6604Methods of treating factor VIIa-associated conditions with compounds having an amine nucleus
#6605Heteroaryl substituted spirocyclic sulfamides for inhibition of gamma secretase
#6606Inhibitors of c-jun -terminal kinases
#6607Heterocyclic amides, method for the production thereof, substances containing said heterocyclic amides, and use thereof as pesticides
#6608Heteroaryl sulfonamides and CCR2
#6609Compounds for inflammation and immune-related uses
#6610Heteroaryl compounds as P2Yreceptor inhibitors
#6611Methods and compositions of novel triazine compounds
#6612Protection against and treatment of hearing loss
#6613Sulfonamide inhibitors of aspartyl protease
#6614Compounds and methods for the inhibition of compounds cruzi
#6615Stereoisomerically enriched 3-aminocarbonyl bicycloheptene pyrimidinediamine compounds and their uses
#6616Process to prepare pioglitazone via several novel intermediates
#6617Compounds for the treatment of CNS and amyloid associated diseases
#6618Heteroarylcarbamoylbenzene derivative
#6619Monocyclic substituted phenyl methanones
#6620Pyrrolydin-2-one derivatives as inhibitors of thrombin and factor xa
#6621Indole derivatives as ppar modulators
#6622N-(substituted arylmethyl)-4-(disubstituted methyl)piperidines and piperazines
#6623Tetrahydrocarbazole derivatives and their pharmaceutical use
#66243-phenylpropionic acid derivatives
#6625Thiazole-4-carboxyamide derivatives
#6626Tetrahydroisoquinolines as factor Xa inhibitors
#6627Nitrogen-containing aromatic derivatives
#6628Phosphodiesterase 10 inhibitors
#6629Carboxylic acid derivatives, their preparation and their use
#6630Pyrimidinone derivatives as therapeutic agents against acute and chronic inflammatory, ischaemic and remodelling processes
#6631Transcription factor modulating compounds and methods of use thereof
#6632Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
#6633Tachykinin receptor antagonists
#6634Optical recording materials having high storage density
#6635Modulators of cytokine mediated signaling pathways and integrin alphabeta3 receptor antagonists for combination therapy
#6636Fungicidal 1,2,3 triazole derivatives
#6637Phthalazinone derivatives
#6638Compounds that modulate PPARγ type receptors and cosmetic/pharmaceutical compositions comprised thereof
#6639Carboxamide derivatives
#6640Coumarin-amide derivatives and its preparation, said drug composition and its use
#66415-Phenylthiazole derivatives and their use as p13 kinase inhibitors
#6642Pyrazole compounds
#6643Therapeutic agents useful for treating pain
#6644Dipeptidyl peptidase IV inhibitors pharmaceutical compositions containing them, and process for their preparation
#6645Benzazole analogues and uses thereof
#6646Polycyclic sulphamate compounds suitable for use as inhibitors of aromatase and/or sulphatase
#6647Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1
#6648Compounds and methods for the treatment or prevention of infections
#6649Piperidine derivative and use thereof
#6650Dual binding site acetylcholinesterase inhibitors for the treatment of alzheimer's disease
#6651Oxy substituted chalcones as antihyperglycemic and antidyslipidemic agents
#6652Phthalazinone derivatives
#6653Therapeutic agent for senile dementia
#6654Amide derivatives
#6655Benzazole analogues and uses thereof
#6656N-acyl nitrogen heterocycles as ligands of peroxisome proliferator-activated receptors
#66571h-Indazole-3-carboxamide compounds as cyclin dependent kinase (cdk) inhibitors
#6658Heterocyclic inhibitors of kinases
#66592-acylamino-4-phenylthiazole derivatives, preparation thereof and therapeutic application thereof
#6660Benzothiazole-4,7-diones and benzoxazole-4,7-diones with substituents in position 5 or 6 and method for production thereof
#66612,4-Pyrimidinediamine compounds and their uses
#6662Phosphodiesterase 4 inhibitors
#6663Platelet adenosine diphosphate receptor antagonists
#6664Fused heterocyclic compounds as peptidase inhibitors
#66655-ARYLTETRAZOLE COMPOUNDS AND COMPOSITIONS THEREOF
#6666N-(substituted arylmethyl)-4-(disubstituted methyl) piperidines and pyridines
#66671,2,4-thiadiazole derivatives as melanocortin receptor modulators
#6668Thiazole derivatives
#6669Tubulysins, method for producing the same and tubulysin preparations
#6670Biaryl compounds having anti-infective activity
#6671Lactam glycogen phosphorylase inhibitors and method of use
#6672Heterocyclic compounds having inhibitory activity against HIV integrase
#66739-ketospinosyn derivatives
#6674Computer program code size partitioning method for multiple memory multi-processing systems
#6675Aryl piperidine derivatives and use thereof to reduce elevated levels of ldl-cholesterol
#6676Biaryloxymethylarenecarboxylic acids as glycogen synthase activators
#6677Inhibitors of IMPDH enzyme
#66782-aryloxy-2-arylalkanoic acids for diabetes and lipid disorders
#6679Substituted biaryl-carboxylate derivatives
#66804,5-diarylthiazole derivatives as cb-1 ligands
#6681Quinoline and quinoxaline compounds
#6682Heterocycle substituted carboxylic acids
#6683Fused heteroaryl derivatives for use as P38 kinase inhibitors
#6684Uracil-thioether
#6685Sulphonamide compounds that modulate chemokine receptor activity (ccr4)
#6686N-(indolethyl-)cycloamine compounds
#6687Platelet adenosine diphosphate receptor antagonists
#6688Heteroaromatic pentacyclic compound and medicinal use thereof
#6689Substituted iminoazines
#6690Pyrido[2,3-D]pyrimidine inhibitors of phosphodiesterase (PDE) 7
#6691Process for the purification of meloxicam
#6692Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
#6693Thrombopoietin activity modulating compounds and methods
#6694N-substituted benzothiophenesulfonamide derivatives
#6695Amide derivatives
#66967-(1,3-thiazol-2-YL)thio-coumarin derivatives and their use as leukotriene biosynthesis inhibitors
#6697Indol derivatives and their use as 5-HT ligands
#6698Hepatitis c virus inhibitors
#66991-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
#6700Integrin antagonists useful as anticancer agents
#67014-Piperidinecarboxamide modulators of vanilloid VR1 receptor
#6702Azabicyclo derivatives as muscarinic receptor antagonists
#6703Substituted 5-oxo pyrazoles and [1,2,4]triazoles as antiviral agents
#67041-phenyl1-3,4-dihydropyrimidin-2(1H)-one derivatives and their use
#6705Substituted arylcyclopropylacetamides as glucokinase activators
#6706Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient
#6707Substituted hydroxyethylamines
#6708Process for the preparation of thiazolidinedione derivatives
#6709Benzimidazole acetic acids exhibiting CRTH2 receptor antagonism and uses thereof
#6710Benzothiazole derivatives having beta-2-adrenoreceptor agonist activity
#6711Drug efflux pump inhibitor
#6712Heterocyclyls as selective melanin concentrating hormone receptor antagonists for the treatment of obesity and related disorders
#6713Aminopyridine derivatives having Aurora A selective inhibitory action
#6714Novel use of benzothiazole derivatives
#6715Mitotic kinesin inhibitors
#6716Furan or thiophene derivative and medicinal use thereof
#6717Process for the preparation of substituted triazole compounds
#6718Substituted biphenyl-4-carboxylic acid arylamide analogues
#6719Inhibitors of HIV-1 capsid formation: substituted aryl aminomethyl thiazole ureas and analogues thereof
#67202,4-diaminopyrimidine derivatives
#67212-Thiopyrimidinones as therapeutic agents
#6722Heteroaryl guanidines; inhibitors of viral replication
#6723Bradykinin-B1 antagonists, process for their preparation and their use as medicaments
#6724Factor Xa inhibitors
#6725Mitotic kinesin inhibitors and methods of use thereof
#67263-Aryl-3-hydroxy-2-methylenepropionic acid esters as fungicides
#6727Combination of a SRC kinase inhibitor and a BCR-ABL inhibitor for the treatment of proliferative diseases
#6728NK1 antagonists
#6729Indole, azaindole and related heterocyclic ureido and thioureido piperazine derivatives
#6730Benzothiadiazine compounds
#6731Quetiapine analogs and methods of use thereof
#6732Heterocyclic compounds and thrombopoietin receptor activators
#6733Ziprasidone process
#6734Heteroaryl substituted biphenyl derivatives as p38 kinase inhibitors
#67358-hydroxy quinoline derivatives
#6736Substituted thiazines as material protecting agents
#6737Neuropeptide receptor modulators
#6738Lactams and uses thereof
#6739Substituted (thioxo)carbonylaminophenyluracils
#6740Compounds as PDE IV and TNF-inhibitors
#6741Isoxazole derivatives
#6742Aromatic sulfone hydroxamic acid metalloprotease inhibitor
#6743Quinoline derivatives as H3R inverse agonists
#6744Derivatives of amidines, their preparation, their use as medicaments and the pharmaceutical compositions containing them
#6745Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound
#6746Cyclic protein tyrosine kinase inhibitors
#6747Diarylmethylidene piperidine derivatives, preparations thereof and uses thereof
#6748Quinoline derivatives as glucokinase ligands
#6749Anilino-pyrimidine analogs
#6750Morpholin-acetamide derivatives for the treatment of inflammatory diseases
#6751Thiazolidinones and the use therof as polo-like kinase inhibitors
#6752Hydroxamic acid and amide compounds and their use as protease inhibitors
#6753Cyclic AMP-specific phosphodiesterase inhibitors
#6754Inhibitors of soluble adenylate cyclase
#6755Modulators of ATP-binding cassette transporters
#6756Substituted arylamides
#6757Sulfonamide compounds
#6758Ophthalmic compositions for treating ocular hypertension
#6759Sulfonamides, sulfamates and sulfamides as gamma-secretase inhibitors
#6760Thiazole-based nitric oxide donors capable of releasing two or more nitric oxide molecules and uses thereof
#6761Thiazole-based nitric oxide donors having alkyl substituent(s) and uses thereof
#6762Chemokine receptor binding heterocyclic compounds
#676317β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
#6764Heterocyclic NF-κB inhibitors
#6765Prodrugs of protein tyrosine kinase inhibitors
#6766Bicyclic compound
#6767Triazine compounds
#6768Histamine-3 receptor antagonists
#6769Receptor-type kinase modulators and methods of use
#6770Compounds for the treatment of inflammatory disorders
#6771Substituted hydantoins
#67723-Hetero arylmethoxy ! pyridines and their analogues as p38 map kinase inhibitors
#6773Pyridyl inhibitors of hedgehog signalling
#6774Use of aryl- and heteroaryl-substituted tetrahydroisoquinolines to block reuptake of norepinephrine, dopamine, and serotonin
#6775Morpholinyl-urea derivatives for use in the treatment of inflammatory diseases
#67762-substituted heteroaryl compounds
#6777Quinazoline compounds
#6778Benzofuran derivatives, process for their preparation and intermediates thereof
#6779Vanilloid receptor ligands and their use in treatments
#67802,4-pyrimidinediamine compounds and their uses
#6781CA IX-specific inhibitors
#6782Substituted heterocyclic compounds
#6783Process for preparing substituted phenoxy-acetic acids from phenols
#6784HDAC inhibitor
#6785Aryloxyalkylamine derivatives as h3 receptor ligands
#6786Acylaminothiazole derivatives, their preparation and their therapeutic use
#6787Conjugation agent
#6788Thiazolo-naphthyl acids
#67892-Amido-thiazole-based compounds exhibiting ATP-utilizing enzyme inhibitory activity, and compositions, and uses thereof
#6790Pyridone derivatives having a binding activity to the cannabinoid type 2 receptor
#6791Capped pyrazinoylguanidine sodium channel blockers
#6792Capped pyrazinoylguanidine sodium channel blockers
#6793Isoindoline derivative
#6794Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
#6795Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
#6796Amino-tetrazole analogues and methods of use
#6797Pyridine derivatives as fungicidal compounds
#6798Modulators of ATP-binding cassette transporters
#6799Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
#6800Substituted quinazoline derivatives and their use as inhibitors
#6801Gamma-lactams as beta-secretase inhibitors
#6802Substituted hydantoins
#6803PDE4B inhibitors and uses therefor
#6804Benzothiazole-and benzoxazole-4, 7-dione derivatives and their use as dcd25 phosphatase inhibitors
#6805Substituted amide beta secretase inhibitors
#68065-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazolidine-2,4-dione Mesylate salt
#6807Antiinflammatory 3-arylthio-3-thiazolyl-alkylamines
#6808Thiobenzimidazole derivatives
#6809Compounds with anti-bacterial activity
#6810Benzazepine derivatives for the treatment of neurological disorders
#6811Piperazine urea derivatives as melanocortin-4 receptor agonists
#6812Substituted indole compounds, their preparation and use in medicaments
#68132,4-pyrimidinediamine compounds and their uses
#6814Cycloalkyl substituted pyrimidinediamine compounds and their uses
#6815Azo-metal chelate dye and optical recording medium
#6816N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation
#6817PNA monomer and precursor
#6818Vanilloid receptor ligands and their use in treatments
#6819Novel 1,2,4-thiadiazolium derivatives as melanocortin receptor modulators
#6820Thiazolyl inhibitors of Tec family tyrosine kinases
#6821Substituted N-acyl-2-aminothiazoles
#6822Heteroaryl urea neuropeptide Y Y5 receptor antagonists
#6823Cyclopropyl-thienyl-carboxamide as fungicides
#6824Sulfonamides as inhibitors of histone deacetylase for the treatment of disease
#6825Uracils having a herbicidal activity
#6826Compounds and methods for inhibiting the interaction of BCL proteins with binding partners
#6827Hydroxyethylamine derivatives for the treatment of Alzheimer's disease
#6828Isothiazole dioxides as CXC- and CC-chemokine receptor ligands
#6829Pyrimidyl sulphone amide derivatives as chemokine receptor modulators
#6830Remedy for integration dysfunction syndrome
#6831Substituted aryl acylthioureas and related compounds; inhibitors of viral replication
#6832Compositions useful as inhibitors of voltage-gated sodium channels
#68332,4-pyrimidinediamine compounds and their uses
#6834Process for the preparation of crystalline form-1 of 4-hydroxy-2-methyl-N-(5-methyl-2-thiazolyl)-2H-1,2-benzothiazine-3-carboxamide-1,1-dioxide
#68351,2,3,4-tetrahydropyrazin-2-yl acetamides and methods of use
#6836Chemical linkers and conjugates thereof
#6837Processes and intermediates
#6838Compounds, compositions and methods
#6839Ophthalmic compositions for treating ocular hypertension
#6840Histamine-3 receptor antagonist
#6841Methods and compositions for the treatment of neuroleptic and related disorders using ziprasidone metabolites
#6842Gonadotropin releasing hormone receptor antagonists
#6843Benzothiazole derivatives
#6844Therapeutic chromone compounds
#6845Hepatitis C inhibitor peptide analogs
#6846Bicyclic and tricyclic amines as modulators of chemokine receptor activity
#6847Thiadiazole compound and use thereof
#68484-Aminothiazole derivatives
#6849Substituted aryl thioureas and related compounds; inhibitors of viral replication
#6850CXCR1 and CXCR2 chemokine antagonists
#6851Heterocyclo inhibitors of potassium channel function
#6852BICYCLIC, SUBSTITUTED TRIAZOLES AS MODULATORS OF PPAR AND METHODS OF THEIR PREPARATION
#6853Sulfonylamino-acetic acid derivatives
#6854Thiazole, imidazole and oxazole compounds and treatments of disorders associated with protein aging
#6855Compounds, compositions and methods
#6856Methods for the use of inhibitors of cytosolic phospholipase A2
#685717 β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
#6858Inhibitors of IAP
#6859Azo compound, tautomer thereof, and azo dye
#6860N-(2-Arylethyl) benzylamines as antagonists of the 5-HTreceptor
#6861Substituted imidazole derivatives
#6862PNA monomer and precursor
#6863Isothiazoloanthrones, isoxazoloanthrones, isoindolanthrones and derivatives thereof a JNK inhibitors and compositions and methods related thereto
#6864Agent for preventing or treating neuropathy
#6865Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
#6866Sodium salts of 5-'4-'2-(N-methyl-N-(2-pyridyl) amino) ethoxy!benzyl!thiazolidine -2, 4-dione
#68673-glyoxylamideindoles for treating cancer
#6868Compounds for treatment of neurodegenerative diseases
#6869Pyrimidine derivatives as modulators of chemokine receptor activity
#6870Quinazoline derivatives as angiogenesis inhibitors
#6871Cinnamide compound
#6872Indazolecarboxamide derivatives, preparation and use thereof as CDK1, CDK2 and CDK4 inhibitors
#6873Benzothiazole derivatives with activity as adenosine receptor ligands
#6874Method of making PNA oligomers
#68751,3-Oxazole compounds for the treatment of cancer
#6876Substituted thiazolidinedione derivative, process for its preparation and its pharmaceutical use
#6877Use of 2-amino-thiazoline derivatives as inhibitors of inducible no-synthase
#68783-amino-2-phenylpyrrolidine derivatives
#6879Certain triazole-based compounds, compositions, and uses thereof
#6880Cysteine protease inhibitors
#68812,4-diaminoquinazolines for spinal muscular atrophy
#6882N-biarylmethyl aminocycloalkanecarboxamide derivatives
#6883Cyclic protein tyrosine kinase inhibitors
#6884Anti-inflammatory medicaments
#6885Compounds as inhibitors of hepatitis C virus NS3 serine protease
#6886PNA monomer and precursor
#68873-(3,5-Disubstituted-4-hydroxyphenyl)propionamide derivatives as cathepsin b inhibitors
#6888Hydrochloride salt of 5-[4-[2-(N-methyl-N-(2-pyridyl)amino)ethoxy]benzyl]thiazo-lidine-2,4-dione
#6889Heterocyclic substituted indane derivatives and related compounds for the treatment of schizophrenia
#6890Ubiquitin ligase inhibitors
#6891Aminobenzamide derivative
#6892Sodium salts of 5-'4-'2-(N-methyl-N-(2-pyridyl)amino)ethoxy!benzyl!thiazolidine-2, 4-dione
#6893M3muscarinic acetylcholine receptor antagonists
#68943-Aryl-3-hydroxy-and 3-aryl-3-oxopropionic acid esters as fungicides
#6895Preparation of an anhydrate form of 5-[2-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]ethyl]-6-chloro-1,3-dihydro-2H-indol-2-one hydrochloride (ziprasidone hydrochloride)
#6896Vanilloid receptor ligands and their use in treatments
#6897Vanilloid receptor ligands and their use in treatments
#6898Substituted thiophene carboxamides
#6899Vanilloid receptor ligands and their use in treatments
#6900Phosphodiesterase 4 inhibitors