ClassID:

95375 āŽ˜

C07D473/08 - CPC Classification

Classification description:

Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3 with methyl radicals in positions 1 and 3, e.g. theophylline

Recent Application in this class:
#1
20260151398
2026-06-04

COMPOUNDS FOR REDUCING CHOLESTEROL AND TREATING LIVER AND KIDNEY DISEASE

#2
20260062414
2026-03-05

NOVEL COCRYSTALS OF METHYLXANTHINES, THEIR POLYMORPHS AND PROCESS THEREOF

#3
20260035361
2026-02-05

COMPOUNDS FOR MODULATING HUR (ELAVL1)

#4
20250353850
2025-11-20

CYCLIC AMIDE-CONTAINING PYRIDYL XANTHINES AS A2B ANTAGONISTS

#5
20240415937
2024-12-19

THEOPHYLLINE-LOADED COLLAGEN NANOPARTICLES

#6
20240360095
2024-10-31

NOVEL KINASE MODULATORS

#7
20240124457
2024-04-18

Cyclic amide-containing pyridyl xanthines as AB antagonists

#8
20240109892
2024-04-04

POLY(ADP-RIBOSE) GLYCOHYDROLASE (PARG) INHIBITORS AGAINST COVID MACRODOMAIN AND METHODS OF USING THE SAME

#9
20230219957
2023-07-13

SMALL MOLECULE CB002-ANALOGES RESTORE THE P53 PATHWAY AND TARGET S-PHASE CHECKPOINT

#10
20230174533
2023-06-08

PURINE DIONES AS WNT PATHWAY MODULATORS

#11
20220402919
2022-12-22

Cyclic amide-containing pyridyl xanthines as Aantagonists

#12
20220104495
2022-04-07

THEOPHYLLINE DERIVATIVES WITH NEMATOCIDAL ACTIVITY, THEIR AGRONOMIC COMPOSITIONS AND RELATIVE USE

#13
20220073519
2022-03-10

Compounds For Repressing Cancer Cell Growth

#14
20210391038
2021-12-16

SPECIFICALLY-SHAPED CRYSTAL OF COMPOUND AND METHOD FOR PRODUCING SAME

#15
20210313015
2021-10-07

SPECIFICALLY-SHAPED CRYSTAL OF COMPOUND AND METHOD FOR PRODUCING SAME

#16
20210155623
2021-05-27

Purine diones as Wnt pathway modulators

#17
20210128566
2021-05-06

NOVEL FUNCTIONALIZED PURINE-2,6-DIONES AND THEIR USE IN MEDICINE

#18
20210037826
2021-02-11

Microbiocidal oxadiazole derivatives

#19
20200399271
2020-12-24

Xanthine analogs as potent anti-West Nile viral agents

#20
20200239427
2020-07-30

Kinase modulators

#21
20200190086
2020-06-18

Purine diones as Wnt pathway modulators

#22
20200002340
2020-01-02

Oxadiazole transient receptor potential channel inhibitors

#23
20190330212
2019-10-31

Inhibiting the transient receptor potential A1 ion channel

#24
20190297892
2019-10-03

Microbiocidal oxadiazole derivatives

#25
20190248791
2019-08-15

NOVEL MODULATORS OF CALCIUM RELEASE-ACTIVATED CALCIUM CHANNEL AND METHODS FOR TREATMENT OF NON-SMALL CELL LUNG CANCER

#26
20190225613
2019-07-25

Compounds for repressing cancer cell growth

#27
20180325906
2018-11-15

THEOBROMINE COMPOSITIONS USEFUL FOR INCREASING FETAL WEIGHT GAIN AND ENHANCING BONE PROPERTIES

#28
20180291025
2018-10-11

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#29
20180230149
2018-08-16

Inhibiting the transient receptor potential A1 ion channel

#30
20180170932
2018-06-21

Purine diones as Wnt pathway modulators

#31
20180127631
2018-05-10

Anti-ice nucleation activator

#32
20180093986
2018-04-05

Methods and compositions for treating pain

#33
20180057495
2018-03-01

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#34
20170334912
2017-11-23

Purine diones as Wnt pathway modulators

#35
20170326148
2017-11-16

Prevention or treatment of uratic or gouty diseases

#36
20170312285
2017-11-02

Compounds for the treatment of myotonic dystrophy

#37
20170275285
2017-09-28

Inhibiting the transient receptor potential A1 ion channel

#38
20170050966
2017-02-23

INHIBITING THE TRANSIENT RECEPTOR POTENTIAL A1 ION CHANNEL

#39
20160318890
2016-11-03

Kinase modulators

#40
20160229823
2016-08-11

Deuterated compounds useful for treating neurodegenerative diseases

#41
20160194327
2016-07-07

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and thier use as pharmaceutical compositions

#42
20160145257
2016-05-26

SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF

#43
20160090386
2016-03-31

Purine diones as Wnt pathway modulators

#44
20160038499
2016-02-11

Composition useful for treating disorders related to TRPA1

#45
20160030434
2016-02-04

Theobromine compositions useful for increasing fetal weight gain and enhancing bone properties

#46
20160002239
2016-01-07

Flagellar and needle complex (injectosome) loop as anti bacterial drug target

#47
20150307503
2015-10-29

Small molecule bicyclic and tricyclic CFTR correctors

#48
20150291627
2015-10-15

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#49
20150291588
2015-10-15

Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer

#50
20150218166
2015-08-06

Process for the preparation of acebrophylline

#51
20150183788
2015-07-02

Xanthine derivative

#52
20150018321
2015-01-15

Derivatives of 1-phenyl-2-pyridinyl alkyl alcohols as phosphodiesterase inhibitors

#53
20140275528
2014-09-18

SUBSTITUTED XANTHINES AND METHODS OF USE THEREOF

#54
20140221401
2014-08-07

Methods and compositions for treating pain

#55
20140206650
2014-07-24

Inhibiting the transient receptor potential A1 ion channel

#56
20140194447
2014-07-10

Caffeinated compounds and compositions for treatment of amyloid diseases and synucleinopathies

#57
20140163048
2014-06-12

COMPOSITIONS WITH INCREASED STABILITY FOR INHIBITING TRANSIENT RECEPTOR POTENTIAL ION CHANNEL TRPA1

#58
20140158116
2014-06-12

INHIBITING TRPA1 FOR THE TREATMENT OF ASTHMA

#59
20140142307
2014-05-22

Azolium and purinium salt anticancer and antimicrobial agents

#60
20140128604
2014-05-08

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#61
20140100224
2014-04-10

NEUROTROPHIN MIMETICS AND USES THEREOF

#62
20140073656
2014-03-13

SERMs for the treatment of estrogen receptor-mediated disorders

#63
20140057901
2014-02-27

XANTHINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS

#64
20140045824
2014-02-13

Method for producing complex crystal and method for screening complex crystal

#65
20140005208
2014-01-02

Compositions useful for treating disorders related to TRPA1

#66
20130310404
2013-11-21

Inhibitors of p75 receptor and their uses

#67
20130310347
2013-11-21

MULTI-MODALITY MOLECULAR IMAGING HIGH-THROUGHPUT ASSAY FOR IDENTIFYING HEAT SHOCK PROTEIN 90 (HSP90) INHIBITORS

#68
20130310345
2013-11-21

Use of TRPA1 antagonists to prevent or treat infections caused by biological-warfare agents

#69
20130303491
2013-11-14

Antiviral drugs for treatment or prevention of dengue infection

#70
20130274273
2013-10-17

Inhibiting transient receptor potential ion channel TRPA1

#71
20130202549
2013-08-08

USE OF DPAS AND CO-POLYMERS FOR HYPERLIPIDEMIA AND ATHEROSCLEROSIS ALONG WITH REDUCING FEEDING RATE AND ADIPOSE TISSUE WEIGHT OF OBESITY ANIMAL

#72
20130165428
2013-06-27

XANTHINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS

#73
20130137648
2013-05-30

DERIVATIVES OF 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOLS AS PHOSPHODIESTERASE INHIBITORS

#74
20130123283
2013-05-16

Methods and compositions for treating pain

#75
20130059869
2013-03-07

METHODS AND COMPOSITIONS FOR TREATING DISORDERS

#76
20130036938
2013-02-14

Azo compound, azo pigment, pigment dispersion, coloring composition, color filter, ink for inkjet recording, and printing ink

#77
20120322799
2012-12-20

DEUTERATED COMPOUNDS USEFUL FOR TREATING NEURODEGENERATIVE DISEASES

#78
20120252783
2012-10-04

Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions

#79
20120252782
2012-10-04

Xanthine Derivatives, the Preparation Thereof and Their Use as Pharmaceutical Compositions

#80
20120251482
2012-10-04

USE FOR IMPROVING 5-HT FUNCTION AND ENOS EXPRESSION OF KMUPS AMINE SALTS

#81
20120208831
2012-08-16

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#82
20120116097
2012-05-10

Process for preparing heteroaromatic ring compound having N-Rf group

#83
20120116091
2012-05-10

Derivatives of 1-phenyl-2-pyridinyl alkyl alcohols as phosphodiesterase inhibitors

#84
20120095013
2012-04-19

USE OF KMUP-3 FOR MYOCARDIAL INFARCTION

#85
20120059001
2012-03-08

4H-chromen-4-one compounds as modulators of protein kinases

#86
20120040982
2012-02-16

Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions

#87
20120035158
2012-02-09

Xanthine Derivatives, the Preparation Thereof and Their Use as Pharmaceutical Compositions

#88
20110230479
2011-09-22

NEUROTROPHIN MIMETICS AND USES THEREOF

#89
20110144095
2011-06-16

Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions

#90
20110144083
2011-06-16

Xanthine Derivatives, the Preparation Thereof and Their Use as Pharmaceutical Compositions

#91
20110144075
2011-06-16

DERIVATIVES OF 1-PHENYL-2-PYRIDINYL ALKYL ALCOHOLS AS PHOSPHODIESTERASE INHIBITORS

#92
20110144070
2011-06-16

Derivatives of 1-phenyl-2-pyridinyl alkyl alcohols as phosphodiesterase inhibitors

#93
20110118464
2011-05-19

HALOGENATED XANTHINE DERIVATIVES AND PRECURSORS THEREOF FOR ANTI-CANCER AND ANTI-METASTASIS ACTIVITY AND PREPARING METHOD THEREOF

#94
20110118257
2011-05-19

2,3-disubstituted chromen-4-one compounds as modulators of protein kinases

#95
20110112058
2011-05-12

Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer

#96
20110086868
2011-04-14

SPECIFIC INHIBITORS FOR VASCULAR ENDOTHELIAL GROWTH FACTOR RECEPTORS

#97
20110009430
2011-01-13

Methods and compositions for treating asthma

#98
20100317671
2010-12-16

XANTHINE-BASED CYCLIC GMP-ENHANCING RHO-KINASE INHIBITOR INHIBITS PHYSIOLOGICAL ACTIVITIES OF LUNG EPITHELIAL CELL LINE

#99
20100280040
2010-11-04

SYNTHESIS AND PHARMACOKINETIC ACTIVITIES OF PULMODIL AND PULMODIL-1, TWO CHLOROPHENYLPIPERAZINE SALT DERIVATIVES

#100
20100273780
2010-10-28

SUBSTITUTED 8-HETEROARYL XANTHINES

#101
20100267750
2010-10-21

Methods and compositions for treating pain

#102
20100249154
2010-09-30

Compositions useful for treating disorders related to TRPA1

#103
20100222598
2010-09-02

Process for preparing heteroaromatic ring compound having N-Rf group

#104
20100204250
2010-08-12

Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions

#105
20100189685
2010-07-29

Antiviral drugs for treatment or prevention of dengue infection

#106
20100173916
2010-07-08

Xanthine Derivatives, the Preparation Thereof and Their Use as Pharmaceutical Compositions

#107
20100087455
2010-04-08

SUBSTITUTED XANTHINE COMPOUNDS

#108
20100016329
2010-01-21

XANTHINE-BASED CYCLIC GMP-ENHANCING RHO-KINASE INHIBITOR INHIBITS PHYSIOLOGICAL ACTIVITIES OF LUNG EPITHELIAL CELL LINE

#109
20090298744
2009-12-03

Heterocyclic compounds as adenosine receptor antagonist

#110
20090209560
2009-08-20

ANTI-INFLAMMATION ACTIVITY OF NEWLY SYNTHESIZED XANTHINE DERIVATIVES KMUP-1 AND KMUP-3

#111
20090143377
2009-06-04

Methods and compositions for treating disorders

#112
20090137802
2009-05-28

A2B ADENOSINE RECEPTOR ANTAGONISTS

#113
20090048220
2009-02-19

Derivatives of 1-phenyl-2-pyridinyl alkyl alcohols as phosphodiesterase inhibitors

#114
20090018148
2009-01-15

Xanthine Derivatives, Processes For Preparing Them And Their Uses

#115
20080318983
2008-12-25

A2B ADENOSINE RECEPTOR ANTAGONISTS

#116
20080255159
2008-10-16

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#117
20080249089
2008-10-09

8-[3-amino-piperidin-1-yl]-xanthines, the preparation thereof and their use as pharmaceutical compositions

#118
20080200456
2008-08-21

Substituted 8-heteroaryl xanthines

#119
20080194593
2008-08-14

A2B ADENOSINE RECEPTOR ANTAGONISTS

#120
20080139585
2008-06-12

Specific inhibitors for vascular endothelial growth factor receptors

#121
20080113993
2008-05-15

BARBITURIC ACID ANALOGS AS THERAPEUTIC AGENTS

#122
20080081816
2008-04-03

ANTI-INFLAMMATION ACTIVITY OF NEWLY SYNTHESIZED XANTHINE DERIVATIVES KMUP-1 AND KMUP-3

#123
20080064705
2008-03-13

Theophylline-based nitophenylpiperazine derivatives for enhancing aortic smooth muscle relaxation

#124
20080058354
2008-03-06

Xanthine phosphodiesterase V inhibitors

#125
20080045549
2008-02-21

Adenosine A2B receptor antagonists

#126
20070265284
2007-11-15

Substituted 8-aminoalkylthioxanthines, and their use as inhibitors of dipeptidyl peptidase IV

#127
20070219222
2007-09-20

Methods and compositions for treating pain

#128
20070213316
2007-09-13

N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives

#129
20070179297
2007-08-02

Chemical compounds

#130
20070161663
2007-07-12

Agents for treating migraine

#131
20070142631
2007-06-21

Conjugates of mycophenolic acid

#132
20060281921
2006-12-14

Aadenosine receptor antagonists

#133
20060247226
2006-11-02

XANTHINE DERIVATIVES, THE PREPARATION THEREOF AND THEIR USE AS PHARMACEUTICAL COMPOSITIONS

#134
20060205711
2006-09-14

Xanthine derivatives, the preparation thereof and their use as pharmaceutical compositions

#135
20060142309
2006-06-29

8-heteroaryl xanthine adenosine Areceptor antagonists

#136
20060084667
2006-04-20

Derivatives of amidines, their preparation, their use as medicaments and the pharmaceutical compositions containing them

#137
20050261269
2005-11-24

Derivatives of amidines, their preparation, their use as medicaments and the pharmaceutical compositions containing them

#138
20050209243
2005-09-22

Theophylline-based soluble guanylyl cyclase activators KMUP-1 analogues enhanced cyclic GMP and K+ channel activities on rabbit corpus cavernosum smooth muscle and intercavernous pressure activities

#139
20050209242
2005-09-22

Theophylline and 3-isobutyl-1 methylxanthine based N-7 substituted derivatives displaying inhibitory activities on PDE-5 phospodiesterase

#140
20050182077
2005-08-18

Xanthine phosphodiesterase V inhibitors

#141
20050171092
2005-08-04

Chemical compounds

#142
20050106652
2005-05-19

Electrochemiluminescent assays

#143
20050101778
2005-05-12

Aadenosine receptor antagonists

#144
20050075349
2005-04-07

Xanthine phosphodiesterase V inhibitors

#145
20050065341
2005-03-24

Substituted 8-heteroaryl xanthines

#146
20050038045
2005-02-17

Aadenosine receptor antagonists

#147
20050009829
2005-01-13

Benzimidazole-derivatives as factor Xa inhibitors

#148
20050009076
2005-01-13

Conjugates of mycophenolic acid