ClassID:

96227

C07F9/65583 - CPC Classification

Classification description:

Compounds containing elements of Groups 5 or 15 of the Periodic System; Phosphorus compounds; Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing at least two different or differently substituted hetero rings neither condensed among themselves nor condensed with a common carbocyclic ring or ring system each of the hetero rings containing nitrogen as ring hetero atom

Recent Application in this class:
#1
20260137698
2026-05-21

CYCLIN-DEPENDENT KINASE 7 INHIBITORS

#2
20260132160
2026-05-14

IRON REPLACEMENT TREATMENTS

#3
20260132158
2026-05-14

PHENYL OXY AMIDE KINASE INHIBITORS

#4
20260132121
2026-05-14

INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF

#5
20260125370
2026-05-07

SULFOXIMINE COMPOUNDS AS HISTONE DEACETYLASE 6 INHIBITOR, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME

#6
20260116903
2026-04-30

AROMATIC HETEROCYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION, AND USE THEREOF

#7
20260103480
2026-04-16

NUCLEOTIDE PRECURSORS, NUCLEOTIDE ANALOGS AND OLIGOMERIC COMPOUNDS CONTAINING THE SAME

#8
20260103479
2026-04-16

PRODRUGS OF OPICAPONE

#9
20260103456
2026-04-16

COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, SYNTHESIS METHOD THEREFOR AND USE THEREOF

#10
20260098043
2026-04-09

POLYCYCLIC COMPOUND AND USE THEREOF

#11
20260085082
2026-03-26

KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE

#12
20260085050
2026-03-26

TRIPLE KINASE INHIBITORS

#13
20260055126
2026-02-26

SMALL MOLECULE COMPOUNDS WITH PHOSPHORYLATED ARYL STRUCTURES AND USE THEREOF

#14
20260042734
2026-02-12

HETEROCYCLIC RING-SUBSTITUTED AROMATIC COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF

#15
20260035393
2026-02-05

INHIBITORS OF CYCLIN-DEPENDENT KINASE 7 (CDK7)

#16
20260035357
2026-02-05

THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION

#17
20260028365
2026-01-29

TYROSINE KINASE 2 INHIBITORS AND USES THEREOF

#18
20260022135
2026-01-22

ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 (ENPP1) INHIBITORS AND USES THEREOF

#19
20260001898
2026-01-01

Heteroaryl compounds as inhibitors of TYK2/JAK1, composition and application thereof

#20
20260000692
2026-01-01

Substituted N-(Pyridin-2-yl)Acetamide Derivatives as CDK12/13 Inhibitors

#21
20250388571
2025-12-25

AMP-ACTIVATED PROTEIN KINASE MODULATOR COMPOUNDS AND USES THEREOF

#22
20250368666
2025-12-04

INDAZOLE COMPOUNDS

#23
20250346616
2025-11-13

ROCK INHIBITORS AND USES THEREOF

#24
20250346591
2025-11-13

THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS AND USES THEREOF

#25
20250346590
2025-11-13

THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS AND USES THEREOF

#26
20250346574
2025-11-13

PYRIDINYL SUBSTITUTED OXOISOINDOLINE COMPOUNDS FOR THE TREATMENT OF CANCER

#27
20250339566
2025-11-06

INHIBITORS OF FIBROBLAST ACTIVATION PROTEIN

#28
20250333428
2025-10-30

COT MODULATORS AND METHODS OF USE THEREOF

#29
20250333398
2025-10-30

MONOARYL AND HETARYL SUBSTITUTED INDAZOLES AND BENZIMIDAZOLES AS STING ANTAGONISTS AND THE USE THEREOF AS MEDICAMENT

#30
20250326744
2025-10-23

PIPERAZINE DERIVATIVE OR SALT THEREOF, AND PHARMACEUTICAL COMPOSITION

#31
20250320241
2025-10-16

OXYGEN SENSING MATERIALS AND METHODS OF USE

#32
20250304608
2025-10-02

PHOSPHORUS COMPOUND AND USE THEREOF

#33
20250304555
2025-10-02

SULFONE PYRIDINE ALKYL AMIDE-SUBSTITUTED HETEROARYL COMPOUNDS

#34
20250296946
2025-09-25

NUCLEIC ACID-POLYPEPTIDE COMPOSITIONS AND USES THEREOF

#35
20250288595
2025-09-18

TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS

#36
20250282746
2025-09-11

HALOGEN-SUBSTITUTED ISOINDOLINE COMPOUND AND USE THEREOF

#37
20250276988
2025-09-04

PROCESSES FOR PREPARING PHOSPHORODIAMIDATE MORPHOLINO OLIGOMERS

#38
20250257086
2025-08-14

EGFR DEGRADATION AGENT

#39
20250243228
2025-07-31

PHOSPHORUS PRODRUGS OF PYRAZOLO-SUBSTITUTED PYRIMIDINE sGC STIMULATORS

#40
20250236611
2025-07-24

PYRAZOLE COMPOUNDS AND USES THEREOF

#41
20250230180
2025-07-17

LPXC INHIBITORS AND USES THEREOF

#42
20250223307
2025-07-10

MDM2/MDMX DOUBLE-TARGET INHIBITOR COMPOUND, PRODRUG, PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#43
20250214940
2025-07-03

HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHOLOGICAL DISORDERS

#44
20250197568
2025-06-19

PHOSPHORUS CONTAINING OLIGOMERS AND POLYMERS

#45
20250197375
2025-06-19

PYRIMIDINES AND METHODS OF THEIR USE

#46
20250188102
2025-06-12

TRIAZINE COMPOUND, INTERMEDIATE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF

#47
20250186432
2025-06-12

SPLEEN TYROSINE KINASE INHIBITOR, COMPOSITION, AND METHODS OF USE

#48
20250171475
2025-05-29

CHIRAL REAGENTS FOR PREPARATION OF HOMOGENEOUS OLIGOMERS

#49
20250171473
2025-05-29

Phosphorous Containing BCL Inhibitors and Senolytic Compounds and Uses Thereof

#50
20250171417
2025-05-29

HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL USE THEREOF

#51
20250171400
2025-05-29

AZA-HETEROCYCLYL CARBOXAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS

#52
20250163086
2025-05-22

Crystalline Forms

#53
20250154105
2025-05-15

POLYCYCLIC COMPOUND AND USE THEREOF

#54
20250145597
2025-05-08

INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF

#55
20250134890
2025-05-01

ANTIMALARIAL HEXAHYDROPYRIMIDINE ANALOGUES

#56
20250127800
2025-04-24

PYRIMIDINE OR PYRIDINE DERIVATIVE AND MEDICINAL USE THEREOF

#57
20250115608
2025-04-10

HORMONE RECEPTOR MODULATORS FOR TREATING METABOLIC CONDITIONS AND DISORDERS

#58
20250102497
2025-03-27

CYANINE DYES AND THEIR BIOLOGICAL CONJUGATES

#59
20250101052
2025-03-27

COMPOUND FOR EGFR KINASE INHIBITOR, COMPOSITION, AND USE THEREOF

#60
20250101012
2025-03-27

HETEROCYCLE SUBSTITUTED PYRIDINE DERIVATIVE ANTIFUNGAL AGENTS

#61
20250099493
2025-03-27

PHOSPHONATES AS INHIBITORS OF ENPP1 AND CDNP

#62
20250092017
2025-03-20

2-PIPERIDYL OR 2-PYRAZOLYL SUBSTITUTED PYRIMIDINE COMPOUND SERVING AS EGFR INHIBITOR

#63
20250066397
2025-02-27

PROTEIN PROXIMITY ASSAY IN FORMALIN FIXED PAFFAFIN EMBEDDED TISSUE USING CAGED HAPTENS

#64
20250066344
2025-02-27

BENZOTHIAZOLE, BENZOISOXAZOLE, AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS

#65
20250064787
2025-02-27

Heterocyclic Carboxylate Compounds as Glycolate Oxidase Inhibitors

#66
20250059218
2025-02-20

ENPP1 Inhibitors and Methods of Modulating Immune Response

#67
20250042926
2025-02-06

THERAPEUTIC COMPOUNDS FOR HIV

#68
20250034185
2025-01-30

PYRIDOXAL-5-PHOSPHATE (P5P) ANALOGS

#69
20250026773
2025-01-23

MONO-P-TOLUENESULFONATE OF AXL KINASE INHIBITOR AND CRYSTAL FORM THEREOF

#70
20250011353
2025-01-09

PROCESS OF PREPARING HIV CAPSID INHIBITOR

#71
20250011352
2025-01-09

SOLID FORMS

#72
20250011348
2025-01-09

Synthesis Process of X-IPM, Stable Crystal Form and Application Thereof

#73
20250002512
2025-01-02

NOVEL ANTI-DEPRESSANT AND NEUROPLASTIC AGENTS AND THERAPEUTIC USES THEREOF

#74
20240425484
2024-12-26

INHIBITORS OF TYK2

#75
20240417396
2024-12-19

INHIBITORS OF TYK2

#76
20240409609
2024-12-12

REVERSIBLE LYSINE COVALENT MODIFIERS OF EGFR AND USES THEREOF

#77
20240400590
2024-12-05

SYNTHESIS OF BACKBONE MODIFIED MORPHOLINO OLIGONUCLEOTIDES AND CHIMERAS USING PHOSPHORAMIDITE CHEMISTRY

#78
20240391940
2024-11-28

FUSED RING-CONTAINING COMPOUND, APPLICATION THEREOF, AND COMPOSITION CONTAINING SAME

#79
20240385182
2024-11-21

MASKED FLUOROGENIC LIPID COMPOUNDS, LIPID PARTICLES COMPRISING THE SAME, AND METHODS OF USE THEREOF

#80
20240383932
2024-11-21

Phenol Prodrugs

#81
20240376138
2024-11-14

Crystal Forms, Preparation Method And Application Of Aryl Phosphine Oxide Compound

#82
20240376137
2024-11-14

NUCLEOTIDE PRECURSORS, NUCLEOTIDE ANALOGS AND OLIGOMERIC COMPOUNDS CONTAINING THE SAME

#83
20240376070
2024-11-14

GPR52 MODULATOR COMPOUNDS

#84
20240374582
2024-11-14

SELECTIVE INHIBITORS OF ROCK1 AND ROCK2 PROTEIN KINASES AND THEIR USES THEREOF

#85
20240368203
2024-11-07

DEGRADATION OF (EGFR) BY CONJUGATION OF EGFR INHIBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE

#86
20240368144
2024-11-07

N-substituted-dioxocyclobutenylamino-3-hydroxy-picolinamides useful as CCR6 inhibitors

#87
20240368122
2024-11-07

JAK2 INHIBITORS AND METHODS OF USE THEREOF

#88
20240368113
2024-11-07

AMIDE COMPOUND AND USE THEREOF

#89
20240360165
2024-10-31

INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7)

#90
20240360164
2024-10-31

PHOSPHORUS PRODRUGS OF PYRAZOLO-SUBSTITUTED PYRIMIDINE SGC STIMULATORS

#91
20240360146
2024-10-31

BRUTON'S TYROSINE KINASE AND MUTANT DEGRADER, COMPOSITION AND APPLICATION THEREOF

#92
20240352053
2024-10-24

SALT AND CRYSTAL FORM OF EGFR INHIBITOR, AND COMPOSITION AND USE THEREOF

#93
20240352046
2024-10-24

ECTONUCLEOTIDE PYROPHOSPHATASE-PHOSPHODIESTERASE-1 (ENPP1) INHIBITORS AND USES THEREOF

#94
20240350655
2024-10-24

THIOL-CONJUGATION WITH UNSATURATED PHOSPHORUS(V) COMPOUNDS

#95
20240343747
2024-10-17

Heteroaryl compounds as inhibitors of TYK2, composition and application thereof

#96
20240336643
2024-10-10

BIFUNCTIONAL COMPOUNDS THAT DEGRADE ALK AND USES THEREOF

#97
20240335462
2024-10-10

SULFUR/PHOSPHORUS-CONTAINING ARYL COMPOUND AND APPLICATION THEREOF

#98
20240327399
2024-10-03

THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS AND USES THEREOF

#99
20240317784
2024-09-26

PROCESS FOR THE SYNTHESIS OF 4-((R)-2-{[6-((S)-3-METHOXY-PYRROLIDIN-1-YL)-2-PHENYL-PYRIMIDINE-4-CARBONYL]-AMINO}-3-PHOSPHONO-PROPIONYL)-PIPERAZINE-1-CARBOXYLIC ACID BUTYL ESTER

#100
20240317741
2024-09-26

NAPHTHYRIDINE DERIVATIVE AS ATR INHIBITOR AND METHOD FOR PREPARING SAME

#101
20240316047
2024-09-26

Inhibitors of RNA helicase DHX9 and uses thereof

#102
20240298524
2024-09-05

N-Doped Semiconducting Material Comprising Phosphine Oxide Matrix and Metal Dopant

#103
20240286999
2024-08-29

AZABICYCLO[3.1.0]HEXANE COMPOUND

#104
20240279258
2024-08-22

MODULATORS OF TNF-ALPHA ACTIVITY

#105
20240270773
2024-08-15

LpxC inhibitors and uses thereof

#106
20240270772
2024-08-15

PHOSPHONATE-CONTAINING CROSSLINKERS

#107
20240270771
2024-08-15

Compound containing phosphate group, pharmaceutical composition containing same, preparation method therefor and use thereof

#108
20240270722
2024-08-15

POLO LIKE KINASE 4 INHIBITORS

#109
20240270698
2024-08-15

NOVEL PYRIMIDINE DERIVATIVE AND USE THEREOF

#110
20240255514
2024-08-01

ULTRA BRIGHT DIMERIC OR POLYMERIC DYES WITH SPACING LINKER GROUPS

#111
20240248094
2024-07-25

ULTRA BRIGHT DIMERIC OR POLYMERIC DYES WITH SPACING LINKER GROUPS

#112
20240228520
2024-07-11

PHOSPHORUS PRODRUGS OF PYRAZOLO-SUBSTITUTED PYRIMIDINE SGC STIMULATORS

#113
20240228469
2024-07-11

PCSK9 INHIBITORS AND METHODS OF USE THEREOF

#114
20240228458
2024-07-11

PYRIMIDINE DERIVATIVE HAVING PROTEIN KINASE INHIBITORY ACTIVITY, AND THERAPEUTIC PHARMACEUTICAL COMPOSITION COMPRISING SAME

#115
20240209363
2024-06-27

OLIGONUCLEOTIDES FOR TREATING EXPANDED REPEAT DISEASES

#116
20240208954
2024-06-27

OXADIAZOLE COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF

#117
20240199654
2024-06-20

CTLA-4 SMALL MOLECULE DEGRADATION AGENT AND APPLICATION THEREOF

#118
20240199583
2024-06-20

ARYL, HETEROARYL, AND HETEROCYCLIC COMPOUNDS FOR TREATMENT OF IMMUNE AND INFLAMMATORY DISORDERS

#119
20240190903
2024-06-13

COMPOUNDS FOR PROGRAMMABLE PROTEIN DEGRADATION AND METHODS OF USE FOR THE TREATMENT OF DISEASE

#120
20240189322
2024-06-13

Tropomyosin-related kinase (trk) inhibitors

#121
20240182504
2024-06-06

BISPHOSPHONATE QUINOLONE CONJUGATES AND USES THEREOF

#122
20240174702
2024-05-30

SOLID FORMS OF A COMPOUND FOR MODULATING COT

#123
20240150313
2024-05-09

TRI-SUBSTITUTED INDOLE BINDING FUNCTION 3 (BF3) COMPOUNDS AND METHODS FOR THEIR USE

#124
20240132528
2024-04-25

PHOSPHORUS PRODRUGS OF PYRAZOLO-SUBSTITUTED PYRIMIDINE SGC STIMULATORS

#125
20240132489
2024-04-25

AROMATIC HETEROCYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION, AND USE THEREOF

#126
20240124504
2024-04-18

AROMATIC HETEROCYCLIC COMPOUND, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF

#127
20240124426
2024-04-18

Polo like kinase 4 inhibitors

#128
20240092788
2024-03-21

MASP-2 INHIBITORS AND METHODS OF USE

#129
20240091200
2024-03-21

Heterocyclic carboxylate compounds as glycolate oxidase inhibitors

#130
20240083925
2024-03-14

Prodrugs of 2-(3,5-Dichloro-1-methyl-indazol-4-yl)-1-[(1S,3R)-3-(hydroxymethyl)-5-(1-hydroxy-1-methyl-ethyl)-1-methyl-3,4-dihydro-1H-isoquinolin-2-yl]ethanone

#131
20240076306
2024-03-07

Modulators of TNF-α activity

#132
20240051978
2024-02-15

3-CYCLIC AMINE-INDOLE DERIVATIVES AS SEROTONERGIC AGENTS FOR THE TREATMENT OF CNS DISORDERS

#133
20240043458
2024-02-08

COT MODULATORS AND METHODS OF USE THEREOF

#134
20240043457
2024-02-08

CRYSTALLINE FORMS OF 5-CHLORO-N4-[-2-(DIMETHYLPHOSPHORYL) PHENYL]-N2-{2-METHOXY-4-[4[(4-METHYLPIPERAZIN-1-YL) PIPERIDIN-1-YL] PHENYL} PYRIMIDINE-2,4-DIAMINE

#135
20240043456
2024-02-08

Crystalline Solid Meglumine Salt Inhibitor of BCL and Methods of Making and Using Same

#136
20240043395
2024-02-08

COMPOUNDS AND COMPOSITIONS AS MODULATORS OF TLR SIGNALING

#137
20240034742
2024-02-01

DOSING REGIMENS FOR CYCLIN-DEPENDENT KINASE 7 (CDK7) INHIBITORS

#138
20240018174
2024-01-18

QUINONE METHIDE ANALOG SIGNAL AMPLIFICATION

#139
20240002364
2024-01-04

SULFONE PYRIDINE ALKYL AMIDE-SUBSTITUTED HETEROARYL COMPOUNDS

#140
20230416287
2023-12-28

Chemical Compounds

#141
20230416257
2023-12-28

TOLL-LIKE RECEPTOR AGONIST

#142
20230416204
2023-12-28

AMINOPYRIDINE COMPOUND AND APPLICATION THEREOF

#143
20230373935
2023-11-23

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR

#144
20230366045
2023-11-16

NUCLEIC ACID CROSSLINKING REAGENTS AND USES THEREOF

#145
20230357253
2023-11-09

AGONISTS OF STIMULATOR OF INTERFERON GENES STING

#146
20230348426
2023-11-02

OXOPYRROLIDINE FPR2 AGONISTS

#147
20230348399
2023-11-02

NOVEL PYRIMIDINE DERIVATIVE AND USE THEREOF

#148
20230339896
2023-10-26

HPK1 INHIBITORS AND USES THEREOF

#149
20230322822
2023-10-12

ARYL PHOSPHOROUS OXIDE COMPOUNDS AND USE THEREOF

#150
20230303503
2023-09-28

CELL ACTIVATABLE IRON CHELATORS

#151
20230295200
2023-09-21

STAT5 and STAT6 Inhibitors and Uses Thereof

#152
20230286947
2023-09-14

COMPLEMENT FACTOR B INHIBITOR, AND PHARMACEUTICAL COMPOSITION, PREPARATION METHOD AND USE THEREOF

#153
20230271986
2023-08-31

Crystalline or Amorphous form of Bcl-2/Bcl-xL inhibitor compound or its salts

#154
20230265116
2023-08-24

DEGRADATION OF (EGFR) BY CONJUGATION OF EGFR INHIBITORS WITH E3 LIGASE LIGAND AND METHODS OF USE

#155
20230234978
2023-07-27

NUCLEIC ACID-POLYPEPTIDE COMPOSITIONS AND USES THEREOF

#156
20230227484
2023-07-20

PYRIMIDINE COMPOUND AS AXL INHIBITOR

#157
20230227483
2023-07-20

PYRIMIDINE COMPOUNDS FOR USE AS MAP4K1 INHIBITORS

#158
20230227437
2023-07-20

IMMUNOMODULATOR

#159
20230219986
2023-07-13

NOVEL AMINOPYRIMIDINE EGFR INHIBITOR

#160
20230212148
2023-07-06

THERAPEUTIC COMPOUNDS FOR HIV VIRUS INFECTION

#161
20230183276
2023-06-15

PYRROLE INHIBITORS OF ERK PROTEIN KINASE, SYNTHESIS THEREOF AND INTERMEDIATES THERETO

#162
20230167142
2023-06-01

METHODS FOR THE MONO-AMIDATION OF PHOSPHATES AND PHOSPHONATES

#163
20230159489
2023-05-25

PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND USE

#164
20230159458
2023-05-25

SOLID SUPPORTS AND PHOSPHORAMIDITE BUILDING BLOCKS FOR OLIGONUCLEOTIDE CONJUGATES

#165
20230151037
2023-05-18

GPR40 AGONISTS

#166
20230150941
2023-05-18

Heterocyclic compounds for the treatment of neurological and psychological disorders

#167
20230145793
2023-05-11

SUBSTITUTED PYRIMIDINE OR PYRIDINE AMINE DERIVATIVE, COMPOSITION THEREOF, AND MEDICAL USE THEREOF

#168
20230139597
2023-05-04

Hormone receptor modulators for treating metabolic conditions and disorders

#169
20230139502
2023-05-04

Aza-heterocyclyl carboxamide and related compounds and their use in treating medical conditions

#170
20230129481
2023-04-27

ULTRA BRIGHT DIMERIC OR POLYMERIC DYES WITH SPACING LINKER GROUPS

#171
20230102829
2023-03-30

Heteroaryl compounds for kinase inhibition

#172
20230082993
2023-03-16

Selective inhibitors of ROCK1 and ROCK2 protein kinases and uses thereof

#173
20230080874
2023-03-16

Tropomyosin-related kinase (Trk) inhibitors

#174
20230071675
2023-03-09

Heterocyclic amides useful as protein modulators

#175
20230071620
2023-03-09

Pharmaceutical compounds for treatment of medical disorders

#176
20230065881
2023-03-02

Heterocycle substituted pyridine derivative antifungal agents

#177
20230062491
2023-03-02

INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7)

#178
20230062100
2023-03-02

SUBSTITUTED AMINOQUINOLONES AS DGKALPHA INHIBITORS FOR IMMUNE ACTIVATION

#179
20230046407
2023-02-16

New-type oxazolidinone compounds and preparation method therefor

#180
20230045831
2023-02-16

Phosphorodiamidate morpholino oligomers

#181
20230039185
2023-02-09

PHOSPHATE DERIVATIVES OF RORGAMMA MODULATORS AND USES THEREOF

#182
20230030115
2023-02-02

RHO-ASSOCIATED PROTEIN KINASE INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND PREPARATION METHOD AND USE THEREOF

#183
20230026840
2023-01-26

COMPOUND USED AS EGFR KINASE INHIBITOR AND USE THEREOF

#184
20230014962
2023-01-19

Quinoline compound and use thereof

#185
20230002397
2023-01-05

SMALL MOLECULE DEGRADERS OF HELIOS AND METODS OF USE

#186
20220389037
2022-12-08

HPK1 INHIBITORS AND USES THEREOF

#187
20220340605
2022-10-27

Processes for preparing phosphorodiamidate morpholino oligomers

#188
20220315995
2022-10-06

THIOL-CONTAINING CLEAVE REAGENTS AND OXIDATIVE WASH

#189
20220315562
2022-10-06

Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders

#190
20220312770
2022-10-06

PYRIDAZINOL COMPOUNDS AND DERIVATIVES, PREPARATION METHODS, HERBICIDAL COMPOSITIONS AND APPLICATIONS THEREOF

#191
20220306659
2022-09-29

COMPOUND INHIBITING AND INDUCING DEGRADATION OF EGFR AND ALK

#192
20220306617
2022-09-29

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Phosphatidylinositol 3-kinase inhibitors

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STAT3 PROTEIN DEGRADERS

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MAGL inhibitors

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Antiviral agents

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Quinone methide analog signal amplification

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Anti-viral compounds

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Inhibitors of cyclin dependent kinase 7 (CDK7)

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Inhibitors of cyclin-dependent kinase 7 (CDK7)

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Phosphorus containing oligomers and polymers

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Phenylpyrrolidinone formyl peptide 2 receptor agonists

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Protein proximity assay in formalin fixed paffafin embedded tissue using caged haptens

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Benzimidazol derivatives for treating filovirus infection

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Sulfone pyridine alkyl amide-substituted heteroaryl compounds

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ANTI-INFECTIVE HETEROCYCLIC COMPOUNDS AND USES THEREOF

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PROTEIN PROXIMITY ASSAY IN FORMALIN FIXED PARAFFIN EMBEDDED TISSUE USING CAGED HAPTENS

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N-substituted-dioxocyclobutenylamino-3-hydroxy-picolinamides useful as CCR6 inhibitors

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N-Doped Semiconducting Material Comprising Phosphine Oxide Matrix and Metal Dopant

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Processes for preparing oligomers

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Cannabinoid receptor modulators

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EXON SKIPPING OLIGOMERS FOR MUSCULAR DYSTROPHY

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CHIRAL REAGENTS FOR PREPARATION OF HOMOGENEOUS OLIGOMERS

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MASP-2 inhibitors and methods of use

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Tropomyosin-related kinase (TRK) inhibitors

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Heterocycle substituted pyridine derivative antifungal agents

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QUINAZOLINE COMPOUND SERVING AS EGFR TRIPLE MUTATION INHIBITOR AND APPLICATIONS THEREOF

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Cot modulators and methods of use thereof

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Phenylacetamides as inhibitors of rock

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OLIGONUCLEOTIDE ANALOGUES HAVING MODIFIED INTERSUBUNIT LINKAGES AND/OR TERMINAL GROUPS

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Heterocyclic amides useful as protein modulators

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Heterocyclic carboxylate compounds as glycolate oxidase inhibitors

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Skeletal removal of bisphosphonates

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NOVEL OXAZOLIDINONE DERIVATIVES

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Nucleotide precursors, nucleotide analogs and oligomeric compounds containing the same

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Amide compounds for treatment of immune and inflammatory disorders

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Bisphosphonate quinolone conjugates and uses thereof

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Ultra bright dimeric or polymeric dyes with spacing linker groups

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OLIGONUCLEOTIDES COMPRISING ACYCLIC AND ABASIC NUCLEOSIDES AND ANALOGS

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Dianilinopyrimidine compound for inhibiting kinase activity

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COT MODULATORS AND METHODS OF USE THEREOF

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Mito-lonidamine, compositions and methods of use

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Phosphate derivatives and use thereof

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Phospholipidation of imidazoquinolines and oxoadenines

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HORMONE RECEPTOR MODULATORS FOR TREATING METABOLIC CONDITIONS AND DISORDERS

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Crystalline forms

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ARYLPHOSPHINE OXIDES FOR INHIBITING KINASE ACTIVITY

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Heterocyclic compounds for the treatment of neurological and psychological disorders

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Cot modulators and methods of use thereof

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Nucleic acid-polypeptide compositions and uses thereof

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Chiral tetradentate ligand, method for producing same and transition metal complex of said chiral tetradentate ligand

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Biaryl monobactam compounds and methods of use thereof for the treatment of bacterial infections

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S1PR2 ANTAGONISTS AND USES THEREFOR

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Prodrugs of substituted triazole derivatives and uses thereof

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PHOSPHOROUS DERIVATIVES AS KINASE INHIBITORS

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(R)-3-((3S,4S)-3-FLUORO-4-(4-HYDROXYPHENYL)PIPERIDIN-1-YL)-1-(4-METHYLBENZYL)PYRROLIDIN-2-ONE AND ITS PRODRUGS FOR THE TREATMENT OF PSYCHIATRIC DISORDERS

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Acylsulfonamide derivatives for treating senescence-associated diseases and disorders

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Ultra bright dimeric or polymeric dyes with spacing linker groups

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Solid supports and phosphoramidite building blocks for oligonucleotide conjugates

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PRODRUGS OF 2,4-PYRIMIDINEDIAMINE COMPOUNDS AND THEIR USES

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Soluble C5aR antagonists

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Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders

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Phenylpyrrolidinone formyl peptide 2 receptor agonists

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Organic compound and organic electroluminescent device using the same

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Morpholino modified oligomeric compounds

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Electrochromic compound, electrochromic composition, and display element

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COMPOSITIONS AND METHODS FOR INHIBITION OF THE JAK PATHWAY

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POMALIDOMIDE DERIVATIVE AND PREPARATION METHOD THEREFOR

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Inhibitors of cyclin-dependent kinase 7 (CDK7)

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Organic electronic device comprising an organic semiconductor layer

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Aminothiazole Derivatives Useful As Antiviral Agents

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Functionally-modified oligonucleotides and subunits thereof

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Substituted phosphorodiamidate morpholino oligomers

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Compositions and methods for inhibition of the JAK pathway

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Organic electronic device comprising an organic semiconductor layer and a device

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N-substituted-dioxocyclobutenylamino-3-hydroxy-picolinamides useful as CCR6 inhibitors

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Aziridine containing DNA alkylating agents

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NOVEL OXAZOLIDINONE DERIVATIVES