96671 ⎘
Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)3-C(=0)-, e.g. statine or derivatives thereof
NOVEL AURISTATIN ANALOGS AND IMMUNOCONJUGATES THEREOF
#2MAGNETIC RESONANCE IMAGE PROCESSING APPARATUS AND METHOD TO WHICH IMPROVEMENT IN SLICE RESOLUTION IS APPLIED
#3IMMUNOGLOBULINS AND USES THEREOF
#4CONJUGATES AND METHODS OF USING THE SAME
#5DECARBOXYLATIVE CONJUGATE ADDITIONS AND APPLICATIONS THEREOF
#6HEMIASTERLIN DERIVATIVES FOR CONJUGATION AND THERAPY
#7XTEN CONJUGATE COMPOSITIONS AND METHODS OF MAKING SAME
#8CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPEPTIDE Y RECEPTORS
#9Cytotoxic and anti-mitotic compounds, and methods of using the same
#10ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPEPTIDE Y RECEPTORS
#11Cytotoxic and anti-mitotic compounds, and methods of using the same
#12EFFICIENT PREPARATION OF DOLASTATIN AND AURISTATIN ANALOGS THROUGH A COMMON INTERMEDIATE
#13AURISTATIN-RELATED COMPOUNDS, CONJUGATED AURISTATIN-RELATED COMPOUNDS, AND METHODS OF USE THEREOF
#14DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS
#15COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES
#16DERIVATIVES OF DOLAPROINE-DOLAISOLEUINE PEPTIDES
#17METHOD FOR PREPARING DRUG-LINKER MC-MMAF FOR ANTIBODY DRUG CONJUGATE, AND INTERMEDIATES THEREIN
#18PROSTATE-SPECIFIC MEMBRANE ANTIGEN ANTIBODY DRUG CONJUGATES
#19Decarboxylative conjugate additions and applications thereof
#20XTEN CONJUGATE COMPOSITIONS AND METHODS OF MAKING SAME
#21Heteroaryl sulfone-based conjugation handles, methods for their preparation, and their use in synthesizing antibody drug conjugates
#22Compositions containing, methods involving, and uses of non-natural amino acid linked dolastatin derivatives
#23HEMIASTERLIN DERIVATIVES FOR CONJUGATION AND THERAPY
#24Cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#25Hemiasterlin derivatives for conjugation and therapy
#26Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#27Conjugates and methods of using the same
#28DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS
#29Immunoglobulins and uses thereof
#30Immunoglobulins and uses thereof
#31Albumin-binding prodrugs of auristatin E derivatives
#32Derivatives of dolaproine-dolaisoleucine peptides
#33ANTI-CANCER COMPOUNDS AND CONJUGATES THEREOF
#34CD48 ANTIBODIES AND CONJUGATES THEREOF
#35Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#36Hemiasterlin derivatives and antibody-drug conjugates including same
#37N-acyldipeptide derivatives and their uses
#38Cytotoxic and anti-mitotic compounds, and methods of using the same
#39Tripeptide epoxy ketone protease inhibitors
#40Peptide-Based Quorum Sensing Inhibitors for the Attenuation of Virulence in Staphylococcus Aureus
#41PRODRUG OF AN ICE INHIBITOR
#42Growth Hormone Releasing Peptides
#43DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS
#44MALT1 inhibitors and uses thereof
#45Cytotoxic peptides and conjugates thereof
#46Immunoglobulins and uses thereof
#47CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME
#48Cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#49Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#50Cytotoxic and anti-mitotic compounds, and methods of using the same
#51Immunoglobulins and uses thereof
#52Difluoroketamide derivatives as HTRA1 inhibitors
#53XTEN conjugate compositions and methods of making same
#54CHIRAL COMPOUNDS OF VARYING CONFORMATIONAL RIGIDITY AND METHODS OF SYNTHESIS
#55Quinstatin compounds
#56MONOMETHYLVALINE COMPOUNDS HAVING PHENYLALANINE SIDE-CHAIN MODIFICATIONS AT THE C-TERMINUS
#57PRODRUG OF AN ICE INHIBITOR
#58Combination of N-acyldipeptide derivatives and retinol, and methods of use thereof
#59Anti-cancer compounds and conjugates thereof
#60MALT1 inhibitors and uses thereof
#61Cytotoxic peptides and conjugates thereof
#62DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS
#63Cytotoxic and anti-mitotic compounds, and methods of using the same
#64Decarboxylative conjugate additions and applications thereof
#65Cytotoxic peptides and conjugates thereof
#66Cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#67Immunoglobulins and uses thereof
#68Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors
#69CD48 antibodies and conjugates thereof
#70Difluoroketamide derivatives
#71Compositions containing, methods involving, and uses of non-natural amino acid linked dolastatin derivatives
#72Growth Hormone Releasing Peptides
#73METHOD OF MAKING PRODRUGS AND TARGETED THERAPEUTIC COMPOUNDS
#74ANTIBODY-DRUG CONJUGATE OF AN ANTI-GLYPICAN-3 ANTIBODY AND A TUBULYSIN ANALOG, PREPARATION AND USES
#75Cytotoxic and anti-mitotic compounds, and methods of using the same
#76HCV NS-3 serine protease inhibitors
#77DERIVATIVES OF DOLAPROINE-DOLAISOLEUINE PEPTIDES
#78N-acyldipeptide derivatives and their uses
#79Hydroxystatin derivatives for the treatment of arthrosis
#80Prodrug of an ICE inhibitor
#81Tripeptide epoxy ketone protease inhibitors
#82Cytotoxic peptides and conjugates thereof
#83Gamma amino acid building blocks
#84Hemiasterlin derivatives for conjugation and therapy
#85Aminostatin derivatives for the treatment of arthrosis
#86PEPTIDE-BASED QUORUM SENSING INHIBITORS FOR THE ATTENUATION OF VIRULENCE IN STAPHYLOCOCCUS AUREUS
#87Chromobacterium bioactive compositions and metabolites
#88Cytotoxic and anti-mitotic compounds, and methods of using the same
#89DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS
#90DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS
#91Compositions containing, methods involving, and uses of non-natural amino acid linked dolastatin derivatives
#92Cytotoxic and anti-mitotic compounds, and methods of using the same
#93Dipeptide and tripeptide epoxy ketone protease inhibitors
#94Auristatin tyramine phosphate salts and auristatin aminoquinoline derivatives and prodrugs thereof
#95Prodrug of an ice inhibitor
#96Dolastatin-10 derivative, method of producing the same and anticancer drug composition containing the same
#97Hydroxystatin derivatives for the treatment of arthrosis
#98Prostate-specific membrane antigen antibody drug conjugates
#99Gamma amino acid building blocks
#100Methods of using monomethylvaline compositions having phenylalanine carboxy modifications at the C-terminus
#101XTEN conjugate compositions and methods of making same
#102Growth hormone releasing peptides
#103Cytotoxic peptides and antibody drug conjugates thereof
#104Cytotoxic and anti-mitotic compounds, and methods of using the same
#105Chiral oligomeric pentenoate amides as bio-oligomer mimetics
#106Chromobacterium bioactive compositions and metabolites
#107Crystal structures of dolastatin 16, dolamethylleuine and dolaphenvaline, and methods for preparing dolamethylleuine and dolaphenvaline
#108N-carboxyalkylauristatins and use thereof
#109Auristatin drug linker conjugates
#110Auristatin tyramine phosphate salts and auristatin aminoquinoline derivatives and prodrugs thereof
#111Oligopeptides and process for preparation thereof
#112Prodrug of an ice inhibitor
#113Aminostatin derivatives for the treatment of arthrosis
#114Selective inhibitors of prolylcarboxypeptidase
#115N-carboxyalkyl-auristatin and the use thereof
#116Cytotoxic peptides and antibody drug conjugates thereof
#117Monomethylvaline compounds having phenylalanine side-chain modification at the C-terminus
#118Growth hormone releasing peptides
#119NEW BINDER-DRUG CONJUGATES (ADCS) AND USE THEREOF
#120Peptidomimetic protease inhibitors
#121Process for and intermediates in the preparation of canfosfamide and its salts
#122bioactive compositions and metabolites
#123Peptidomimetic protease inhibitors
#124ACETYLATED AMINO ACIDS AS ANTI-PLATELET AGENTS, NUTRITIONAL AND VITAMIN SUPPLEMENTS
#125Prodrug of an ICE inhibitor
#126Dipeptoid prodrugs and the use thereof
#127Acetylated amino acids as anti-platelet agents, nutritional and vitamin supplements
#128Inhibitors of Cancer Cell, T-Cell and Keratinocyte Proliferation
#129Gamma amino acid building blocks
#130Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease
#131Inhibitors for the soluble epoxide hydrolase
#132Auristatin drug linker conjugates
#133Prodrugs of GABA analogs, compositions and uses thereof
#134HCV NS-3 SERINE PROTEASE INHIBITORS
#135Peptidomimetic protease inhibitors
#136INTEGRIN TARGETED CYCLOPEPTIDE LIGANDS, THEIR PREPARATION AND USE
#137Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease
#138Depsipeptides and their therapeutic use
#139Depsipeptides and their therapeutic use
#140CYCLIC MALONAMIDES AS INHIBITORS OF A BETA PROTEIN PRODUCTION
#141CYCLIC MALONAMIDES AS INHIBITORS OF ABETA PROTEIN PRODUCTION
#142HCV NS-3 Serine Protease Inhibitors
#143Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease
#144RADIOFLUORINATION METHODS
#145Methods of treating using conjugates transported by a PEPT2 transporter
#146HEMIASTERLIN ANALOGS
#147CYCLIC MALONAMIDES AS INHIBITORS OF Abeta PROTEIN PRODUCTION
#148STILBENE DERIVATIVES AND METHODS OF INHIBITING CANCER CELL GROWTH AND MICROBIAL GROWTH
#149SMALL PEPTIDIC AND PEPTIDO-MIMETIC AFFINITY LIGANDS FOR FACTOR VIII AND FACTOR VIII-LIKE PROTEINS
#150INHIBITORS OF CANCER CELL, T-CELL AND KERATINOCYTE PROLIFERATION
#151Monomethylvaline compounds having phenylalanine carboxy modifications at the C-terminus
#152Biologically active peptides and compositions, their use
#153Anti-cancer compounds
#154Monomethylvaline compounds having phenylalanine side-chain replacements at the C-terminus
#155Prodrug of an ICE inhibitor
#156Cyclic malonamides as inhibitors of aβ protein production
#157Alkene Mimics
#158COMPOUNDS FOR SUSTAINED RELEASE OF ORALLY DELIVERED DRUGS
#159Use of Derivatives of Dipeptides for the Manufacture of of a Medicament for the Treamtent of Microbial Infections
#160Growth hormone releasing peptides
#161Novel Drugs for Dementia
#162Amino acid conjugates providing for sustained systemic concentrations of GABA analogues
#163Compounds for treating tumors
#164RECOMBINANT ANTI-CD30 ANTIBODIES AND USES THEREOF
#165Hemiasterlin Derivatives and Uses Thereof
#166Myd88 Homodimerization Inhibitors
#167Cyclic malonamides as inhibitors of Aβ protein production
#168Synthetic methods for aplidine and new antitumoral derivatives, methods of making and using them
#169Depeptidized inhibitors of hepatitis C virus NS3 protease
#170HCV NS-3 serine protease inhibitors
#171HCV NS-3 serine protease inhibitors
#172Tamandarin analogs and fragments thereof and methods of making and using
#173Inhibitors of hepatitis C virus NS3 protease
#174Deoxo-proline-containing tamandarin and didemnin analogs, dehydro-proline-containing tamandarin and didemnin analogs, and methods of making and using them
#175Acetylated amino acids as anti-platelet agents, nutritional and vitamin supplements
#176Didemnin analogs and fragments and methods of making and using them
#177Ketoamides with cyclic P4's as inhibitors of NS3 serine protease of hepatitis C virus
#178Inhibitors of cancer cell, T-cell and keratinocyte proliferation
#179Hemiasterlin affinity probes and their uses
#180Bile-acid derived compounds for enhancing oral absorption and systemic bioavailability of drugs
#181Prodrugs of GABA analogs, compositions and uses thereof
#182Administration of HCV protease inhibitors in combination with food to improve bioavailability
#183Inhibitors for the soluble epoxide hydrolase
#184Pentapeptide compounds and uses related thereto
#185Anti-cancer compounds
#186Bile-acid conjugates providing for sustained systemic concentration of drugs
#187Statine derivatives for the treatment of Alzheimer's disease II
#188Process for the manufacture of disubstituted amines
#189Hemiasterlin derivatives and uses thereof
#190Synthesis of epoxide based inhibitors of cysteine proteases
#191Cyclic malonamides as inhibitors of Aβ protein protection
#192Process for and intermediates in the preparation of canfosfamide and its salts
#1933-Pyrrolidin-2-yl-propionic acid derivatives
#194Statine derivatives for the treatment of Alzheimer's disease III
#195Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease
#196Low molecular weight peptidomimetic growth hormone secretagogues
#197Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
#198Hybrid molecules QA, wherein Q is an aminoquinoline and a is an antibiotic or a resistance enzyme inhibitor, their synthesis and their uses as antibacterial agent
#199Hepatitis C inhibitor peptide analogs
#200Novel amide derivatives as growth hormone secretagogues
#201Process for the synthesis of intermediates useful for the synthesis of tubulin inhibitors
#202Bile-acid conjugates for providing sustained systemic concentrations of drugs
#203Diamines as modulators of chemokine receptor activity
#204Bile-acid derived compounds for providing sustained systemic concentrations of drugs after oral administration
#205Substituted prolines as inhibitors of hepatitis C virus NS3 serine protease
#206Inhibitors of hepatitis C virus NS3 protease
#207Method of making tetrapeptide derivative TZT-1027 crystal
#208Ketoamides with cyclic P4'S as inhibitors of NS3 protease of hepatitis C virus
#209Derivatives of dehydrodidemnin B
#210Methods for identifying RNA binding compounds
#211Methods of screening agents, conjugates or conjugate moieties for transport by a PEPT2 transporter
#212Depsipeptide compound
#213Peptidomimetic protease inhibitors
#214Dipeptide inhibitors of β-secretase
#215Biologically active peptides and compositions, their use
#216Conjugates of ligand linker and cytotoxic agent and related composition and methods of use
#217Depeptidized inhibitors of hepatitis C virus NS3 protease
#218Vitronectin receptor antagonist pharmaceuticals
#219Bile-acid conjugates providing for sustained systemic concentration of drugs
#220Growth hormone releasing peptides
#221Pentapeptide compounds and uses related thereto
#222Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis
#223Novel statine derivatives for the treatment of Alzheimer's disease
#224Compounds for sustained release of orally delivered drugs
#225Compounds for treating tumors
#226Cyclic malonamides as inhibitors of A-β protein production
#227Pentapeptide compounds and uses related thereto
#228Bivalent inhibitors of Glutathione-S-Transferases
#229Modified polynucleotides and uses thereof