ClassID:

96671

C07K5/0205 - CPC Classification

Classification description:

Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -NH-(X)3-C(=0)-, e.g. statine or derivatives thereof

Recent Application in this class:
#1
20260131016
2026-05-14

NOVEL AURISTATIN ANALOGS AND IMMUNOCONJUGATES THEREOF

#2
20250188121
2025-06-12

MAGNETIC RESONANCE IMAGE PROCESSING APPARATUS AND METHOD TO WHICH IMPROVEMENT IN SLICE RESOLUTION IS APPLIED

#3
20250026803
2025-01-23

IMMUNOGLOBULINS AND USES THEREOF

#4
20240398966
2024-12-05

CONJUGATES AND METHODS OF USING THE SAME

#5
20240287129
2024-08-29

DECARBOXYLATIVE CONJUGATE ADDITIONS AND APPLICATIONS THEREOF

#6
20240254163
2024-08-01

HEMIASTERLIN DERIVATIVES FOR CONJUGATION AND THERAPY

#7
20240091315
2024-03-21

XTEN CONJUGATE COMPOSITIONS AND METHODS OF MAKING SAME

#8
20240018208
2024-01-18

CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPEPTIDE Y RECEPTORS

#9
20230390354
2023-12-07

Cytotoxic and anti-mitotic compounds, and methods of using the same

#10
20230365644
2023-11-16

ANTIBODY-COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE COMPOUNDS AS MODULATORS OF NEUROPEPTIDE Y RECEPTORS

#11
20230317700
2023-10-05

Cytotoxic and anti-mitotic compounds, and methods of using the same

#12
20230129674
2023-04-27

EFFICIENT PREPARATION OF DOLASTATIN AND AURISTATIN ANALOGS THROUGH A COMMON INTERMEDIATE

#13
20230071763
2023-03-09

AURISTATIN-RELATED COMPOUNDS, CONJUGATED AURISTATIN-RELATED COMPOUNDS, AND METHODS OF USE THEREOF

#14
20230002316
2023-01-05

DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS

#15
20220411469
2022-12-29

COMPOSITIONS CONTAINING, METHODS INVOLVING, AND USES OF NON-NATURAL AMINO ACID LINKED DOLASTATIN DERIVATIVES

#16
20220204557
2022-06-30

DERIVATIVES OF DOLAPROINE-DOLAISOLEUINE PEPTIDES

#17
20220119441
2022-04-21

METHOD FOR PREPARING DRUG-LINKER MC-MMAF FOR ANTIBODY DRUG CONJUGATE, AND INTERMEDIATES THEREIN

#18
20220033518
2022-02-03

PROSTATE-SPECIFIC MEMBRANE ANTIGEN ANTIBODY DRUG CONJUGATES

#19
20220002342
2022-01-06

Decarboxylative conjugate additions and applications thereof

#20
20210322518
2021-10-21

XTEN CONJUGATE COMPOSITIONS AND METHODS OF MAKING SAME

#21
20210308276
2021-10-07

Heteroaryl sulfone-based conjugation handles, methods for their preparation, and their use in synthesizing antibody drug conjugates

#22
20210277056
2021-09-09

Compositions containing, methods involving, and uses of non-natural amino acid linked dolastatin derivatives

#23
20210261611
2021-08-26

HEMIASTERLIN DERIVATIVES FOR CONJUGATION AND THERAPY

#24
20210206822
2021-07-08

Cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#25
20210198314
2021-07-01

Hemiasterlin derivatives for conjugation and therapy

#26
20210163566
2021-06-03

Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#27
20210162057
2021-06-03

Conjugates and methods of using the same

#28
20210107868
2021-04-15

DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS

#29
20210094998
2021-04-01

Immunoglobulins and uses thereof

#30
20200385439
2020-12-10

Immunoglobulins and uses thereof

#31
20200385421
2020-12-10

Albumin-binding prodrugs of auristatin E derivatives

#32
20200325170
2020-10-15

Derivatives of dolaproine-dolaisoleucine peptides

#33
20200316214
2020-10-08

ANTI-CANCER COMPOUNDS AND CONJUGATES THEREOF

#34
20200289661
2020-09-17

CD48 ANTIBODIES AND CONJUGATES THEREOF

#35
20200283491
2020-09-10

Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#36
20200247845
2020-08-06

Hemiasterlin derivatives and antibody-drug conjugates including same

#37
20200237637
2020-07-30

N-acyldipeptide derivatives and their uses

#38
20200207865
2020-07-02

Cytotoxic and anti-mitotic compounds, and methods of using the same

#39
20200207809
2020-07-02

Tripeptide epoxy ketone protease inhibitors

#40
20200140489
2020-05-07

Peptide-Based Quorum Sensing Inhibitors for the Attenuation of Virulence in Staphylococcus Aureus

#41
20200048306
2020-02-13

PRODRUG OF AN ICE INHIBITOR

#42
20200017548
2020-01-16

Growth Hormone Releasing Peptides

#43
20200010414
2020-01-09

DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS

#44
20190389904
2019-12-26

MALT1 inhibitors and uses thereof

#45
20190382441
2019-12-19

Cytotoxic peptides and conjugates thereof

#46
20190367577
2019-12-05

Immunoglobulins and uses thereof

#47
20190345254
2019-11-14

CYTOTOXIC AND ANTI-MITOTIC COMPOUNDS, AND METHODS OF USING THE SAME

#48
20190345214
2019-11-14

Cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#49
20190298849
2019-10-03

Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#50
20190269785
2019-09-05

Cytotoxic and anti-mitotic compounds, and methods of using the same

#51
20190263879
2019-08-29

Immunoglobulins and uses thereof

#52
20190185427
2019-06-20

Difluoroketamide derivatives as HTRA1 inhibitors

#53
20190083577
2019-03-21

XTEN conjugate compositions and methods of making same

#54
20180371014
2018-12-27

CHIRAL COMPOUNDS OF VARYING CONFORMATIONAL RIGIDITY AND METHODS OF SYNTHESIS

#55
20180371012
2018-12-27

Quinstatin compounds

#56
20180355025
2018-12-13

MONOMETHYLVALINE COMPOUNDS HAVING PHENYLALANINE SIDE-CHAIN MODIFICATIONS AT THE C-TERMINUS

#57
20180327449
2018-11-15

PRODRUG OF AN ICE INHIBITOR

#58
20180303741
2018-10-25

Combination of N-acyldipeptide derivatives and retinol, and methods of use thereof

#59
20180296688
2018-10-18

Anti-cancer compounds and conjugates thereof

#60
20180251489
2018-09-06

MALT1 inhibitors and uses thereof

#61
20180244717
2018-08-30

Cytotoxic peptides and conjugates thereof

#62
20180222858
2018-08-09

DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS

#63
20180208667
2018-07-26

Cytotoxic and anti-mitotic compounds, and methods of using the same

#64
20180179248
2018-06-28

Decarboxylative conjugate additions and applications thereof

#65
20180155281
2018-06-07

Cytotoxic peptides and conjugates thereof

#66
20180127476
2018-05-10

Cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#67
20180125998
2018-05-10

Immunoglobulins and uses thereof

#68
20180117170
2018-05-03

Antibody-coupled cyclic peptide tyrosine tyrosine compounds as modulators of neuropeptide Y receptors

#69
20180092984
2018-04-05

CD48 antibodies and conjugates thereof

#70
20180057526
2018-03-01

Difluoroketamide derivatives

#71
20180009845
2018-01-11

Compositions containing, methods involving, and uses of non-natural amino acid linked dolastatin derivatives

#72
20170362275
2017-12-21

Growth Hormone Releasing Peptides

#73
20170342106
2017-11-30

METHOD OF MAKING PRODRUGS AND TARGETED THERAPEUTIC COMPOUNDS

#74
20170326249
2017-11-16

ANTIBODY-DRUG CONJUGATE OF AN ANTI-GLYPICAN-3 ANTIBODY AND A TUBULYSIN ANALOG, PREPARATION AND USES

#75
20170247408
2017-08-31

Cytotoxic and anti-mitotic compounds, and methods of using the same

#76
20170196849
2017-07-13

HCV NS-3 serine protease inhibitors

#77
20170190735
2017-07-06

DERIVATIVES OF DOLAPROINE-DOLAISOLEUINE PEPTIDES

#78
20170119646
2017-05-04

N-acyldipeptide derivatives and their uses

#79
20170081361
2017-03-23

Hydroxystatin derivatives for the treatment of arthrosis

#80
20170022249
2017-01-26

Prodrug of an ICE inhibitor

#81
20160368946
2016-12-22

Tripeptide epoxy ketone protease inhibitors

#82
20160311853
2016-10-27

Cytotoxic peptides and conjugates thereof

#83
20160280632
2016-09-29

Gamma amino acid building blocks

#84
20160257709
2016-09-08

Hemiasterlin derivatives for conjugation and therapy

#85
20160228493
2016-08-11

Aminostatin derivatives for the treatment of arthrosis

#86
20160194360
2016-07-07

PEPTIDE-BASED QUORUM SENSING INHIBITORS FOR THE ATTENUATION OF VIRULENCE IN STAPHYLOCOCCUS AUREUS

#87
20160095323
2016-04-07

Chromobacterium bioactive compositions and metabolites

#88
20160075735
2016-03-17

Cytotoxic and anti-mitotic compounds, and methods of using the same

#89
20160068567
2016-03-10

DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS

#90
20160068566
2016-03-10

DERIVATIVES OF DOLASTATIN 10 AND AURISTATINS

#91
20160052966
2016-02-25

Compositions containing, methods involving, and uses of non-natural amino acid linked dolastatin derivatives

#92
20160038606
2016-02-11

Cytotoxic and anti-mitotic compounds, and methods of using the same

#93
20160031934
2016-02-04

Dipeptide and tripeptide epoxy ketone protease inhibitors

#94
20150344522
2015-12-03

Auristatin tyramine phosphate salts and auristatin aminoquinoline derivatives and prodrugs thereof

#95
20150284426
2015-10-08

Prodrug of an ice inhibitor

#96
20150225455
2015-08-13

Dolastatin-10 derivative, method of producing the same and anticancer drug composition containing the same

#97
20150225451
2015-08-13

Hydroxystatin derivatives for the treatment of arthrosis

#98
20150152190
2015-06-04

Prostate-specific membrane antigen antibody drug conjugates

#99
20150148523
2015-05-28

Gamma amino acid building blocks

#100
20150044238
2015-02-12

Methods of using monomethylvaline compositions having phenylalanine carboxy modifications at the C-terminus

#101
20150037359
2015-02-05

XTEN conjugate compositions and methods of making same

#102
20150031615
2015-01-29

Growth hormone releasing peptides

#103
20140363452
2014-12-11

Cytotoxic peptides and antibody drug conjugates thereof

#104
20140315954
2014-10-23

Cytotoxic and anti-mitotic compounds, and methods of using the same

#105
20140271488
2014-09-18

Chiral oligomeric pentenoate amides as bio-oligomer mimetics

#106
20140199269
2014-07-17

Chromobacterium bioactive compositions and metabolites

#107
20140179897
2014-06-26

Crystal structures of dolastatin 16, dolamethylleuine and dolaphenvaline, and methods for preparing dolamethylleuine and dolaphenvaline

#108
20140080763
2014-03-20

N-carboxyalkylauristatins and use thereof

#109
20140050746
2014-02-20

Auristatin drug linker conjugates

#110
20140023666
2014-01-23

Auristatin tyramine phosphate salts and auristatin aminoquinoline derivatives and prodrugs thereof

#111
20140005121
2014-01-02

Oligopeptides and process for preparation thereof

#112
20130331310
2013-12-12

Prodrug of an ice inhibitor

#113
20130316955
2013-11-28

Aminostatin derivatives for the treatment of arthrosis

#114
20130310311
2013-11-21

Selective inhibitors of prolylcarboxypeptidase

#115
20130261064
2013-10-03

N-carboxyalkyl-auristatin and the use thereof

#116
20130129753
2013-05-23

Cytotoxic peptides and antibody drug conjugates thereof

#117
20130123465
2013-05-16

Monomethylvaline compounds having phenylalanine side-chain modification at the C-terminus

#118
20130123170
2013-05-16

Growth hormone releasing peptides

#119
20130066055
2013-03-14

NEW BINDER-DRUG CONJUGATES (ADCS) AND USE THEREOF

#120
20120282219
2012-11-08

Peptidomimetic protease inhibitors

#121
20120238772
2012-09-20

Process for and intermediates in the preparation of canfosfamide and its salts

#122
20120100236
2012-04-26

bioactive compositions and metabolites

#123
20120064034
2012-03-15

Peptidomimetic protease inhibitors

#124
20110312890
2011-12-22

ACETYLATED AMINO ACIDS AS ANTI-PLATELET AGENTS, NUTRITIONAL AND VITAMIN SUPPLEMENTS

#125
20110301096
2011-12-08

Prodrug of an ICE inhibitor

#126
20110294719
2011-12-01

Dipeptoid prodrugs and the use thereof

#127
20110275713
2011-11-10

Acetylated amino acids as anti-platelet agents, nutritional and vitamin supplements

#128
20110263486
2011-10-27

Inhibitors of Cancer Cell, T-Cell and Keratinocyte Proliferation

#129
20110118440
2011-05-19

Gamma amino acid building blocks

#130
20110064753
2011-03-17

Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease

#131
20110021448
2011-01-27

Inhibitors for the soluble epoxide hydrolase

#132
20110020343
2011-01-27

Auristatin drug linker conjugates

#133
20100267946
2010-10-21

Prodrugs of GABA analogs, compositions and uses thereof

#134
20100166706
2010-07-01

HCV NS-3 SERINE PROTEASE INHIBITORS

#135
20100137583
2010-06-03

Peptidomimetic protease inhibitors

#136
20100093612
2010-04-15

INTEGRIN TARGETED CYCLOPEPTIDE LIGANDS, THEIR PREPARATION AND USE

#137
20100062008
2010-03-11

Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease

#138
20100056435
2010-03-04

Depsipeptides and their therapeutic use

#139
20100056434
2010-03-04

Depsipeptides and their therapeutic use

#140
20100041639
2010-02-18

CYCLIC MALONAMIDES AS INHIBITORS OF A BETA PROTEIN PRODUCTION

#141
20100009965
2010-01-14

CYCLIC MALONAMIDES AS INHIBITORS OF ABETA PROTEIN PRODUCTION

#142
20100003216
2010-01-07

HCV NS-3 Serine Protease Inhibitors

#143
20090324621
2009-12-31

Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease

#144
20090317326
2009-12-24

RADIOFLUORINATION METHODS

#145
20090306036
2009-12-10

Methods of treating using conjugates transported by a PEPT2 transporter

#146
20090264487
2009-10-22

HEMIASTERLIN ANALOGS

#147
20090264419
2009-10-22

CYCLIC MALONAMIDES AS INHIBITORS OF Abeta PROTEIN PRODUCTION

#148
20090221666
2009-09-03

STILBENE DERIVATIVES AND METHODS OF INHIBITING CANCER CELL GROWTH AND MICROBIAL GROWTH

#149
20090215025
2009-08-27

SMALL PEPTIDIC AND PEPTIDO-MIMETIC AFFINITY LIGANDS FOR FACTOR VIII AND FACTOR VIII-LIKE PROTEINS

#150
20090176716
2009-07-09

INHIBITORS OF CANCER CELL, T-CELL AND KERATINOCYTE PROLIFERATION

#151
20090111756
2009-04-30

Monomethylvaline compounds having phenylalanine carboxy modifications at the C-terminus

#152
20090088573
2009-04-02

Biologically active peptides and compositions, their use

#153
20090088454
2009-04-02

Anti-cancer compounds

#154
20090018086
2009-01-15

Monomethylvaline compounds having phenylalanine side-chain replacements at the C-terminus

#155
20090012149
2009-01-08

Prodrug of an ICE inhibitor

#156
20080275024
2008-11-06

Cyclic malonamides as inhibitors of aβ protein production

#157
20080261923
2008-10-23

Alkene Mimics

#158
20080255073
2008-10-16

COMPOUNDS FOR SUSTAINED RELEASE OF ORALLY DELIVERED DRUGS

#159
20080255055
2008-10-16

Use of Derivatives of Dipeptides for the Manufacture of of a Medicament for the Treamtent of Microbial Infections

#160
20080242619
2008-10-02

Growth hormone releasing peptides

#161
20080227806
2008-09-18

Novel Drugs for Dementia

#162
20080226716
2008-09-18

Amino acid conjugates providing for sustained systemic concentrations of GABA analogues

#163
20080221181
2008-09-11

Compounds for treating tumors

#164
20080213289
2008-09-04

RECOMBINANT ANTI-CD30 ANTIBODIES AND USES THEREOF

#165
20080108820
2008-05-08

Hemiasterlin Derivatives and Uses Thereof

#166
20080064643
2008-03-13

Myd88 Homodimerization Inhibitors

#167
20080021014
2008-01-24

Cyclic malonamides as inhibitors of Aβ protein production

#168
20080009435
2008-01-10

Synthetic methods for aplidine and new antitumoral derivatives, methods of making and using them

#169
20070258947
2007-11-08

Depeptidized inhibitors of hepatitis C virus NS3 protease

#170
20070203072
2007-08-30

HCV NS-3 serine protease inhibitors

#171
20070161574
2007-07-12

HCV NS-3 serine protease inhibitors

#172
20070149446
2007-06-28

Tamandarin analogs and fragments thereof and methods of making and using

#173
20070142301
2007-06-21

Inhibitors of hepatitis C virus NS3 protease

#174
20070129289
2007-06-07

Deoxo-proline-containing tamandarin and didemnin analogs, dehydro-proline-containing tamandarin and didemnin analogs, and methods of making and using them

#175
20070112060
2007-05-17

Acetylated amino acids as anti-platelet agents, nutritional and vitamin supplements

#176
20070111928
2007-05-17

Didemnin analogs and fragments and methods of making and using them

#177
20070093430
2007-04-26

Ketoamides with cyclic P4's as inhibitors of NS3 serine protease of hepatitis C virus

#178
20070037753
2007-02-15

Inhibitors of cancer cell, T-cell and keratinocyte proliferation

#179
20070026478
2007-02-01

Hemiasterlin affinity probes and their uses

#180
20070015716
2007-01-18

Bile-acid derived compounds for enhancing oral absorption and systemic bioavailability of drugs

#181
20070010453
2007-01-11

Prodrugs of GABA analogs, compositions and uses thereof

#182
20060281688
2006-12-14

Administration of HCV protease inhibitors in combination with food to improve bioavailability

#183
20060270609
2006-11-30

Inhibitors for the soluble epoxide hydrolase

#184
20060229253
2006-10-12

Pentapeptide compounds and uses related thereto

#185
20060183772
2006-08-17

Anti-cancer compounds

#186
20060166858
2006-07-27

Bile-acid conjugates providing for sustained systemic concentration of drugs

#187
20060160747
2006-07-20

Statine derivatives for the treatment of Alzheimer's disease II

#188
20060155110
2006-07-13

Process for the manufacture of disubstituted amines

#189
20060154872
2006-07-13

Hemiasterlin derivatives and uses thereof

#190
20060154325
2006-07-13

Synthesis of epoxide based inhibitors of cysteine proteases

#191
20060135762
2006-06-22

Cyclic malonamides as inhibitors of Aβ protein protection

#192
20060135409
2006-06-22

Process for and intermediates in the preparation of canfosfamide and its salts

#193
20060128970
2006-06-15

3-Pyrrolidin-2-yl-propionic acid derivatives

#194
20060100158
2006-05-11

Statine derivatives for the treatment of Alzheimer's disease III

#195
20060074008
2006-04-06

Drug conjugates and their use for treating cancer, an autoimmune disease or an infectious disease

#196
20060063807
2006-03-23

Low molecular weight peptidomimetic growth hormone secretagogues

#197
20060046966
2006-03-02

Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis

#198
20060025327
2006-02-02

Hybrid molecules QA, wherein Q is an aminoquinoline and a is an antibiotic or a resistance enzyme inhibitor, their synthesis and their uses as antibacterial agent

#199
20060019905
2006-01-26

Hepatitis C inhibitor peptide analogs

#200
20060014701
2006-01-19

Novel amide derivatives as growth hormone secretagogues

#201
20050288486
2005-12-29

Process for the synthesis of intermediates useful for the synthesis of tubulin inhibitors

#202
20050288228
2005-12-29

Bile-acid conjugates for providing sustained systemic concentrations of drugs

#203
20050282882
2005-12-22

Diamines as modulators of chemokine receptor activity

#204
20050272710
2005-12-08

Bile-acid derived compounds for providing sustained systemic concentrations of drugs after oral administration

#205
20050272663
2005-12-08

Substituted prolines as inhibitors of hepatitis C virus NS3 serine protease

#206
20050267043
2005-12-01

Inhibitors of hepatitis C virus NS3 protease

#207
20050267041
2005-12-01

Method of making tetrapeptide derivative TZT-1027 crystal

#208
20050222047
2005-10-06

Ketoamides with cyclic P4'S as inhibitors of NS3 protease of hepatitis C virus

#209
20050222015
2005-10-06

Derivatives of dehydrodidemnin B

#210
20050221368
2005-10-06

Methods for identifying RNA binding compounds

#211
20050214853
2005-09-29

Methods of screening agents, conjugates or conjugate moieties for transport by a PEPT2 transporter

#212
20050209134
2005-09-22

Depsipeptide compound

#213
20050197299
2005-09-08

Peptidomimetic protease inhibitors

#214
20050182138
2005-08-18

Dipeptide inhibitors of β-secretase

#215
20050171137
2005-08-04

Biologically active peptides and compositions, their use

#216
20050171014
2005-08-04

Conjugates of ligand linker and cytotoxic agent and related composition and methods of use

#217
20050164921
2005-07-28

Depeptidized inhibitors of hepatitis C virus NS3 protease

#218
20050154185
2005-07-14

Vitronectin receptor antagonist pharmaceuticals

#219
20050148564
2005-07-07

Bile-acid conjugates providing for sustained systemic concentration of drugs

#220
20050148515
2005-07-07

Growth hormone releasing peptides

#221
20050113308
2005-05-26

Pentapeptide compounds and uses related thereto

#222
20050101651
2005-05-12

Antipicornaviral compounds and compositions, their pharmaceutical uses, and materials for their synthesis

#223
20050090449
2005-04-28

Novel statine derivatives for the treatment of Alzheimer's disease

#224
20050054559
2005-03-10

Compounds for sustained release of orally delivered drugs

#225
20050037977
2005-02-17

Compounds for treating tumors

#226
20050009807
2005-01-13

Cyclic malonamides as inhibitors of A-β protein production

#227
20050009751
2005-01-13

Pentapeptide compounds and uses related thereto

#228
20050004038
2005-01-06

Bivalent inhibitors of Glutathione-S-Transferases

#229
17176617
2023-11-07

Modified polynucleotides and uses thereof