Inventor profile of:

Andrew P. Combs

City:

Kennett Square, Pennsylvania

Country:

United States

Published Applications:

147

Last publication date:

2025-12-25

Top Assignees for applications by Andrew P. Combs

The entities that hold a legal rights for patent applications filed by inventor Combs Andrew P.:

Recent patent applications by Combs Andrew P.

Andrew P. Combs from Kennett Square, US has applied for patents for these inventions. The list has both pending applications and granted patents:

#1 | 2025-12-25
US20250388553A1
Chemistry; metallurgy

AMINOPYRAZINE DERIVATIVES AS PI3K-y INHIBITORS

#2 | 2025-10-23
US20250325550A1
Human necessities

HETEROCYCLYLAMINES AS PI3K INHIBITORS

#3 | 2025-10-09
US20250313550A1
Chemistry; metallurgy

AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS

#4 | 2025-09-18
US20250289823A1
Chemistry; metallurgy

USE OF PYRAZOLOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PI3K-DELTA RELATED DISORDERS

#5 | 2025-07-31
US20250243206A1
Chemistry; metallurgy

CRYSTALLINE FORMS OF A PHOSPHOINOSITIDE 3-KINASE (PI3K) INHIBITOR

#6 | 2025-05-08
US20250145621A1
Chemistry; metallurgy

1H-PYRROLO[2,3-c]PYRIDIN-7(6H)-ONES AND PYRAZOLO[3,4-c]PYRIDIN-7(6H)-ONES AS INHIBITORS OF BET PROTEINS

#7 | 2025-04-24
US20250129098A1
Chemistry; metallurgy

BICYCLIC HETEROARYLAMINOALKYL PHENYL DERIVATIVES AS PI3K INHIBITORS

#8 | 2024-12-05
US20240400541A1
Chemistry; metallurgy

AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS

#9 | 2024-07-11
US20240228498A1
Chemistry; metallurgy

TERTIARY ALCOHOLS AS PI3K-y INHIBITORS

#10 | 2024-07-04
US20240216377A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#11 | 2024-05-30
US20240173303A1
Human necessities

1,2,5-Oxadiazoles As Inhibitors Of Indoleamine 2,3- Dioxygenase

#12 | 2024-04-18
US20240124422A1
Chemistry; metallurgy

MUTANT PI3K-ALPHA INHIBITORS AND THEIR USE AS PHARMACEUTICALS

#13 | 2024-01-04
US20240002381A1
Chemistry; metallurgy

1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c] pyridin-7(6H)-ones as inhibitors of BET proteins

#14 | 2023-08-24
US20230265083A1
Chemistry; metallurgy

Heterocycle CDK Inhibitors And Their Use Thereof

#15 | 2023-04-20
US20230121440A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#16 | 2023-01-12
US20230009843A1
Chemistry; metallurgy

HETEROCYCLIC COMPOUNDS AS PI3K-y INHIBITORS

#17 | 2022-12-29
US20220411383A1
Chemistry; metallurgy

AMINOPYRAZINE DERIVATIVES AS PI3K-y INHIBITORS

#18 | 2022-10-27
US20220340544A1
Chemistry; metallurgy

SUBSTITUTED HETEROCYCLIC DERIVATIVES AS PI3K INHIBITORS

#19 | 2022-10-20
US20220331296A1
Human necessities

1,2,5-Oxadiazoles As Inhibitors Of Indoleamine 2,3- Dioxygenase

#20 | 2022-08-11
US20220251087A1
Chemistry; metallurgy

Substituted imidazo[2,1-f][1,2,4]triazines as PI3K-gamma inhibitors

#21 | 2022-07-21
US20220227736A1
Chemistry; metallurgy

Pyridine and pyridimine compounds as PI3K-gamma inhibitors

#22 | 2022-07-07
US20220213107A1
Chemistry; metallurgy

Tertiary alcohols as PI3K-γ inhibitors

#23 | 2022-07-07
US20220213065A1
Chemistry; metallurgy

Aminopyrazine diol compounds as PI3K-γ inhibitors

#24 | 2022-06-09
US20220177491A1
Chemistry; metallurgy

Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors

#25 | 2022-04-21
US20220119393A1
Chemistry; metallurgy

USE OF PYRAZOLOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PI3K-DELTA RELATED DISORDERS

#26 | 2022-04-14
US20220112198A1
Chemistry; metallurgy

Crystalline forms of a phosphoinositide 3-kinase (PI3K) inhibitor

#27 | 2022-04-07
US20220106318A1
Chemistry; metallurgy

Use of pyrazolopyrimidine derivatives for the treatment of PI3K-δ related disorders

#28 | 2021-12-23
US20210395258A1
Chemistry; metallurgy

Heterocyclic derivatives as PI3K inhibitors

#29 | 2021-10-28
US20210332059A1
Chemistry; metallurgy

USE OF PYRAZOLOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PI3K-DELTA RELATED DISORDERS

#30 | 2021-09-30
US20210300925A1
Chemistry; metallurgy

1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins

#31 | 2021-08-19
US20210253601A1
Chemistry; metallurgy

Pyrimidinones as PI3K inhibitors

#32 | 2021-06-24
US20210188872A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#33 | 2021-02-04
US20210030722A1
Human necessities

1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

#34 | 2020-12-10
US20200385392A1
Chemistry; metallurgy

Tertiary alcohols as PI3K-γ inhibitors

#35 | 2020-12-03
US20200377502A1
Chemistry; metallurgy

1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins

#36 | 2020-10-29
US20200339542A1
Chemistry; metallurgy

AMINOPYRAZINE DIOL COMPOUNDS AS PI3K-y INHIBITORS

#37 | 2020-10-22
US20200331903A1
Chemistry; metallurgy

3-(5-amino-pyrazin-2-yl)-benzenesulfonamide derivatives and related compounds as PI3K-gamma kinase inhibitors

#38 | 2020-10-15
US20200323858A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#39 | 2020-08-06
US20200247820A1
Chemistry; metallurgy

Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors

#40 | 2020-05-14
US20200148689A1
Chemistry; metallurgy

Heterocyclic derivatives as PI3K inhibitors

#41 | 2020-05-14
US20200148671A1
Chemistry; metallurgy

Heterocyclic derivatives as PI3K inhibitors

#42 | 2020-05-14
US20200148667A1
Chemistry; metallurgy

Substituted heterocyclic derivatives as PI3K inhibitors

#43 | 2020-04-30
US20200131195A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#44 | 2020-04-23
US20200123176A1
Chemistry; metallurgy

Pyrimidinones as PI3K inhibitors

#45 | 2020-04-02
US20200102315A1
Chemistry; metallurgy

Imidazo[2,1-f][1,2,4]triazine compounds as pi3k-y inhibitors

#46 | 2020-03-05
US20200071335A1
Chemistry; metallurgy

Crystalline forms of a phosphoinositide 3-kinase (PI3K) inhibitor

#47 | 2020-02-13
US20200048251A1
Chemistry; metallurgy

1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins

#48 | 2020-01-30
US20200031837A1
Chemistry; metallurgy

Heterocyclic compounds as PI3K-y inhibitors

#49 | 2020-01-02
US20200002295A1
Chemistry; metallurgy

Aminopyrazine derivatives as PI3K-γ inhibitors

#50 | 2019-11-28
US20190359592A1
Chemistry; metallurgy

Pyridine and pyridimine compounds as PI3K-gamma inhibitors

#51 | 2019-10-03
US20190298724A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#52 | 2019-10-03
US20190298700A1
Human necessities

1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

#53 | 2019-09-12
US20190276435A1
Chemistry; metallurgy

Aminopyrazine diol compounds as PI3K-γ inhibitors

#54 | 2019-08-01
US20190233435A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#55 | 2019-07-11
US20190210985A1
Chemistry; metallurgy

Modulators of indoleamine 2,3-dioxygenase and methods of using the same

#56 | 2019-05-23
US20190152975A1
Chemistry; metallurgy

Tertiary alcohols as PI3K-γ inhibitors

#57 | 2019-05-09
US20190134040A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#58 | 2019-04-25
US20190119287A1
Chemistry; metallurgy

Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors

#59 | 2019-03-21
US20190084997A1
Chemistry; metallurgy

Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors

#60 | 2019-02-28
US20190062336A1
Chemistry; metallurgy

Heterocyclic compounds as PI3K-γ inhibitors

#61 | 2019-02-28
US20190060331A1
Human necessities

Aza-heteroaryl compounds as PI3K-gamma inhibitors

#62 | 2019-02-07
US20190040067A1
Chemistry; metallurgy

USE OF PYRAZOLOPYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PI3K-DELTA RELATED DISORDERS

#63 | 2019-01-03
US20190002470A1
Chemistry; metallurgy

Bicyclic azaheterocyclobenzylamines as PI3K inhibitors

#64 | 2018-12-20
US20180362546A1
Chemistry; metallurgy

Pyrimidinones as PI3K inhibitors

#65 | 2018-12-06
US20180346481A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#66 | 2018-11-01
US20180312506A1
Chemistry; metallurgy

1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins

#67 | 2018-08-09
US20180222920A1
Chemistry; metallurgy

Tricyclic heterocycles as bet protein inhibitors

#68 | 2018-06-28
US20180177769A1
Human necessities

1,2,5-Oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

#69 | 2018-02-01
US20180030006A1
Chemistry; metallurgy

Modulators of indoleamine 2,3-dioxygenase and methods of using the same

#70 | 2018-01-11
US20180009816A1
Chemistry; metallurgy

Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-γ inhibitors

#71 | 2017-12-07
US20170349579A1
Chemistry; metallurgy

Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b] pyrimidin-5-yl-amines as Janus kinase inhibitors

#72 | 2017-12-07
US20170348289A1
Human necessities

1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

#73 | 2017-11-30
US20170340641A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#74 | 2017-08-17
US20170232016A1
Human necessities

Aza-heteroaryl compounds as PI3K-gamma inhibitors

#75 | 2017-08-03
US20170217985A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#76 | 2017-07-27
US20170210754A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#77 | 2017-07-06
US20170190689A1
Chemistry; metallurgy

PYRIDINE AND PYRIDIMINE COMPOUNDS AS PI3K-GAMMA INHIBITORS

#78 | 2017-06-08
US20170158710A1
Chemistry; metallurgy

Tricyclic heterocycles as bet protein inhibitors

#79 | 2017-06-08
US20170158696A1
Chemistry; metallurgy

N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors

#80 | 2017-06-08
US20170158689A1
Chemistry; metallurgy

1H-pyrrolo[2,3,c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins

#81 | 2017-05-11
US20170129899A1
Chemistry; metallurgy

Heterocyclic compounds as PI3K-γ inhibitors

#82 | 2017-02-23
US20170050987A1
Chemistry; metallurgy

Pyrimidinones as PI3K inhibitors

#83 | 2017-01-19
US20170014418A1
Human necessities

Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors

#84 | 2016-09-15
US20160264580A1
Chemistry; metallurgy

Bicyclic azaheterocyclobenzylamines as PI3K inhibitors

#85 | 2016-08-11
US20160229843A1
Chemistry; metallurgy

Aza-heteroaryl compounds as PI3K-gamma inhibitors

#86 | 2016-08-04
US20160220543A1
Human necessities

1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

#87 | 2016-07-28
US20160213654A1
Human necessities

Bicyclic heterocycles as bet protein inhibitors

#88 | 2016-06-09
US20160159817A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#89 | 2016-03-17
US20160075721A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#90 | 2016-02-18
US20160046650A1
Chemistry; metallurgy

Tricyclic heterocycles as BET protein inhibitors

#91 | 2016-01-28
US20160024117A1
Chemistry; metallurgy

Heterocyclylamines as PI3K inhibitors

#92 | 2016-01-28
US20160022685A1
Human necessities

Heterocyclylamines as PI3K inhibitors

#93 | 2015-12-17
US20150361094A1
Chemistry; metallurgy

Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors

#94 | 2015-11-05
US20150315185A1
Chemistry; metallurgy

Pyrrolo[2,3-b]pyridin-4-yl-amines and pyrrolo[2,3-b]pyrimidin-5-yl-amines as Janus kinase inhibitors

#95 | 2015-10-29
US20150307493A1
Chemistry; metallurgy

1H-pyrrolo[2,3-c]pyridin-7(6H)-ones and pyrazolo[3,4-c]pyridin-7(6H)-ones as inhibitors of BET proteins

#96 | 2015-10-08
US20150284390A1
Chemistry; metallurgy

N-(1-(substituted-phenyl)ethyl)-9H-purin-6-amines as PI3K inhibitors

#97 | 2015-07-09
US20150190378A1
Human necessities

1,2,5-oxadiazoles as inhibitors of indoleamine 2,3-dioxygenase

#98 | 2015-05-28
US20150148375A1
Chemistry; metallurgy

Bicyclic heterocycles as BET protein inhibitors

#99 | 2015-05-28
US20150148372A1
Chemistry; metallurgy

BICYCLIC HETEROCYCLES AS BET PROTEIN INHIBITORS

#100 | 2015-05-28
US20150148342A1
Chemistry; metallurgy

Substituted pyrrolo[2,3-c]pyridines and pyrazolo[3,4-c]pyridines as BET protein inhibitors

InventorID:

128957 ⎘