ClassID:

20412

A61K31/4985 - CPC Classification

Classification description:

Medicinal preparations containing organic active ingredients; Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two nitrogen atoms as the only ring heteroatoms, e.g. piperazine Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems

Recent Application in this class:
#1
20260152505
2026-06-04

CHEMOKINE RECEPTOR MODULATORS AND USES THEREOF

#2
20260152499
2026-06-04

COMPOUNDS AND USES THEREOF

#3
20260152484
2026-06-04

HETEROCYCLIC COMPOUNDS AS TRIGGERING RECEPTOR EXPRESSED ON MYELOID CELLS 2 AGONISTS

#4
20260146035
2026-05-28

FUSED BICYCLIC COMPOUNDS AND THEIR USE AS MER AND AXL INHIBITORS

#5
20260138990
2026-05-21

TRICYCLIC FUSED IMIDAZOLE COMPOUNDS AS CD38 MODULATORS AND USES THEREOF

#6
20260138978
2026-05-21

POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M1

#7
20260138956
2026-05-21

NOVEL COMPOUNDS AND USES THEREOF

#8
20260137706
2026-05-21

METHODS OF TREATING INFLAMMATORY DISEASES

#9
20260137689
2026-05-21

INTEGRATION OF MOLECULAR MECHANISMS IN THE STRIATUM AS A COMBINATION DRUG STRATEGY FOR THE TREATMENT OF PSYCHIATRIC AND NEUROLOGICAL DISORDERS IN WHICH ANHEDONIA OR MOTIVATION-RELATED DYSFUNCTION EXISTS

#10
20260137681
2026-05-21

EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE INHIBITORS IN COMBINATION WITH HGF-RECEPTOR INHIBITORS FOR THE TREATMENT OF CANCER

#11
20260137679
2026-05-21

GCN2 INHIBITOR FOR TREATING METASTASES

#12
20260137666
2026-05-21

N-methyl-D-aspartic Acid Receptor Modulators

#13
20260137665
2026-05-21

COMBINATION THERAPIES FOR THE TREATMENT OF CANCER

#14
20260132140
2026-05-14

IMIDAZOLYL-AMINO-PYRAZINE-CARBONITRILS AS CHK-1 INHIBITORS

#15
20260132136
2026-05-14

Pyrazolo[5,1-f][1,2,4]triazin-4-ones as inhibitors of NOX4

#16
20260132128
2026-05-14

COMPOUND FOR RECOVERING P53 MUTATION FUNCTION AND USE THEREOF

#17
20260132127
2026-05-14

NOVEL SPIRO COMPOUND

#18
20260131140
2026-05-14

MODIFYING EARLY-STAGE PARKINSON'S DISEASE PROGRESSION WITH DEEP BRAIN STIMULATION

#19
20260130886
2026-05-14

EXTRUDED SOFT CHEW CONTAINING A NON-ANIMAL BASED PALATANT AND ACTIVE PHARMACEUTICAL INGREDIENTS

#20
20260130859
2026-05-14

PALATABLE FORMULATIONS

#21
20260130856
2026-05-14

LIPOSOME COMPOSITIONS FOR DELIVERY OF COMPOUNDS AND METHODS THEREOF

#22
20260125398
2026-05-07

5,6-FUSED BICYCLIC ALCOHOL COMPOUNDS AS 15-PROSTAGLANDIN DEHYDROGENASE MODULATORS

#23
20260125384
2026-05-07

INDAZOLE INHIBITORS OF CYCLIC GMP-AMP SYNTHASE AND USES THEREOF

#24
20260125383
2026-05-07

INDAZOLE INHIBITORS OF CYCLIC GMP-AMP SYNTHASE AND USES THEREOF

#25
20260124214
2026-05-07

HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER

#26
20260124209
2026-05-07

INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

#27
20260124198
2026-05-07

ANTIVIRAL PYRAZOLOPYRIDINONE COMPOUNDS

#28
20260116884
2026-04-30

PROTAC CHIMERIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF

#29
20260116881
2026-04-30

KIF MODULATOR COMPOUNDS AND METHODS OF USE

#30
20260116871
2026-04-30

Tyrosine Kinase Inhibitors and Uses Thereof

#31
20260115226
2026-04-30

PHARMACEUTICAL COMPOSITION

#32
20260115188
2026-04-30

METHODS OF TREATING CENTERAL NERVOUS SYSTEM DISORDERS COMPRISING ADMINISTERING DEUTERATED LUMATEPERONE AND A NITRIC OXIDE DONOR

#33
20260115182
2026-04-30

PAPD5 INHIBITORS AND METHODS OF USE THEREOF

#34
20260115174
2026-04-30

PHARMACOLOGICAL CORRECTORS OF RHODOPSIN AND USES THEREOF

#35
20260109709
2026-04-23

2-AMINO IMIDAZOLE DERIVATIVES AS PRMT5 INHIBITORS

#36
20260109704
2026-04-23

5-MEMBERED HETEROARYL INDAZOLE CGAS INHIBITORS AND USES THEREOF

#37
20260109699
2026-04-23

AZOLE DERIVATIVES AS SHP2 INHIBITORS

#38
20260108546
2026-04-23

GIP RECEPTOR AGONIST COMPOUNDS

#39
20260108510
2026-04-23

PYRAZOLYL INDAZOLE CGAS INHIBITORS AND USES THEREOF

#40
20260108509
2026-04-23

6-MEMBERED HETEROARYL INDAZOLE CGAS INHIBITORS AND USES THEREOF

#41
20260108496
2026-04-23

METHODS FOR REPROGRAMING EXHAUSTED T CELLS AND BOOSTING IMMUNE CHECKPOINT BLOCKADE THERAPY FOR CANCER

#42
20260102395
2026-04-16

INHIBITING HISTONE DEACETYLASE 6

#43
20260102394
2026-04-16

PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS

#44
20260097056
2026-04-09

SYK ACTIVATORS AND INHIBITORS IN NEURODEGENERATIVE DISEASES

#45
20260097033
2026-04-09

TREATING SPONDYLOARTHRITIC AND PSORIATIC CONDITIONS WITH UPADACITINIB

#46
20260097032
2026-04-09

PHARMACEUTICAL COMPOSITION, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#47
20260092076
2026-04-02

NOVEL COMPOUNDS

#48
20260092074
2026-04-02

Annelated Pyridines as Steroidogenesis Inhibitors, Preparation Method and Use Thereof

#49
20260091048
2026-04-02

GIP RECEPTOR AGONIST COMPOUNDS

#50
20260091032
2026-04-02

AMORPHOUS SOLID DISPERSIONS

#51
20260085083
2026-03-26

NOVEL COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF

#52
20260085073
2026-03-26

PYRAZOLYLCARBOXAMIDE COMPOUNDS AND THEIR USE IN THERAPY

#53
20260085071
2026-03-26

NOVEL CRYSTALLINE FORM OF 1-(8-BROMOPYRIDO[2,3- E][1,2,4]TRIAZOLO[4,3-A]PYRAZIN-4-YL)-NMETHYLAZETIDIN- 3-AMINE

#54
20260085045
2026-03-26

NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF

#55
20260083759
2026-03-26

Combinations Comprising Psychedelics for the Treatment of Schizophrenia and Other Neuropsychiatric and Neurologic Disorders

#56
20260083732
2026-03-26

UPADACITINIB FORMULATION

#57
20260078130
2026-03-19

NAMPT MODULATORS, PREPARATIONS, AND USES THEREOF

#58
20260078122
2026-03-19

INDAZOLE COMPOUNDS AS PKMYT1 KINASE INHIBITORS

#59
20260078103
2026-03-19

ISOQUINOLONES AS PI3K INHIBITORS

#60
20260070922
2026-03-12

PYRAZOLE AND IMIDAZOLE DERIVATIVES AS DUAL OREXIN AND KAPPA-OPIOID RECEPTORS MODULATORS COMPOSITION, METHODS FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS

#61
20260070902
2026-03-12

SULFONYL DERIVATIVES AS CCR6 INHIBITORS

#62
20260062416
2026-03-05

INHIBITORS OF KIF18A AND USES THEREOF

#63
20260062409
2026-03-05

Composition and Method for Treating Metabolic Disorders

#64
20260060943
2026-03-05

OVARIAN CANCER VACCINES

#65
20260060941
2026-03-05

ENGAGING THE CERVICAL SPINAL CORD CIRCUITRY TO RE-ENABLE VOLITIONAL CONTROL OF HAND FUNCTION IN TETRAPLEGIC SUBJECTS

#66
20260055121
2026-02-26

TYK2 INHIBITORS AND USES THEREOF

#67
20260055100
2026-02-26

INDANE AND COUMARAN DERIVATIVES AS FAST SKELETAL MUSCLE MYOSIN INHIBITORS

#68
20260055090
2026-02-26

OXADIAZOLE HDAC6 INHIBITORS AND USES THEREOF

#69
20260053797
2026-02-26

METHOD AND FORMULATION FOR TREATING MALE PREMATURE EJACULATION

#70
20260053748
2026-02-26

NOVEL METHODS

#71
20260049145
2026-02-19

ANTI-PD-L1 COMBINATIONS FOR TREATING TUMORS

#72
20260049082
2026-02-19

AMIDO PYRIDO[3,4-B]INDOLE-1,4-DIONE COMPOUNDS FOR TREATMENT OF PORPHYRIAS

#73
20260049080
2026-02-19

WILD TYPE KIT INHIBITORS

#74
20260049061
2026-02-19

SMALL MOLECULES AS KCNQ2/3 (KV7.2/3) CHANNEL ACTIVATORS AND THEIR MEDICAL USE THEREOF

#75
20260048062
2026-02-19

FUSED AMINO PYRIMIDINE COMPOUNDS FOR TREATMENT OF PSYCHOSIS AND PSYCHOTIC DISORDERS

#76
20260048056
2026-02-19

SOLID PHARMACEUTICAL COMPOSITIONS COMPRISING BIOPTERIN DERIVATIVES AND USES OF SUCH COMPOSITIONS

#77
20260048019
2026-02-19

USE OF CO-PROCESSED EXCIPIENTS IN CONTINUOUS MANUFACTURING OF SOLID DOSAGE FORMS

#78
20260042760
2026-02-12

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH CALCITONIN RECEPTOR AND/OR AMYLIN RECEPTOR ACTIVITY

#79
20260041684
2026-02-12

ORGANIC COMPOUNDS

#80
20260041639
2026-02-12

GEPOTIDACIN FORMULATION

#81
20260035387
2026-02-05

COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE

#82
20260035367
2026-02-05

PKC-Theta Modulators

#83
20260034125
2026-02-05

N-PHENYL-1-(PHENYLSULFONYL)PIPERIDIN-4-AMINE DERIVATIVES AS CCR6 INHIBITORS

#84
20260034124
2026-02-05

NOVEL SALTS AND CRYSTALS

#85
20260034123
2026-02-05

CDK2 INHIBITORS AND METHODS OF USING THE SAME

#86
20260028354
2026-01-29

TETRAHYDRONAPHTHALENE DERIVATIVES AS ESTROGEN RECEPTOR DEGRADERS

#87
20260028343
2026-01-29

Substituted Imidazopyrazine Compounds as Ligand Directed Degraders of IRAK3

#88
20260028334
2026-01-29

N-(3-(BENZO[B]THIOPHENE-2-CARBOXAMIDO)-PHENYL)-2,3-DIHYDROBENZO[B][1,4]DIOXINE-6-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS LACTATE/ATP PRODUCTION INHIBITORS FOR THE TREATMENT OF CANCER

#89
20260028328
2026-01-29

HETEROARYL DERIVATIVES AS DDRs INHIBITORS

#90
20260027123
2026-01-29

Compositions for Modulating Lipoxygenase and Methods of Using Same

#91
20260027108
2026-01-29

PHARMACEUTICAL COMPOSITION OF HETEROARYL DERIVATIVE AND MEDICAL USE THEREOF

#92
20260027088
2026-01-29

Inhibitors of Glutathione S-Transferases (GSTS) and NAD(P)H:Quinone Oxidoreductase 1 (NQO1), Pharmaceutical Compositions, and Uses in Managing Cancer

#93
20260026529
2026-01-29

MATERIALS AND METHODS FOR THE MANUFACTURE OF AN ANIMAL FEED

#94
20260022118
2026-01-22

HETEROCYCLIC COMPOUNDS AS NRAS INHIBITORS

#95
20260021100
2026-01-22

METHODS FOR TREATING ALZHEIMER DISEASE AND FOR REDUCING AMYLOID BETA FORMATION

#96
20260021091
2026-01-22

PHARMACEUTICAL COMPOSITIONS

#97
20260021071
2026-01-22

SMALL MOLECULE BROAD-SPECTRUM ANTIBIOTICS

#98
20260015360
2026-01-15

BIARYL DERIVATIVES AND RELATED USES

#99
20260015354
2026-01-15

Solid State Forms of Ensifentrine

#100
20260014164
2026-01-15

COMBINATION THERAPY FOR PI3K-ASSOCIATED DISEASE OR DISORDER

#101
20260014162
2026-01-15

REHYDRATION COMPOSITION AND METHOD OF USE

#102
20260014161
2026-01-15

Uses of JAK Inhibitors in the Management of Inflammation-Associated Depression and Central Nervous System (CNS) Pathologies

#103
20260014159
2026-01-15

DEVELOPMENT OF ALPHA-1A-ADRENERGIC RECEPTOR AGONISTS AS A THERAPY TO TREAT HEART FAILURE

#104
20260014156
2026-01-15

TREATMENT OF A DISEASE OF THE GASTROINTESTINAL TRACT WITH A JAK OR OTHER KINASE INHIBITOR

#105
20260014147
2026-01-15

STAT6 DEGRADERS

#106
20260009079
2026-01-08

BIOMARKERS OF PREGNANCY LOSS

#107
20260008780
2026-01-08

SUBSTITUTED 3,4-DIHYDROISOQUINOLIN-1(2H)-ONE DERIVATIVES AND RELATED USES

#108
20260008770
2026-01-08

CBL-B INHIBITORS AND METHODS OF USES THEREOF

#109
20260007662
2026-01-08

COMPOSITIONS COMPRISING TIGOLANER FOR CONTROLLING PARASITES

#110
20260007661
2026-01-08

EXTENDED RELEASE UPADACITINIB FORMULATIONS

#111
20260001892
2026-01-01

COMPOUND FOR REGULATING AND CONTROLLING ACTIVITY OF 15-PGDH AND PREPARATION METHOD THEREFOR

#112
20260001885
2026-01-01

4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDES AS BTK INHIBITORS

#113
20260001879
2026-01-01

COMPOUNDS AS MYT1 INHIBITORS

#114
20260001876
2026-01-01

Compounds and Their Use as PDE4 Activators

#115
20250388604
2025-12-25

Compounds and Their Use as PDE4 Activators

#116
20250388603
2025-12-25

ANTIMALARIAL COMPOUNDS

#117
20250388585
2025-12-25

PRMT5 INHIBITORS AND USES THEREOF

#118
20250388583
2025-12-25

COMPOUNDS AND METHOD FOR PKMYT1 INHIBITION

#119
20250388581
2025-12-25

ORGANIC COMPOUNDS

#120
20250388578
2025-12-25

NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#121
20250387397
2025-12-25

SUBSTITUTED AMINO TRIAZOLOPYRIMIDINE AND AMINO TRIAZOLOPYRAZINE ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE

#122
20250387364
2025-12-25

ARSINOTHRICIN AND METHODS OF TREATING INFECTIONS USING ARSINOTHRICIN

#123
20250387343
2025-12-25

Nanoparticle Compositions and Methods for Synthesis Thereof

#124
20250382306
2025-12-18

HETEROCYCLIC COMPOUND AS TAAR1 LIGAND AGONIST

#125
20250382302
2025-12-18

Anticancer polyheterocyclic compounds and associated methods

#126
20250382298
2025-12-18

NITROGEN-CONTAINING COMPOUND AND USE THEREOF

#127
20250382297
2025-12-18

INHIBITORS OF FGFR2 AND FGFR3 AND USES THEREOF

#128
20250382296
2025-12-18

NITROGEN-CONTAINING FUSED THREE RING PRMT5 INHIBITOR, AND PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF

#129
20250381187
2025-12-18

KRAS G12C INHIBITORS AND METHODS OF USING THE SAME

#130
20250381181
2025-12-18

CANCER TREATMENT AGENT INCLUDING MALT1 INHIBITING DRUG AS ACTIVE INGREDIENT

#131
20250376473
2025-12-11

PRMTS INHIBITOR AND USE THEREOF

#132
20250376461
2025-12-11

INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS

#133
20250375428
2025-12-11

CBL-B INHIBITORS AND ANTI-PD1/ANTI-PD-L1 FOR USE IN THE TREATMENT OF CANCER

#134
20250368651
2025-12-04

ANTIVIRAL COMPOUNDS USEFUL AGAINST SARS-COV-2

#135
20250367192
2025-12-04

BICYCLIC COMPOUNDS AND METHODS FOR THEIR USE IN TREATING PITT HOPKINS SYNDROME

#136
20250367191
2025-12-04

TREATMENT OF MITOCHONDRIAL DISEASES WITH A CNS-PENETRANT SGC STIMULATOR ZAGOCIGUAT

#137
20250361239
2025-11-27

PROTEIN DEGRADERS AND USES THEREOF

#138
20250360145
2025-11-27

CSF-1R INHIBITORS AND USES THEREOF

#139
20250360140
2025-11-27

NOVEL METHODS

#140
20250360136
2025-11-27

Treatment or Reversal of Treatment Resistant Depression and Related Central Nervous System (CNS) Inflammatory Conditions with a JAK Inhibitor

#141
20250360126
2025-11-27

TARGETING AN ENZYME REQUIRED FOR ACUTE MYELOID LEUKEMIA

#142
20250360103
2025-11-27

METHODS OF TREATING WHSC1-OVEREXPRESSING CANCERS BY INHIBITING SETD2

#143
20250353864
2025-11-20

INDAZOLE CONTAINING MACROCYCLES AND THEIR USE

#144
20250353862
2025-11-20

C-MYC MRNA TRANSLATION MODULATORS AND USES THEREOF IN THE TREATMENT OF CANCER

#145
20250353859
2025-11-20

COMPOUNDS AS CCR6 INHIBITORS

#146
20250353853
2025-11-20

FLAVIVIRUS INHIBITORS

#147
20250353841
2025-11-20

HETEROCYCLIC COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE

#148
20250352548
2025-11-20

BTK Reducing Molecules for Treatment of Cancers and Immune System Disorders

#149
20250352518
2025-11-20

A BENZIMIDAZOLE COMPOUND WITH ANTIHELMINTHIC ACTIVITY FOR USE IN REVERSING, ARRESTING OR SLOWING DOWN CELLULAR AGEING IN A VERTEBRATE SUBJECT

#150
20250352469
2025-11-20

NOVEL COMPOSITIONS, DEVICES, AND METHODS

#151
20250346571
2025-11-13

BICYCLIC DERIVATIVE PARP INHIBITOR AND USE THEREOF

#152
20250345345
2025-11-13

METHODS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS

#153
20250340532
2025-11-06

HETEROCYCLIC COMPOUND CCR4 INHIBITOR AND USER THEREOF

#154
20250339520
2025-11-06

COMPOSITIONS AND METHODS FOR USE IN KRAS-TARGETED THERAPIES FOR THE TREATMENT OF CANCER

#155
20250339427
2025-11-06

AMORPHOUS SOLID DISPERSIONS

#156
20250339426
2025-11-06

GCN2 MODULATOR FOR TREATING CANCER

#157
20250333423
2025-10-30

SMALL MOLECULE MODULATORS OF GP130 SIGNALING PATHWAYS

#158
20250332173
2025-10-30

COMPOUNDS AND METHODS FOR MODULATING NUCLEIC ACID SPLICING

#159
20250332171
2025-10-30

PDE5 INHIBITOR POWDER FORMULATIONS AND METHODS RELATING THERETO

#160
20250332165
2025-10-30

PHARMACEUTICAL COMPOSITIONS OF NILOTINIB

#161
20250332164
2025-10-30

METHODS AND COMPOSITIONS FOR SLEEP DISORDERS AND OTHER DISORDERS

#162
20250332159
2025-10-30

REACTIVE OXYGEN SPECIES MODULATION THROUGH BINDING OF LIGANDS AT THE NQ-BINDING SITE OF THE RESPIRATORY COMPLEX III

#163
20250332155
2025-10-30

SUBSTITUTED TETRAHYDROQUINOLINONE COMPOUNDS AS ROR GAMMA MODULATORS

#164
20250332143
2025-10-30

COMPOSITION COMPRISING ALOX5 INHIBITOR FOR PREVENTING OR TREATING SARCOPENIA

#165
20250326761
2025-10-23

sGC STIMULATORS

#166
20250326755
2025-10-23

CYCLIC QUATERNARY AMMONIUM SALT COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#167
20250326722
2025-10-23

NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF

#168
20250320224
2025-10-16

NOVEL PAR-2 INHIBITORS

#169
20250320214
2025-10-16

ORGANIC COMPOUNDS

#170
20250320213
2025-10-16

Nitrogen-Containing Heterocyclic Compounds

#171
20250319081
2025-10-16

Compositions, Devices, and Methods for Treating or Preventing Headaches

#172
20250319060
2025-10-16

METHODS FOR THE PROPHYLAXIS AND TREATMENT OF COVID AND COVID-19

#173
20250313576
2025-10-09

COMPOUND FOR PHOTOOXYGENATION CATALYST AND MEDICINAL COMPOSITION CONTAINING SAME

#174
20250313564
2025-10-09

ACIDIC SALT OR CRYSTAL FORM OF NITROGEN-CONTAINING FUSED RING DERIVATIVE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#175
20250313563
2025-10-09

GLYCOGEN SYNTHASE KINASE 3 INHIBITORS AND USES THEREOF

#176
20250312456
2025-10-09

TREATMENT FOR DIABETES IN PATIENTS INAPPROPRIATE FOR METFORMIN THERAPY

#177
20250312353
2025-10-09

DRUG REPURPOSING FOR TREATMENT OF CONGENITAL VASCULAR MALFORMATIONS

#178
20250312352
2025-10-09

GLP-1R MODULATING COMPOUNDS

#179
20250312350
2025-10-09

INHIBITORS OF RLIP76

#180
20250312340
2025-10-09

METHODS OF TREATING NEUROPATHIC PAIN

#181
20250312339
2025-10-09

METHODS AND COMPOSITIONS COMPRISING A SHP2 INHIBITOR AND A PD-LI BINDING ANTAGONIST

#182
20250312338
2025-10-09

TREATMENT OF NEUROLOGICAL DISORDERS

#183
20250304600
2025-10-02

PHARMACEUTICAL COMPOUNDS AND COMPOSITIONS AS c-KIT KINASE INHIBITORS

#184
20250302954
2025-10-02

METHODS TO OVERCOME DRUG RESISTANCE BY RE-SENSITIZING CANCER CELLS TO TREATMENT WITH A PRIOR THERAPY VIA TREATMENT WITH A T CELL THERAPY

#185
20250302852
2025-10-02

COMPOSITIONS COMPRISING METHYLXANTHINES AND DISACCHARIDES DERIVED FROM ENZYMATIC CONVERSION OF SUCROSE

#186
20250302842
2025-10-02

HETEROCYCLIC COMPOUNDS USEFUL FOR TREATMENT OF CANCERS

#187
20250302830
2025-10-02

METHOD FOR TREATING HIV WITH CABOTEGRAVIR AND RILPIVIRINE

#188
20250302829
2025-10-02

METHOD FOR TREATING HIV WITH CABOTEGRAVIR AND RILPIVIRINE

#189
20250302828
2025-10-02

ORAL GLIPTIN COMPOSITIONS AND METHOD FOR PREPARATION THEREOF

#190
20250296988
2025-09-25

COMBINATION THERAPY

#191
20250296916
2025-09-25

BICYCLIC PIPERAZINONES AND THERAPEUTIC USES THEREOF

#192
20250295655
2025-09-25

BRUTON'S KINASE INHIBITORS FOR THE TREATMENT OF A SUDDEN ALLERGIC REACTION

#193
20250295642
2025-09-25

FLUOROQUINOXALINONE DERIVATIVE FOR SELECTIVELY INHIBITING PARP1

#194
20250289789
2025-09-18

REVERSIBLE LYSINE COVALENT MODIFIERS OF CDK2 AND USES THEREOF

#195
20250282798
2025-09-11

HETEROARYL-SUBSTITUTED BICYCLIC COMPOUND AND USE THEREOF

#196
20250282797
2025-09-11

CRYSTALLINE FORM OF FGFR4 INHIBITOR AND USE THEREOF

#197
20250282785
2025-09-11

PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE

#198
20250282782
2025-09-11

PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS

#199
20250282749
2025-09-11

COMPOUNDS AND METHODS OF USE

#200
20250281482
2025-09-11

BILE ACID RECYCLING INHIBITORS FOR TREATMENT OF PEDIATRIC CHOLESTATIC LIVER DISEASES

#201
20250281473
2025-09-11

CDK Inhibitors And Their Use As Pharmaceuticals

#202
20250281470
2025-09-11

COMPOSITIONS FOR THE TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE AND NON-ALCOHOLIC STEATOHEPATITIS

#203
20250276972
2025-09-04

COMPOUNDS AS CASEIN KINASE INHIBITORS

#204
20250275963
2025-09-04

DRY EYE TREATMENTS

#205
20250275962
2025-09-04

TRANSMUCOSAL METHODS FOR TREATING PSYCHIATRIC AND NEUROLOGICAL CONDITIONS

#206
20250275961
2025-09-04

BROMOCRIPTINE FORMULATIONS

#207
20250270224
2025-08-28

POLYCYCLIC POLY(ADP-RIBOSE) POLYMERASE SELECTIVE INHIBITOR

#208
20250270208
2025-08-28

BICYCLIC HETEROCYCLES AS MRGPRX2 ANTAGONISTS

#209
20250268893
2025-08-28

PHARMACEUTICAL COMPOSITIONS

#210
20250263415
2025-08-21

TERTIARY AMIDE DERIVATIVES SUBSTITUTED WITH 4-MEMBERED RING STRUCTURE

#211
20250263410
2025-08-21

NK3 MODULATORS AND USES THEREOF

#212
20250263394
2025-08-21

COMPOUNDS, PREPARATION METHODS AND USES THEREOF

#213
20250262268
2025-08-21

Methods and Compositions for Inhibiting Viral Infection

#214
20250262206
2025-08-21

USE OF TACHYKININ RECEPTOR 3 INHIBITÓR

#215
20250262194
2025-08-21

PHARMACEUTICAL FOR TREATING OR PREVENTING CANCER

#216
20250257067
2025-08-14

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH CALCITONIN RECEPTOR AND/OR AMYLIN RECEPTOR ACTIVITY

#217
20250257062
2025-08-14

GLP-1R Agonist and Therapeutic Method Thereof

#218
20250257055
2025-08-14

TERTIARY AMIDE DERIVATIVES SUBSTITUTED WITH 4-MEMBERED RING STRUCTURE

#219
20250255870
2025-08-14

METHODS FOR TREATING HAIR LOSS AND NAIL BRITTLENESS, FRAGILITY, OR PITTING

#220
20250255865
2025-08-14

METHODS OF TREATING OCULAR CONDITIONS

#221
20250250277
2025-08-07

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#222
20250249026
2025-08-07

PHARMACEUTICAL COMPOSITION FOR PRODUCING SAFE AMOUNT OF NITRIC OXIDE AND USE THEREOF

#223
20250249019
2025-08-07

METHOD OF TREATMENT INCLUDING KRAS G12C INHIBITORS AND AURORA A INHIBITORS

#224
20250249005
2025-08-07

INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

#225
20250243201
2025-07-31

ORGANIC COMPOUNDS

#226
20250241996
2025-07-31

COMBINATORIAL, AND ROTATIONAL COMBINATORIAL THERAPIES

#227
20250241992
2025-07-31

COMPOSITIONS AND METHODS FOR TREATING METABOLIC DISEASES

#228
20250241924
2025-07-31

TREATMENT OF ERECTILE DYSFUNCTION AND OTHER INDICATIONS

#229
20250241911
2025-07-31

TADALAFIL ORAL SUSPENSION

#230
20250241885
2025-07-31

ARSINOTHRICIN AND METHODS OF TREATING INFECTIONS USING ARSINOTHRICIN

#231
20250236627
2025-07-24

CERTAIN OCTAHYDROFURO[3,4- B]PYRAZINES AS GLP-1 RECEPTOR MODULATORS

#232
20250236619
2025-07-24

FUSED BICYCLIC COMPOUND CONTAINING PYRROLINONE

#233
20250235449
2025-07-24

METHODS OF TREATING OCULAR CONDITIONS

#234
20250230172
2025-07-17

SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF

#235
20250230166
2025-07-17

OXADIAZOLE HDAC6 INHIBITORS AND USES THEREOF

#236
20250230165
2025-07-17

HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF CANCER

#237
20250230138
2025-07-17

COMPOUNDS HAVING A T-STRUCTURE FORMED BY AT LEAST FOUR CYCLES FOR USE IN THE TREATMENT OF CANCER AND OTHER INDICATIONS

#238
20250228848
2025-07-17

PROCESS FOR MAKING A KRAS G12C INHIBITOR

#239
20250228778
2025-07-17

PLATFORM DRUG DELIVERY SYSTEM UTILIZING CRYSTAL ENGINEERING AND THEANINE DISSOLUTION

#240
20250221990
2025-07-10

TOPICAL ADMINISTRATION TO THE ORAL CAVITY

#241
20250221989
2025-07-10

PHARMACEUTICAL COMPOSITION, USE THEREOF, AND METHOD FOR TREATING CANCER

#242
20250221987
2025-07-10

PIPERAZINO RING-CONTAINING DERIVATIVE, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#243
20250221979
2025-07-10

NOVEL HETEROCYCLIC COMPOUND

#244
20250215016
2025-07-03

ISOXAZOLE-HETEROCYCLIC DERIVATIVE, PHARMACEUTICAL COMPOSITION AND USE

#245
20250215013
2025-07-03

SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND THE USE THEREOF

#246
20250214991
2025-07-03

BICYCLIC HETEROARYL-CONTAINING COMPOUNDS AS IKZF2 DEGRADERS

#247
20250214977
2025-07-03

STAT6 INHIBITORS AND USES THEREOF

#248
20250214951
2025-07-03

3-PHENYLISOXAZOLE DERIVATIVE, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING EYE DISEASE, CONTAINING SAME AS ACTIVE INGREDIENT

#249
20250214942
2025-07-03

INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATMENT OF DISEASE

#250
20250206749
2025-06-26

PRMT5 INHIBITING COMPOUNDS AND USES THEREOF

#251
20250206738
2025-06-26

WRN INHIBITORS

#252
20250206722
2025-06-26

SMALL MOLECULE INHIBITORS OF TEA DOMAIN FAMILY MEMBERS

#253
20250205518
2025-06-26

PULMONARY HYPERTENSION TREATMENT

#254
20250197406
2025-06-19

INDAZOLES AS HEMATOPOIETIC PROGENITOR KINASE 1 (HPK1) INHIBITORS AND METHODS FOR USING SAME

#255
20250197397
2025-06-19

ORGANIC COMPOUNDS

#256
20250195521
2025-06-19

USE OF SOS1 INHIBITORS TO TREAT MALIGNANCIES WITH SHP2 MUTATIONS

#257
20250195511
2025-06-19

INDAZOLE DERIVATIVES USEFUL AS INHIBITORS OF NOD-LIKE RECEPTOR PROTEIN 3

#258
20250195510
2025-06-19

NOVEL METHODS

#259
20250188091
2025-06-12

PYRIDONE COMPOUND HAVING INTEGRASE INHIBITORY ACTIVITY AND PHARMACEUTICAL USE THEREOF

#260
20250188088
2025-06-12

COMPOUND AND USE THEREOF

#261
20250186432
2025-06-12

SPLEEN TYROSINE KINASE INHIBITOR, COMPOSITION, AND METHODS OF USE

#262
20250186363
2025-06-12

Pharmaceutical Compositions and Methods for Treating Parkinson's Disease

#263
20250179079
2025-06-05

HEXAHYDROPYRIDO[4,3-B]INDOLYL KETONE DERIVATIVES USEFUL AS CGAS MODULATORS

#264
20250179027
2025-06-05

CYCLOALKYL OR HETEROCYCLYL SUBSTITUTED HETEROARYL COMPOUND, AND COMPOSITION AND USE THEREOF

#265
20250177478
2025-06-05

G ALPHA Q/11 INHIBITORS FOR USE AS AN ANALGESIC

#266
20250177408
2025-06-05

INHIBITOR OF INTERACTION BETWEEN YAP/TAZ AND TEAD, PREPARATION THEREOF, PHARMACEUTICAL COMPOSITION THEREOF AND USE THEREOF

#267
20250177389
2025-06-05

METHOD OF TREATMENT INCLUDING KRAS G12C INHIBITORS AND SHP2 INHIBITORS

#268
20250177374
2025-06-05

BCL-XL Inhibitory Compounds Having Low Cell Permeability and Antibody Drug Conjugates Including the Same

#269
20250171459
2025-05-29

2-METHYL-4',5'-DIHYDROSPIRO[PIPERIDINE-4,7'-THIENO[2,3-C]PYRAN] DERIVATIVES AS INHIBITORS OF APOL1 AND METHODS OF USING SAME

#270
20250171442
2025-05-29

WRN INHIBITORS

#271
20250171441
2025-05-29

WRN INHIBITORS

#272
20250171440
2025-05-29

WRN INHIBITORS

#273
20250170127
2025-05-29

RE-SENSITIZING MULTIDRUG-RESISTANT (MDR) GRAM-NEGATIVE BACTERIA TO COLISTIN USING IONOPHORES

#274
20250170124
2025-05-29

METHODS OF DIAGNOSING AND TREATING NEURODEGENERATIVE DISEASES

#275
20250163077
2025-05-22

MEMBRANE-ASSOCIATED TYROSINE- AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF

#276
20250163071
2025-05-22

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3,-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#277
20250163067
2025-05-22

NUCLEOBASE-SUBSTITUTED PIPERIDINYL-PYRIDINES AND RELATED COMPOUNDS AND THEIR USE IN TREATING DISEASES AND CONDITIONS

#278
20250161302
2025-05-22

EXTENDED RELEASE UPADACITINIB FORMULATIONS

#279
20250161301
2025-05-22

COMPOSITION FOR PREVENTING, AMELIORATING OR TREATING OBESITY AND DIABETES COMPRISING ZINC GLUCONATE AND CYCLO-HISPRO AS ACTIVE INGREDIENTS

#280
20250161278
2025-05-22

CBL-B INHIBITOR, COMPOSITIONS COMPRISING A CBL-B INHIBITOR IN A METHOD OF TREATING A DISEASE ASSOCIATED WITH CELL PROLIFERATION

#281
20250154174
2025-05-15

BICYCLIC HETEROCYCLES AS MRGPRX2 ANTAGONISTS

#282
20250154169
2025-05-15

COMPOUNDS AND METHODS FOR MODULATING SPLICING

#283
20250154149
2025-05-15

PHARMACEUTICAL COMPOSITION AND METHOD FOR PREPARING ACTIVE INGREDIENT COMPOUND THEREOF

#284
20250154144
2025-05-15

MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF

#285
20250154107
2025-05-15

3,4-Dihydroisoquinolin-1(2H)-Ones Derivatives as STING Antagonists and the Use Thereof

#286
20250154105
2025-05-15

POLYCYCLIC COMPOUND AND USE THEREOF

#287
20250152507
2025-05-15

SUBLINGUAL COMPOSITIONS FOR ERECTILE DYSFUNCTION

#288
20250145619
2025-05-08

KHK INHIBITOR, PREPARATION METHOD THEREFOR AND USE THEREOF

#289
20250145606
2025-05-08

THIAZOLE COMPOUNDS AND METHODS OF USE THEREOF

#290
20250145597
2025-05-08

INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF

#291
20250144091
2025-05-08

SITAGLIPTIN PREPARATION AND METHOD OF STORAGE THEREOF

#292
20250137057
2025-05-01

ADRM1/RPN13 SPLICED VARIANT IN THE PROGNOSIS AND TREATMENT OF HEPATOCELLULAR CARCINOMA

#293
20250136607
2025-05-01

PAD4 INHIBITORS AND USE THEREOF

#294
20250136601
2025-05-01

CYCLOPIPERIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF

#295
20250136596
2025-05-01

MEMBRANE-ASSOCIATED TYROSINE- AND THREONINE-SPECIFIC CDC2-INHIBITORY KINASE (PKMYT1) INHIBITORS AND USES THEREOF

#296
20250136581
2025-05-01

SUBSTITUTED TRIAZOLE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF

#297
20250136577
2025-05-01

HETEROCYCLIC DERIVATIVES AS MALT1 INHIBITORS

#298
20250136568
2025-05-01

FUSED HETEROCYCLIC COMPOUNDS AS PI3KALPHA INHIBITORS

#299
20250134806
2025-05-01

PHARMACEUTICAL COMPOSITION FOR DRY POWDER INHALATION AND PREPARATION METHOD THEREOF

#300
20250129093
2025-04-24

COMPOSITIONS AND METHODS RELATING TO ATP/P2X7R SIGNALING INHIBITION