ClassID:

20412

A61K31/4985 - page 2 - CPC Classification

Classification description:

Medicinal preparations containing organic active ingredients; Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two nitrogen atoms as the only ring heteroatoms, e.g. piperazine Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems

Recent Application in this class:
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MASP-2 INHIBITORS AND METHODS OF USE

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SIX-MEMBERED CYCLOTHIAZOLE COMPOUND AND USE THEREOF

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NITROGEN-CONTAINING TETRACYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF

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ADENOSINE RECEPTOR ANTAGONISTS

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ORAL FILM FORMULATION FOR MODULATING ABSORPTION PROFILE

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CERTAIN 2,5-DIAZABICYCLO[4.2.0]OCTANES AND OCTAHYDROFURO[3,4-B]PYRAZINES AS GLP-1 RECEPTOR MODULATORS

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AROMATIC HETEROCYCLIC COMPOUNDS, PREPARATION METHOD THEREFOR AND USES THEREOF

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SULFOXIMINE GLYCOSIDASE INHIBITORS

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BIFUNCTIONAL ARYLSULPHONAMIDE COMPOUNDS

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SULFONAMIDE COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL CONDITIONS

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cGAS ANTAGONIST COMPOUNDS

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BIPHENYL-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS

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TRICYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF

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DOSAGE FORM COMPOSITIONS COMPRISING AN INHIBITOR OF BRUTON'S TYROSINE KINASE

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COMBINATION THERAPIES

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STING AGONIST COMPOUNDS AND CONJUGATES

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ORGANIC COMPOUNDS

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SALT CRYSTAL FORM AND FREE BASE CRYSTAL FORM OF KINASE INHIBITOR

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GEPOTIDACIN AND VANCOMYCIN FOR USE IN THE TREATMENT OF AN INFECTION CAUSED BY STAPHYLOCOCCUS SAPROPHYTICUS

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TIP60 NEURO-EPIGENETIC MODULATORS

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ORGANIC COMPOUNDS

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PHARMACEUTICAL COMPOSITIONS

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Sustained Release Pharmaceutical Composition of Upadacitinib

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Certain Triazolopyridines and Triazolopyrazines, Compositions Thereof and Methods of Use Therefor

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COMBINATION OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE AND ITS DERIVATIVES WITH A JAK INHIBITOR

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COMPOUNDS FOR USE IN TREATING NEUROLOGICAL DISORDERS

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2-(INDAZOL-5-YL)-6-(PIPERIDIN-4-YL)-1,7-NAPHTHYRIDINE DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS FOR SPLICING NUCLEIC ACIDS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES

#333
20250092050
2025-03-20

1-AMINOBENZO[4,5]IMIDAZO[1,2-A]PYRAZINE-3-FORMAMIDE COMPOUND, AND PREPARATION THEREFOR AND USE THEREOF

#334
20250091989
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SMALL MOLECULE PROTEIN SYNTHESIS MODULATORS

#335
20250090543
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CXCR7 INHIBITORS FOR THE TREATMENT OF CANCER

#336
20250090534
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Phosphodiesterase-5 Inhibitor Combinations, Methods of Making, and Methods of Use Thereof

#337
20250090525
2025-03-20

Methods of Treating Cancers, Immune and Autoimmune Diseases, and Inflammatory Diseases Based on BTK Occupancy and BTK Resynthesis Rate

#338
20250090524
2025-03-20

BTK INHIBITORS

#339
20250084078
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FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#340
20250082648
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COMPOSITIONS AND METHODS FOR ENHANCING KRAS INHIBITOR OR SHP2 INHIBITOR EFFICACY

#341
20250082633
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COMPOUNDS AND METHODS FOR MODULATING SPLICING

#342
20250082631
2025-03-13

SLEEP IMPROVING AGENT

#343
20250082629
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ANTIPROLIFERATIVE COMPOUNDS AND SECOND ACTIVE AGENTS FOR COMBINED USE

#344
20250074913
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PYRAZOLE DERIVATIVES AS STING AGONISTS

#345
20250074911
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MACROCYCLIC BTK INHIBITORS

#346
20250074907
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INHIBITORS OF SARS-COV-2

#347
20250066473
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TREATMENT OF CANCER WITH COMBINATIONS OF IMMUNOREGULATORY AGENTS

#348
20250066389
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HETEROCYCLIC AMIDES AND METHODS OF USING THE SAME

#349
20250066368
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DNA POLYMERASE THETA INHIBITOR AND USE THEREOF

#350
20250066349
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CYCLIC COMPOUNDS AND THEIR USE FOR THE TREATMENT OF NEUROLOGICAL DISORDERS

#351
20250066344
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BENZOTHIAZOLE, BENZOISOXAZOLE, AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS

#352
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HETEROCYCLIC COMPOUNDS AS DYRK1A INHIBITORS

#353
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BACTERIAL COMPOSITIONS AND METHODS FOR TREATING CANCER AND IMMUNE DISEASES

#354
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USES OF DPP IV INHIBITORS

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CD73 INHIBITOR AND A2A/A2B ADENOSINE RECEPTOR INHIBITOR COMBINATION THERAPY

#356
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FUSED RING COMPOUND ACTING AS SHP2 INHIBITOR

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ARYLSULPHONAMIDE COMPOUNDS

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BICYCLIC HETEROCYCLIC COMPOUNDS USEFUL AS MONOACYLGLYCEROL LIPASE INHIBITORS

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Pharmaceutical Compounds and Compositions as C-Kit Kinase Inhibitors

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COMPOUNDS AND METHODS FOR MODULATING STAT3

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Intestine-Targeted Drug Delivery Compositions and Preparation Methods Thereof

#362
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POLYMORPH OF KRAS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF

#363
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PARP INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF

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TREATMENT OF NEUROLOGICAL DISORDERS

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METHODS OF TREATING ALOPECIA ARAETA

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POLYMORPH FORMS OF A 5H-PYRROLO[2,3-b]PYRAZINE DERIVATIVE, METHODS OF PREPARATION, AND USES THEREFORE

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HETEROCYCLIC SUBSTITUTED 1,3,4-THIADIAZOLE AND PYRIDAZINE COMPOUNDS AND METHODS OF USING THE SAME

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SOS1 Inhibitor With Pyrido-Fused Six-Membered Ring Structure

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Combination Therapy Comprising A2A/A2B and PD-1/PD-L1 Inhibitors

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BRUTON'S TYROSINE KINASE INHIBITORS AS ANTIVIRAL AGENTS

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Synergistic compositions for use in the treatment of cancer

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AN IGF1R INHIBITOR AND AN AKT INHIBITOR FOR USE IN THE TREATMENT OF CANCER

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REGULATING T CELL IMMUNE RESPONSE THROUGH IGF-I RECEPTOR (IGF-1R)

#374
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SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF

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NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE PARP INHIBITOR AND USE THEREOF

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PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

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BTK INHIBITORS

#378
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Compounds and Compositions as C-Kit Kinase Inhibitors

#379
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WRN INHIBITORS

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COMPOSITIONS AND METHODS FOR TREATING WITH A COMBINATION OF ALTERNATING ELECTRIC FIELDS AND DNA-DEPENDENT PROTEIN KINASE INHIBITORS

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TREATMENT OF HIDRADENITIS WITH JAK INHIBITORS

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APPLICATION OF IMIDAZO [1,2-A] PYRAZINE COMPOUNDS OR THEIR PHARMACEUTICALLY ACCEPTABLE SALTS IN THE PREPARATION OF ANTI-CORONAVIRUS DRUGS

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THERAPEUTIC TARGETS AND AGENTS FOR THE TREATMENT OF POSTTRAUMATIC STRESS DISORDER

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N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (THIAZOLYL)])(SUBSTITUTED)CARBOXAMIDE COMPOUNDS AND USE THEREOF FOR INHIBITING HUMAN POLYMERASE THETA

#385
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METHODS FOR TREATING ALZHEIMER DISEASE AND FOR REDUCING AMYLOID BETA FORMATION

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TREATMENT OF NEURODEGENERATIVE DISEASES VIA ADMINISTRATION OF BUNTANETAP AND A PHOSPHODIESTERASE INHIBITOR

#387
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COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES

#388
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PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF

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Antiviral Therapy

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PHARMACEUTICAL COMPOSITIONS

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PHARMACEUTICAL COMPOSITIONS

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PYRAZOLO FUSED RING COMPOUND AND USE THEREOF

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HPK1 ANTAGONISTS AND USES THEREOF

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Imidazo[1,2- a]pyrazine and Imidazo[1,2- a]pyridine Based Tyrosyl-DNA Phosphodiesterase I (TDP1) Inhibitors

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NOVEL COMPOSITIONS AND METHODS

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6-SUBSTITUTED INDOLE COMPOUNDS

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NITROGEN-CONTAINING COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

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NOVEL COMPOUND AND PHARMACEUTICAL COMPOSITION COMPRISING SAME

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USE OF GCN2 INHIBITORS IN TREATING CANCER

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COMBINATION THERAPIES FOR HIV INFECTIONS AND USES THEREOF

#401
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PARG INHIBITORY COMPOUNDS

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HETEROARYL COMPOUNDS USEFUL IN THE TREATMENT OF COGNITIVE DISORDERS

#403
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NITROGEN-CONTAINING TRICYCLIC COMPOUND AND PHARMACEUTICAL USE THEREOF

#404
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TETRAHYDRONAPTHYRIDINE AND RELATED ANALOGS FOR INHIBITING YAP/TAZ-TEAD

#405
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METHOD OF INJECTING DIHYDROERGOTAMINE INTO THE BODY

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NOVEL METHODS

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CONTINUOUS DELIVERY PREPARATION CAPABLE OF BEING STABLY RELEASED AND PREPARATION METHOD THEREFOR

#408
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BENZOPIPERAZINE AND RELATED ANALOGS FOR INHIBITING YAP/TAZ-TEAD

#409
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Solid Forms of Upadacitinib

#410
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NK3 modulators and uses thereof

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SUBSTITUTED TRIAZOLOHETEROARYL COMPOUNDS AS USP1 INHIBITORS AND THE USE THEREOF

#412
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COMPOUNDS AND METHODS FOR MODULATING SPLICING

#413
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NOVEL ENTEROCOCCUS FAECIUM LCM001 STRAIN, AND USE THEREOF

#414
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COMPOSITIONS FOR ENHANCING SEXUAL PLEASURE WITH REDUCED PHARMACEUTICAL LOAD OF PDE5 INHIBITOR

#415
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HETEROARYL DERIVATIVE PARP INHIBITOR AND USE THEREOF

#416
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2024-12-05

COMPOUNDS AND METHODS FOR MODULATING SPLICING

#417
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2024-12-05

Compounds, Compositions and Methods for Attenuation of Mammalian Translation of C-MYC or N-MYC Proteins of the MYC Proto-Oncogene Family of BHLH Transcription Factors

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NOVEL NANOPARTICLES OF ANTIRETROVIRAL DRUGS, THEIR PREPARATION AND THEIR USE FOR THE TREATMENT OF VIRAL INFECTIONS

#419
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THERAPEUTIC AGENT COMPOSITION AND METHOD OF USE, FOR TREATING, RELIEVING, OR ALLEVIATING ALZHEIMER'S DISEASE

#420
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HETEROARYL HETEROCYCLIC COMPOUNDS AND USES THEREOF

#421
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TREATING SPONDYLOARTHRITIC CONDITIONS WITH UPADACITINIB

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METHODS OF TREATING RBP4 RELATED DISEASES WITH TRIAZOLOPYRIDINES

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TREATMENT OF SCLERODERMA AND RAYNAUD'S SYNDROME

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INHIBITORS OF THE MTDH-SND1 PROTEIN COMPLEX FOR CANCER THERAPY

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Combination methods and compositions including sleep therapeutics for treating mood

#426
20240391937
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BICYCLIC DERIVATIVE PARP INHIBITOR AND USE THEREOF

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2024-11-28

TETRAHYDROTHIENO PYRIDINE DERIVATIVES AS DDRS INHIBITORS

#428
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METHIONINE ADENOSYLTRANSFERASE 2A INHIBITOR FOR TREATING MTAP DELETION-TYPE CANCER

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Substituted Quinoxalines

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CHIMERIC MODIFIED ION CHANNELS AND USES THEREOF FOR TREATMENT OF TRIGEMINAL NERVE DISORDERS

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2024-11-28

PHOSPHORYLATED TRISTETRAPROLIN AS A BIOMARKER AND THERAPEUTIC TARGET FOR ANTIAGING DRUGS

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INHIBITOR OF BTK AND MUTANTS THEREOF

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METHODS OF TREATING VITILIGO WITH UPADACITINIB

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IRHOM2 INHIBITORS AND USES THEREOF

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THIOPHENE RING COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#436
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AZAINDAZOLE MACROCYCLE COMPOUNDS AND USES THEREOF

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20240383906
2024-11-21

5-SUBSTITUTED PYRIDINE-2(1H)-KETONE COMPOUND AND USE THEREOF

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2024-11-21

SUBSTITUTED HYDANTOIN COMPOUNDS, METHODS FOR PREPARATION THEREOF AND USE THEREOF IN THE TREATMENT AND/OR PREVENTION OF A CORONA VIRUS DISEASE

#439
20240383868
2024-11-21

SMARCA DEGRADERS AND USES THEREOF

#440
20240376126
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PRMT5 INHIBITOR AND THE USE THEREOF

#441
20240376123
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KRAS G12D INHIBITORS AND USES THEREOF

#442
20240376115
2024-11-14

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#443
20240376110
2024-11-14

PRMT5 INHIBITORS AND USES THEREOF

#444
20240376090
2024-11-14

ISOXAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERED RELATED THERETO

#445
20240376056
2024-11-14

PHENYL ACETAMIDE BASED IL-17A MODULATORS AND USES THEREOF

#446
20240374627
2024-11-14

A PHARMACEUTICAL COMPOSITION COMPRISING COMBINATION OF SITAGLIPTIN AND EMPAGLIFLOZIN

#447
20240374586
2024-11-14

NOVEL METHODS

#448
20240374575
2024-11-14

METHODS AND COMPOSITIONS FOR TREATING CANCER

#449
20240374541
2024-11-14

ENGAGING THE CERVICAL SPINAL CORD CIRCUITRY TO RE-ENABLE VOLITIONAL CONTROL OF HAND FUNCTION IN TETRAPLEGIC SUBJECTS

#450
20240374527
2024-11-14

Pharmaceutical Composition Comprising Lumateperone

#451
20240368188
2024-11-07

Positive allosteric modulators of the muscarinic acetylcholine receptor M4

#452
20240368169
2024-11-07

SUBSTITUTED TRICYCLIC COMPOUNDS AS PARP INHIBITORS AND USE THEREOF

#453
20240366648
2024-11-07

NAD-AUGMENTATION THERAPY FOR PARKINSON'S DISEASE

#454
20240366582
2024-11-07

TREATMENT OF RAYNAUD'S DISEASE

#455
20240366511
2024-11-07

ORAL SOLID DOSE FORMULATIONS

#456
20240360154
2024-10-31

AROYL SUBSTITUTED TRICYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF

#457
20240358699
2024-10-31

METHOD OF REDUCING PULMONARY EXACERBATIONS IN RESPIRATORY DISEASE PATIENTS

#458
20240358693
2024-10-31

METHODS OF TREATING PAIN

#459
20240358692
2024-10-31

TREATMENT OF SCLERODERMA

#460
20240351997
2024-10-24

NOVEL PARP7 INHIBITOR AND USE THEREOF

#461
20240351986
2024-10-24

UREA COMPOUND CONTAINING 2-HETEROAROMATIC RING SUBSTITUTION, PREPARATION METHOD THEREFOR AND USE THEREOF

#462
20240350486
2024-10-24

Regimens for treating HIV infections and aids

#463
20240343726
2024-10-17

PYRROLOPYRIDINE-3- AND 4-CARBOXAMIDE COMPOSITIONS AND METHODS FOR CELLULAR PROLIFERATION

#464
20240343716
2024-10-17

COMPOUNDS FOR PREVENTING, INHIBITING, OR TREATING CANCER, AIDS AND/OR PREMATURE AGING

#465
20240342168
2024-10-17

SMALL MOLECULE INHIBITORS FOR ANTI-CANCER COMBINATION THERAPY

#466
20240342106
2024-10-17

NANOPARTICLES AND USES THEREOF FOR TREATMENT OF HUMAN IMMUNODEFICIENCY VIRUS

#467
20240336624
2024-10-10

PARP INHIBITOR CONTAINING PIPERAZINE STRUCTURE, PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF

#468
20240335455
2024-10-10

MITOFUSIN ACTIVATORS AND USES THEREOF

#469
20240327416
2024-10-03

Further Substituted Triazolo Quinoxaline Derivatives

#470
20240327412
2024-10-03

FACTOR XIIA INHIBITORS

#471
20240327411
2024-10-03

SIRT6 ACTIVATORS

#472
20240327407
2024-10-03

NOVEL INHIBITORS OF AUTOTAXIN

#473
20240327364
2024-10-03

THERAPEUTIC TARGETING OF GPR68 TO INDUCE FERROPTOSIS

#474
20240325311
2024-10-03

ORAL COMPLEX TABLET COMPRISING SITAGLIPTIN, DAPAGLIFLOZIN, AND METFORMIN

#475
20240317770
2024-09-26

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#476
20240317767
2024-09-26

PYRAZOLE DERIVATIVES USEFUL AS 5-LIPOXYGENASE ACTIVATING PROTEIN (FLAP) INHIBITORS

#477
20240317764
2024-09-26

SALTS AND SOLID FORMS OF A COMPOUND HAVING APJ RECEPTOR ACTIVITY

#478
20240317756
2024-09-26

INHIBITORS OF BRUTON'S TYROSINE KINASE

#479
20240317735
2024-09-26

HYDROISOQUINOLINE OR HYDRONAPHTHYRIDINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE

#480
20240317721
2024-09-26

PYRAZOLYL DERIVATIVES AS INHIBITORS OF THE KRAS MUTANT PROTEIN

#481
20240316047
2024-09-26

Inhibitors of RNA helicase DHX9 and uses thereof

#482
20240316042
2024-09-26

METHODS OF TREATING PEDIATRIC PATIENTS WITH UPADACITINIB

#483
20240316041
2024-09-26

PROCESS FOR THE PREPARATION OF SITAGLIPTIN FREE FROM GENOTOXIC IMPURITIES

#484
20240316040
2024-09-26

EXTENDED RELEASE UPADACITINIB FORMULATIONS

#485
20240316034
2024-09-26

Chemokine CXCR4 Receptor Modulators and Uses Related Thereto

#486
20240315994
2024-09-26

SMALL MOLECULE MODULATORS OF FERROPTOSIS

#487
20240315978
2024-09-26

PHARMACEUTICAL COMPOSITIONS COMPRISING ACALABRUTINIB

#488
20240309006
2024-09-19

NOVEL BICYCLIC COMPOUNDS

#489
20240309003
2024-09-19

HETEROCYCLIC COMPOUNDS AS TRIGGERING RECEPTOR EXPRESSED ON MYELOID CELLS 2 AGONISTS AND METHODS OF USE

#490
20240308992
2024-09-19

DRAK2 INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#491
20240307387
2024-09-19

Pharmaceutical compositions

#492
20240307386
2024-09-19

NOVEL METHODS

#493
20240307382
2024-09-19

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#494
20240299538
2024-09-12

AGENT FOR USE IN THE TREATMENT OF GLIOMA

#495
20240299397
2024-09-12

REHYDRATION COMPOSITION AND METHOD OF USE

#496
20240299396
2024-09-12

Liquid oral formulations for tadalafil

#497
20240299380
2024-09-12

APPLICATION OF COMPOUND IN PREPARATION OF DRUG FOR TREATING MYELOFIBROSIS AND RELATED SYMPTOMS/SIGNS THEREOF, AND USE OF COMPOUND

#498
20240299357
2024-09-12

PHARMACEUTICAL COMBINATION, COMPOSITION AND COMPOUND PREPARATION COMPRISING GLUCOKINASE ACTIVATOR AND DPP-IV INHIBITOR, AND PREPARATION METHOD AND USE THEREOF

#499
20240294530
2024-09-05

MULTI-CYCLIC IRAK AND FLT3 INHIBITING COMPOUNDS AND USES THEREOF

#500
20240294524
2024-09-05

HETEROCYCLIC COMPOUNDS USEFUL AS PDK1 INHIBITORS

#501
20240294523
2024-09-05

HETEROCYCLIC LACTAM COMPOUND, AND PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF

#502
20240293489
2024-09-05

PLANT EXTRACTS WITH ANTI-DIABETIC AND OTHER USEFUL ACTIVITIES

#503
20240293444
2024-09-05

PHARMACEUTICAL COMPOSITION

#504
20240287094
2024-08-29

NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINES

#505
20240287093
2024-08-29

HIGH ACTIVITY STING PROTEIN AGONIST

#506
20240287070
2024-08-29

FUSED HETEROCYCLIC DERIVATIVES

#507
20240285820
2024-08-29

Intratumoral Alpha-Emitter Radiation in Combination with Immune Checkpoint Regulators

#508
20240285645
2024-08-29

MODULATORS OF TOLL-LIKE RECEPTORS FOR THE TREATMENT OF HIV

#509
20240285619
2024-08-29

Oral gliptin compositions and method for preparation thereof

#510
20240285618
2024-08-29

PHARMACEUTICAL COMPOSITIONS OF LUMATEPERONE

#511
20240285617
2024-08-29

Heterocyclic derivatives useful as SHP2 inhibitors

#512
20240285611
2024-08-29

APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES

#513
20240285572
2024-08-29

COMPOSITIONS COMPRISING NITRIC OXIDE-RELEASING COMPOUNDS FOR TREATING CHOROIDAL VASCULAR DISEASES AND METHODS OF THEIR USE

#514
20240279238
2024-08-22

POLYCYCLIC CARBAMOYLPYRIDONE DERIVATIVE HAVING HIV INTEGRASE INHIBITORY ACTIVITY

#515
20240279237
2024-08-22

FUSED BICYCLIC HETEROARYL COMPOUNDS USEFUL AS NLRP3 INHIBITORS

#516
20240279228
2024-08-22

NOVEL SALTS AND CRYSTALS

#517
20240279227
2024-08-22

FUSED HETEROCYCLIC DERIVATIVES

#518
20240277705
2024-08-22

DOSAGE REGIMENS FOR ECUBECTEDIN

#519
20240270756
2024-08-15

Integrase Inhibitor and Use Thereof

#520
20240270747
2024-08-15

HETEROARYL PYRIDONE AND AZA-PYRIDONE COMPOUNDS

#521
20240270741
2024-08-15

COMPOUNDS FOR FGFRS INHIBITORS

#522
20240269329
2024-08-15

GENE THERAPY FOR DUCHENNE MUSCULAR DYSTROPHY

#523
20240269194
2024-08-15

COMPOSITIONS AND METHODS FOR ISLET CELL TRANSPLANTS

#524
20240262835
2024-08-08

PRMT5 inhibiting compounds and uses thereof

#525
20240262832
2024-08-08

SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF

#526
20240262826
2024-08-08

Wild type kit inhibitors

#527
20240262821
2024-08-08

PKC-Theta Modulators

#528
20240261436
2024-08-08

GENE EDITING THERAPY FOR HIV INFECTION VIA DUAL TARGETING OF HIV GENOME AND CCR5

#529
20240254139
2024-08-01

FUSED ISOXAZOLYL COMPOUNDS AS KAT6A INHIBITORS

#530
20240254136
2024-08-01

COMPOUNDS TARGETING RNA-BINDING PROTEINS OR RNA-MODIFYING PROTEINS

#531
20240254134
2024-08-01

AGELASTATIN A DERIVATIVES AND RELATED METHODS

#532
20240254131
2024-08-01

NOVEL HETEROCYCLIC COMPOUNDS, COMPOSITIONS, METHODS OF PREPARATION AND USES THEREOF

#533
20240252491
2024-08-01

NOVEL METHODS

#534
20240252490
2024-08-01

Combination Therapies Comprising Kras Inhibitors and SPH2 Inhibitors

#535
20240252489
2024-08-01

REPEATED ADMINISTRATION OF DIHYDROERGOTAMINE FOR TREATMENT OF FREQUENT MIGRAINE HEADACHES

#536
20240246992
2024-07-25

MACROCYCLIC LRRK2 KINASE INHIBITORS

#537
20240246984
2024-07-25

HETEROCYCLIC JAK INHIBITOR

#538
20240246969
2024-07-25

HETEROCYCLIC DERIVATIVES AS CAMKK2 INHIBITORS

#539
20240246968
2024-07-25

SMALL MOLECULE INHIBITORS OF KRAS G12C MUTANT

#540
20240246952
2024-07-25

SMALL MOLECULE MODULATORS OF GLUCOCEREBROSIDASE ACTIVITY AND USES THEREOF

#541
20240245806
2024-07-25

TREATMENT OF NEURODEGENERATIVE DISEASE USING CSA- AND INDY-TYPE COMPOUNDS

#542
20240245716
2024-07-25

ADENOSINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME

#543
20240245689
2024-07-25

Liquid oral formulations for sildenafil

#544
20240245688
2024-07-25

LIQUID ORAL FORMULATIONS FOR TADALAFIL

#545
20240245685
2024-07-25

PHOSPHODIESTERASE-5 INHIBITOR COMBINATIONS, METHODS OF MAKING, AND METHODS OF USE THEREOF

#546
20240245681
2024-07-25

HETEROCYCLIC DERIVATIVES USEFUL AS SHP2 INHIBITORS

#547
20240245610
2024-07-25

NOVEL METHODS

#548
20240245547
2024-07-25

INTRAVAGINAL RING DEVICES

#549
20240239811
2024-07-18

5-(5-(PIPERIDIN-4-YL)THIENO[3,2-C]PYRAZOL-2-YL]INDAZOLE DERIVATIVES AND RELATED COMPOUNDS AS MODULATORS FOR SPLICING NUCLEIC ACIDS AND FOR THE T

#550
20240238286
2024-07-18

COMPOSITIONS FOR USE IN THE PREVENTION AND/ OR TREATMENT OF INTELLECTUAL DISABILITY AND NEURODEGENERATIVE DISEASES IN A SUBJECT WITH DOWN SYNDROME

#551
20240238285
2024-07-18

POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE

#552
20240238259
2024-07-18

COMBINATION THERAPY FOR PULMONARY HYPERTENSION

#553
20240228506
2024-07-11

RIPK1 INHIBITORS AND METHODS OF USE

#554
20240228501
2024-07-11

IMIDAZOLE-CONTAINING CONDENSED RING DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF IN MEDICINE

#555
20240228497
2024-07-11

Pyrrolo[2, 3-b]Pyrazine-Based Bifunctional Compounds as HPK1 Degraders and the Use Thereof

#556
20240228491
2024-07-11

METHIONINE ADENOSYLTRANSFERASE INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#557
20240226097
2024-07-11

METHODS OF CANCER TREATMENT USING A COMBINATION OF BTK INHIBITORS AND PI3 KINASE INHIBITORS

#558
20240226035
2024-07-11

Precision Medicine Approach to Treating Parkinson's Disease with a Monoamine Oxidase Inhibitor, an Antioxidant, or Both

#559
20240226002
2024-07-11

SOFT CHEWABLE FORMULATIONS WITH ACTIVE INGREDIENTS

#560
20240217967
2024-07-04

INDOLINE DERIVATIVES AS DDRS INHIBITORS

#561
20240217951
2024-07-04

PCSK9 INHIBITORS AND METHODS OF USE THEREOF

#562
20240216476
2024-07-04

COMBINATION OF BITTER RECEPTOR AGONIST AND GUT-SIGNALING COMPOUND

#563
20240216383
2024-07-04

FORMULATIONS AND METHODS FOR TREATING ERECTILE DYSFUNCTION

#564
20240216380
2024-07-04

BTK Inhibitors to Treat Solid Tumors Through Modulation of the Tumor Microenvironment

#565
20240216368
2024-07-04

Pharmaceutical capsules comprising lumateperone mono-tosylate

#566
20240216367
2024-07-04

TREATING SPONDYLOARTHRITIC AND PSORIATIC CONDITIONS WITH UPADACITINIB

#567
20240216357
2024-07-04

POLYCYCLIC COMPOUND AND APPLICATION THEREOF

#568
20240216330
2024-07-04

COMBINATION TREATMENT METHODS OF MULTIPLE SCLEROSIS

#569
20240208993
2024-06-27

Five- and six-membered compound, and preparation method therefor and pharmaceutical composition and use thereof

#570
20240208974
2024-06-27

NOVEL COMPOUNDS AND METHODS

#571
20240208970
2024-06-27

SUBSTITUTED HYDANTOIN COMPOUNDS, METHODS FOR PREPARATION THEREOF AND USE THEREOF IN THE TREATMENT AND/OR PREVENTION OF A CORONA VIRUS DISEASE

#572
20240208942
2024-06-27

METAP-2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS AND THERAPEUTIC METHODS THEREOF

#573
20240207300
2024-06-27

COMBINATION THERAPIES INCLUDING MYT1 INHIBITORS

#574
20240207273
2024-06-27

TREATMENT OF AUTISM SPECTRUM DISORDERS, OBSESSIVE-COMPULSIVE DISORDER AND ANXIETY DISORDERS

#575
20240207259
2024-06-27

NOVEL METHODS

#576
20240199622
2024-06-20

Crystal Forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)-pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide

#577
20240199620
2024-06-20

CHEMOKINE RECEPTOR MODULATORS AND USES THEREOF

#578
20240199610
2024-06-20

TYK2 INHIBITORS AND USES THEREOF

#579
20240199584
2024-06-20

KRAS INHIBITORS

#580
20240199554
2024-06-20

Inhibitors of receptor interacting protein kinase I for the treatment of disease

#581
20240197744
2024-06-20

TREATING SEX STEROID DEPENDENT CANCER WITH BMX INHIBITORS

#582
20240197742
2024-06-20

Therapeutic Combinations of a CD19 Inhibitor and a BTK Inhibitor

#583
20240190887
2024-06-13

COMPOUND USED AS SHP2 INHIBITOR AND USE THEREOF

#584
20240190864
2024-06-13

Bruton's Tyrosine Kinase (BTK) INHIBITOR AND APPLICATION THEREOF

#585
20240189320
2024-06-13

HIGHLY ACTIVE STING PROTEIN AGONIST COMPOUND

#586
20240189309
2024-06-13

TYK2 INHIBITORS AND USES THEREOF

#587
20240182495
2024-06-06

ANTIBACTERIAL COMPOUNDS

#588
20240182477
2024-06-06

HETEROCYCLIC COMPOUNDS AS TRIGGERING RECEPTOR EXPRESSED ON MYELOID CELLS 2 AGONISTS AND METHODS OF USE

#589
20240182468
2024-06-06

COMPOUNDS FOR THE ACTIVATION OF AMPK

#590
20240181066
2024-06-06

Anti-cancer nuclear hormone receptor-targeting compounds

#591
20240180924
2024-06-06

BCL-2 INHIBITORS

#592
20240180913
2024-06-06

THE THERAPEUTIC REGIMEN

#593
20240180904
2024-06-06

Methods of treating chronic lymphocytic leukemia and small lymphocytic leukemia using a BTK inhibitor

#594
20240180903
2024-06-06

INJECTABLE PHARMACEUTICAL COMPOSITION, PREPARATION METHOD THEREFOR AND USE THEREOF

#595
20240180880
2024-06-06

METHODS OF USING EHMT2 INHIBITORS IN TREATING OR PREVENTING BLOOD DISORDERS

#596
20240174682
2024-05-30

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#597
20240173318
2024-05-30

DRY EYE TREATMENTS

#598
20240173208
2024-05-30

PRESERVATIVE REMOVAL FROM EYE DROPS

#599
20240166657
2024-05-23

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#600
20240166648
2024-05-23

Novel Crystalline Form Of 1-(8-Bromopyrido[2,3-E][1,2,4]triazolo[4,3-A]pyrazin-4-Yl)-Nmethylazetidin-3-Amine Hydrogen Sulfate Monohydrate