ClassID:

90494

C07B2200/13 - page 13 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#3601
20190135848
2019-05-09

Amine solvate of sodium-glucose linked transporter inhibitor, and preparation method and application thereof

#3602
20190135846
2019-05-09

Crystal of 3'-sialyllactose sodium salt n-hydrate, and process for producing same

#3603
20190135831
2019-05-09

POLYMORPHIC FORMS ALPHA, BETA AND GAMMA OF RIFAXIMIN

#3604
20190135830
2019-05-09

PHARMACEUTICAL COMPOSITIONS COMPRISING POLYMORPHIC FORMS ALPHA, BETA, AND GAMMA OF RIFAXIMIN

#3605
20190135806
2019-05-09

Solid state forms of Venetoclax and processes for preparation of Venetoclax

#3606
20190135792
2019-05-09

Crystalline form of compound suppressing protein kinase activity, and application thereof

#3607
20190135787
2019-05-09

PYRIMIDINE COMPOSITIONS, ULTRA-PURE COMPOSITIONS AND SALTS THEREOF, METHODS OF MAKING THE SAME, AND METHODS OF USING THE SAME FOR TREATING HISTAMINE H4 RECEPTOR (H4) MEDIATED DISEASES AND CONDITIONS

#3608
20190135779
2019-05-09

Crystals of quinazoline derivative and preparation method therefor

#3609
20190135755
2019-05-09

CRYSTAL POLYMORPHISM OF KCNQ2-5 CHANNEL ACTIVATOR

#3610
20190135732
2019-05-09

Crystal forms and methods of synthesis of (2R, 6R)-hydroxynorketamine and (2S, 6S)-hydroxynorketamine

#3611
20190135719
2019-05-09

Method for the continuous manufacture of bisphenol A

#3612
20190134038
2019-05-09

Salt of fused heterocyclic derivative and crystal thereof

#3613
20190127417
2019-05-02

Crystalline polymorph of 15B-hydroxy-osaterone acetate

#3614
20190127416
2019-05-02

Squalamine solid forms and methods of making the same

#3615
20190127404
2019-05-02

TH-302 solid forms and methods related thereto

#3616
20190127369
2019-05-02

Process for preparing (4S)- 4-(4-cyano-2-methoxyphenyl)-5-ethoxy-2,8-dimethyl-1,4-dihydro-1,6-naphthyridine-3-carboxamide and purification thereof for use as a pharmaceutical active ingredient

#3617
20190127364
2019-05-02

Pyrimidine compound as JAK kinase inhibitor

#3618
20190127334
2019-05-02

Polymorphic form of crystalline rosuvastatin calcium and novel processes for crystalline as well as amorphous rosuvastatin calcium

#3619
20190119310
2019-04-25

Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use

#3620
20190119306
2019-04-25

Process for the preparation of tavaborole, its novel polymorphic forms and the polymorphs thereof

#3621
20190119287
2019-04-25

Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines and substituted imidazo[1,2-b]pyridazines as PI3K-gamma inhibitors

#3622
20190119262
2019-04-25

Crystal form of brexpiprazole and preparation method therefor

#3623
20190119253
2019-04-25

Crystalline forms and compositions of CFTR modulators

#3624
20190119226
2019-04-25

Crystalline form E of tafamidis meglumine, process for preparation and use thereof

#3625
20190117662
2019-04-25

Therapeutically active compounds and their methods of use

#3626
20190117536
2019-04-25

Oral care composition zinc-lysine complex

#3627
20190112327
2019-04-18

Crystal form of fludarabine phosphate, preparation method therefor, and application thereof

#3628
20190112313
2019-04-18

Salts of TAM inhibitors

#3629
20190112310
2019-04-18

Co-crystals of 1-(4-fluoro-phenyl)-4-((6bR,1OaS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H- pyrido[3′,4′:4,51_pyrrolo [1,2,3-delqcuinoxalin-8-yl)-butan-1-one with nicotinamide or isonicotinamide

#3630
20190112309
2019-04-18

Salts and crystals of ITI-007

#3631
20190112304
2019-04-18

Treatment of osteoarthritis

#3632
20190112277
2019-04-18

Process for the preparation of diphenylpyrazine derivatives

#3633
20190112270
2019-04-18

Polymorphic form of N-{6-(hydroxypropan-2-yl)-2-[2-(methylsulphonyl)ethyl]-2H-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide

#3634
20190106421
2019-04-11

Pharmaceutical forms of diazabicyclooctane derivatives and manufacturing method thereof

#3635
20190106410
2019-04-11

Plinabulin compositions

#3636
20190106408
2019-04-11

Method for preparing the anhydrous crystalline form of isoniazid-derived hydrazone, thus produced crystalline polymorph of the anyhydrous form, use thereof for the treatment of alzheimer's disease, parkinsonism and other neurodegenerative disorders, and pharamceutical composition

#3637
20190106407
2019-04-11

Synthesis of indazoles

#3638
20190106405
2019-04-11

Solid forms of 2-(4-chlorophenyl)-N-((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-5-yl)methyl)-2,2-difluoroacetamide, and their pharmaceutical compositions and uses

#3639
20190106404
2019-04-11

Process for synthesizing 2-hydroxy-6-((2-(1-isopropyl-1H-pyrazol-5-yl)-pyridin-3-yl)methoxy)benzaldehyde

#3640
20190106402
2019-04-11

Physical form of a SGR modulator

#3641
20190106401
2019-04-11

COFORMER SALTS OF (2S,3S)-METHYL 7-FLUORO-2-(4-FLUOROPHENYL)-3-(1-METHYL-1H-1,2,4-TRIAZOL-5-YL)-4-OXO-1,2,3,4-TETRAHYDROQUINOLINE-5-CARBOXYLATE AND METHODS OF PREPARING THEM

#3642
20190106389
2019-04-11

NOVEL FORMS OF APREMILAST

#3643
20190105390
2019-04-11

Formulations of a PI3K/mTOR-inhibitor for intravenous administration

#3644
20190100550
2019-04-04

Polymorphic forms of sofosbuvir

#3645
20190100542
2019-04-04

Crystal form of tenofovir alafenamide salt, preparation method and use thereof

#3646
20190100529
2019-04-04

Polymorph of DPPIV inhibitor maleate and preparation method therefor

#3647
20190100519
2019-04-04

HYDROCHLORIDE SALT CRYSTAL OF DRUG FOR TREATING OR PREVENTING JAK-ASSOCIATED DISEASE AND PREPARATION METHOD THEREOF

#3648
20190100513
2019-04-04

Crystalline form of (2S,3S,6S,7R,10R,E)-7,10-dihydroxy-3,7-dimethyl-12-oxo-2-((R,2E,4E)-6-(piridin-2-yl)hepta-2,4-dien-2-yl)oxacyclododec-4-en-6-yl-4-methylpiperazine-1-carboxylate and methods of use thereof

#3649
20190100512
2019-04-04

SOLID FORMS COMPRISING (1E, 4E)-2-AMINO-N,N-DIPROPYL-8-(4-(PYRROLIDINE-1-CARBONYL)PHENYL)-3H-BENZO[B]AZEPINE-4-CARBOXAMIDE, COMPOSITIONS THEREOF, AND USES THEREOF

#3650
20190100498
2019-04-04

CRYSTALLINE FORM

#3651
20190092792
2019-03-28

VINORELBINE MONOTARTRATE AND ITS PHARMACEUTICAL USE

#3652
20190092773
2019-03-28

Crystalline forms of diazabicyclooctane derivatives and production process thereof

#3653
20190092766
2019-03-28

Crystalline forms of (3-Amino-oxetan-3-ylmethyl)-[2-(5,5-dioxo-5,6,7,9-tetrahydro-5lambda*6*-thia-8-aza-benzocyclohepten-8-yl)-6-methyl-quinazolin-4-yl]-amine

#3654
20190092753
2019-03-28

Crystalline forms of mesylate salt of pyridinyl amino pyrimidine derivative, preparation methods therefor, and applications thereof

#3655
20190092748
2019-03-28

Crystalline 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione hemihydrate, compositions and methods of use thereof

#3656
20190092747
2019-03-28

Crystalline 4-amino-2-(2,6-dioxopiperidine-3-YL)isoindoline-1,3-dione monohydrate, compositions and methods of use thereof

#3657
20190092734
2019-03-28

Crystalline form of Eluxadoline

#3658
20190085009
2019-03-21

Crystal forms of beta-nicotinamide mononucleotide

#3659
20190084963
2019-03-21

Solid forms of an HIV capsid inhibitor

#3660
20190084935
2019-03-21

Polymorph of pimavanserin tartrate and preparation method thereof and use of same

#3661
20190083511
2019-03-21

Enzymatic process for obtaining 17 alpha-monoesters of cortexolone and/or its 9,11-dehydroderivatives

#3662
20190077810
2019-03-14

Crystalline forms of therapeutic compounds and uses thereof

#3663
20190077791
2019-03-14

EGFR inhibitor free base or acid salt polycrystalline form, preparation method therefor, and application

#3664
20190077775
2019-03-14

Process for the preparation of Trisodium (4- {[1S,3R)-1-([1,1′-biphenyl]-4-ylmethyl)-4-ethoxy-3-methyl-4-oxobutyl]amino}-4-oxobutanoate)-(N-petanoyl-N-{[2′-(1H-tetrazol-1-1D-5-yl)[1,1′-biphenyl]-4-yl]methyl}- L-valinate) and its polymorphs thereof

#3665
20190077747
2019-03-14

Chlorhexidine crystal forms and uses thereof in medicine

#3666
20190071449
2019-03-07

Solid state forms of spiro-oxindole compounds

#3667
20190071442
2019-03-07

Crystal forms of palbociclib, and preparation method and use therefor

#3668
20190071440
2019-03-07

Indazole inhibitors of the Wnt signal pathway and therapeutic uses thereof

#3669
20190071426
2019-03-07

Solid state forms of Nilotinib salts

#3670
20190071414
2019-03-07

Crystalline 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione dihydrate, compositions and methods of use thereof

#3671
20190071402
2019-03-07

Solid forms of 2-(5-(4-(2-morpholinoethoxy)phenyl)pyridin-2-yl)-N-benzylacetamide

#3672
20190070162
2019-03-07

Solid forms of N-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide

#3673
20190064785
2019-02-28

Method and system for transporting inventory items

#3674
20190062346
2019-02-28

Method for producing 7h-pyrrolo[2, 3-d]pyrimidine derivative and intermediate thereof

#3675
20190062295
2019-02-28

Process for the preparation of optically active Beraprost

#3676
20190062263
2019-02-28

Crystalline Forms of (-)-(1R,2R)-3-(3-dimethylamino-1-ethyl-2-methylpropyl)-phenol hydrochloride

#3677
20190060274
2019-02-28

D-proline derivatives as SAP depleting agent

#3678
20190055263
2019-02-21

Polymorphic form of TG02

#3679
20190055255
2019-02-21

Crystalline forms of (6-(1H-indazol-6-yl)-N-[4-(4-(4-morpholinyl)phenyl]imidazo[1,2-A]pyrazin-8-amine) methanesulfonate

#3680
20190055237
2019-02-21

Crystalline forms of a FGFR inhibitor and processes for preparing the same

#3681
20190055197
2019-02-21

Crystalline modifications of methyl (3Z)-3-{[(4-{methyl[(4-methylpiperazin-1-yl)acetyl]amino}phenyl)amino](phenyl)methylidene}-2-oxo-2,3-dihydro-1H-indole-6-carboxylate salts and methods of preparation thereof

#3682
20190048023
2019-02-14

Crystal of compound having JAK-inhibiting activity

#3683
20190048010
2019-02-14

Mercaptopurine hemihydrate

#3684
20190047996
2019-02-14

Crystalline forms

#3685
20190047994
2019-02-14

Anhydrate-free polymorphically pure micronized crystalline brexpiprazole di-hydrate for use in intramuscular injectable sustained release formulations

#3686
20190047983
2019-02-14

Modified process for the preparation of Ceritinib and amorphous form of Ceritinib

#3687
20190047956
2019-02-14

Trans-isomeric heterocyclic compounds and preparation thereof

#3688
20190047953
2019-02-14

Crystalline form of 1-(5-(2,4-difluorophenyl)-1-((3-fluorophenyl)sulfonyl)-4-methoxy-1H-pyrrol-3-yl)-N-methylmethanamine salt

#3689
20190046534
2019-02-14

Salts of the Janus kinase inhibitor (R)-3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-cyclopentylpropanenitrile

#3690
20190040228
2019-02-07

Zinc oxide complexes

#3691
20190040096
2019-02-07

CRYSTALLINE FORMS OF A MACROLIDE, AND USES THEREFOR

#3692
20190040092
2019-02-07

Crystalline forms of ethyl ((S)-((((2R,5R)-5-(6-amino-9H-purin-9-yl)-4-fluoro-2,5-dihydrofuran-2-yl)oxy)methyl)(phenoxy)phosphoryl(-L-alaninate

#3693
20190040071
2019-02-07

Crystal form A of 2-butoxy-7-(4-(pyrrolidin-1-ylmethyl)benzyl)-5H-pyrrolo[3,2-D] pyrimidin-4-amine, preparation process and use thereof

#3694
20190040043
2019-02-07

Pyrazolo and triazolo bicyclic compounds as JAK kinase inhibitors

#3695
20190040015
2019-02-07

Sodium salt of uric acid transporter inhibitor and crystalline form thereof

#3696
20190040014
2019-02-07

Solid forms of an S-Nitrosoglutathione reductase inhibitor

#3697
20190040002
2019-02-07

CRYSTALLINE SALTS OF (4S,4AS,5AR,12AS)-4-DIMETHYLAMINO-3,10,12,12A-TETRAHYDROXY-7-[(METHOXY(METHYL)AMINO)-METHYL]-1,11-DIOXO-1,4,4A,5,5A,6,11,12A-OCTAHYDRO-NAPHTHACENE-2-CARBOXYLIC ACID AMIDE AND METHODS OF USING THE SAME

#3698
20190038607
2019-02-07

CHEMICAL COMPOUNDS

#3699
20190031687
2019-01-31

Polymorphs

#3700
20190031678
2019-01-31

Salt form of DPPIV inhibitor and preparation method thereof

#3701
20190031674
2019-01-31

Quantification and preparation of pharmaceutical grade cantharidin

#3702
20190031666
2019-01-31

TLR7 agonist trifluoroacetate salt and crystalline form B thereof, preparation methods and uses

#3703
20190031659
2019-01-31

Processes for producing diazabicyclooctane compounds

#3704
20190031654
2019-01-31

Formulations of a compound modulating kinases

#3705
20190030000
2019-01-31

Pharmaceutical composition comprising sacubitril and valsartan

#3706
20190023719
2019-01-24

Substituted tetrahydrocarbazole and carbazole carboxamide compounds

#3707
20190023718
2019-01-24

Polymorphs of dolutegravir and salts thereof

#3708
20190023714
2019-01-24

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-alpha]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#3709
20190023693
2019-01-24

Solid forms of Selinexor and process for their preparation

#3710
20190023655
2019-01-24

Solid state forms of N-[2-[(1S)-1-(3-ethoxy-4-methoxyphenyl)-2-(methylsulfonyl)ethyl]-2,3-dihydro-1,3-dioxo-1H-isoindol-4-yl]acetamide and process for preparation thereof

#3711
20190022080
2019-01-24

Crystalline forms of a prolyl hydroxylase inhibitor

#3712
20190016737
2019-01-17

Mechanically interlocked air-stable radicals

#3713
20190016729
2019-01-17

Process for making beta 3 agonists and intermediates

#3714
20190016725
2019-01-17

Forms of a PI3K delta selective inhibitor for use in pharmaceutical formulations

#3715
20190016718
2019-01-17

Salts of morpholine derivative, crystal forms thereof, processes for producing the same, pharmaceutical compositions including the same, and use thereof

#3716
20190016661
2019-01-17

Powdery 1,4-cyclohexanedicarboxylic acid

#3717
20190015420
2019-01-17

CRYSTALLINE FORMS OF (2R,5S,13AR)-8-HYDROXY-7,9-DIOXO-N-(2,4,6-TRIFLUOROBENZYL)-2,3,4,5,7,9,13,13A-OCTAHYDRO-2,5-METHANOPYRIDO[1',2':4,5]PYRAZINO[2,1-B][1,3]OXAZEPINE-10-CARBOXAMIDE

#3718
20190015337
2019-01-17

Formulations, methods, kit, and dosage forms for improved stability of an active pharmaceutical ingredient

#3719
20190010161
2019-01-10

Crystalline form of BTK kinase inhibitor and preparation method thereof

#3720
20190010160
2019-01-10

Salt of quinolone compound, polymorphs thereof, preparation method therefor, composition, and applications

#3721
20190010147
2019-01-10

Process for making crystalline form a of gefitinib

#3722
20190010142
2019-01-10

Crystalline forms of 1-(4-{[6-amino-5-(4-phenoxy-phenyl)-pyrimidin-4-ylamino]-methyl}-piperidin-1-yl)-propenone

#3723
20190010123
2019-01-10

Process for the preparation of apremilast

#3724
20190002483
2019-01-03

Crystalline forms

#3725
20190002471
2019-01-03

Crystalline Form Of Ticagrelor

#3726
20190002468
2019-01-03

Crystalline forms of ibrutinib

#3727
20190002461
2019-01-03

Polymorph of Riociguat and its process for the preparation

#3728
20190002449
2019-01-03

Crystallization procedure for obtaining canagliflozin hemihydrate crystals

#3729
20190002444
2019-01-03

CRYSTALLINE FORMS OF VILAZODONE HYDROCHLORIDE AND VILAZODONE FREE BASE

#3730
20190002434
2019-01-03

Crystals of quinazoline derivative and preparation method therefor

#3731
20190002421
2019-01-03

Process and novel polymorphic form of vortioxetine and its pharmaceutically acceptable salts

#3732
20190002416
2019-01-03

Crystalline(2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-bipheny]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2-methylpentanoic acid and uses thereof

#3733
20190002405
2019-01-03

Preparation of latanoprostene bunod of desired, pre-defined quality by gravity chromatography

#3734
20180371002
2018-12-27

Crystalline form A of rebaudioside D, and preparation method and application therefor

#3735
20180370980
2018-12-27

Crystal form of substituted aminopyran derivativek

#3736
20180370960
2018-12-27

Solid Oral Formulations and Crystalline Forms of an Inhibitor of Apoptosis Protein

#3737
20180370951
2018-12-27

Therapeutically active compounds and their methods of use

#3738
20180370948
2018-12-27

P-TOLUENESULFONATE FOR MEK KINASE INHIBITOR, METHOD OF PREPARATION THEREOF, AND METHOD OF USE THEREOF

#3739
20180370926
2018-12-27

PROCESS OF PREPARING TYROSINE KINASE INHIBITOR

#3740
20180370902
2018-12-27

Solabegron zwitterion and uses thereof

#3741
20180370901
2018-12-27

Gamma-aminobutyric acid hemihydrate crystal and preparation method thereof

#3742
20180368407
2018-12-27

2-(3-ethanesulfonylpyridine-2-yl)-5-(trifluoromethanesulfonyl) benzoxazole crystal

#3743
20180362580
2018-12-20

CRYSTALLINE AND AMORPHOUS FORMS OF CARFILZOMIB

#3744
20180362536
2018-12-20

Crystalline forms of a Bruton's tyrosine kinase inhibitor

#3745
20180362535
2018-12-20

Crystalline forms of a Bruton's tyrosine kinase inhibitor

#3746
20180362534
2018-12-20

CRYSTALLINE FORMS OF A BRUTON'S TYROSINE KINASE INHIBITOR

#3747
20180362529
2018-12-20

Solid forms of (1S,4S)-4-(2-(((3S,4R)-3-fluorotetrahydro-2H-pyran-4-yl)amino)-8-((2,4,6-trichlorophenyl)amino)-9H-purin-9-yl)-1-methylcyclohexane-1-carboxamide and methods of their use

#3748
20180362523
2018-12-20

Process for the preparation of aclidinium bromide

#3749
20180362522
2018-12-20

Inhibiting agents for Bruton's tyrosine kinase

#3750
20180362498
2018-12-20

Forms and compositions of an ERK inhibitor

#3751
20180362459
2018-12-20

Method of preparing (3R,4S)-3-acetamido-4-allyl-N-(tert-butyl)pyrrolidine-3-carboxamide

#3752
20180362444
2018-12-20

Process for the preparation of enclomiphene citrate having needle shaped crystal habit

#3753
20180362427
2018-12-20

Crystalline polymorphs of 1,6-dibromo-1,6-dideoxy-dulcitol

#3754
20180354974
2018-12-13

Crystalline solvate comprising 3-((1R,3s,5S)-3-((7-((5-methyl-1H-pyrazol-3-yl)amino)-1,6-naphthyridin-5-yl)amino-8-azabicyclo[3.2.1]octan-8-yl)propanenitrile, methanol, N-N-dimethylformamide, and water

#3755
20180354971
2018-12-13

Solvated crystal form of rifaximin, production, compositions and uses thereof

#3756
20180354938
2018-12-13

Solid forms of (Z)-4-(5-((3-benzyl-4-oxo-2-thioxothiazolidin-5-ylidene)methyl)furan-2-yl)benzoic acid

#3757
20180354917
2018-12-13

Crystalline forms of (S)-afoxolaner

#3758
20180354916
2018-12-13

Preparation method for eutectic hydrate crystal form II of AHU-377 and diovan trisodium salt

#3759
20180354893
2018-12-13

Method and system for transporting inventory items

#3760
20180353499
2018-12-13

Piperidin-4-yl azetidine derivatives as JAK1 inhibitors

#3761
20180346506
2018-12-06

METHOD FOR PREPARING SOFOSBUVIR CRYSTAL FORM-6

#3762
20180346504
2018-12-06

Crystalline forms of (S)-2-ethylbutyl 2-(((S)-(((2R,3S,4R,5R)-5- (4-aminopyrrolo[2,1-f] [1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxytetrahydrofuran-2-yl)methoxy)(phenoxy) phosphoryl)amino)propanoate

#3763
20180346494
2018-12-06

Chlorosilylarylgermanes, method for preparation thereof and use thereof

#3764
20180346472
2018-12-06

Synergistic compositions comprising (R)-dimiracetam (1) and (S)-dimiracetam (2) in a non-racemic ratio

#3765
20180346442
2018-12-06

Crystalline fumarate salt of (S)-[3,4-difluoro-2-(2-fluoro-4-iodophenylamino)phenyl] [3-hydroxy-3-(piperidin-2-yl) azetidin-1-yl]methanone

#3766
20180346436
2018-12-06

Crystal of a heterocyclidene acetamide derivative

#3767
20180346425
2018-12-06

CRYSTALLINE FORMS OF PITAVASTATIN CALCIUM

#3768
20180346400
2018-12-06

POLYMORPHIC FORMS OF SODIUM BENZOATE AND USES THEREOF

#3769
20180339997
2018-11-29

POLYMORPHS AND SOLID FORMS OF (S)-2-((2-((S)-4-(DIFLUOROMETHYL)-2-OXOOXAZOLIDIN-3-YL)-5,6-DIHYDROBENZO[F]IMIDAZO[1,2-D][1,4]OXAZEPIN-9-YL)AMINO)PROPANAMIDE, AND METHODS OF PRODUCTION

#3770
20180339984
2018-11-29

5-methyl-1,3,4-oxadiazol-2-yl compounds

#3771
20180339962
2018-11-29

Polymorphic forms of minocycline base and processes for their preparation

#3772
20180334466
2018-11-22

Crystals of thiadiazole derivative DPP-IV inhibitors and uses thereof

#3773
20180334457
2018-11-22

SUBSTANTIALLY PURE VEMURAFENIB AND ITS SALTS

#3774
20180334449
2018-11-22

Process for the preparation of pure nilotinib and its salt

#3775
20180334443
2018-11-22

Process for synthesis of lenalidomide

#3776
20180333425
2018-11-22

Crystallization method and bioavailability

#3777
20180327415
2018-11-15

Crystalline forms of a Bruton's tyrosine kinase inhibitor

#3778
20180327386
2018-11-15

Crystalline forms of (R)-N-((4-methoxy-6-methyl-2-oxo-1,2-dihydropyridin-3-yl)methyl)-2-methyl-1-(1-(1-(2,2,2-trifluoroethyl)piperidin-4-yl)ethyl)-1H-indole-3-carboxamide

#3779
20180327384
2018-11-15

3-methyl-pyrrolidine-2,5-dione derivatives useful as CGRP receptor antagonists

#3780
20180327383
2018-11-15

Process for the preparation of crystalline dexlansoprazole

#3781
20180327356
2018-11-15

Process and novel polymorphic form of Apremilast

#3782
20180327344
2018-11-15

Crystal of monovalent cation salt of 3-hydroxyisovaleric acid and process for producing the crystal

#3783
20180325911
2018-11-15

NOVEL COMPOUNDS

#3784
20180325897
2018-11-15

Co-crystals and pharmaceutical compositions comprising the same

#3785
20180319806
2018-11-08

Crystalline forms of a bruton's tyrosine kinase inhibitor

#3786
20180319805
2018-11-08

CRYSTALLINE FORMS OF A BRUTON'S TYROSINE KINASE INHIBITOR

#3787
20180319803
2018-11-08

Salt and polymorphic forms of (3R,4S)-L-((4-amino-5H-pyrrolo[3,2,-D]pyrimidin-7-yl)methyl)-4(methylthiomethyl)pyrodin-3-ol(MTDIA)

#3788
20180319799
2018-11-08

Pyrido[1,2-A]pyrimidone analog, crystal form thereof, intermediate thereof and preparation method therefor

#3789
20180319792
2018-11-08

Pyrroloquinoline quinone B crystal form and preparation method therefor

#3790
20180319770
2018-11-08

EGFR inhibitor and pharmaceutically acceptable salt and polymorph thereof, and use thereof

#3791
20180319766
2018-11-08

CO-CRYSTALS OF BENZIMIDAZOLE COMPOUNDS

#3792
20180319754
2018-11-08

Thermodynamically stable crystal modification of 2-methyl-N-(5-methyl-1, 3, 4-oxadiazol-2-yl)-3-(methylsulfonyl)-4-(trifluoromethyl)benzamide

#3793
20180318292
2018-11-08

2-(1H-indazol-3-yl)-3H-imidazo[4,5-C]pyridines and their anti-inflammatory uses thereof

#3794
20180312543
2018-11-01

CYCLOSPORIN A FORM 2 AND METHOD OF MAKING SAME

#3795
20180312512
2018-11-01

Crystal form, preparation method and intermediate of dihydropyrido ring compound

#3796
20180312510
2018-11-01

Pharmaceutical salts, physical forms, and compositions of pyrrolopyrimidine kinase inhibitors, and methods of making same

#3797
20180312494
2018-11-01

Polymorphic forms of Afatinib free base and Afatinib dimaleate

#3798
20180312474
2018-11-01

KDM1A inhibitors for the treatment of disease

#3799
20180312472
2018-11-01

Quinazolin crotyl compound dimaleate crystals and preparation methods and uses thereof

#3800
20180312465
2018-11-01

Heat-sensitive recording material and diphenylsulfone

#3801
20180305397
2018-10-25

Preparation and Uses of Obeticholic Acid

#3802
20180305388
2018-10-25

Crystal of 6′-sialyllactose sodium salt, and process for producing same

#3803
20180305365
2018-10-25

Pharmaceutical compositions of compound

#3804
20180305361
2018-10-25

Crystal form A of 7-(cyclopropylmethyl)-1-((()-4-hydroxy-4-methylcyclohexyl)methyl)-3-methyl-1H-purine-2,6-(3H,7H)-dione for treating liver diseases

#3805
20180305349
2018-10-25

1, 3, 4-thiadiazole compounds and their use in treating cancer

#3806
20180305297
2018-10-25

DTPA PRODRUGS, COMPOSITIONS THEREOF, AND METHODS OF USING THE SAME

#3807
20180305296
2018-10-25

Acetylsalicylic acid derivative crystal, its preparation method and use

#3808
20180303825
2018-10-25

Polymorphic forms of naltrexone

#3809
20180298025
2018-10-18

Processes for preparing ACC inhibitors and solid forms thereof

#3810
20180298016
2018-10-18

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-A]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#3811
20180297992
2018-10-18

Inhibiting agents for bruton's tyrosine kinase

#3812
20180297956
2018-10-18

CRYSTAL FORM OF QUINOLINE COMPOUND AND PROCESS FOR ITS PRODUCTION

#3813
20180297933
2018-10-18

PROCESS FOR PREPARING A DIAMINE/DICARBOXYLIC ACID SALT

#3814
20180296533
2018-10-18

Preparation of and formulation comprising a MEK inhibitor

#3815
20180296519
2018-10-18

Sacubitril calcium salts

#3816
20180291049
2018-10-11

Crystalline Forms of Fosnetupitant

#3817
20180291032
2018-10-11

POLYMORPHOUS FORMS OF RIFAXIMIN, PROCESSES FOR THEIR PRODUCTION AND USE THEREOF IN THE MEDICINAL PREPARATIONS

#3818
20180291010
2018-10-11

Fumagillol derivatives and polymorphs thereof

#3819
20180291005
2018-10-11

Stable crystal form of tipiracil hydrochloride and crystallization method for the same

#3820
20180291001
2018-10-11

Inhibitors of Bruton's tyrosine kinase

#3821
20180290964
2018-10-11

CRYSTALLINE SOLID FORMS OF THE ACETATE SALT OF (1S,3S,4R)-4-((3AS,4R,5S,7AS)-4-(AMINOMETHYL)-7A-METHYL-1-METHYLENEOCTAHYDRO-1H-INDEN-5-YL)-3-(HYDROXYMETHYL)-4-METHYLCYCLOHEXANOL

#3822
20180289800
2018-10-11

PYRAZOLOPYRIMIDINE COMPOUNDS

#3823
20180289662
2018-10-11

Pharmaceutical co-crystal and use thereof

#3824
20180282619
2018-10-04

Reversible Continuous Variable Chromogenic Material, Preparation Method and Application thereof

#3825
20180282366
2018-10-04

Crystalline and amorphous forms of 17-alpha-hydroxyprogesterone caproate

#3826
20180282362
2018-10-04

Crystal forms of β-nicotinamide mononucleotide

#3827
20180282351
2018-10-04

Amorphous Ixazomib Citrate

#3828
20180282342
2018-10-04

Salt of pyrrolo[2,3-D]pyrimidine compound and novel polymorph of salt

#3829
20180282339
2018-10-04

PROCESS FOR THE PREPARATION OF THE AMORPHOUS FORM OF IBRUTINIB AND NOVEL CRYSTALLINE FORM

#3830
20180282312
2018-10-04

Hydrochloride salt form for EZH2 inhibition

#3831
20180282310
2018-10-04

FORMS AND COMPOSITIONS OF BIARYL INHIBITORS OF BRUTON'S TYROSINE KINASE

#3832
20180282300
2018-10-04

Crystal form of a potassium-competitive acid blocker and preparation method thereof

#3833
20180282266
2018-10-04

(S)-CSA salt of S-ketamine, (R)-CSA salt of S-ketamine and processes for the preparation of S-ketamine

#3834
20180282260
2018-10-04

1-AMINOCYCLOPROPANE-1-CARBOXYLIC ACID POLYMORPHS

#3835
20180273592
2018-09-27

Highly crystalline spherical silk fibroin micro-particles and a process for preparation thereof

#3836
20180273526
2018-09-27

CRYSTAL FORM OF PYRROLOQUINOLINE QUINONE SODIUM SALT AND PREPARATION METHOD AND USE THEREOF

#3837
20180273522
2018-09-27

Salts and solid forms of a monobactam antibiotic

#3838
20180273507
2018-09-27

CRYSTAL FORMS OF A M1 RECEPTOR POSITIVE ALLOSTERIC MODULATOR

#3839
20180273501
2018-09-27

Methods for purification of non-psychoactive isoprenoid compounds from biological extracts

#3840
20180273499
2018-09-27

SALTS AND SOLID STATE FORMS OF VORTIOXETINE

#3841
20180273493
2018-09-27

Amorphous trisodium sacubitril valsartan and a process for the preparation thereof

#3842
20180273490
2018-09-27

Process for the Preparation of Eltrombopag Olamine

#3843
20180273483
2018-09-27

Dibenzo azepine compounds and their use in the treatment of otic diseases and disorders

#3844
20180273481
2018-09-27

Polymorphic forms of pitavastatin sodium

#3845
20180265530
2018-09-20

Crystalline forms of tenofovir alafenamide

#3846
20180265513
2018-09-20

Process for the preparation of dipeptidyl peptidase-4 (DPP-4) enzyme inhibitor

#3847
20180265495
2018-09-20

Crystal form of neratinib maleate and preparation method therefor

#3848
20180265492
2018-09-20

Antifungal compounds and processes for making

#3849
20180265474
2018-09-20

Polymorphic compounds and uses thereof

#3850
20180258105
2018-09-13

Crystalline forms of a PI3K inhibitor

#3851
20180258093
2018-09-13

Salt type and crystal type of 4H-pyrazolo [1, 5-alpha] benzimidazole compound and preparation method and intermediate thereof

#3852
20180258086
2018-09-13

TYK2 inhibitors, uses, and methods for production thereof

#3853
20180258081
2018-09-13

DIACYLGLYCEROL ACYL TRANSFERASE 2 INHIBITORS

#3854
20180258078
2018-09-13

Process for the preparation of Daclatasvir dihydrochloride and its intermediates

#3855
20180258069
2018-09-13

NEW CRYSTAL OF PIPERAZINE COMPOUND

#3856
20180258068
2018-09-13

Antifungal compound process

#3857
20180258064
2018-09-13

SOLID FORMS OF 3-(5-AMINO-2-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERIDINE-2,6-DIONE, AND THEIR PHARMACEUTICAL COMPOSITIONS AND USES

#3858
20180258055
2018-09-13

Solid forms of substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine compounds

#3859
20180251575
2018-09-06

Process for preparation and purification of Sugammades sodium

#3860
20180251464
2018-09-06

Inhibitors of bruton'S tyrosine kinase

#3861
20180251463
2018-09-06

Ibrutinib solid forms and production process therefor

#3862
20180251462
2018-09-06

DOSAGE FORM COMPOSITIONS COMPRISING AN INHIBITOR OF BRUTON'S TYROSINE KINASE

#3863
20180251430
2018-09-06

1-(4-(2-((1-(3,4-difluorophenyl)-1H-pyrazol-3-Yl)methoxy)ethyl)piperazin-1- Yl)ethanone salts

#3864
20180244711
2018-08-30

CRYSTAL FORM OF FLUDARABINE PHOSPHATE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#3865
20180244701
2018-08-30

Phosphoramidate compound and preparation method and crystal thereof

#3866
20180244700
2018-08-30

METHODS OF TREATING A FATTY ACID AMIDE HYDROLASE-MEDIATED CONDITION

#3867
20180244696
2018-08-30

Polymorphic forms and co-crystals of a c-Met inhibitor

#3868
20180244675
2018-08-30

Purinone derivative hydrochloride

#3869
20180244661
2018-08-30

Process for the preparation of amorphous (1S)-1,5-anhydro-1-[3-[[5-(4 fluorophenyl)-2-thienyl]-4-methylphenyl]-D-glucitol and its polymorphs thereof

#3870
20180244649
2018-08-30

Pyridine substituted 2-aminopyridine protein kinase inhibitor crystal

#3871
20180244647
2018-08-30

Crystals of 5-cyclopropyl-2-((1-(3-fluorobenzyl)-1H-indol-5-yl)amino)nicotinic acid

#3872
20180244628
2018-08-30

Crystalline form of androgen receptor inhibitor and preparation method thereof

#3873
20180244608
2018-08-30

Process for the preparation of the compound N-(3,5-dimethylphenyl)-N′-(2-trifluoromethylphenyl) guanidine

#3874
20180237445
2018-08-23

Medical use of compound III

#3875
20180237443
2018-08-23

Chemical compounds

#3876
20180237438
2018-08-23

Crystal form of bisulfate of JAK inhibitor and preparation method therefor

#3877
20180237396
2018-08-23

Process for preparing AG-10, its intermediates, and salts thereof

#3878
20180235955
2018-08-23

Acetate salt of buprenorphine and methods for preparing buprenorphine

#3879
20180235933
2018-08-23

Crystalline form of lorlatinib free base

#3880
20180230158
2018-08-16

[1,2,4]triazolo[4,3-B]pyridazines for use in the treatment of proliferative diseases

#3881
20180230149
2018-08-16

Inhibiting the transient receptor potential A1 ion channel

#3882
20180230147
2018-08-16

Hydroxyethyl sulfonate of cyclin-dependent protein kinase inhibitor, crystalline form thereof and preparation method therefor

#3883
20180230140
2018-08-16

MULTICOMPONENT CRYSTALS OF DASATINIB WITH MENTHOL OR VANILLIN

#3884
20180230136
2018-08-16

Crystal form of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxole-5-yl)cyclopropane formamido)-3-methylpyridine-2-yl)benzoic acid and preparation method thereof

#3885
20180230082
2018-08-16

Crystalline Forms of (-)-(1R,2R)-3-(3-dimethylamino-1-ethyl-2-methylpropyl)-phenol hydrochloride

#3886
20180228807
2018-08-16

Methods of synthesizing thyroid hormone analogs and polymorphs thereof

#3887
20180228774
2018-08-16

(2R,4R)-5-(5′-chloro-2′-fluorobiphenyl-4-yl)-2-hydroxy-4-[(5-methyloxazole-2-carbonyl)amino]pentanoic acid

#3888
20180228754
2018-08-16

Co-crystals of substituted glycine and uses thereof

#3889
20180228753
2018-08-16

Co-crystals of substituted glycine and uses thereof

#3890
20180222914
2018-08-09

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#3891
20180222913
2018-08-09

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#3892
20180222845
2018-08-09

LEVALBUTEROL SALT

#3893
20180215776
2018-08-02

Nucleotide hemi-sulfate salt for the treatment of hepatitis C virus

#3894
20180215756
2018-08-02

Processes for preparing an FGFR inhibitor

#3895
20180215751
2018-08-02

5-methyl-1,2,4-oxadiazol-3-yl compounds

#3896
20180215744
2018-08-02

Salts of quinazoline derivative or crystals thereof, and the process for producing thereof

#3897
20180215733
2018-08-02

Polymorphs of Selinexor

#3898
20180215715
2018-08-02

Solid state forms of netarsudil mesylate

#3899
20180208623
2018-07-26

CRYSTALLINE SOLVATE FORMS OF A PHARMACEUTICAL

#3900
20180208622
2018-07-26

STABLE CRYSTALLINE FORM OF REGADENOSON