ClassID:

90494

C07B2200/13 - page 14 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#3901
20180208614
2018-07-26

Crystal of cyclic phosphonic acid sodium salt and method for manufacturing same

#3902
20180208599
2018-07-26

Polymorphs of ponatinib hydrochloride

#3903
20180208596
2018-07-26

Pharmaceutical composition comprising a crystal form of (S)-4-(8-amino-3-(1-(but-2-ynoyl) pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-N-(pyridin-2-yl)benzamide

#3904
20180208563
2018-07-26

THERMODYNAMICALLY STABLE CRYSTAL MODIFICATION OF 2-CHLORO-3-(METHYLSULFANYL)-N-(1-METHYL-1H-TETRAZOL-5-YL)-4-(TRIFLUOROMETHYL)BENZAMIDE

#3905
20180208530
2018-07-26

Process for the synthesis of 9,9-bis(hydroxymethyl)fluorene

#3906
20180201603
2018-07-19

Substituted tetrahydroisoquinoline compounds as factor XIa inhibitors

#3907
20180201594
2018-07-19

Compound pac-1 or salt thereof and pharmaceutical composition comprising same

#3908
20180201589
2018-07-19

Crystalline forms of trisodium supramolecular complex comprising valsartan and AHU-377 and methods thereof

#3909
20180200252
2018-07-19

Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-(trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino [2,3-b]pyrazin-2(1H)-one, a solid form thereof and methods of their use

#3910
20180200245
2018-07-19

Solid forms comprising 4-amino-2-(2,6-dioxopiperidine-3-yl)isoindoline-1,3-dione and a coformer, compositions and methods of use thereof

#3911
20180194777
2018-07-12

Diaryl macrocycle polymorph

#3912
20180194754
2018-07-12

Polymorphs and process for the preparation of quinazolinyl derivatives

#3913
20180194752
2018-07-12

Ledipasvir crystal form and preparation method thereof

#3914
20180194749
2018-07-12

Plinabulin compositions

#3915
20180194734
2018-07-12

Process for the preparation of Lorcaserin hydrochloride

#3916
20180194719
2018-07-12

Crystal forms of verapamil hydrochloride

#3917
20180193292
2018-07-12

Process for preparation of cysteamine bitartrate

#3918
20180186822
2018-07-05

Pharmaceutical co-crystal composition and use thereof

#3919
20180186805
2018-07-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-#a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-#carboxamide and solid state forms thereof

#3920
20180186803
2018-07-05

Short-acting benzodiazepine salts and their polymorphic forms

#3921
20180186784
2018-07-05

Crystalline forms of N-(2-chloro-6-methy]phenvn-2-[F6-[4-(2-hvdroxvethvl)-L-piperazin-vil-2-methvil-4-pvrimidinvllaminol-5-thiazolecarboxamide and their process thereof

#3922
20180186740
2018-07-05

Crystalline freebase forms of a biphenyl compound

#3923
20180186738
2018-07-05

Crystalline L-arginine salt of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclo-penta [b]indol-3-yl)acetic acid(Compund1) for use in SIPI receptor-associated disorders

#3924
20180186726
2018-07-05

Polymorphic forms of RAD1901-2HCL

#3925
20180179240
2018-06-28

Pharmaceutical composition of carboplatin based co-crystals and use thereof

#3926
20180179215
2018-06-28

Crystalline forms of a bruton's tyrosine kinase inhibitor

#3927
20180179214
2018-06-28

Crystalline forms of a Bruton's tyrosine kinase inhibitor

#3928
20180179196
2018-06-28

Crystalline forms of cadazolid

#3929
20180170958
2018-06-21

Crystalline form A of obeticholic acid and preparation method thereof

#3930
20180170945
2018-06-21

Crystalline forms of darunavir

#3931
20180170940
2018-06-21

CRYSTALLINE FORMS OF A BRUTON'S TYROSINE KINASE INHIBITOR

#3932
20180170926
2018-06-21

Crystal of 5-hydroxy-4-(trifluoromethyl)pyrazolopyridine derivative

#3933
20180170919
2018-06-21

Crystaline forms of N-[6-(cis-2,6-dimethylmorpholine-4-yl)pyridine-3-yl]-2-Methyl-4′-(trifluoromethoxy) [1,1′-biphenyl]-3-Methanamide monophosphate, and process of preparation thereof

#3934
20180170907
2018-06-21

Salts of a Pim kinase inhibitor

#3935
20180170880
2018-06-21

Method for producing 1-(acyloxy)alkyl carbamate derivative

#3936
20180170871
2018-06-21

Crystalline forms of (R)-1-(1-(methylsulfonyl)propan-2-yl)-4-(trifluoromethyl)-1H-indole-5-carbonitrile

#3937
20180170023
2018-06-21

Composite for neutral layer

#3938
20180169245
2018-06-21

Premix of crystalline raltegravir potassium salt and a process for the preparation thereof

#3939
20180162900
2018-06-14

Polymorphic forms of an oxysterol and methods of making them

#3940
20180162866
2018-06-14

Acetate salt of buprenorphine and methods for preparing buprenorphine

#3941
20180162865
2018-06-14

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluorethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#3942
20180162839
2018-06-14

Modulator of the cystic fibrosis transmembrane conductance regulator, pharmaceutical compositions, methods of treatment, and process for making the modulator

#3943
20180162820
2018-06-14

Method for the preparation of highly pure ivabradine base and salts thereof

#3944
20180155364
2018-06-07

Process for the preparation of dolutegravir and pharmaceutically acceptable salts thereof

#3945
20180155358
2018-06-07

Ertugliflozin co-crystals and process for their preparation

#3946
20180155356
2018-06-07

Crystals of dispiropyrrolidine derivatives

#3947
20180155355
2018-06-07

Crystals of dispiropyrrolidine derivatives

#3948
20180155352
2018-06-07

CRYSTALLINE FORMS OF A BRUTON'S TYROSINE KINASE INHIBITOR

#3949
20180155337
2018-06-07

Crystalline forms of (3-amino-oxetan-3-ylmethyl)-[2-(5,5-dioxo-5,6,7,9-tetrahydro-5lambda*6*-thia-8-aza-benzocyclohepten-8-yl)-6-methyl-quinazolin-4-yl]-amine

#3950
20180155300
2018-06-07

Solid state forms of trisodium valsartan: sacubitril

#3951
20180155291
2018-06-07

Crystal form of lenvatinib methanesulfonate salt and preparation method thereof

#3952
20180155273
2018-06-07

Crystalline solid forms of the acetate salt of (1S,3S,4R)-4-((3AS,4R,5S,7AS)-4-(aminomethyl)-7A-methyl-1-methyleneoctahydro-1H-inden-5-YL)-3- (hydroxymethyl)-4-methylcyclohexanol

#3953
20180153895
2018-06-07

Crystalline forms of ibrutinib

#3954
20180148443
2018-05-31

Crystals of azabicyclic compound

#3955
20180148436
2018-05-31

Pyridone derivatives having tetrahydropyranylmethyl groups

#3956
20180148432
2018-05-31

Heteroarylphenoxy benzamide kappa opioid ligands

#3957
20180148409
2018-05-31

Crystal of salt of novel 3-azabicyclo[3.1.0]hexane derivative and pharmaceutical use thereof

#3958
20180148403
2018-05-31

Fenfluramine compositions and methods of preparing the same

#3959
20180148402
2018-05-31

Crystalline inhibitor of 4-hydroxyphenylpyruvate dioxygenase

#3960
20180142365
2018-05-24

METHOD FOR REDUCING CARBON DIOXIDE ELECTROCHEMICALLY TO GENERATE ETHYLENE SELECTIVELY

#3961
20180141955
2018-05-24

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-alpla]pyrrolo[2,3-e]-pyrazin-8-YL)-N-(2,2,2-Trifluoroethyl)pyrrol and solid state forms thereof

#3962
20180141950
2018-05-24

Crystal (6S,9aS)-N-benzyl-8-({6-[3-(4-ethylpiperazin-1-yl)azetidin-1-yl]pyridin-2-yl}methyl)-6-(2-fluoro-4-hydroxybenzyl)-4,7-dioxo-2-(prop-2-en-1-yl)hexahydro-2H-pyrazino[2,1-c][1,2,4]triazine-1(6H)-carboxamide

#3963
20180141940
2018-05-24

Salt form and crystal form of 1,2,5-thiadiazolidin-1,1-dioxide, preparation method thereof and intermediate

#3964
20180141939
2018-05-24

SOLID FORMS OF A BET INHIBITOR

#3965
20180141915
2018-05-24

Crystal form A of 1-isobutyryl-1′-((1-(4,4,4-trifluorobutyl)-4,5,6,7-tetrahydro-1H-benzo [d]imidazol-2-yl)methyl)spiro[azetidine-3,3′-indolin]-2′-one

#3966
20180134745
2018-05-17

METHODS OF SYNTHESIZING SUBSTITUTED PURINE COMPOUNDS

#3967
20180134744
2018-05-17

METHODS OF SYNTHESIZING SUBSTITUTED PURINE COMPOUNDS

#3968
20180134743
2018-05-17

Efficient and scalable syntheses of nicotinoyl ribosides and reduced nicotinoyl ribosides, modified derivatives thereof, phosphorylated analogs thereof, adenylyl dinucleotide conjugates thereof, and novel crystalline forms thereof

#3969
20180134742
2018-05-17

Crystalline forms of nicotinoyl ribosides, modified derivatives thereof, and phosphorylated analogs thereof, and methods of preparation thereof

#3970
20180134711
2018-05-17

Stable formulations of 5,10-methylene-(6R)-tetrahydrofolic acid

#3971
20180134687
2018-05-17

1-pyrazolyl-3-(4-((2-anilinopyrimidin-4-yl) oxy) napththalen-I-yl) ureas as P38 mapkinase inhibitors

#3972
20180134668
2018-05-17

Quinazolin crotyl compound dimaleate crystals and preparation methods and uses thereof

#3973
20180134666
2018-05-17

Crystal of uracil compound

#3974
20180134663
2018-05-17

Sodium salt of uric acid transporter inhibitor and crystalline form thereof

#3975
20180127452
2018-05-10

Polymorph of regadenoson and process for preparation thereof

#3976
20180127446
2018-05-10

Co-crystals, salts and solid forms of tenofovir alafenamide

#3977
20180127428
2018-05-10

Salt of fused pyrimidine compound and crystal thereof

#3978
20180127417
2018-05-10

Intermediates for preparing CGRP receptor antagonists

#3979
20180127412
2018-05-10

Maleate salts of a B-RAF kinase inhibitor, crystalline forms, methods of preparation, and uses therefore

#3980
20180127398
2018-05-10

Solid forms of 3-(6-(1-(2,2-difluorobenzo[D][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid

#3981
20180127376
2018-05-10

NOVEL CRYSTALLINE FORM OF ESLICARBAZEPINE

#3982
20180127359
2018-05-10

Nitrite salts of 1,1-dimethylbiguanide, pharmaceutical compositions, and methods of use

#3983
20180127349
2018-05-10

5-bromo-2-(α-hydroxypentyl)benzoic acid sodium salts in different crystal forms, and preparation method thereof

#3984
20180127344
2018-05-10

Solubilization of pterostilbene and resveratrol for aqueous beverages

#3985
20180118726
2018-05-03

LFA-1 inhibitor and methods of preparation and polymorph thereof

#3986
20180118715
2018-05-03

P-toluenesulfonate for MEK kinase inhibitor, and crystal form thereof and preparation method therefor

#3987
20180118714
2018-05-03

Process for the preparation of Efinaconazole

#3988
20180118701
2018-05-03

Process for the preparation of substituted oxiranes and triazoles

#3989
20180118686
2018-05-03

Process for the preparation of a PDE4 inhibitor

#3990
20180118662
2018-05-03

Tranilast compositions and cocrystals

#3991
20180111949
2018-04-26

NOVEL INDUSTRIAL CRYSTALLIZATION METHOD OF CEFUROXIME SODIUM AND PREPARATION THEREOF

#3992
20180111932
2018-04-26

Naphthyridinone derivatives and their use in the treatment of arrhythmia

#3993
20180111930
2018-04-26

COMPOSITIONS AND USES THEREOF

#3994
20180111915
2018-04-26

Polymorphic form X of nilotinib dihydrochloride hydrate

#3995
20180111903
2018-04-26

Crystalline forms of cabozantinib phosphate and cabozantinib hydrochloride

#3996
20180111891
2018-04-26

Polymorphic forms of sodium benzoate and uses thereof

#3997
20180111890
2018-04-26

Process for the preparation of ethacrynic acid

#3998
20180110773
2018-04-26

Polymorphic forms of naltrexone

#3999
20180105543
2018-04-19

Oriented perovskite crystals and methods of making the same

#4000
20180105517
2018-04-19

Process for the preparation of aclidinium bromide

#4001
20180104262
2018-04-19

SALTS AND POLYMORPHS OF A TETRACYCLINE COMPOUND

#4002
20180099991
2018-04-12

SALTS OF OBETICHOLIC ACID

#4003
20180099976
2018-04-12

Compounds as rearranged during transfection (RET) inhibitors

#4004
20180099969
2018-04-12

Polymorphs

#4005
20180099948
2018-04-12

Crystalline salts of (S)-6-((1-acetylpiperidin-4-yl)amino)-N-(3-(3,4-dihydroisoquinolin-2(1H)-yl)-2-hydroxypropyl)pyrimidine-4-carboxamide

#4006
20180099944
2018-04-12

Crystal forms of immunomodulatory drug pomalidomide and co-crystal with gentisic acid

#4007
20180099924
2018-04-12

Metabolites of (1R-trans)-N-[[2-(2,3-dihydro-4-benzofuranyl)cyclopropyl]methyl]propanamide

#4008
20180094020
2018-04-05

2,2-DIFLUOROPROPIONAMIDE DERIVATIVES OF BARDOXOLONE METHYL, POLYMORPHIC FORMS AND METHODS OF USE THEREOF

#4009
20180094014
2018-04-05

Method of producing epirubicin and novel production intermediate thereof

#4010
20180093998
2018-04-05

Chemical compounds

#4011
20180092898
2018-04-05

PROCESSES OF MAKING AND CRYSTALLINE FORMS OF A MDM2 INHIBITOR

#4012
20180086783
2018-03-29

Crystalline form of nicotinamide riboside

#4013
20180086762
2018-03-29

Beta-lactamase inhibitors

#4014
20180086731
2018-03-29

Crystalline forms of 1-((2R,4R)-2-(1H-benzo[d]imidazol-2-yl)-1-methylpiperidin-4-yl)-3-(4-cyanophenyl)urea maleate

#4015
20180086695
2018-03-29

Crystalline form of AHU377, preparation method and use thereof

#4016
20180086692
2018-03-29

Solid forms

#4017
20180079762
2018-03-22

Carbidopa and L-dopa prodrugs and methods of use

#4018
20180079758
2018-03-22

Substituted tetrahydrocarbazole and carbazole carboxamide compounds

#4019
20180079705
2018-03-22

METHOD FOR PURIFICATION OF AN AROMATIC DIACID OR THE CORRESPONDING ANHYDRIDE

#4020
20180078660
2018-03-22

Crystalline contrast agent for magnetic resonance imaging, kit and composition comprising it and their use

#4021
20180073049
2018-03-15

Method of converting RB to RD by using cutinase under stepwise changing temperatures

#4022
20180072748
2018-03-15

Crystal of 6,7-unsaturated-7-carbamoyl morphinan derivative and method for producing the same

#4023
20180072737
2018-03-15

Co-crystals of ibrutinib with carboxylic acids

#4024
20180072733
2018-03-15

Crystalline form alpha of IPI-145 and preparation method thereof

#4025
20180072700
2018-03-15

POLYMORPHIC FORMS OF 3-(4-AMINO-1-OXO-1,3 DIHYDRO-ISOINDOL-2-YL)-PIPERIDINE-2,6-DIONE

#4026
20180072685
2018-03-15

Method for producing (4S)-4-[4-cyano-2-(methylsulfonyl)phenyl]-3,6-dimethyl-2-oxo-1-[3-(trifluoromethyl)phenyl]-1,2,3,4-tetrohydro pyrimidine-5-carbonitrile

#4027
20180072676
2018-03-15

CRYSTAL FORM OF QUINOLINE COMPOUND AND PROCESS FOR ITS PRODUCTION

#4028
20180072667
2018-03-15

Selective FKBP51 ligands for treatment of psychiatric disorders

#4029
20180071287
2018-03-15

Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3-yl)-1-((trans)-4-methoxycyclohexyl)-3,4-dihydropyrazino[2,3- ]pyrazin-2(1)-one, a solid form there of and methods of their use

#4030
20180065988
2018-03-08

PHARMACEUTICAL COMPOSITIONS COMPRISING POLYMORPHIC FORMS ALPHA, BETA, AND GAMMA OF RIFAXIMIN

#4031
20180065987
2018-03-08

POLYMORPHIC FORMS ALPHA, BETA AND GAMMA OF RIFAXIMIN

#4032
20180065986
2018-03-08

Sodium (2R,5S,13aR)-7,9-dioxo-10-((2,4,6-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13a-octahydro-2,5-methanopyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]oxazepin-8-olate

#4033
20180065979
2018-03-08

Crystalline forms of therapeutic compounds and uses thereof

#4034
20180065978
2018-03-08

Crystalline forms of therapeutic compounds and uses thereof

#4035
20180065977
2018-03-08

Crystalline forms of therapeutic compounds and uses thereof

#4036
20180065973
2018-03-08

Process for making beta 3 agonists and intermediates

#4037
20180065963
2018-03-08

Inhibitors of influenza viruses replication

#4038
20180065942
2018-03-08

Crystalline substituted 5-fluoro-1H-pyrazolopyridines and process for preparing

#4039
20180065939
2018-03-08

Process for the preparation of clobazam and its intermediate

#4040
20180065937
2018-03-08

Methods for preparing substituted 5,6-dihydro-6-phenylbenzo[F]isoquinolin-2-amine

#4041
20180057503
2018-03-01

Pharmaceutically acceptable salts and polymorphic forms of hydrocodone benzoic acid enol ester and processes for making same

#4042
20180057502
2018-03-01

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-alpha]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#4043
20180057498
2018-03-01

Co-crystal of a CDK inhibitor and an MEK inhibitor and process of preparation thereof

#4044
20180057481
2018-03-01

Solid forms of cenicriviroc mesylate and processes of making solid forms of cenicriviroc mesylate

#4045
20180057469
2018-03-01

Crystalline forms of tyrosine kinase inhibitors and their salts

#4046
20180055836
2018-03-01

Process for the preparation of benzhydrocodone hydrochloride

#4047
20180051026
2018-02-22

POLYMORPHS OF IBRUTINIB

#4048
20180051012
2018-02-22

Diacylglycerol acyl transferase 2 inhibitors

#4049
20180051004
2018-02-22

Crystalline forms of a biphenyl compound

#4050
20180051002
2018-02-22

Nicotine salts, co-crystals, and salt co-crystal complexes

#4051
20180050991
2018-02-22

Crystalline forms of olaparib and manufacturing processes therefor

#4052
20180050057
2018-02-22

Crystal-water-free calcium dibutyryladenosine cyclophosphate crystal form and preparation method and application thereof

#4053
20180049995
2018-02-22

HIF-2-ALPHA INHIBITOR POLYMORPHS

#4054
20180044366
2018-02-15

NOVEL CRYSTALLINE FORMS OF AN ANTIVIRAL BENZIMIDAZOLE COMPOUND

#4055
20180044356
2018-02-15

Crystalline form of a proteasome inhibitor

#4056
20180044353
2018-02-15

4-substituted benzoxaborole compounds and uses thereof

#4057
20180044351
2018-02-15

Crystalline methyl (4R,12aS)-7-(benzyloxy)-4-methyl-6,8-dioxo-3,4,6,8,12,12a-hexahydro-2H-pyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxylate

#4058
20180044348
2018-02-15

CRYSTALLINE SALTS OF MORPHINE SULFATE

#4059
20180044347
2018-02-15

CRYSTALLINE SALTS OF HYDROCODONE BITARTRATE

#4060
20180044342
2018-02-15

Crystal form of JAK inhibitor and preparation method thereof

#4061
20180044323
2018-02-15

Deuterated diaminopyrimidine compounds and pharmaceutical compositions comprising such compounds

#4062
20180044317
2018-02-15

Benzimidazole derivatives as bromodomain inhibitors

#4063
20180042914
2018-02-15

Bromodomain inhibitor

#4064
20180037597
2018-02-08

Crystalline forms of 5-chloro-N4-[-2-(dimethylphosphoryl)phenyl]-N2-{2-methoxy-4-[4-(4-methylpiperazin-1-YL) piperidin-1-YL]phenyl}pyrimidine-2,4-diamine

#4065
20180037595
2018-02-08

BENZOXABOROLE COMPOUNDS AND USES THEREOF

#4066
20180037593
2018-02-08

Method of producing (3S,11aR)-6,8-dihalo-3-methyl-2,3,11,11a-tetrahydrooxazolo[3,2-a]pyrido[1,2-d]pyrazine-5,7-diones

#4067
20180037592
2018-02-08

Crystalline methyl (4R,12aS)-7-(benzyloxy)-4-methyl-6,8-dioxo-3,4,6,8,12,12a-hexahydro-2H-pyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]oxazine-9-carboxylate

#4068
20180037591
2018-02-08

Crystalline dimethyl 3-(benzyloxy)-1-(2,2-dimethoxyethyl)-4-oxo-1,4-dihydropyridine-2,5-dicarboxylate

#4069
20180037560
2018-02-08

Crystalline forms of neurotrophin mimetic compounds and their salts

#4070
20180037559
2018-02-08

Crystalline forms of neurotrophin mimetic compounds and their salts

#4071
20180037549
2018-02-08

Processes and intermediates for the preparation of Pimavanserin

#4072
20180036247
2018-02-08

Pharmaceutical compositions

#4073
20180030085
2018-02-01

Crystal form of Abiraterone propionate and preparation method therefor

#4074
20180030079
2018-02-01

Crystalline form of nicotinamide riboside

#4075
20180030067
2018-02-01

Crystal of imidazo-oxazine, pharmaceutical composition containing said crystal, and method for producing said crystal

#4076
20180030066
2018-02-01

Crystal form A of compound and preparation method thereof

#4077
20180030058
2018-02-01

Crystal of 5-((2-(6-amino)-9H-purin-9-yl)ethyl)amino)pentan-1-o1

#4078
20180030038
2018-02-01

Polymorphic Forms of Afatinib Dimaleate

#4079
20180030008
2018-02-01

Process for the preparation of vortioxetine

#4080
20180029994
2018-02-01

Process for the preparation of intermediates useful in the synthesis of Eluxadoline

#4081
20180029987
2018-02-01

CRYSTALLINE FORMS OF PITAVASTATIN CALCIUM

#4082
20180029986
2018-02-01

POLYMORPHIC FORMS OF THE SODIUM SALT OF 4-TERT- BUTYL -N-[4-CHLORO-2-(1-OXY-PYRIDINE-4-CARBONYL)-PHENYL]-BENZENE SULFONAMIDE

#4083
20180029977
2018-02-01

Polymorphic forms of minocycline base and processes for their preparation

#4084
20180029976
2018-02-01

Crystalline Forms of (-)-(1R,2R)-3-(3-dimethylamino-1-ethyl-2-methylpropyl)-phenol hydrochloride

#4085
20180028539
2018-02-01

Therapeutically active compounds and their methods of use

#4086
20180028476
2018-02-01

STABLE DOSAGE FORMS OF LEVOMILNACIPRAN

#4087
20180022775
2018-01-25

Preparations of hydrophobic therapeutic agents, methods of manufacture and use thereof

#4088
20180022711
2018-01-25

Crystal forms of the monosodium salt of foramsulfuron

#4089
20180022708
2018-01-25

Processes for preparing ASK1 inhibitors

#4090
20180022704
2018-01-25

Process for the preparation of histamine H3 receptor modulators

#4091
20180022674
2018-01-25

Process for preparation of ospemifene

#4092
20180022136
2018-01-25

Crystalline modification of N-(2-(3-phenylureido)phenyl)benzenesulfonamide and recording material using same

#4093
20180021310
2018-01-25

Mebendazole polymorph for treatment and prevention of tumors

#4094
20180016297
2018-01-18

Crystalline forms of S-[4-(3-fluoro-3-methylbutyryloxy)but-2-ynyl] 6-α,9-α-difluoro-17-α-(furan-2-yl)carbonyloxy-11-β-hydroxy-16-α-methyl-3-oxoandrosta-1,4-diene-17-β-carbothioate

#4095
20180016284
2018-01-18

Polymorphs

#4096
20180016283
2018-01-18

Solid state forms of spiro-oxindole compounds

#4097
20180016264
2018-01-18

Salt forms of 4-cyano-N-(2-(4,4-dimethylcyclohex-1-en-1-yl)-6-(2,2,6,6-tetramethyltetrahydro-2H-pyran-4-yl)pyridin-3-yl)-1H-imidazole-2-carboxamide

#4098
20180016246
2018-01-18

Process for preparation of polymorphic form of Mirabegron

#4099
20180016230
2018-01-18

Salts of Prostaglandin Analog Intermediates

#4100
20180009831
2018-01-11

PROCESS FOR THE PREPARATION OF NOVEL POLYMORPHIC FORMS OF 5-FLUORO-1,3-DIHYDRO-1-HYDROXY-2,1- BENZOXABOROLE

#4101
20180009824
2018-01-11

Crystalline forms of therapeutic compounds and uses thereof

#4102
20180009816
2018-01-11

Substituted imidazo[2,1-f][1,2,4]triazines, substituted imidazo[1,2-a]pyridines, substituted imidazo[1,2-b]pyridazines and substituted imidazo[1,2-a]pyrazines as PI3K-γ inhibitors

#4103
20180009804
2018-01-11

Hydroxyethyl sulfonate of cyclin-dependent protein kinase inhibitor, crystalline form thereof and preparation method therefor

#4104
20180009803
2018-01-11

High-solubility acetone-added pyrroloquinoline quinone salt

#4105
20180009801
2018-01-11

Salts of aza-bicyclic di-aryl ethers and methods to make them or their precursors

#4106
20180009753
2018-01-11

METHOD FOR PREPARING AN ANTIFIBROTIC AGENT

#4107
20180002364
2018-01-04

Crystal of ammonium N-acetylneuraminate anhydrate, and process for producing same

#4108
20180002341
2018-01-04

Asymmetric synthesis of funapide

#4109
20180002338
2018-01-04

Short-acting benzodiazepine salts and their polymorphic forms

#4110
20180002326
2018-01-04

Production method of thiazole derivative

#4111
20180002317
2018-01-04

Crystalline salt form of (S)-(2-(6 chloro-7-methyl-1H-benzo[d]imidazol-2-yl)-2-methylpyrrolidin-1-yl)(5-methoxy-2-(2H-1,2,3-triazol-2-yl)phenyl)methanone as orexin receptor antagonist

#4112
20180002310
2018-01-04

CRYSTALLINE FORMS OF EFINACONAZOLE

#4113
20180002282
2018-01-04

Mono- or di-substituted indole derivatives as dengue viral replication inhibitors

#4114
20180002273
2018-01-04

Solid forms of desvenlafaxine

#4115
20180002247
2018-01-04

METHODS FOR CHIRAL RESOLUTION OF TROLOX

#4116
20180000879
2018-01-04

Methods of purifying cannabinoids, compositions and kits thereof

#4117
20180000845
2018-01-04

Complexes of celecoxib and its salts and derivatives, process for the preparation thereof and pharmaceutical compositions containing them

#4118
20180000749
2018-01-04

Polymorphic and amorphous forms of (R)-2-hydroxy-2-methyl-4-(2,4,5-trimethyl-3,6-dioxocyclohexa-1,4-dienyl)butanamide

#4119
20170369475
2017-12-28

Flibanserin Hydrate

#4120
20170369423
2017-12-28

Crystalline modification of propanil

#4121
20170362247
2017-12-21

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl and solid state forms thereof

#4122
20170362229
2017-12-21

Crystalline solid forms of a BET inhibitor

#4123
20170362212
2017-12-21

Process for preparation of luliconazole

#4124
20170362189
2017-12-21

Crystalline forms of trisodium supramolecular complex comprising valsartan and AHU-377 and methods thereof

#4125
20170362175
2017-12-21

Forms of apremilast

#4126
20170362159
2017-12-21

Method for enhancing uniformity of crystallized succinic acid and purified succinic acid produced by the same

#4127
20170360935
2017-12-21

Formulations of a PI3K/mTor-inhibitor for intravenous administration

#4128
20170360730
2017-12-21

Modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

#4129
20170355684
2017-12-14

Crystalline isoxazole hydroxamic acid compounds

#4130
20170355666
2017-12-14

POLYMORPHS OF CDDO ETHYL ESTER AND USES THEREOF

#4131
20170355665
2017-12-14

(2S,4R)-5-(5′-chloro-2′-fluorobiphenyl-4-yl)-4-(ethoxyoxalylamino)-2-hydroxymethyl-2-methylpentanoic acid

#4132
20170349609
2017-12-07

Crystalline form of cefamandole nafate compound, preparation and preparing method thereof

#4133
20170349608
2017-12-07

Crystalline form of rifaximin and process for its preparation

#4134
20170349603
2017-12-07

Efficient method for producing and purifying anhydrous sugar alcohol

#4135
20170349592
2017-12-07

Polymorphic substance of yonkenafil hydrochloride, preparation method therefor, and composition and use thereof

#4136
20170349584
2017-12-07

Process for preparing N-(5-(3-(7-(3-fluorophenyl)-3H-imidazo [4,5-C]pyridin-2-yl)-1H-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide

#4137
20170349533
2017-12-07

STABLE SOLID FORMS OF ENCLOMIPHENE AND ENCLOMIPHENE CITRATE

#4138
20170349518
2017-12-07

Crystalline form of cannabidiol

#4139
20170349517
2017-12-07

Crystalline cannabidivarin

#4140
20170342084
2017-11-30

REDUCTION OF ALPHA, BETA-UNSATURATED KETONE LEVELS IN MORPHINAN DERIVATIVE COMPOSITIONS

#4141
20170342083
2017-11-30

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#4142
20170342075
2017-11-30

Salt of pyrrolo[2,3-D]pyrimidine compound and novel polymorph of salt

#4143
20170342061
2017-11-30

CRYSTAL FORM I OF CANAGLIFLOZIN AND PREPARATION METHOD THEREOF

#4144
20170342037
2017-11-30

Crystal form of neptinib di-p-methylbenzenesulfonate, preparation method thereof, and pharmaceutical composition containing same

#4145
20170340584
2017-11-30

MODIFIED TAURINE, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING METABOLIC DISEASES CONTAINING SAME

#4146
20170334929
2017-11-23

Diaryl macrocycles as modulators of protein kinases

#4147
20170334921
2017-11-23

Crystalline forms of a bruton's tyrosine kinase inhibitor

#4148
20170334881
2017-11-23

Nicotine salts, co-crystals, and salt co-crystal complexes

#4149
20170334877
2017-11-23

Revaprazan hydrochloride polymorphs and preparation method therefor

#4150
20170334860
2017-11-23

Polymorphs of Ivacaftor, process for its preparation and pharmaceutical composition thereof

#4151
20170333438
2017-11-23

Crystalline forms of (2R,5S,13AR)-8-hydroxy-7,9-dioxo-N-(2,4,6-trifluorobenzyl)-2,3,4,5,7,9,13,13A- octahydro-2,5-methanopyrido[1′,2′:4,5]pyrazino[2,1-B] [1,3] oxazepine-10-carboxamide

#4152
20170333311
2017-11-23

Oral care composition comprising zinc-lysine complex

#4153
20170327499
2017-11-16

Lyophilized composition of a diazabicyclooctane compound and process of producing the same

#4154
20170327486
2017-11-16

Methods for the preparation of charged crosslinkers

#4155
20170327484
2017-11-16

Process for synthesizing 2-hydroxy-6-((2-(1-isopropyl-1H-pyrazol-5-yl)-pyridin-3-yl)methoxy)benzaldehyde

#4156
20170327467
2017-11-16

Cocrystal of lorcaserin, preparation methods, pharmaceutical compositions and uses thereof

#4157
20170327464
2017-11-16

CRYSTALS OF LAQUINIMOD SODIUM AND IMPROVED PROCESS FOR THE MANUFACTURE THEREOF

#4158
20170326115
2017-11-16

Chemical compounds

#4159
20170320872
2017-11-09

Substantially pure vemurafenib and its salts

#4160
20170320850
2017-11-09

Crystalline CHClNOmalonate

#4161
20170320845
2017-11-09

Preparation of dialkyl esters of 2,5-furandicarboxylic acid

#4162
20170320822
2017-11-09

Crystalline (3Z,5S)-5-(hydroxymethyl)-1-[(2′-methyl-1,1′-biphenyl-4-yl)carbonyl]pyrrolidin-3-one O-methyloxime, and methods of using the same

#4163
20170319588
2017-11-09

Salt of fused heterocyclic derivative and crystal thereof

#4164
20170313724
2017-11-02

Crystalline forms of a therapeutic compound and uses thereof

#4165
20170313709
2017-11-02

Crystalline form of JAK kinase inhibitor bisulfate and a preparation method thereof

#4166
20170313706
2017-11-02

Purinone derivative hydrochloride

#4167
20170313694
2017-11-02

Crystalline Form of (R)-7-Chloro-N-(Quinuclidin-3-YL)benzo[B]thiophene-2-Carboxamide Hydrochloride Monohydrate

#4168
20170313678
2017-11-02

Crystalline form of a substituted quinoline compound and pharmaceutical compositions thereof

#4169
20170313666
2017-11-02

Crystalline forms of tyrosine kinase inhibitors and their salts

#4170
20170313664
2017-11-02

NOVEL FORM OF PYRIMIDINE COMPOUND HAVING DIBENZYLAMINE STRUCTURE

#4171
20170305958
2017-10-26

Crystalline forms of 5α-androstane-3β,5,6β-triol and preparation methods therefor

#4172
20170305957
2017-10-26

Crystalline forms of 5α-androstane-3β,5,6β-triol and preparation methods therefor

#4173
20170305936
2017-10-26

SOLID STATE FORMS OF CRISABOROLE

#4174
20170305934
2017-10-26

Crystalline form of 3-((1R,3s,5S)-3-((7-((5-methyl-1H-pyrazol-3-yl)amino)-1,6-naphthyridin-5-yl)amino)-8-azabicyclo[3.2.1]octan-8-yl)propanenitrile

#4175
20170305919
2017-10-26

CRYSTALLINE FORMS OF A BRUTON'S TYROSINE KINASE INHIBITOR

#4176
20170305914
2017-10-26

Acid addition salt of ibrutinib

#4177
20170305905
2017-10-26

CRYSTALLINE FORM OF AN ANXIOLYTIC COMPOUND

#4178
20170305885
2017-10-26

Therapeutically active compounds and their methods of use

#4179
20170305858
2017-10-26

Amorphous form of lomitapide mesylate

#4180
20170305841
2017-10-26

Crystal forms of verapamil hydrochloride

#4181
20170298087
2017-10-19

L-proline complex of sodium-glucose cotransporter 2 inhibitor, monohydrate and crystal form thereof

#4182
20170298074
2017-10-19

Compounds as rearranged during transfection (RET) inhibitors

#4183
20170298073
2017-10-19

SALTS, CO-CRYSTALS, AMORPHOUS FORMS, AND CRYSTALLINE FORMS OF A CO-ACTIVATOR-ASSOCIATED ARGININE METHYLTRANSFERASE 1 (CARM1) INHIBITOR

#4184
20170298071
2017-10-19

Crystalline solid state form of the benzene sulphonic acid salt of 2-[(4S)-6-(4-chlorophenyl)-1-methyl-8-(methyloxy)-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepin-4-yl]-N-ethylacetamide

#4185
20170297999
2017-10-19

METHOD FOR PRODUCING TRIPHENYLBUTENE DERIVATIVE

#4186
20170296570
2017-10-19

High Drug Load Tablets Comprising Sofosbuvir

#4187
20170291883
2017-10-12

Salt of dicarboxylic acid compound

#4188
20170284986
2017-10-05

Metal coordination complex for detection of vapors and anions and process for the preparation thereof

#4189
20170283418
2017-10-05

Solid forms of (1S,4S)-4-(2-(((3S,4R)-3-fluorotetrahydro-2H-pyran-4-yl)amino)-8-((2,4,6-trichlorophenyl)amino)-9H-purin-9-yl)-1-methylcyclohexane-1-carboxamide and methods of their use

#4190
20170283404
2017-10-05

CRYSTALLINE FORMS OF 2-(4-(4-ETHOXY-6-OXO-1,6-DIHYDROPYRIDIN-3-YL)-2-FLUOROPHENYL)-N-(5-(1,1,1-TRIFLUORO-2-METHYLPROPAN-2-YL)ISOXAZOL-3-YL)ACETAMIDE

#4191
20170283399
2017-10-05

Crystalline forms of 6-((6,7-dimethoxyquinazolin-4-yl)oxy)-N,2-dimethylbenzofuran-3-carboxamide

#4192
20170283372
2017-10-05

Method for producing high-purity aqueous urea solution in urea production process

#4193
20170283354
2017-10-05

Process for the preparation of vitamin K2

#4194
20170275326
2017-09-28

IDIOPATHIC PULMONARY FIBROSIS-DETECTION, MONITORING, PREDICTION METHODS

#4195
20170275299
2017-09-28

Preparation method for benzoxazoleoxazine ketone compound and intermediate and crystal form thereof

#4196
20170275264
2017-09-28

CARBAMATE/UREA DERIVATIVES

#4197
20170275259
2017-09-28

Crystalline(2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2-methylpentanoic acid and uses thereof

#4198
20170275229
2017-09-28

Process for preparation of acitrecin

#4199
20170273953
2017-09-28

Crystalline solid forms of 6-carboxy-2-(3,5-dichlorophenyl)-benzoxazole

#4200
20170267810
2017-09-21

Crystal polymorphism of inclusion compound and method for producing same, and curable resin composition