ClassID:

90494

C07B2200/13 - page 3 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#601
20240150352
2024-05-09

Crystalline imidazo[4,5-b]pyridine compound, pharmaceutical compositions, and their use in treating medical conditions

#602
20240150299
2024-05-09

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#603
20240150289
2024-05-09

CRYSTALLINE CARBAZOLE DERIVATIVE

#604
20240148742
2024-05-09

METHOD OF SYNTHESIZING THYROID HORMONE ANALOGS AND POLYMORPHS THEREOF

#605
20240140990
2024-05-02

Crystalline salt forms of Boc-D-Arg-DMT-Lys-(Boc)-Phe-NH

#606
20240140985
2024-05-02

SALTS AND CRYSTAL FORMS OF GABA-A POSITIVE ALLOSTERIC MODULATOR

#607
20240140967
2024-05-02

Process for preparing 7H-pyrrolo[2,3-d]pyrimidine derivatives and synthetic intermediates thereof

#608
20240140964
2024-05-02

DIARYL MACROCYCLES AS MODULATORS OF PROTEIN KINASES

#609
20240140911
2024-05-02

CRYSTALLINE L-ARGININE SALT OF (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMETHYL)BENZYLOXY)-1,2,3, 4-TETRAHYDROCYCLO-PENTA [B]INDOL-3-YL)ACETIC ACID(COMPOUND1) FOR USE IN SIPI RECEPTOR-ASSOCIATED DISORDERS

#610
20240140908
2024-05-02

A PHARMACEUTICAL SALT OF AN ARYLPYRROLE DERIVATIVE

#611
20240140897
2024-05-02

CO-CRYSTAL OF COENZYME QH AND NICOTINAMIDE, PREPARATION METHOD THEREFOR AND USE THEREOF

#612
20240132523
2024-04-25

SALTS AND CRYSTALLINE FORMS OF A PD-1/PD-L1 INHIBITOR

#613
20240132520
2024-04-25

NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS

#614
20240132512
2024-04-25

CRYSTAL FORMS OF AN ANTI-SARS COV-2 AGENT

#615
20240132510
2024-04-25

Crystalline forms of (S)-1-(4-fluorophenyl)-1-(2-(4-(6-(1-methyl-1H-pyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl)piperazinyl)-pyrimidin-5-yl)ethan-1-amine and methods of making

#616
20240132503
2024-04-25

SALT FORM AND CRYSTAL FORM OF PYRAZOLE SUBSTITUTED IMIDAZO[1,2- A]QUINOXALINE DERIVATIVE

#617
20240132501
2024-04-25

ION CHANNEL MODULATORS

#618
20240132498
2024-04-25

CRYSTALLINE FORMS OF 5-(3,4-DIFLUOROBENZYL)-8-((1R,4R)-4-METHYLCYCLOHEXYL)-6,9-DIOXO-2,5,8-TRIAZASPIRO[3.5]NONANE-2-CARBALDEHYDE

#619
20240132478
2024-04-25

COCRYSTAL

#620
20240132474
2024-04-25

THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE

#621
20240132472
2024-04-25

NOVEL CRYSTALLINE FORMS OF 1-(4-{[6-AMINO-5-(4-PHENOXY-PHENYL)-PYRIMIDIN-4-YLAMINO]-METHYL}-4-FLUORO-PIPERIDIN-1-YL)-PROPENONE, SALT FORMS THEREOF, AND PROCESSES TO OBTAIN

#622
20240132447
2024-04-25

Polymorphs of (2S,5R)-5-(2-chlorophenyl)-1-(2′-methoxy-[1,1′-biphenyl]-4-carbonyl)pyrrolidine-2-carboxylic acid and preparation processes thereof

#623
20240132442
2024-04-25

BRANCHED-CHAIN AMINO ACID CRYSTALLIZATION METHOD CAPABLE OF SUSTAINABLY CYCLING AMMONIA

#624
20240132352
2024-04-25

BIS(FLUOROSULFONYL)IMIDE SALTS AND PREPARATION METHOD THEREOF

#625
20240128076
2024-04-18

Enhanced perovskite materials for photovoltaic devices

#626
20240124461
2024-04-18

PROCESSES FOR THE PREPARATION OF ZANUBRUTINIB AND INTERMEDIATES THEREOF

#627
20240124458
2024-04-18

POLYMORPHS OF AVAPRITINIB AND METHODS FOR PREPARING THE POLYMORPHS

#628
20240124456
2024-04-18

AZA-ERGOLINE DERIVATIVE AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#629
20240124441
2024-04-18

POLYMORPH OF LATREPIRDINE DIHYDROCHLORIDE

#630
20240124437
2024-04-18

INJECTABLE LURASIDONE SUSPENSION AND PREPARATION METHOD THEREFOR

#631
20240124425
2024-04-18

Solid state forms of Belumosudil and Belumosudil salts

#632
20240124398
2024-04-18

PHARMACEUTICALLY ACCEPTABLE SALTS OF PSILOCIN AND USES THEREOF

#633
20240124391
2024-04-18

SOLABEGRON ZWITTERION AND USES THEREOF

#634
20240122936
2024-04-18

Method of synthesizing thyroid hormone analogs and polymorphs thereof

#635
20240122925
2024-04-18

SHP2 PHOSPHATASE INHIBITORS AND METHODS OF MAKING AND USING THE SAME

#636
20240122910
2024-04-18

SOLID FORMS OF {[5-(3-CHLOROPHENYL)-3-HYDROXYPYRIDINE-2-CARBONYL]AMINO}ACETIC ACID, COMPOSITIONS, AND USES THEREOF

#637
20240116953
2024-04-11

PHTHALOCYANINE COMPOUND

#638
20240116940
2024-04-11

Crystalline form of (s)-7-(1-acryloylpiperidin-4-yl)- 2-(4-phenoxyphenyl)-4,5,6,7-tetra- hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#639
20240116937
2024-04-11

Polymorph of (1S,2S,3S,5R)-3-((6-(difluoromethyl)-5-fluoro-1,2,3,4-tetrahydroisoquinolin-8-yl)oxy)-5-(4-methyl-7H-pyrrolo[2,3-D]pyrimidin-7-yl)cyclopentane-1,2-diol

#640
20240116932
2024-04-11

COCRYSTALLINE FORMS OF FGFR3 INHIBITORS

#641
20240116927
2024-04-11

INDAZOLE INHIBITORS OF THE WNT SIGNAL PATHWAY AND THERAPEUTIC USES THEREOF

#642
20240116925
2024-04-11

SALT OF NITROGEN-CONTAINING FUSED HETEROCYCLIC COMPOUND OR CRYSTAL FORM THEREOF, AND PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF

#643
20240116913
2024-04-11

A CRYSTALLINE FORM OF (4-METHYL-2-[1,2,3]TRIAZOL-2-YL-PHENYL)-[(R)-3-(3-[1,2,3]TRIAZOL-2-YL-BENZYL)-MORPHOLIN-4-YL]-METHANONE

#644
20240116904
2024-04-11

Polymorphisms of HM30181 mesylate

#645
20240116891
2024-04-11

MARALIXIBAT SOLID FORMS, INTERMEDIATES AND PROCESSES OF MAKING SAME

#646
20240116884
2024-04-11

Salts of Viloxazine

#647
20240116880
2024-04-11

CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS

#648
20240116853
2024-04-11

2-HYDROXY-5-[2-(4-(TRIFLUOROMETHYLPHENYL)ETHYLAMINO)]BENZOIC ACID CRYSTAL FORMS AND PREPARATION METHOD THEREFOR

#649
20240116850
2024-04-11

COMPOSITIONS AND METHODS RELATED TO BICYCLO[2.2.1] HEPTANAMINE-CONTAINING COMPOUNDS

#650
20240115552
2024-04-11

MEBENDAZOLE POLYMORPH FOR TREATMENT AND PREVENTION OF TUMORS

#651
20240109932
2024-04-04

Crystalline solids of nicotinic acid mononucleotide and esters thereof and methods of making and use

#652
20240109876
2024-04-04

COMPOSITIONS FOR TREATMENT OF OCULAR DISEASES

#653
20240109844
2024-04-04

CRYSTALLINE SALTS OF A PLASMA KALLIKREIN INHIBITOR

#654
20240108622
2024-04-04

INHALABLE IMATINIB FORMULATIONS, MANUFACTURE, AND USES THEREOF

#655
20240101564
2024-03-28

SALTS OF A PI3Kdelta INHIBITOR, CRYSTALLINE FORMS, METHODS OF PREPARATION, AND USES THEREFORE

#656
20240101551
2024-03-28

CRYSTAL FORM AND SALT FORM OF BROMINE DOMAIN PROTEIN INHIBITOR AND PREPARATION METHOD THEREFOR

#657
20240101530
2024-03-28

HDAC INHIBITOR SOLID STATE FORMS

#658
20240101520
2024-03-28

PYRIMETHAMINE CRYSTAL FORM

#659
20240101514
2024-03-28

Pharmaceutically acceptable salts and compositions thereof

#660
20240101505
2024-03-28

SALTS AND ESTERS OF APX3330 AND THERAPEUTIC USES THEREOF

#661
20240101504
2024-03-28

HYDROXYALKANOIC ACID CRYSTAL PRODUCTION METHOD AND HYDROXYALKANOIC ACID CRYSTAL POLYMORPH

#662
20240092825
2024-03-21

CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS

#663
20240092787
2024-03-21

PHARMACEUTICAL PROCESS AND INTERMEDIATES

#664
20240092786
2024-03-21

Crystalline form of (S)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra-hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#665
20240092772
2024-03-21

CRYSTALLINE FORM OF A PIPERAZINYL-THIAZOLE DERIVATIVE

#666
20240092771
2024-03-21

CRYSTAL FORM OF LANIFIBRANOR, PREPARATION METHOD THEREFOR, AND USE THEREOF

#667
20240092768
2024-03-21

CRYSTAL FORM OF ANTI-INFLUENZA VIRUS COMPOUND, PREPARATION METHOD FOR CRYSTAL FORM, AND USE OF CRYSTAL FORM

#668
20240092748
2024-03-21

PHARMACEUTICAL FORMULATION OF ODEVIXIBAT

#669
20240092727
2024-03-21

CRYSTALLINE 4-((L-VALYL)OXY)BUTANOIC ACID

#670
20240091226
2024-03-21

Forms and Formulations Of A Tyrosine Kinase Non-Receptor 1 (TNK1) Inhibitor

#671
20240090532
2024-03-21

COMPOSITIONS AND METHODS FOR SOLIDIFIED FERMENTED ANIMAL FEED

#672
20240083935
2024-03-14

CYTOSINE-TYPE BRIDGED NUCLEOSIDE AMIDITE CRYSTALS AND METHOD FOR PRODUCING SAME

#673
20240083914
2024-03-14

Crystalline Polymorphs of a Muscarinic Acetylcholine Receptor Agonist

#674
20240083911
2024-03-14

Method for preparing heterocyclic derivative compound, composition containing same compound, and hydrate of same compound

#675
20240083902
2024-03-14

CRYSTALLINE FORMS OF 3-(IMIDAZO[1,2-B]PYRIDAZIN-3-YLETHYNYL)-4-METHYL-N-{4-[(4-METHYLPIPERAZIN-1-YL)METHYL]-3-(TRIFLUOROMETHYL)PHENYL}BENZAMIDE AND ITS MONO HYDROCHLORIDE SALT

#676
20240083870
2024-03-14

SALTS OF PYRIDINYLMETHYLENEPIPERIDINE DERIVATIVES AND USES THEREOF

#677
20240083856
2024-03-14

Polymorphs of pyrimidine cyclohexyl glucocorticoid receptor modulators

#678
20240082335
2024-03-14

PROCESSES AND SYSTEMS FOR CONVERTING CANNABINOIDS INTO CANNABINOID DERIVATIVES AND ISOLATING THE SAME

#679
20240082248
2024-03-14

PROCESS FOR PREPARATION OF MAVACAMTEN AND SOLID STATE FORMS THEREOF

#680
20240082210
2024-03-14

CROMOLYN METAL COMPLEXES AS ENHANCED PHARMACEUTICAL FORMULATIONS AND METHOD OF USING THE SAME

#681
20240076365
2024-03-07

GREMLIN-1 CRYSTAL STRUCTURE AND INHIBITORY ANTIBODY

#682
20240076342
2024-03-07

De novo design of potent and selective interleukin mimetics

#683
20240076290
2024-03-07

SOLID FORMS OF A MODULATOR OF HEMOGLOBIN

#684
20240076275
2024-03-07

OXAZOLE COMPOUND CRYSTAL

#685
20240076268
2024-03-07

Polypeptide Integrin Antagonists

#686
20240076265
2024-03-07

Phenylcarbamate crystalline form and method for manufacturing the same

#687
20240076261
2024-03-07

METHOD FOR PREPARING HIGH-BULK-DENSITY IBUPROFEN SPHERICAL CRYSTAL AND PRODUCT THEREOF

#688
20240067659
2024-02-29

Method for preparing heterocyclic derivative compound, composition containing same compound, and hydrate of same compound

#689
20240067647
2024-02-29

SOLID STATE FORMS

#690
20240067644
2024-02-29

POLYMORPHS OF THE HYDROCHLORIDE SALT OF LINAPRAZAN GLURATE

#691
20240067628
2024-02-29

SSTR4 AGONIST SALTS

#692
20240067609
2024-02-29

LAUROLACTAM PREPARATION METHOD, SYNTHESIZING DEVICE THEREFOR, LAUROLACTAM COMPOSITION PREPARED THEREBY, AND POLYLAUROLACTAM PREPARATION METHOD USING SAME

#693
20240059699
2024-02-22

Crystalline form of (S)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra-hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#694
20240059683
2024-02-22

SOLID FORMS OF AN SGC STIMULATOR

#695
20240059679
2024-02-22

GLP-1 Receptor Agonists and Uses Thereof

#696
20240059669
2024-02-22

COCRYSTAL OF A CDK INHIBITOR

#697
20240059666
2024-02-22

PROCESSES AND INTERMEDIATE FOR THE LARGE-SCALE PREPARATION OF 2,4,6-TRIFLUORO-N-[6-(1-METHYL-PIPERIDINE-4-CARBONYL)-PYRIDIN-2-YL]-BENZAMIDE HEMISUCCINATE, AND PREPARATION OF 2,4,6-TRIFLUORO-N-[6-(1-METHYL-PIPERIDINE-4-CARBONYL)-PYRIDIN-2-YL]-BENZAMIDE ACETATE

#698
20240059662
2024-02-22

SOLID FORMS OF A COMPOUND

#699
20240059652
2024-02-22

AMORPHOUS MELANOCORTIN RECEPTOR AGONIST AND METHOD FOR PREPARING SAME

#700
20240051984
2024-02-15

METHOD FOR PREPARING DISODIUM 5'-GUANYLATE HEPTAHYDRATE CRYSTAL

#701
20240051962
2024-02-15

SOLID FORMS OF A NUCLEOSIDE ANALOGUE AND USES THEREOF

#702
20240051957
2024-02-15

CRYSTALLINE FORM OF HETEROCYCLIC COMPOUND AS PROTEIN KINASE INHIBITOR

#703
20240051944
2024-02-15

CRYSTALLINE FORM II OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD THEREFOR

#704
20240051942
2024-02-15

Solid form of compound

#705
20240051941
2024-02-15

CAPSID INHIBITORS FOR THE PREVENTION OF HIV

#706
20240051926
2024-02-15

SOLID FORMS OF AN N-TERMINAL DOMAIN ANDROGEN RECEPTOR INHIBITOR AND USES THEREOF

#707
20240051924
2024-02-15

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#708
20240051921
2024-02-15

CRYSTALLINE FORM OF A PHENOLIC TRPV1 AGONIST PRODRUG

#709
20240051920
2024-02-15

AN IMPROVED HIGHLY EFFICIENT PROCESS FOR THE PREPARATION OF NINTEDANIB AND PHARMACEUTICALLY ACCEPTABLE SALT THEREOF

#710
20240051919
2024-02-15

CRYSTALLINE FORM III OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD THEREFOR

#711
20240051913
2024-02-15

Cage silicate and method for producing the same

#712
20240043466
2024-02-08

SOLID FORMS OF A NUCLEOSIDE ANALOGUE AND USES THEREOF

#713
20240043465
2024-02-08

CO-CRYSTAL FORMS OF A NOVOBIOCIN ANALOG AND PROLINE

#714
20240043459
2024-02-08

Crystalline forms and methods of producing crystalline forms of a compound

#715
20240043457
2024-02-08

CRYSTALLINE FORMS OF 5-CHLORO-N4-[-2-(DIMETHYLPHOSPHORYL) PHENYL]-N2-{2-METHOXY-4-[4[(4-METHYLPIPERAZIN-1-YL) PIPERIDIN-1-YL] PHENYL} PYRIMIDINE-2,4-DIAMINE

#716
20240043456
2024-02-08

Crystalline Solid Meglumine Salt Inhibitor of BCL and Methods of Making and Using Same

#717
20240043437
2024-02-08

Crystal form of compound, and preparation method therefor and use thereof

#718
20240043434
2024-02-08

COCRYSTALS OF UPADACITINIB

#719
20240043432
2024-02-08

CRYSTALLINE COMPOSITION OF TILDACERFONT AND METHODS OF USE AND PREPARATION THEREOF

#720
20240043416
2024-02-08

SALT AND CRYSTAL FORM OF HA INHIBITOR COMPOUND

#721
20240043409
2024-02-08

CRYSTALLINE FORMS OF 5-[(1,1-DIOXIDO-4-THIOMORPHOLINYL)METHYL]-2-PHENYL-N-(TETRAHYDRO-2H-PYRAN-4-YL)-1H-INDOL-7-AMINE

#722
20240043408
2024-02-08

CRYSTAL FORM OF FIBROBLAST GROWTH FACTOR RECEPTOR INHIBITOR AND PREPARATION METHOD THEREFOR

#723
20240043407
2024-02-08

CRYSTALLINE FORM I OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND METHOD FOR PREPARING SAME

#724
20240043383
2024-02-08

Method of preparing indolin-2-one compound and method of using indolin-2-one

#725
20240043381
2024-02-08

Crystalline 5-methoxy-dipropyl tryptamine compounds

#726
20240041879
2024-02-08

INHALABLE IMATINIB FORMULATIONS, MANUFACTURE, AND USES THEREOF

#727
20240041874
2024-02-08

METHOD OF TREATING SCLC AND MANAGING NEUTROPENIA

#728
20240041873
2024-02-08

METHOD OF TREATING SCLC AND MANAGING HEPATOTOXICITY

#729
20240041872
2024-02-08

STABLE LURBINECTEDIN COMPOSITION

#730
20240034741
2024-02-01

METHODS FOR CRYSTALLIZATION OF DRUGS

#731
20240034740
2024-02-01

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#732
20240034738
2024-02-01

SOLID STATE FORMS OF SUBSTITUTED PYRAZOLOPYRIMIDINES AND USES THEREOF

#733
20240034718
2024-02-01

Salts and solid forms of (R)-1-(5-methoxy-1H-indol-1-yl)-N,N-dimethylpropan-2-amine

#734
20240025938
2024-01-25

NOVEL FORMS OF ANTIVIRAL NUCLEOSIDES

#735
20240025920
2024-01-25

SALT FORM USED AS CDC7 INHIBITOR AND CRYSTAL FORM THEREOF

#736
20240025915
2024-01-25

SOLID FORMS OF 4-(3,3-DIFLUORO-2,2-DIMETHYL-PROPANOYL)-3,5-DIHYDRO-2H-PYRIDO[3,4-F][1,4]OXAZEPINE-9-CARBONITRILE

#737
20240025897
2024-01-25

Crystalline hydrate of a JAK inhibitor compound

#738
20240025855
2024-01-25

TABLET COMPRISING MODOFLANER AS AN ACTIVE COMPONENT

#739
20240025841
2024-01-25

METHOD FOR OBTAINING CRYSTALLINE DIETHYLAMINO HYDROXYBENZOYL HEXYL BENZOATE

#740
20240024305
2024-01-25

Methods and compositions for treating retina-associated disease using CCR3-inhibitors

#741
20240018179
2024-01-18

Nucleotide hemi-sulfate salt for the treatment of hepatitis c virus

#742
20240018147
2024-01-18

SALT OF COMPOUND FOR DEGRADING BTK, CRYSTAL FORM THEREOF, AND USE THEREOF IN MEDICINE

#743
20240018143
2024-01-18

PROCESS FOR THE PREPARATION OF (9S)-N-[3-(6-METHYLPYRIMIDIN-4-YL)-3-AZABICYCLO[3.2.1]OCTAN-8-YL]-9-(2,3,4-TRIFLUOROPHENYL)-6,7,8,9-TETRAHYDRO-5H-[1,2,4]TRIAZOLO[1,5-A]AZEPIN-2-AMINE AND ITS SOLID FORM

#744
20240018142
2024-01-18

Crystal and amorphous form of tolebrutinib, preparation method therefor, and use thereof

#745
20240018091
2024-01-18

Polymorphic compounds and uses thereof

#746
20240010663
2024-01-11

Psilocybin and O-acetylpsilocin, salts and solid state forms thereof

#747
20240010656
2024-01-11

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#748
20240010654
2024-01-11

CRYSTALLINE FORMS OF A TYK2 INHIBITOR

#749
20240010653
2024-01-11

Crystalline Forms of 4-amino-N-[4-(methoxymethyl)phenyl]-7-(1-methylcyclopropyl)-6-(3-morpholinoprop-1-yn-1-yl)-7H-pyrrolo[2,3-d]pyrimidine-5-carboxamide

#750
20240010651
2024-01-11

Processes for the Preparation of Multicomponent Crystalline Forms of Active Pharmaceutical Ingredients Using Solvent Vapour

#751
20240010649
2024-01-11

CRYSTALLINE FORMS OF AN S1P RECEPTOR MODULATOR

#752
20240010646
2024-01-11

Urea Co-Crystal of Apixaban, and Preparation Method Therefor

#753
20240010633
2024-01-11

CRYSTALLINE FORM IV OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD THEREFOR

#754
20240010632
2024-01-11

SOLID STATE FORMS OF ERDAFITINIB SALTS AND PROCESSES FOR PREPARATION OF ERDAFITINIB

#755
20240010630
2024-01-11

Salts of obicetrapib and processes for their manufacture and intermediates thereof

#756
20240010629
2024-01-11

SOLID STATE FORM OF LEMBOREXANT

#757
20240010621
2024-01-11

Crystalline solid forms of salts of N-{4-[(6,7-dimethoxyquinolin-4-yl)oxy]phenyl}-N'-(4-fluorophenyl) cyclopropane-1,1-dicarboxamide, processes for making, and methods of use

#758
20240010617
2024-01-11

Crystalline forms of a cannabinoid receptor type 1 (CB1) modulator and methods of use and preparation thereof

#759
20240010616
2024-01-11

SIPONIMOD SALTS AND COCRYSTALS

#760
20240002413
2024-01-04

TITANIUM HETEROMETALLIC METAL-ORGANIC SOLIDS, METHOD FOR OBTAINING THEM AND THEIR USES

#761
20240002404
2024-01-04

SALT OF PYRROLOPYRIMIDINE COMPOUND, CRYSTALLINE FORM THEREOF, AND APPLICATION THEREOF

#762
20240002386
2024-01-04

SOLID FORMS OF 4-(5-(4-FLUOROPHENYL)-6-(TETRAHYDRO-2H-PYRAN-4-YL)-1,5-DIHYDROPYRROLO[2,3-F]INDAZOL-7-YL)BENZOIC ACID

#763
20240002356
2024-01-04

CRYSTALLINE PPAR-DELTA AGONIST

#764
20240002338
2024-01-04

Crystalline forms of compositions comprising psilocin and psilocybin

#765
20240002337
2024-01-04

SALTS AND SOLID FORMS OF (R)-1-(5-METHOXY-1H-INDOL-1-YL)-N,N-DIMETHYLPROPAN-2-AMINE

#766
20240002322
2024-01-04

METHOD FOR PREPARING INTERMEDIATE FOR SYNTHESIS OF SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST

#767
20230416276
2023-12-28

LYOPHILIZED PHARMACEUTICAL COMPOSITION AND USES OF A CRYSTALLIZED FORM OF LURBINECTEDIN

#768
20230416267
2023-12-28

Solid forms of Alpha-1062 gluconate

#769
20230416253
2023-12-28

Folate salts

#770
20230416252
2023-12-28

PROCESS TOWARD THE MANUFACTURE OF (6R,10S)-10-{4-[5-CHLORO-2-(4-CHLORO-1H-1,2,3-TRIAZOL-1-YL)PHENYL]-6-OXO-1(6H)-PYRIMIDINYL}- 1-(DIFLUOROMETHYL)-6-METHYL-1,4,7,8,9,10-HEXAHYDRO-11,15-(METHENO)PYRAZOLO[4,3-B][1,7]DIAZACYCLOTETRADECIN-5(6H)-ONE

#771
20230416250
2023-12-28

METHODS OF PREPARING HETEROARYL-KETONE FUSED AZADECALIN GLUCOCORTICOID RECEPTOR MODULATORS

#772
20230416234
2023-12-28

CRYSTAL FORM OF RESMETIROM, PREPARATION METHOD THEREFOR, AND USE THEREOF

#773
20230416223
2023-12-28

Niraparib Compositions

#774
20230416219
2023-12-28

R-MDMA CRYSTAL FORMS

#775
20230416212
2023-12-28

Crystalline forms of eravacycline

#776
20230416207
2023-12-28

CRYSTALLINE FORMS OF QUINAZOLINONE COMPOUND AND PROCESS FOR PREPARING THE SAME

#777
20230416197
2023-12-28

HIGH-EFFICIENCY CYCLIC PREPARATION METHOD FOR COLUMNAR TAURINE

#778
20230414547
2023-12-28

METHODS OF TREATING SYSTEMIC SCLEROSIS AND IDIOPATHIC PULMONARY FIBROSIS

#779
20230406866
2023-12-21

CRYSTALLINE FORMS OF IRAK DEGRADERS

#780
20230406865
2023-12-21

CRYSTAL FORM OF FREE BASE OF INHIBITOR CONTAINING BICYCLIC RING DERIVATIVE AND PREPARATION METHOD AND APPLICATION OF CRYSTAL FORM

#781
20230406857
2023-12-21

Salts and pharmaceutical compositions thereof for the treatment of inflammatory disorders

#782
20230406850
2023-12-21

CRYSTALLINE FORM OF HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#783
20230406827
2023-12-21

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#784
20230406823
2023-12-21

4-pivaloyloxy-n-methyltryptammonium chloride

#785
20230406815
2023-12-21

Crystalline prostacyclin (IP) receptor agonist and uses thereof

#786
20230404984
2023-12-21

Formulations of RBP4 inhibitors and methods of use

#787
20230404954
2023-12-21

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#788
20230399357
2023-12-14

CRYSTALLINE 19-NOR C3,3-DISUBSTITUTED C21-N-PYRAZOLYL STEROID

#789
20230399347
2023-12-14

CRYSTAL FORM OF L-GLUFOSINATE AND PREPARATION METHOD AND USE THEREOF

#790
20230399345
2023-12-14

CRYSTALLIZED FORM OF LURBINECTEDIN AND METHOD OF MAKING THE SAME

#791
20230399344
2023-12-14

A LYOPHILIZED PHARMACEUTICAL COMPOSITION

#792
20230399334
2023-12-14

PROCESS FOR PURIFYING NOROXYMORPHONE

#793
20230399333
2023-12-14

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#794
20230399331
2023-12-14

SOLID FORMS OF JAK INHIBITOR AND PROCESS OF PREPARING THE SAME

#795
20230399325
2023-12-14

SUCCINATE AND CRYSTAL FORM THEREOF AS THERAPEUTICS

#796
20230399321
2023-12-14

CRYSTALLINE FORM II OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD THEREFOR

#797
20230399316
2023-12-14

CRYSTAL FORMS OF 5-FLUORO-1-(4-FLUORO-3-(4-(PYRIMIDIN-2-YL)PIPERAZINE-1-CARBONYL)BENZYL)QUINAZOLINE-2,4(1H,3H)-DIONE AND PREPARATION THEREOF

#798
20230399313
2023-12-14

BIOLOGICAL ACTIVITIES OF 5-(2-(4-(4-FLUORO-2-METHYL-1H-INDOL-5-YLOXY)-6-METHOXYQUINOLIN-7-YLOXY)ETHYL)-5-AZASPIRO[2.4]-HEPTAN-7-OL CRYSTALLINE, PHOSPHORIC ACID SALT AND ITS ENANTIOMERS

#799
20230399311
2023-12-14

POLYMORPHS OF SUBSTITUTED ISOQUINOLINE-BASED RHO KINASE INHIBITORS

#800
20230399309
2023-12-14

DEUTERATED HPK1 KINASE INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#801
20230398086
2023-12-14

Methods of manufacturing 14,15-epoxyeicosatrienoic acid analogs and improved therapeutic delivery of same

#802
20230391815
2023-12-07

Efficient and scalable syntheses of nicotinoyl ribosides and reduced nicotinoyl ribosides, modified derivatives thereof, phosphorylated analogs thereof, adenylyl dinucleotide conjugates thereof, and novel crystalline forms thereof

#803
20230391791
2023-12-07

Compositions and methods for oral delivery of crystalline PRX-3140 potassium salt

#804
20230391771
2023-12-07

PROCESS FOR RACEMIZING AND ISOLATING ATROPISOMERS OF 7-CHLORO-6-FLUORO-1-(2-ISOPROPYL-4-METHYLPYRIDIN-3-YL)PYRIDO[2,3-D]PYRIMIDINE-2,4(1H,3H)-DIONE

#805
20230391759
2023-12-07

Solid forms of a dual RAF/MEK inhibitor

#806
20230391757
2023-12-07

Crystalline forms of a 4-pyrimidinesulfamide derivative aprocitentan

#807
20230391755
2023-12-07

Solid state forms of Belumosudil and Belumosudil salts

#808
20230391754
2023-12-07

CRYSTALLINE FORM OF SELINEXOR

#809
20230391749
2023-12-07

CRYSTALLINE AND AMORPHOUS FORMS OF A DELTA-OPIOID MODULATOR

#810
20230391746
2023-12-07

SOLID STATE FORMS OF PRALSETINIB AND PROCESS FOR PREPARATION THEREOF

#811
20230391737
2023-12-07

PROCESS FOR PREPARATION OF TAFAMIDIS AND SALTS THEREOF

#812
20230391729
2023-12-07

SUCCINATE SALTS OF N-(3-(4-(3-(DIISOBUTYLAMINO)PROPYL)PIPERAZIN-1-YL)PROPYL)-1H-BENZO[D]IMIDAZOL-2-AMINE, PREPARATION THEREOF AND USE OF THE SAME

#813
20230391724
2023-12-07

Crystalline forms of a pharmaceutical compound

#814
20230390286
2023-12-07

METHOD OF TREATING SCLC AND MANAGING THROMBOCYTOPENIA

#815
20230390285
2023-12-07

Lurbinectedin Composition and Methods Making the Same

#816
20230389586
2023-12-07

FUNCTIONAL CRYSTALLINE SWEETENER

#817
20230383439
2023-11-30

Nonlinear optical crystal of guanidinium tetrafluoroborate, preparation method and use thereof

#818
20230382944
2023-11-30

NOVEL COCRYSTALS OF DEXAMETHASONE

#819
20230382942
2023-11-30

Crystalline forms of a CD73 inhibitor and uses thereof

#820
20230382922
2023-11-30

Method of treatment of symptoms of menopause

#821
20230382914
2023-11-30

SOLID STATE FORMS OF LUMATEPERONE DITOSYLATE SALT

#822
20230382899
2023-11-30

CRYSTAL FORMS OF GLP-1R AGONISTS AND USES THEREOF

#823
20230382898
2023-11-30

CRYSTAL FORM OF MULTI-SUBSTITUTED BENZENE RING COMPOUND MALEATE, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#824
20230382897
2023-11-30

CRYSTALLINE FORM OF LIFITEGRAST, AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME

#825
20230382896
2023-11-30

ENANTIOMERICALLY PURIFIED GPER AGONIST FOR USE IN TREATING DISEASE STATES AND CONDITIONS

#826
20230382895
2023-11-30

CRYSTALLINE FORM III OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD THEREFOR

#827
20230382877
2023-11-30

METHOD FOR REFINING ACESULFAME POTASSIUM

#828
20230382872
2023-11-30

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#829
20230382867
2023-11-30

CRYSTALLINE SOLID FORMS OF N-{4-[(6,7-DIMETHOXYQUINOLIN-4-YL)OXY]PHENYL}-N'-(4-FLUOROPHENYL) CYCLOPROPANE-1,1-DICARBOXAMIDE, PROCESSES FOR MAKING, AND METHODS OF USE

#830
20230382861
2023-11-30

CRYSTALLINE (R)-5-CARBAMOYLPYRIDIN-3-YL-2-METHYL-4-(3-(TRIFLUOROMETHOXY)BENZYL)PIPERAZINE-1-CARBOXYLATE, COMPOSITIONS AND METHODS OF USE THEREOF

#831
20230382859
2023-11-30

Crystalline bis-miprocin fumarate

#832
20230382858
2023-11-30

PHARMACEUTICAL COMPOSITION COMPRISING 5-METHOXY-N,N-DIMETHYLTRYPTAMINE

#833
20230381167
2023-11-30

FREE BASE CRYSTALLINE FORM OF A COMPLEMENT COMPONENT C5a RECEPTOR

#834
20230374028
2023-11-23

SOLID STATE FORMS OF TRILACICLIB AND OF TRILACICLIB SALTS

#835
20230374027
2023-11-23

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#836
20230373990
2023-11-23

Pharmaceutical formulations for the treatment of gastrointestinal disorders

#837
20230373984
2023-11-23

CRYSTALLINE FORM I OF MELANOCORTIN RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD THEREFOR

#838
20230373967
2023-11-23

A STABLE CRYSTALLINE HYDRATE OF CLAZOSENTAN DISODIUM SALT

#839
20230373904
2023-11-23

POLYMORPHIC FORMS OF RAD1901-2HCL

#840
20230365619
2023-11-16

CRYSTALLINE SODIUM CHOLESTERYL SULFATE

#841
20230365618
2023-11-16

CRYSTALLINE THIOCHOLESTEROL

#842
20230365611
2023-11-16

ADVANTAGEOUS MORPHIC FORM OF AT-527 HEMI-SULFATE SALT

#843
20230365596
2023-11-16

CRYSTAL FORMS OF PYRIDOPYRAZOLE COMPOUNDS AND PREPARATION METHOD THEREFOR

#844
20230365564
2023-11-16

COCRYSTALS OF AN ADENOSINE A2B RECEPTOR ANTAGONIST

#845
20230365558
2023-11-16

TETRAHYDROISOQUINOLINE DERIVATIVE AND USE THEREOF

#846
20230365555
2023-11-16

CRYSTALLINE POLYMORPH FORM A OF A JAK INHIBITORAND METHODS FOR ITS PREPARATION

#847
20230365536
2023-11-16

CRYSTAL FORM OF COMPOUND AND FUMARIC ACID, PHARMACEUTICAL COMPOSITION AND METHOD FOR TREATING CORONAVIRUS-INDUCED DISEASES

#848
20230365518
2023-11-16

SALT OF BENZOTHIAZOLE COMPOUND, AND CRYSTAL FORM AND USE THEREOF

#849
20230365513
2023-11-16

TRIAZINE COMPOUND SALT, CRYSTAL FORM THEREOF, AND PRODUCTION METHOD THEREFOR

#850
20230365505
2023-11-16

PROCESSES FOR THE PREPARATION OF IVABRADINE HCl POLYMORPHS

#851
20230365503
2023-11-16

CRYSTAL FORM OF PYRIDINYLPHENYL COMPOUND AND PREPARATION METHOD THEREFOR

#852
20230365490
2023-11-16

Methods for making and using endoxifen

#853
20230364101
2023-11-16

DICLOFENAC PRODRUG AND USE OF THE SAME

#854
20230364093
2023-11-16

PHARMACEUTICAL COMPOSITION CONTAINING PALBOCICLIB AND LETROZOLE

#855
20230364092
2023-11-16

SOLID FORMS OF A TOLL-LIKE RECEPTOR MODULATOR

#856
20230364029
2023-11-16

POLYMORPHIC FORMS OF (R)-2-HYDROXY-2-METHYL-4-(2,4,5-TRIMETHYL-3,6-DIOXOCYCLOHEXA-1,4-DIENYL)BUTANAMIDE

#857
20230357809
2023-11-09

Solid form of (−)-Ambrox formed by a bioconversion of homofarnesol in the presence of a biocatalyst

#858
20230357322
2023-11-09

Method of manufacturing a pharmaceutical composition

#859
20230357318
2023-11-09

Solution phase synthesis of β-turn peptidomimetic cyclic salts

#860
20230357308
2023-11-09

CRYSTALLINE SODIUM CHOLESTERYL SULFONATE

#861
20230357293
2023-11-09

Crystal of Thyroid Hormone B Receptor Agonist, Process for Preparing The Same and Use Thereof

#862
20230357275
2023-11-09

SPIRO-SULFONAMIDE DERIVATIVES AS INHIBITORS OF MYELOID CELL LEUKEMIA-1 (MCL-1) PROTEIN

#863
20230357274
2023-11-09

Salts and polymorphs of certain MCL-1 inhibitors

#864
20230357243
2023-11-09

LSD DERIVATIVES, SYNTHESIS & METHOD FOR TREATMENT OF DISEASES AND DISORDERS

#865
20230357231
2023-11-09

Crystalline forms of a KRas G12C inhibitor

#866
20230357211
2023-11-09

SOLID FORMS OF A CDK4 INHIBITOR

#867
20230357191
2023-11-09

MODULATOR OF THE CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR, PHARMACEUTICAL COMPOSITIONS, METHODS OF TREATMENT, AND PROCESS FOR MAKING THE MODULATOR

#868
20230357190
2023-11-09

CRYSTALLINE FORMS OF A MAGL INHIBITOR

#869
20230357182
2023-11-09

SOLID FORMS OF (S)-1-((2',6-BIS(DIFLUOROMETHYL)-[2,4'-BIPYRIDIN]-5-YL)OXY)-2,4-DIMETHYLPENTAN-2-AMINE AND SALTS THEREOF

#870
20230357167
2023-11-09

POLYMORPHS OF BIS(FLUOROALKYL)-1,4-BENZODIAZEPINONE COMPOUNDS AND USES THEREOF

#871
20230357163
2023-11-09

SOLID STATE FORMS OF GEFAPIXANT AND PROCESS FOR PREPARATION THEREOF

#872
20230357137
2023-11-09

Synthesis of Sulfonamide Intermediates

#873
20230357135
2023-11-09

CRYSTALLINE FORMS OF OMADACYCLINE, METHODS OF SYNTHESIS THEREOF AND METHODS OF USE THEREOF

#874
20230357129
2023-11-09

PROCESS FOR ISOLATING 2-(4'-DIETHYLAMINO-2'-HYDROXYBENZOYL)BENZOIC ACID HEXYL ESTER

#875
20230357121
2023-11-09

CO-CRYSTAL OF KETOPROFEN, LYSINE AND GABAPENTIN, PHARMACEUTICAL COMPOSITIONS AND THEIR MEDICAL USE

#876
20230357113
2023-11-09

TAPINAROF POLYMORPHS

#877
20230355612
2023-11-09

PHARMACEUTICALLY ACCEPTABLE SALT OF CARIPRAZINE AND CRYSTAL FORM THEREOF, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#878
20230348522
2023-11-02

METHOD FOR PRODUCING BICYCLIC PHOSPHORAMIDITE

#879
20230348519
2023-11-02

Crystalline forms of (s)-2-ethylbutyl 2-(((s)-(((2r,3s,4r,5r)-5-(4-aminopyrrolo[2,1-f] [1,2,4]triazin-7-yl)-5-cyano-3,4-dihydroxytetrahydrofuran-2-yl)methoxy) (phenoxy) phosphoryl)amino)propanoate

#880
20230348481
2023-11-02

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#881
20230348446
2023-11-02

Type II crystalline topramezone sodium salt hydrate, preparation method therefor and use thereof

#882
20230348443
2023-11-02

CRYSTAL FORM OF POLYCYCLIC ANAPLASTIC LYMPHOMA KINASE INHIBITOR

#883
20230348433
2023-11-02

Polymorphs of [2-(1H-indol-3-yl)-1H-imidazol-4- yl] (3,4,5-trimethoxyphenyl)methanone and its salts

#884
20230348424
2023-11-02

HETEROCYCLIC COMPOUNDS AND METHODS OF USE

#885
20230348388
2023-11-02

Highly purified batches of pharmaceutical grade migalastat and methods of producing the same

#886
20230348385
2023-11-02

POLYMORPHS OF 5-BROMO-6-CHLORO-3-INDOXYL CAPRYLATE

#887
20230348383
2023-11-02

CRYSTALLINE 5-METHOXY-N,N-DIALLYLTRYPTAMINE COMPOUNDS

#888
20230348382
2023-11-02

Crystalline psilacetin derivatives

#889
20230348381
2023-11-02

COMPOSITION COMPRISING A BENZOATE SALT OF 5-METHOXY-N,N-DIMETHYLTRYPTAMINE

#890
20230348377
2023-11-02

PURE FORMS OF CRYSTALLINE ATICAPRANT

#891
20230348372
2023-11-02

PROCESS FOR SYNTHESIZING TRIARYLMETHANE SULFONE COMPOUNDS

#892
20230348363
2023-11-02

COMPOUNDS AND THEIR USE

#893
20230348352
2023-11-02

METHODS FOR SYNTHESIZING ANHYDROUS LACTIC ACID

#894
20230340010
2023-10-26

PREPARATION AND USES OF OBETICHOLIC ACID

#895
20230339975
2023-10-26

CRYSTALLINE FORM OF SHP2 INHIBITOR, AND COMPOSITION THEREOF, PREPARATION METHOD THEREFOR, AND USE THEREOF

#896
20230339967
2023-10-26

SOLID FORMS OF AN S1P-RECEPTOR MODULATOR

#897
20230339962
2023-10-26

SOLID STATE FORMS OF SEP-363856 AND PROCESS FOR PREPARATION THEREOF

#898
20230339957
2023-10-26

DOSAGE FORM COMPOSITIONS COMPRISING AN INHIBITOR OF BRUTON'S TYROSINE KINASE

#899
20230339933
2023-10-26

Methods for the treatment of gastro-intestinal disorders

#900
20230339928
2023-10-26

Processes and intermediates for the preparation of soluble guanylate cyclase stimulators