ClassID:

90494

C07B2200/13 - page 4 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#901
20230339920
2023-10-26

PREPARATION METHOD FOR AND CRYSTAL FORM OF 3-ARYLOXY-3-FIVE-MEMBERED HETEROARYLPROPYLAMINE COMPOUND

#902
20230339918
2023-10-26

CRYSTAL FORMS OF CRENOLANIB AND METHODS OF USE THEREOF

#903
20230339911
2023-10-26

PYRIDAZINONE COMPOUNDS

#904
20230339901
2023-10-26

SOLID FORMS COMPRISING (S)-2-(2,6-DIOXOPIPERIDIN-3-YL)-4-((2-FLUORO-4-((3-MORPHOLINOAZETIDIN-1-YL)METHYL)BENZYL)AMINO)ISOINDOLINE-1,3-DIONE AND SALTS THEREOF, AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME

#905
20230339899
2023-10-26

PROCESS FOR PREPARING A TETRAZOLE-SUBSTITUTED ANTHRANILIC ACID DIAMIDE DERIVATIVE

#906
20230339880
2023-10-26

COMPOSITIONS OF AJULEMIC ACID AND USES THEREOF

#907
20230339842
2023-10-26

Trientine tetrahydrochloride and a method of preparation and a pharmaceutical composition thereof

#908
20230339836
2023-10-26

METHOD FOR PRODUCING REDUCED COENZYME Q10 FORM II CRYSTALS

#909
20230339835
2023-10-26

2,3,5-TRIMETHYL-6-NONYLCYCLOHEXA-2,5-DIENE-1,4-DIONE FOR SUPPRESSING AND TREATING ALPHA-SYNUCLEINOPATHIES, TAUOPATHIES, AND OTHER DISORDERS

#910
20230331762
2023-10-19

CRYSTALLINE FORM OF ASPACYTARABINE

#911
20230331739
2023-10-19

INDOLO HEPTAMYL OXIME ANALOG CRYSTAL AS PARP INHIBITOR AND METHOD FOR PREPARING SAME

#912
20230331735
2023-10-19

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#913
20230331731
2023-10-19

CRYSTAL FORM OF PYRROLO HETEROCYCLIC DERIVATIVE AND PREPARATION METHOD THEREFOR

#914
20230331730
2023-10-19

CRYSTAL OF PYRIMIDINE COMPOUND

#915
20230331728
2023-10-19

Tebipenem pivoxil crystalline forms, compositions including the same, methods of manufacture, and methods of use

#916
20230331727
2023-10-19

Method for the production of lumateperone and its salts

#917
20230331712
2023-10-19

SOLID FORMS OF (R)-1(2,2-DIFLUOROBENZO[D][1,3]DIOXOL-5-YL)-N-(1-(2,3-DIHYDROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2-YL)-1H-INDOL-5-YL)CYCLOPROPANECARBOXAMIDE

#918
20230331703
2023-10-19

EGFR inhibitors

#919
20230331700
2023-10-19

Compound having cyclic structure

#920
20230331678
2023-10-19

PPARG inverse agonists and uses thereof

#921
20230331677
2023-10-19

Crystal forms of 2-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate

#922
20230331671
2023-10-19

CRYSTALLINE DIMETHYL TRYPTAMINE ANALOGUES

#923
20230330117
2023-10-19

Method for treating anxiety disorders, headache disorders, and eating disorders with psilocybin

#924
20230322812
2023-10-12

CRYSTALLINE FORM OF HETEROBICYCLIC COMPOUND

#925
20230322797
2023-10-12

SOLID FORMS, PHARMACEUTICAL COMPOSITIONS AND PREPARATION OF HETEROAROMATIC MACROCYCLIC ETHER COMPOUNDS

#926
20230322794
2023-10-12

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#927
20230322786
2023-10-12

SOLID STATE FORMS OF AT-001 AND PROCESS FOR PREPARATION THEREOF

#928
20230322760
2023-10-12

Crystal form of azaindole derivative and use thereof

#929
20230322755
2023-10-12

CRYSTAL OF COMPOUND X7 HYDROCHLORIDE AND ITS PREPARATION METHOD AND APPLICATION

#930
20230322737
2023-10-12

Stable salt and crystal forms of 2-[3-({1-[2-(dimethylamino)ethyl]-2-(2,2-dimethylpropyl)-1H-1,3-benzodiazol-5-yl}sulfonyl)azetidin-1-yl]ethan-1-ol

#931
20230322727
2023-10-12

SOLID FORMS OF A COT INHIBITOR COMPOUND

#932
20230322717
2023-10-12

SOLID FORM OF PYRAZINE SUBSTITUTED NICOTINAMIDE, AND PREPARATION AND USE THEREOF

#933
20230322687
2023-10-12

SALT OF ARYLAMINOQUINAZOLINE-CONTAINING COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#934
20230322686
2023-10-12

Olaparib oxalic acid cocrystals and their pharmaceutical use

#935
20230322680
2023-10-12

CRYSTALLINE FORMS OF PITAVASTATIN CALCIUM

#936
20230322679
2023-10-12

CRYSTAL FORM OF QUINOLINE COMPOUND AND PROCESS FOR ITS PRODUCTION

#937
20230322666
2023-10-12

CRYSTALLINE COMPLEXES

#938
20230322657
2023-10-12

CRYSTALLINE EDG-2 RECEPTOR ANTAGONIST AND METHODS OF MAKING

#939
20230313072
2023-10-05

Composite Form of Tetraacetylenediamine

#940
20230312633
2023-10-05

SALTS AND POLYMORPHS OF CETHROMYCIN FOR THE TREATMENT OF DISEASE

#941
20230312606
2023-10-05

MCL-1 INHIBITOR FORMULATIONS

#942
20230312602
2023-10-05

SALT FORMS AND SOLVATES OF MCI-1 ANTAGONISTS

#943
20230312595
2023-10-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#944
20230312594
2023-10-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#945
20230312593
2023-10-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1- carboxamide and solid state forms thereof

#946
20230312584
2023-10-05

SALT OF NUCLEOSIDE ANALOG, AND CRYSTAL FORM, PHARMACEUTICAL COMPOSITION AND USE THEREOF

#947
20230312582
2023-10-05

Salts Of Nitrogen-Containing Heterocyclic Compound, And Solid Forms Of Salts, Pharmaceutical Composition And Use Thereof

#948
20230312573
2023-10-05

NOVEL SALTS, CRYSTALS, AND CO-CRYSTALS

#949
20230312561
2023-10-05

SOLID FORMS OF (Z)-METHYL 3-(((4-(N-METHYL-2-(4-METHYLPIPERAZIN-1-YL)ACETAMIDO)PHENYL)AMINO)(PHENYL)METHYLENE)-2-OXO-2,3-DIHYDRO-1H-PYRROLO[2,3-B]PYRIDINE-6-CARBOXYLATE AND SALTS THEREOF

#950
20230312559
2023-10-05

CRYSTALLINE FORM OF HYDROCHLORIDE SALT OF QUINOLINE DERIVATIVE

#951
20230312551
2023-10-05

SALT OF 2-(SUBSTITUTED PYRIMIDINYL) THIAZOLE CARBOXAMIDE COMPOUND, AND COMPOSITION AND USE THEREOF

#952
20230312530
2023-10-05

SALT OF RHO-ASSOCIATED PROTEIN KINASE INHIBITOR, SOLID FORM OF THE SALT, PREPARATION METHOD FOR SAME, AND USES THEREOF

#953
20230312505
2023-10-05

SOLID STATE FORMS OF CYANTRANILIPROLE

#954
20230312488
2023-10-05

PROCESS FOR THE PREPARATION OF TAUTOMERIC FORMS OF SUNSCREENS

#955
20230312486
2023-10-05

POLYMORPHIC FORMS OF A ROR INHIBITING COMPOUND AND PROCESSES FOR ITS PREPARATION

#956
20230312473
2023-10-05

PROCESS FOR THE PREPARATION OF BIHETEROARYL COMPOUNDS AND CRYSTAL FORMS THEREOF

#957
20230312469
2023-10-05

Crystalline salt forms of mesembrine

#958
20230303589
2023-09-28

CRYSTALLINE FORMS OF CFTR MODULATORS

#959
20230303582
2023-09-28

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#960
20230303572
2023-09-28

18-MC SALT FORMS

#961
20230303557
2023-09-28

CRYSTALLINE FORM OF TLR8 AGONIST

#962
20230303542
2023-09-28

SOLID FORMS OF A PARP14 INHIBITOR

#963
20230303529
2023-09-28

Crystalline forms of carbazole inhibitors of RhoGTPase for the treatment of disease

#964
20230303500
2023-09-28

Crystalline substituted pyrazines as PGI2 receptor agonists

#965
20230303492
2023-09-28

Crystalline freebase forms of a biphenyl compound

#966
20230301983
2023-09-28

BROMODOMAIN INHIBITOR

#967
20230301979
2023-09-28

COMBINATIONS FOR THE TREATMENT OF CANCER

#968
20230301974
2023-09-28

PROCESSES OF MAKING AND CRYSTALLINE FORMS OF A MDM2 INHIBITOR

#969
20230295211
2023-09-21

METHODS OF PRODUCING CRYSTALLINE BETA NICOTINAMIDE RIBOSIDE TRIACETATE CHLORIDE

#970
20230295209
2023-09-21

METHOD FOR PRODUCING ALLULOSE CRYSTALS

#971
20230295208
2023-09-21

D-allose crystal and production method thereof

#972
20230295184
2023-09-21

Diaryl macrocycle polymorph

#973
20230295174
2023-09-21

SALT AND CRYSTAL FORM OF PYRIMIDINE COMPOUND, AND PREPARATION METHODS THEREFOR

#974
20230295160
2023-09-21

SALT FORM AND CRYSTAL FORM OF JAK INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF

#975
20230295156
2023-09-21

CRYSTALLINE FORMS OF 4-[(7-CHLORO-2-METHOXYBENZO[B][1,5]NAPHTHYRIDIN-10-YL)AMINO]-2,6-BIS(PYRROLIDIN-1-YLMETHYL)PHENOL AND SALTS THEREOF

#976
20230295121
2023-09-21

SOLID FORMS OF PRALSETINIB

#977
20230295073
2023-09-21

PROCESS OF MAKING A CRYSTALLINE EDG-2 RECEPTOR ANTAGONIST

#978
20230295069
2023-09-21

RXR agonist salt form, polymorphs thereof, and uses thereof

#979
20230292801
2023-09-21

CRYSTALLINE SUGAR COMPOSITE POWDER AND METHODS FOR MAKING THE SAME

#980
20230287026
2023-09-14

Method for preparing crystalline D-psicose

#981
20230286998
2023-09-14

SUCCINATE SALTS OF OCTAHYDROTHIENOQUINOLINE COMPOUND AND CRYSTALS THEREOF

#982
20230286990
2023-09-14

Solid forms of (R)-N-(2-(5-fluoropyridin-3-yl)-8-isopropylpyrazolo[1,5-a] [1,3,5]triazin-4-yl)-2,3,4,9-tetrahydro-1H-carbazol-3-amine as aryl hydrocarbon receptor (AHR) inhibitors

#983
20230286972
2023-09-14

CRYSTALINE FORMS OF AN O-GLYCOPROTEIN-2-ACETAMIDO-2-DEOXY-3-D-GLUCOPYRANOSIDASE INHIBITOR

#984
20230286969
2023-09-14

AROMATIC SPIRO RING AMIDE DERIVATIVES FOR THE TREATMENT AND PROPHYLAXIS OF HEPATITIS B VIRUS INFECTION

#985
20230286961
2023-09-14

Substituted tetrahydrofurans as modulators of sodium channels

#986
20230286950
2023-09-14

METHODS OF SYNTHESIZING DEUTERATED SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS

#987
20230286939
2023-09-14

IMPROVED CHLORANTRANILIPROLE PROCESS THROUGH USE OF A CRYSTAL INTERMEDIATE

#988
20230286938
2023-09-14

Polymorphs of a dihydroorotate dehydrogenase (DHOD) inhibitor

#989
20230286935
2023-09-14

Dihydromyricetin nanocrystals and preparation method and application thereof

#990
20230286932
2023-09-14

SYNTHETIC METHODS FOR PREPARATION OF 4-(2-CHLORO-4-METHOXY-5-METHYLPHENYL)-N-[(1S)-2-CYCLOPROPYL-1-(3-FLUORO-4-METHYLPHENYL)ETHYL]-5-METHYL-N-PROP-2-YNYL-1,3-THIAZOL-2-AMINE

#991
20230286926
2023-09-14

PROCESS FOR PREPARATION OF TRIAZOLE COMPOUND

#992
20230286924
2023-09-14

CRYSTALLINE FORMS OF 4-(7-HYDROXY-2-ISOPROPYL-4-OXO-4H-QUINAZOLIN-3-YL)-BENZONITRILE AND FORMULATIONS THEREOF

#993
20230286910
2023-09-14

Phenylcarbamate crystalline form and method for manufacturing the same

#994
20230286900
2023-09-14

POLYMORPHIC FORMS OF (R)-OXYBUTYNIN HYDROCHLORIDE

#995
20230286898
2023-09-14

METHOD FOR THE PURIFICATION OF VILANTEROL TRIFENATATE

#996
20230279049
2023-09-07

Crystalline salt forms

#997
20230279036
2023-09-07

Salts of Remdesivir

#998
20230279032
2023-09-07

Co-crystals or salts of psilocybin and methods of treatment therewith

#999
20230279021
2023-09-07

POLYMORPHS OF A GABAA ALPHA5 AGONIST AND METHODS OF USING IN THE TREATMENT OF COGNITIVE IMPAIRMENT

#1000
20230279017
2023-09-07

Solid forms of tabernanthalog monofumarate salt for treating neurological disorders and/or psychiatric disorders

#1001
20230279009
2023-09-07

SOLID STATE FORMS OF AVAPRITINIB SALTS

#1002
20230279004
2023-09-07

SOLID FORMS, SALTS, AND PROCESSES OF PREPARATION OF A CDK2 INHIBITOR

#1003
20230279002
2023-09-07

Polymorphs of Crystalline Forms of 3,10-dimethoxy-5,8,13,13a-tetrahydro-6H-isoquinolino[3,2-a]isoquinolin-9-yl 3-fluorobenzenesulfonate and Salts Thereof

#1004
20230278990
2023-09-07

SOLID STATE FORMS OF N-[2-(2-{4-[2-(6,7-DIMETHOXY-3,4-DIHYDRO-2(1H)-ISOQUINOLINYL)ETHYL]PHENYL}-2H-TETRAZOL-5-YL)-4,5-DIMETHOXYPHENYL]-4-OXO-4H-CHROMENE-2-CARBOXAMIDE MESYLATE SALT

#1005
20230278989
2023-09-07

Isoindolinone inhibitors of the MDM2-P53 interaction and process for making them

#1006
20230278985
2023-09-07

SOLID FORM OF COMPOUND

#1007
20230278977
2023-09-07

STABLE POLYMORPH OF R-MDMA HCL

#1008
20230278970
2023-09-07

Crystalline forms of 3-substituted 1,2,4-oxadiazole

#1009
20230278956
2023-09-07

PREPARATION OF TRIFAROTENE AND INTERMEDIATES AND POLYMORPHS THEREOF

#1010
20230278946
2023-09-07

ALPHA, BETA-UNSATURATED ALDEHYDE PRODUCTION METHOD

#1011
20230277499
2023-09-07

Forms of aticaprant

#1012
20230271986
2023-08-31

Crystalline or Amorphous form of Bcl-2/Bcl-xL inhibitor compound or its salts

#1013
20230271978
2023-08-31

Crystalline forms of (S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydropyrido [3,2-B][1,4]oxazepin-3-yl)-4H-1,2,4-triazole-3-carboxamide

#1014
20230271974
2023-08-31

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms therof

#1015
20230271971
2023-08-31

Crystalline forms of (S)-1-(4-fluorophenyl)-1-(2-(4-(6-(1-methyl-1H-pyrazol-4-yl)pyrrolo[2,1- f][1,2,4]triazin-4-yl)piperazinyl)-pyrimidin-5-yl)ethan-1-amine and methods of making

#1016
20230271967
2023-08-31

SOLID STATE FORMS OF FEZOLINETANT AND SALTS THEREOF

#1017
20230271958
2023-08-31

SALT AND CRYSTAL FORM OF DIHYDROPYRIDO[2,3-d]PYRIMIDINE DERIVATE

#1018
20230271947
2023-08-31

SALT AND CRYSTAL FORM OF KETOHEXOKINASE INHIBITOR AND USE THEREOF

#1019
20230271946
2023-08-31

PROCESS FOR THE PREPARATION OF 6-(CYCLOPROPANEAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE

#1020
20230271945
2023-08-31

Inhibitors of APOL1 and methods of using same

#1021
20230271927
2023-08-31

CRYSTALLINE FORMS OF GSK1278863, PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF

#1022
20230271922
2023-08-31

POLYMORPHS OF PHENYL PYRROLE AMINOGUANDIUM SALTS

#1023
20230271912
2023-08-31

PURIFICATION OF WOOD ACETYLATION FLUID

#1024
20230270753
2023-08-31

COMBINATIONS OF GABAA ALPHA 5 AGONISTS AND SV2A INHIBITORS AND METHODS OF USING IN THE TREATMENT OF COGNITIVE IMPAIRMENT

#1025
20230265097
2023-08-24

SALTS AND FORMS OF A WEE1 INHIBITOR

#1026
20230265095
2023-08-24

Crystalline forms of a MAGL inhibitor

#1027
20230265088
2023-08-24

Method of the preparation of fused multicyclic compounds

#1028
20230265080
2023-08-24

MODULATORS OF ALPHA-1 ANTITRYPSIN

#1029
20230265074
2023-08-24

Solid forms of 1-((S)-4-((R)-7-(6-amino-4-methyl-3-(trifluoromethyl)pyridin-2-yl)-6-chloro-8-fluoro-2-(((S)-1-methylpyrrolidin-2-yl)methoxy)quinazolin-4-yl)-3-methylpiperazin-1-yl)prop-2-en-1-one

#1030
20230265067
2023-08-24

CRYSTALLINE FORM OF LNP023

#1031
20230265059
2023-08-24

SOLID STATE FORMS OF 6-CARBOXY-2-(3, 5-DICHLOROPHENYL)-BENZOXAZOLE OF FORMULA-I AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF

#1032
20230265056
2023-08-24

CRYSTALLINE FORMS OF BENZAMIDE COMPOUND AND PROCESS FOR PREPARING THE SAME

#1033
20230265043
2023-08-24

CRYSTALLINE FORM OF PHENTERMINE HYDROCHLORIDE AND PROCESS FOR OBTAINING SAME

#1034
20230265038
2023-08-24

Crystal of tefluthrin, preparation method therefor and use thereof

#1035
20230263794
2023-08-24

SOLID FORMS OF N-[2,4-BIS(1,1-DIMETHYLETHYL)-5-HYDROXYPHENYL]-1,4-DIHYDRO-4-OXOQUINOLINE-3-CARBOXAMIDE

#1036
20230257391
2023-08-17

METHOD FOR EFFICIENTLY EXTRACTING AND SEPARATING HIGH-PURITY TETRODOTOXIN FROM PUFFERFISH VISCERA

#1037
20230257385
2023-08-17

SALT AND SOLID FORMS OF TABERNANTHALOG

#1038
20230257384
2023-08-17

THE CRYSTALLINE FORMS OR AMORPHOUS FORMS OF BISDIAZABICYCLIC COMPOUNDS OR SALTS THEREOF

#1039
20230257378
2023-08-17

Polymorphs of the hydrochloride salt of linaprazan glurate

#1040
20230257363
2023-08-17

COMPOUNDS, COMPOSITIONS AND METHODS

#1041
20230257361
2023-08-17

Crystalline forms of 3-(5-(2-hydroxy-2-methylpropoxy)-6-methylpyrazin-2-yl)-1H-indole-7-carbonitrile

#1042
20230257360
2023-08-17

Crystalline and salt forms of PPAR agonist compounds

#1043
20230257358
2023-08-17

CRYSTALLIZATION OF CANNABINOIDS

#1044
20230257341
2023-08-17

CIS-PARA-SUBSTITUTED CYCLOHEXYLAMINONITRILE SALT, PREPARATION METHOD THEREFOR AND USE THEREOF, AND METHOD FOR PREPARING PESTICIDE USING SAME

#1045
20230255982
2023-08-17

METHODS OF TREATING COVID-19 USING BARDOXOLONE METHYL OR ANALOGS THEREOF

#1046
20230250116
2023-08-10

CDK9 inhibitors and polymorphs thereof for use as agents for treatment of cancer

#1047
20230250115
2023-08-10

Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use

#1048
20230250087
2023-08-10

SOLID FORMS OF APOL1 INHIBITOR AND METHODS OF USING SAME

#1049
20230250083
2023-08-10

CRYSTALS

#1050
20230250081
2023-08-10

Salt forms and polymorphs of (R)-1-(4-(6-(2-(4-(3,3-difluorocyclobutoxy)-6-methylpyridin-2-yl)acetamido) pyridazin-3-yl)-2-fluorobutyl)-n-methyl-1H-1,2,3-triazole-4-carboxamide

#1051
20230250076
2023-08-10

Processes and intermediate for the large-scale preparation of 2,4,6-trifluoro-N-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide hemisuccinate, and preparation of 2,4,6-trifluoro-N-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide acetate

#1052
20230250075
2023-08-10

Processes and intermediate for the large-scale preparation of 2,4,6-trifluoro-n-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide hemisuccinate, and preparation of 2,4,6-trifluoro-n-[6-(1-methyl-piperidine-4-carbonyl)-pyridin-2-yl]-benzamide acetate

#1053
20230250068
2023-08-10

CRYSTALLINE FORMS OF A JAK2 INHIBITOR

#1054
20230250044
2023-08-10

CRYSTALS OF 3-HYDROXYPROPIONATE AND PROCESS OF RECOVERING 3-HYDROXYPROPIONIC ACID

#1055
20230250043
2023-08-10

Methods of making bempedoic acid and compositions of the same

#1056
20230242542
2023-08-03

COMPOSITIONS COMPRISING (S)-7-(1-ACRYLOYLPIPERIDIN-4-YL)-2-(4-PHENOXYPHENYL)-4,5,6,7-TETRA-HYDROPYRAZOLO[1,5-a]PYRIMIDINE-3-CARBOXAMIDE

#1057
20230242539
2023-08-03

Polymorphs of (1S,2S,3S,5R)-3-((6-(Difluoromethyl)-5-Fluoro-1,2,3,4-Tetrahydroisoquinolin-8-YL)OXY)-5-(4-Methyl-7H-Pyrrolo[2,3-D]Pyrimidin-7-YL)Cyclopentane-1,2-DIOL Mono-Hydrochloride

#1058
20230242517
2023-08-03

Polymorphs of selinexor

#1059
20230242516
2023-08-03

Polymorphs of Selinexor

#1060
20230242515
2023-08-03

Crystalline form of 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyl-D3) pyridazine-3-carboxamide

#1061
20230242505
2023-08-03

PROCESS, COMPOSITIONS, AND CRYSTALLINE FORMS OF SUBSTITUTED PYRIDINONE-PYRIDINYL COMPOUNDS

#1062
20230242485
2023-08-03

Solid forms

#1063
20230242483
2023-08-03

CRYSTALLINE FORMS OF SOLVATES OF TRYPTOPHAN DERIVATIVES, COMPOSITIONS COMPRISING THEM AND USES THEREOF

#1064
20230234983
2023-07-27

SQUALAMINE CRYSTALLINE POLYMORPHS

#1065
20230234974
2023-07-27

Crystal forms of crisaborole in free form and preparation method and use thereof

#1066
20230234972
2023-07-27

Co-crystal compounds comprising lithium ions and isonicotinamide

#1067
20230234961
2023-07-27

CRYSTALLINE SALT OF ERIBULIN

#1068
20230234956
2023-07-27

METHODS OF MAKING WEE1 INHIBITOR COMPOUNDS

#1069
20230234916
2023-07-27

N-[8-(2-HYDROXYBENZOYL)AMINO]POTASSIUM OCTANOATE CRYSTAL POLYMORPH, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#1070
20230233557
2023-07-27

FORMULATIONS COMPRISING HETEROCYCLIC PROTEIN KINASE INHIBITORS

#1071
20230233534
2023-07-27

SYNTHETIC METHODS FOR PREPARATION OF 4-(2-CHLORO-4-METHOXY-5-METHYLPHENYL)-N-[(1S)-2-CYCLOPROPYL-1-(3-FLUORO-4-METHYLPHENYL)ETHYL]-5-METHYL-N-PROP-2-YNYL-1,3-THIAZOL-2-AMINE

#1072
20230227463
2023-07-20

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1073
20230227456
2023-07-20

ORAL FORMULATION COMPRISING A CRYSTALLINE FORM OF RABEXIMOD

#1074
20230227455
2023-07-20

METHOD FOR PREPARING A CRYSTALLINE FORM OF RABEXIMOD

#1075
20230227443
2023-07-20

Solid forms of(Z)-4-(5-((3-benzyl-4-oxo-2-thioxothiazolidin-5-ylidene)methyl)furan-2-yl)benzoic acid

#1076
20230227422
2023-07-20

Phenethylamine compounds salts, polymorphic forms and methods of use thereof

#1077
20230227413
2023-07-20

SOLID STATE FORMS OF ENSARTINIB AND ENSARTINIB SALTS

#1078
20230225325
2023-07-20

CRYSTALLINE FORMS OF DELTAMETHRIN AND METHODS OF USE THEREOF

#1079
20230219977
2023-07-13

Process for the preparation of sodium (2r,5s,13ar)-7,9-dioxo-10-((2,4,6,-trifluorobenzyl)carbamoyl)-2,3,4,5,7,9,13,13A-octahydro-2,5-methanopyrido[1′,2′:4,5]pyrazino[2,1-B] [1,3] oxazepin-8-olate and its polymorphic form

#1080
20230219968
2023-07-13

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1081
20230219955
2023-07-13

LSD DERIVATIVES, SYNTHESIS & METHOD FOR TREATMENT OF DISEASES AND DISORDERS

#1082
20230219936
2023-07-13

PROCESS FOR THE PREPARATION SALTS OF TRIAZOLE COMPOUNDS

#1083
20230219922
2023-07-13

PROCESS FOR SYNTHESIZING 2-HYDROXY-6-((2-(1-ISOPROPYL-1H-PYRAZOL-5-YL)-PYRIDIN-3-YL)METHOXY)BENZALDEHYDE

#1084
20230219910
2023-07-13

CRYSTALLINE FORMS OF {2-[3-CYCLOHEXYL-3-(TRANS-4-PROPOXY-CYCLOHEXYL)-UREIDO]-THIAZOL-5-YLSULFANYL}-ACETIC ACID AND USES THEREOF

#1085
20230219909
2023-07-13

SALTS OR CO-CRYSTALS OF {2-[3-CYCLOHEXYL-3-(TRANS-4-PROPOXY-CYCLOHEXYL)-UREIDO]-THIAZOL-5-YLSULFANYL}-ACETIC ACID AND USES THEREOF

#1086
20230219900
2023-07-13

Sodium 2-[(4S)-8-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[2-methoxy-5-(trifluoromethyl)phenyl]-4H-quinazolin-4-yl]acetate monohydrate, its preparation and use

#1087
20230219899
2023-07-13

A METHOD OF PRODUCING A CRYSTALLINE FORM OF SODIUM 2-[(4S)-8-FLUORO-2-[4-(3-METHOXYPHENYL)PIPERAZIN-1-YL]-3-[2-METHOXY-5-(TRIFLUOROMETHYL)PHENYL]-4H-QUINAZOLINE-4-YL]ACETATE TRIHYDRATE

#1088
20230219892
2023-07-13

FORMS AND COMPOSITIONS OF A BETA ADRENERGIC AGONIST

#1089
20230218623
2023-07-13

SALTS OF NEUROCEUTICALS AND USES THEREOF

#1090
20230218616
2023-07-13

Combinations for Treatment of NAFLD/NASH and Related Diseases

#1091
20230212206
2023-07-06

Complex Containing Betaine, Transition Metal and Sulfate

#1092
20230212193
2023-07-06

CRYSTALLINE RET INHIBITOR

#1093
20230212159
2023-07-06

Process for the Production of Ferroportin Inhibitors

#1094
20230212156
2023-07-06

METHOD FOR PRODUCING NITROFURANTOIN ANHYDRATE, AND PRODUCT THEREOF

#1095
20230212130
2023-07-06

Polymorphs of herbicidal sulfonamides

#1096
20230212128
2023-07-06

Polymorphs of pyrimidine cyclohexyl glucocorticoid receptor modulators

#1097
20230212118
2023-07-06

PREPARATION OF AN SELECTIVE ESTROGEN RECEPTOR DEGRADER

#1098
20230212117
2023-07-06

CRYSTALLINE FORM OF CAPSID PROTEIN ASSEMBLY INHIBITOR CONTAINING N HETERO FIVE-MEMBERED RING, AND APPLICATION THEREOF

#1099
20230212115
2023-07-06

METHODS FOR THE PREPARATION OF SPHINGOSINE 1-PHOSPHATE RECEPTOR MODULATORS AND SOLID FORME THEREOF

#1100
20230203093
2023-06-29

Crystalline dipeptides useful in the synthesis of elamipretide

#1101
20230203051
2023-06-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1- carboxamide and solid state forms thereof

#1102
20230203050
2023-06-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1103
20230203049
2023-06-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1104
20230203040
2023-06-29

CRYSTALLINE FORMS OF A SULFONAMIDE COMPOUND AND PROCESSES FOR PREPARING THE SAME

#1105
20230203023
2023-06-29

SALT AND CRYSTAL FORMS OF GLP-1R AGONISTS AND USES THEREOF

#1106
20230203013
2023-06-29

Method for preparing 2-chloro-n-(1-cyanocyclopropyl)-5-[2'-methyl-5'-(pentafluoroethyl)-4'-(trifluoromethyl)-2'h-1,3'-bipyrazol-4-yl]benzamide

#1107
20230203012
2023-06-29

SOLID FORMS OF A PLASMA KALLIKREIN INHIBITOR AND SALTS THEREOF

#1108
20230203009
2023-06-29

PRALSETINIB PHARMACEUTICAL COMPOSITIONS

#1109
20230203001
2023-06-29

SOLID FORMS OF FASORACETAM

#1110
20230202998
2023-06-29

PHENETHYLAMINE COMPOUNDS SALTS, POLYMORPHIC FORMS AND METHODS OF USE THEREOF

#1111
20230202991
2023-06-29

BENZISOXAZOLE DERIVATIVE

#1112
20230202987
2023-06-29

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#1113
20230202978
2023-06-29

CO-CRYSTAL OR SALT

#1114
20230202975
2023-06-29

PROCESS FOR THE PREPARATION OF CYSTEAMINE BITARTRATE AND PRODUCT SO OBTAINED

#1115
20230202959
2023-06-29

PROCESS FOR THE OXIDATION OF PRIMARY ALCOHOLS TO CARBOXYLIC ACIDS

#1116
20230201797
2023-06-29

TWO-DIMENSIONAL CHALCOGENIDE, AND PREPARATION METHOD AND USE THEREOF

#1117
20230201235
2023-06-29

INHIBITION OF NIDOVIRUSES THAT ENCODE NSP15

#1118
20230192746
2023-06-22

PROCESS FOR CRYSTALLIZING 2'-FUCOSYLLACTOSE AND RELATED COMPOSITIONS

#1119
20230192724
2023-06-22

SUNLIGHT-POWERED ROLLING CRYSTALS

#1120
20230192722
2023-06-22

SALTS AND SOLID FORMS OF AN FGFR INHIBITOR AND PROCESSES OF PREPARING THEREOF

#1121
20230192710
2023-06-22

JAK INHIBITOR COMPOUND AND USE THEREOF

#1122
20230192707
2023-06-22

Solid forms of pyrazolo[3,4-d]pyrimidine compounds

#1123
20230192697
2023-06-22

MESYLATE SALTS OF HETEROCYCLIC CYTOKININS, COMPOSITIONS CONTAINING THESE DERIVATIVES AND USE THEREOF

#1124
20230192694
2023-06-22

Crystal forms of a POL1 inhibitor

#1125
20230192679
2023-06-22

CRYSTALLINE FORMS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE THEREOF

#1126
20230192653
2023-06-22

Novel Therapeutic Methods

#1127
20230192642
2023-06-22

Isotopologues salts, crystalline forms, stereoisomers, of methylone and ethylone and methods of use thereof

#1128
20230192640
2023-06-22

Semi synthetic method for dihydroquercetin

#1129
20230192618
2023-06-22

CRYSTALLINE SALT FORMS OF N-(4-(4-(CYCLOPROPYLMETHYL)PIPERAZINE-1-CARBONYL)PHENYL)QUINOLINE-8-SULFONAMIDE

#1130
20230192612
2023-06-22

Formulations of T-type calcium channel modulators and methods of use thereof

#1131
20230192594
2023-06-22

CRYSTAL FORMS AND METHODS OF SYNTHESIS OF (2R, 6R)-HYDROXYNORKETAMINE AND (2S, 6S)-HYDROXYNORKETAMINE

#1132
20230187700
2023-06-15

1,4-DIOXANE SLOVATE OF LITHIUM DIFLUOROBIS(OXALATO)PHOSPHATE, METHOD FOR PREPARING THE SAME, AND ELECTROLYTE COMPOSITION COMPRISING THE SAME

#1133
20230183274
2023-06-15

SCALABLE POLYPROPIONATE LACTONE STEREOTETRADS

#1134
20230183266
2023-06-15

CRYSTALLINE FORMS OF RET INHIBITOR AND PREPARATION THEREOF

#1135
20230183265
2023-06-15

Crystal Form of Macrocyclic Tyrosine Kinase Inhibitor and Preparation Method therefor

#1136
20230183259
2023-06-15

Crystal Form Of Thiofuran Pyridazine Compound, Preparation Method Therefor And Application Thereof

#1137
20230183257
2023-06-15

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]- pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1138
20230183241
2023-06-15

CRYSTAL OF A HYPOXANTHINE COMPOUND

#1139
20230183236
2023-06-15

CRYSTALLINE FORMS OF AN APOPTOSIS-INDUCING AGENT

#1140
20230183235
2023-06-15

SOLID STATE FORMS OF AMG-510 AND PROCESS FOR PREPARATION THEREOF

#1141
20230183205
2023-06-15

PHARMACEUTICAL COMPOSITION IN WHICH PRODUCTION OF IMPURITIES IS SUPPRESSED

#1142
20230183202
2023-06-15

TETRAHYDROCOCANNABINOLIC ACID COCRYSTALS

#1143
20230183195
2023-06-15

COCRYSTALS OF (1R,3S)-3-(5-CYANO-4-PHENYL-1,3-THIAZOL-2-YLCARBAMOYL)CYCLOPENTANE CARBOXYLIC ACID

#1144
20230183194
2023-06-15

CRYSTALLINE FORM OF OZANIMOD HYDROCHLORIDE

#1145
20230183185
2023-06-15

Olaparib hydroxybenzoic acid cocrystals and their pharmaceutical use

#1146
20230183174
2023-06-15

NOVEL SULFOBETAINE MONOMERS, PROCESS FOR PREPARING SAME, AND USES THEREOF

#1147
20230183172
2023-06-15

Compositions comprising (R)-2-amino-3-phenylpropyl carbamate and uses thereof

#1148
20230183166
2023-06-15

Methods for making and using endoxifen

#1149
20230183164
2023-06-15

Synthesis of Vinyl Cyclobutyl Intermediates

#1150
20230183160
2023-06-15

Methods of making bempedoic acid and compositions of the same

#1151
20230181507
2023-06-15

CO-CRYSTAL OF GABAPENTIN, KETOPROFEN AND LYSINE, PHARMACEUTICAL COMPOSITIONS AND THEIR MEDICAL USE

#1152
20230174562
2023-06-08

RADIO-AND CHEMO-PROTECTIVE COMPOUNDS

#1153
20230174554
2023-06-08

SOLID FORM OF MACROCYCLIC COMPOUND, PREPARATION THEREFOR AND USE THEREOF

#1154
20230174552
2023-06-08

Method of treatment of symptoms of menopause

#1155
20230174549
2023-06-08

SALT AND CRYSTAL FORMS OF 4-AMINO-5-(6-(4-METHYLPIPERAZIN-1-YL)-1H-BENZO[D]IMIDAZOL-2-YL)THIENO[2,3-B]PYRIDIN-6(7H)-ONE

#1156
20230174547
2023-06-08

PHARMACEUTICALLY ACCEPTABLE ACID SALT OF FREE BASE OF GLP1 RECEPTOR AGONIST, AND PREPARATION METHOD THEREFOR

#1157
20230174546
2023-06-08

CRYSTALLINE FORM A OF GLP-1 RECEPTOR AGONIST AND PREPARATION METHOD THEREFOR

#1158
20230174543
2023-06-08

FREE BASE CRYSTALS

#1159
20230174541
2023-06-08

Inhibitors of the menin-MLL interaction

#1160
20230174532
2023-06-08

Methods for antagonizing a melanocortin 4 receptor

#1161
20230174529
2023-06-08

CRYSTALLINE FORMS AND FORMULATIONS OF A VCP/p97 INHIBITOR

#1162
20230174528
2023-06-08

CRYSTAL OF TRIFLUOROMETHYL/CHLORO DISUBSTITUTED SULFONAMIDE SELECTIVE BCL-2 INHIBITOR

#1163
20230174525
2023-06-08

POLYMORPHS OF A HYDROCHLORIDE SALT OF PN6047

#1164
20230174522
2023-06-08

Benzisoxazole Sulfonamide Derivatives

#1165
20230174504
2023-06-08

PROCESS FOR PREPARATION OF 2-HYDROXY-6-((2-(1-ISOPROPYL-1H-PYRAZOL-5-YL)PYRIDIN-3-YL)METHOXY)BENZALDEHYDE

#1166
20230174489
2023-06-08

Crystal form of 2-methyl-2-propanol and amino-substituted aryl compound

#1167
20230174458
2023-06-08

Crystalline Forms of (-)-(1R,2R)-3-(3-dimethylamino-1-ethyl-2-methylpropyl)-phenol hydrochloride

#1168
20230172952
2023-06-08

Fospropofol Salts, Methods And Compositions

#1169
20230167156
2023-06-01

Solid state forms of voclosporin

#1170
20230167132
2023-06-01

FORMS AND COMPOSITIONS OF INHIBITORS OF PLASMA KALLIKREIN

#1171
20230167128
2023-06-01

POLYMORPHS AND SOLID FORMS OF (S)-2-((2-((S)-4-(DIFLUOROMETHYL)-2-OXOOXAZOLIDIN-3-YL)-5,6-DIHYDROBENZO[F]IMIDAZO[1,2-D][1,4]OXAZEPIN-9-YL)AMINO)PROPANAMIDE, AND METHODS OF PRODUCTION

#1172
20230167113
2023-06-01

CRYSTALLINE FORMS OF GEPOTIDACIN

#1173
20230167108
2023-06-01

CRYSTAL OF IMIDAZOPYRIDINONE COMPOUND OR SALT THEREOF

#1174
20230167107
2023-06-01

CRYSTALS, PREPARATION METHOD AND APPLICATION OF A MUSCARINIC RECEPTOR ANTAGONIST

#1175
20230167096
2023-06-01

VORUCICLIB POLYMORPHS AND METHODS OF MAKING AND USING THEREOF

#1176
20230167090
2023-06-01

SOLID STATE FORMS OF APROCITENTAN AND PROCESS FOR PREPARATION THEREOF

#1177
20230167080
2023-06-01

BCKDK INHIBITORS AND/OR DEGRADERS

#1178
20230167077
2023-06-01

Crystal forms of immunomodulators

#1179
20230167069
2023-06-01

Solid state forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide and uses thereof

#1180
20230165857
2023-06-01

AXL KINASE INHIBITORS AND USE OF THE SAME

#1181
20230165260
2023-06-01

Pseudomonas strains and their metabolites to control plant diseases

#1182
20230162974
2023-05-25

Enhanced perovskite materials for photovoltaic devices

#1183
20230159582
2023-05-25

CRYSTALLINE FORMS OF SQUALAMINE

#1184
20230159565
2023-05-25

Solid forms of substituted benzoxaborole and compositions thereof

#1185
20230159549
2023-05-25

Method for preparation of Asenapine

#1186
20230159540
2023-05-25

PYRAZOLO[3,4-d]PYRIMIDIN-3-ONE DERIVATIVE AS WEE-1 INHIBITOR

#1187
20230159539
2023-05-25

CRYSTALLINE FORMS OF 3-CYANO-1-[4-[6-(1-METHYL-1H-PYRAZOL-4-YL)PYRAZOLO[1,5-A]PYRAZIN-4-YL]-1H-PYRAZOL-1-YL]CYCLOBUTANEACETONITRILE, AND USE THEREOF

#1188
20230159533
2023-05-25

Crystalline composition of tildacerfont and methods of use and preparation thereof

#1189
20230159518
2023-05-25

CRYSTALLINE FORMS OR AMORPHOUS FORMS OF N-(PHENYL SULFONYL) BENZAMIDE COMPOUNDS OR ITS SALTS OR SOLVATES

#1190
20230159499
2023-05-25

HDAC inhibitor solid state forms

#1191
20230159494
2023-05-25

HDAC inhibitor solid state forms

#1192
20230159473
2023-05-25

CRYSTALLINE FORMS OF A TYK2 INHIBITOR

#1193
20230159468
2023-05-25

NOVEL FORMS OF PRACINOSTAT DIHYDROCHLORIDE

#1194
20230159462
2023-05-25

METHOD FOR PRODUCING NITROGEN-CONTAINING HETEROARYLCARBOXAMIDE ACETIC ACID DERIVATIVE

#1195
20230159454
2023-05-25

Crystalline form of 1-(5-(2,4-Difluorophenyl)-1-((3-fluorophenyl)sulfonyl)-4-methoxy-1H-pyrrol-3-yl)-n-methylmethanamine salt

#1196
20230159444
2023-05-25

PROCESS FOR SYNTHESIZING SULFONATED TRIARYL METHANE COMPOUNDS

#1197
20230153676
2023-05-18

CHEMICALLY TUNABLE OPTICALLY ADDRESSABLE MOLECULR-SPIN QUBIT AND ASSOCIATED METHODS

#1198
20230151048
2023-05-18

Crystal form, preparation method, and application of 4'-substituted nucleoside

#1199
20230151043
2023-05-18

Compounds and methods for treatment of viral infections

#1200
20230151036
2023-05-18

Psilocybin and O-acetylpsilocin, salts and solid state forms thereof