ClassID:

90494

C07B2200/13 - page 6 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#1501
20220372044
2022-11-24

CRYSTALLINE SOLVATED FORMS OF N-(4-(1-(2,6-DIFLUOROBENZYL)-5- ((DIMETHYLAMINO)METHYL)-3-(6-METHOXY-3-PYRIDAZINYL)-2,4-DIOXO-1,2,3,4- TETRAHYDROTHIENO[2,3-D]PYRIMIDIN-6-YL)PHENYL)-N'-METHOXYUREA

#1502
20220372024
2022-11-24

CRYSTALLINE FORMS OF ENTRECTINIB

#1503
20220372021
2022-11-24

RESMETIROM CRYSTAL, PREPARATION METHOD FOR SAME, AND USES THEREOF

#1504
20220372020
2022-11-24

Crystalline forms of phthalazinone compound

#1505
20220372019
2022-11-24

SALTS AND SOLID STATE FORMS OF PLINABULIN

#1506
20220372006
2022-11-24

SOLID STATE FORMS OF PEMAFIBRATE

#1507
20220372001
2022-11-24

CRYSTAL FORM OF BENZIMIDAZOLE-2-ONE COMPOUND, SOLVATE THEREOF, CRYSTAL FORM OF SOLVATE THEREOF, AND PREPARATION METHOD THEREOF

#1508
20220371998
2022-11-24

Crystalline polymorphs of Rivoceranib and Rivoceranib mesylate

#1509
20220371996
2022-11-24

Salt forms of URAT-1 inhibitors

#1510
20220371994
2022-11-24

CRYSTALLINE POLYMORPHIC FORM OF PSILOCIN

#1511
20220371993
2022-11-24

(C)CRYSTAL COMPOSITION (CC) COMPRISING 4,4'-DICHLORODIPHENYLSULFONE CRYSTALS (C)

#1512
20220371985
2022-11-24

Polymorphic compounds and uses thereof

#1513
20220363705
2022-11-17

METHOD FOR MANUFACTURING REVAUDIOSIDE-D-CONTAINING CRYSTALLIZED PRODUCT, AND REVAUDIOSIDE-D-CONTAINING CRYSTALLIZED PRODUCT

#1514
20220363691
2022-11-17

METHOD FOR PREPARING HETEROCYCLIC DERIVATIVE COMPOUND, COMPOSITION CONTAINING SAME COMPOUND, AND HYDRATE OF SAME COMPOUND

#1515
20220363682
2022-11-17

NOVEL SALTS AND CRYSTALS

#1516
20220363674
2022-11-17

Solid forms of a modulator of hemoglobin

#1517
20220363673
2022-11-17

5-(Thiophen-2-YL)-1 H-Tetrazole Derivative as BCKDK Inhibitors Useful for Treating Various Diseases

#1518
20220363670
2022-11-17

Pyrazolyl derivatives useful as anti-cancer agents

#1519
20220363669
2022-11-17

Crystalline forms of (S)-1-(1-acryloylpyrrolidin-3-yl)-3-((3,5-dimethoxyphenyl)ethynyl)-5-(methylamino)-1H-pyrazole-4-carboxamide

#1520
20220363661
2022-11-17

Cocrystals, pharmaceutical compositions thereof, and methods of treatment involving same

#1521
20220363655
2022-11-17

Salt and solid state forms of escatalopram

#1522
20220363635
2022-11-17

Crystalline forms of psilacetin

#1523
20220363634
2022-11-17

CRYSTALLINE FORM OF CAPSID PROTEIN ASSEMBLY INHIBITOR CONTAINING N HETERO FIVE-MEMBERED RING, AND APPLICATION THEREOF

#1524
20220363629
2022-11-17

Polymorphic forms of N-(4-((4-(3-phenylureido)phenyl)sulfonyl)phenyl)benzolsulfonamide

#1525
20220361526
2022-11-17

Compositions and methods for solidified fermented animal feed

#1526
20220356217
2022-11-10

Polypeptide integrin antagonists

#1527
20220356173
2022-11-10

Polymorphic forms of kinase inhibitor compound, pharmaceutical composition containing same, preparation method therefor and use thereof

#1528
20220356165
2022-11-10

SOLID STATE FORMS OF ROLUPERIDONE AND SALTS THEREOF

#1529
20220348591
2022-11-03

Solid forms of 3-(5-Fluorobenzofuran-3-yl)-4-(5-methyl-5H-[1,3]dioxolo[4,5-f]indol-7-yl)pyrrole-2,5-dione

#1530
20220348582
2022-11-03

Crystal forms of (s)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide

#1531
20220348578
2022-11-03

Crystalline forms of diazabicyclooctane derivative and production process thereof

#1532
20220348575
2022-11-03

LSD SALT CRYSTAL FORMS

#1533
20220348552
2022-11-03

Crystals of tetrahydronaphthyl urea derivative

#1534
20220348545
2022-11-03

Process for the preparation of a PDE4 inhibitor

#1535
20220348543
2022-11-03

SALTS OF OMECAMTIV MECARBIL AND SOLID FORMS THEREOF

#1536
20220348542
2022-11-03

PROCESS FOR SYNTHESIZING APREMILAST

#1537
20220348531
2022-11-03

CRYSTALLINE FORMS OF BEMPEDOIC ACID

#1538
20220348530
2022-11-03

Menaquinol compositions and methods of treatment

#1539
20220340594
2022-10-27

Method for preparing heterocyclic derivative compound, composition containing same compound, and hydrate of same compound

#1540
20220340592
2022-10-27

CHEMICAL COMPOUNDS

#1541
20220340584
2022-10-27

Crystalline form of (S)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra-hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#1542
20220340583
2022-10-27

Crystalline form of (S)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra- hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#1543
20220340574
2022-10-27

Solid polymorphs of a FLNA-binding compound and its hydrochloride salts

#1544
20220340573
2022-10-27

1,2,4-OXADIAZOLE DERIVATIVES AS LIVER X RECEPTOR AGONISTS

#1545
20220340562
2022-10-27

VMAT2 INHIBITOR AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#1546
20220340549
2022-10-27

CRYSTALLINE FORM OF CXCR2 ANTAGONIST AND APPLICATION THEREOF

#1547
20220340542
2022-10-27

SALTS OF OMECAMTIV MECARBIL AND SOLID FORMS THEREOF

#1548
20220340541
2022-10-27

Fumarate salt of (R)-3-(1-(2,3-dichloro-4-(pyrazin-2-yl)phenyl)-2,2,2-trifluoroethyl)-1-methyl-1-(1-methylpiperidin-4-yl)urea, methods of preparation, and uses thereof

#1549
20220340540
2022-10-27

A SALT AND CRYSTAL FORM OF A FAK INHIBITOR

#1550
20220340520
2022-10-27

RREPARATION METHOD OF 3-MERCAPTOPROPIONIC ACID

#1551
20220339132
2022-10-27

Vidofludimus for use in the treatment or prevention of viral diseases

#1552
20220332753
2022-10-20

(17-)-3-Oxoandrost-4-EN-17-YL Dodecanoate Compositions and Methods of Preparation and Use

#1553
20220332745
2022-10-20

D-PSICOSE CRYSTAL AND PREPARATION METHOD THEREFOR

#1554
20220332715
2022-10-20

NEW CRYSTAL FORM OF AN ORGANIC FLUORESCENT COMPOUND

#1555
20220332706
2022-10-20

CRYSTALLINE FORMS OF A JAK2 INHIBITOR

#1556
20220332702
2022-10-20

NON-HYGROSCOPIC CRYSTALLINE SALTS OF A PYRAZOLE COMPOUND, AND PHARMACEUTICAL COMPOSITIONS AND USE THEREOF

#1557
20220332684
2022-10-20

CRYSTAL FORM OF FIVE-MEMBERED N HETEROCYCLIC COMPOUND, AND APPLICATION THEREOF

#1558
20220332682
2022-10-20

CAANABIGEROL PROLINE COCRYSTALS

#1559
20220332680
2022-10-20

Hydrated crystalline form of 2-acrylamido-2-methylpropane sulfonic acid

#1560
20220324901
2022-10-13

Process for the preparation of cortexolone 17α-propionate and new hydrated crystalline form thereof

#1561
20220324897
2022-10-13

CRYSTAL FORM OF SGLT INHIBITOR AND APPLICATION THEREOF

#1562
20220324833
2022-10-13

PROCESS FOR PREPARATION OF 2-HYDROXY-6-((2-(1-ISOPROPYL-1H-PYRAZOL-5-YL)PYRIDIN-3-YL)METHOXY)BENZALDEHYDE

#1563
20220324831
2022-10-13

STABLE CRYSTALLINE APALUTAMIDE IN PURE FORM, AND PROCESS FOR THE PREPARATION THEREOF

#1564
20220324820
2022-10-13

METHODS AND COMPOSITIONS FOR GAMMA-GLUTAMYL CYCLE MODULATION

#1565
20220324816
2022-10-13

Elagolix Sodium Compositions and Processes

#1566
20220324808
2022-10-13

Co-crystal of Compound I Dihydrochloride and Preparation Method and Use Thereof

#1567
20220324802
2022-10-13

METHOD FOR PURIFYING AN ORGANIC COMPOUND

#1568
20220324786
2022-10-13

METHODS FOR RECOVERING ORGANIC ACIDS OR SALTS OR LACTONES THEREOF FROM AQUEOUS SOLUTIONS USING WATER SOLVENT CRYSTALLIZATION AND COMPOSITIONS THEREOF

#1569
20220315618
2022-10-06

Method for producing functional crystalline sweetener

#1570
20220315615
2022-10-06

CONTINUOUS PREPARATION METHOD FOR PENEM INTERMEDIATE MAP

#1571
20220315608
2022-10-06

METFORMIN COMPLEXES WITH TRANSITION METALS AND P GROUP ELEMENTS

#1572
20220315607
2022-10-06

SOLID STATE FORMS OF RISDIPLAM AND PROCESS FOR PREPARATION THEREOF

#1573
20220315605
2022-10-06

IMPROVED PROCESS FOR THE PREPARATON OF PURE (1'R,6R,6aR,7R,13S,14S,16R)-5-(ACETYLOXY)-3',4',6,6a,7,13,14,16-OCTAHYDRO-6',8,14-TRIHYDROXY-7',9-DIMETHOXY-4,10,23-TRIMETHYLSPIRO[6,16-(EPITHIOPROPANOXYMETH ANO)-7,13-IMINO-12H-1,3-DIOXOLO[7,8]ISOQUINO[3,2-b][3]BENZAZOCINE-20,1'(2'H)-ISOQUINOLIN]-19-ONE POLYMORPH THERE OF

#1574
20220315576
2022-10-06

POLYMORPH OF CDK9 INHIBITOR AND PREPARATION METHOD FOR POLYMORPH AND USE THEREOF

#1575
20220315571
2022-10-06

POLYMORPHS OF (R)-N-(5-(5-ETHYL-1,2,4-OXADIAZOL-3-YL)-2,3-DIHYDRO-1H-INDEN-1-YL)-1-METHYL-1H-PYRAZOLE-4-CARBOXAMIDE

#1576
20220315559
2022-10-06

Crystalline form and B crystalline form of pyrazine-2(1H)-ketone compound and preparation method thereof

#1577
20220315558
2022-10-06

POLYMORPHS OF 1-(2-((((TRANS)-3-FLUORO-1-(3-FLUOROPYRIDIN-2-YL)CYCLOBUTYL)METHYL)AMINO)PYRIMIDIN-5-YL)-1H-PYRROLE-3-CARBOXAMIDE

#1578
20220313667
2022-10-06

Sulfasalazine salts, production processes and uses

#1579
20220306650
2022-09-29

PROCESS AND POLYMORPHIC FORMS OF BICTEGRAVIR AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS OR CO-CRYSTALS THEREOF

#1580
20220306643
2022-09-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1581
20220306628
2022-09-29

Crystalline solid forms of a bet inhibitor

#1582
20220306626
2022-09-29

CRYSTALLINE FORM OF A DIHYDROCHLORIDE SALT OF A JAK INHIBITOR COMPOUND

#1583
20220306622
2022-09-29

SALT AND CRYSTAL FORM OF MTORC1/2 DUAL KINASE ACTIVITY INHIBITOR AND PREPARATION METHOD THEREFOR

#1584
20220306594
2022-09-29

Crystalline form of 1,4-bis[1,2-benzisoselenazol-3(2H)-one]-butane, method for preparing same and use thereof

#1585
20220306582
2022-09-29

Anhydrous Crystal of Monosodium N-(2-Ethylsulfonylamino-5-Trifluoromethyl-3-Pyridyl)Cyclohexane Carboxamide

#1586
20220306580
2022-09-29

Crystalline freebase forms of a biphenyl compound

#1587
20220306574
2022-09-29

Process for the preparation of D,L-methionine

#1588
20220306569
2022-09-29

CRYSTALLINE FORMS OF HYDROXYNORKETAMINE

#1589
20220306566
2022-09-29

Two-dimensional coordination polymers

#1590
20220298166
2022-09-22

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1 carboxamide and solid state forms thereof

#1591
20220298165
2022-09-22

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1592
20220298159
2022-09-22

SOLID FORMS OF {6-[(2-AMINO-3-CHLOROPYRIDIN-4-YL)SULFANYL]-3-[(3S,4S)-4-AMINO-3-METHYL-2-OXA-8-AZASPIRO[4.5]DECAN-8-YL]-5-METHYLPYRAZIN-2-YL}METHANOL, A SHP2 INHIBITOR

#1593
20220298158
2022-09-22

POLYMORPH OF VENETOCLAX AND METHOD FOR PREPARING THE POLYMORPH

#1594
20220298117
2022-09-22

CRYSTALLINE FORMS OF [3-(4- {2-BUTYL-1-[4-(4-CHLORO-PHENOXY)-PHENYL]-1H-IMIDAZOL-4-YL} -PHENOXY)-PROPYL]-DIETHYL-AMINE

#1595
20220298116
2022-09-22

PROCESS FOR THE PREPARATION OF KEY INTERMEDIATES FOR THE SYNTHESIS OF ELTROMBOPAG OR SALT THEREOF

#1596
20220298108
2022-09-22

CRYSTALLINE FORM OF SOFPIRONIUM BROMIDE AND PREPARATION METHOD THEREOF

#1597
20220296589
2022-09-22

Formulations of 4-Methyl-5-(Pyrazin-2-yl)-3H-1,2-Dithiole-3-Thione, Taste-Modified Formulations, and Methods of Making and Using Same

#1598
20220296482
2022-09-22

SYNTHESIS AND PURIFICATION OF CANNABIGEROL AND ITS APPLICATION

#1599
20220289837
2022-09-15

Cystic Fibrosis Transmembrane Conductance Regulator Stabilizing Agents

#1600
20220289789
2022-09-15

Hemi-citrate salts of GABA-A positive allosteric modulator and crystalline form thereof

#1601
20220289784
2022-09-15

PROCESS FOR PREPARING AN E-SELECTIN INHIBITOR INTERMEDIATE

#1602
20220289765
2022-09-15

CRYSTAL OF CARCINOGENIC FUSED KINASE INHIBITOR AND APPLICATIONS THEREOF

#1603
20220289764
2022-09-15

CRYSTALLINE LORLATINIB : FUMARIC ACID AND SOLID STATE FORM THEREOF

#1604
20220289761
2022-09-15

CRYSTALLINE FORM B OF TETRAHYDROTHIENOPYRIDINE COMPOUND, PREPARATION METHOD, COMPOSITION AND APPLICATION THEREOF

#1605
20220289760
2022-09-15

Crystalline salt of a multi-tyrosine kinase inhibitor, method of preparation, and use thereof

#1606
20220289741
2022-09-15

STABLE POLYMORPHIC FORM OF 6-FLUORO-9-METHYL-9H-B-CARBOLINE AND USES THEREOF

#1607
20220289722
2022-09-15

Crystal forms C and E of pyrazin-2(1H)-one compound and preparation method therefor

#1608
20220289716
2022-09-15

CRYSTALLINE FORMS OF A CD73 INHIBITOR

#1609
20220289713
2022-09-15

SOLID FORMS COMPRISING (S)-4-(4-(4-(((2-(2,6-DIOXOPIPERIDIN-3-YL)-1-OXOISOINDOLIN-4-YL)OXY)METHYL)BENZYL)PIPERAZIN-1-YL)-3-FLUOROBENZONITRILE AND SALTS THEREOF, AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME

#1610
20220289709
2022-09-15

POLYMORPHIC FORMS OF (R)-4-(1-((3-(DIFLUOROMETHYL)-1-METHYL-1H-PYRAZOL-4-YL)SULFONYL)-1-FLUOROETHYL)-N-(ISOXAZOL-3-YL)PIPERIDINE-1-CARBOXAMIDE

#1611
20220289705
2022-09-15

PROCESS FOR THE PREPARATION OF RIDINILAZOLE AND CRYSTALLINE FORMS THEREOF

#1612
20220289694
2022-09-15

Benzisoxazole derivative

#1613
20220289682
2022-09-15

MOLECULAR COMPLEXES

#1614
20220289680
2022-09-15

METHODS FOR MAKING DIMERIC NAPHTHALIMIDES AND SOLID STATE FORMS OF THE SAME

#1615
20220289675
2022-09-15

SALT AND CRYSTAL FORM OF COMPOUND HAVING AGONISTIC ACTIVITY TO S1P5 RECEPTOR

#1616
20220289674
2022-09-15

A PROCESS FOR PRODUCING 4,4'-DICHLORODIPHENYL SULFONE

#1617
20220289672
2022-09-15

Hydrated crystalline form of 2-acrylamido-2-methylpropane sulfonic acid

#1618
20220289670
2022-09-15

PROCESS FOR THE PREPARATION OF A METASTABLE CRYSTAL MODIFICATION OF N-(AMINOIMINOMETHYL)-2-AMINOETHANOIC ACID (IV)

#1619
20220289659
2022-09-15

METHOD FOR THE PRODUCTION OF A DICARBOXYLIC ACID

#1620
20220288078
2022-09-15

Salts of the Janus Kinase Inhibitor (R)-3-(4-(7h-Pyrrolo[2,3-D]Pyrimidin-4-YL)-1h-Pyrazol-1-Yl)-3- Cyclopentylpropanenitrile

#1621
20220281890
2022-09-08

PHARMACEUTICAL COMPOSITIONS CONTAINING SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVES AND PRODRUG THEREOF

#1622
20220281882
2022-09-08

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#1623
20220281881
2022-09-08

Crystalline form of (S)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra- hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#1624
20220281880
2022-09-08

CRYSTALLINE FORMS OF PYRIMIDINO DIAZEPINE DERIVATIVE

#1625
20220281879
2022-09-08

SALT AND CRYSTAL FORMS OF AN ACTIVIN RECEPTOR-LIKE KINASE INHIBITOR

#1626
20220281867
2022-09-08

Lumateperone bis-tosylate salts and crystals and methods for manufacture thereof

#1627
20220281858
2022-09-08

CRYSTALLINE FORM OF ATR INHIBITOR AND USE THEREOF

#1628
20220281853
2022-09-08

Crystal form D of pyrazine-2(1H)-ketone compound and preparation method therefor

#1629
20220281847
2022-09-08

EGFR INHIBITOR FREE BASE OR ACID SALT POLYCRYSTALLINE FORM, PREPARATION METHOD THEREFOR, AND APPLICATION

#1630
20220281836
2022-09-08

PROCESS FOR THE PREPARATION OF APALUTAMIDE

#1631
20220281832
2022-09-08

Crystal modifications of odevixibat

#1632
20220281830
2022-09-08

SALT

#1633
20220281795
2022-09-08

Methods of making bempedoic acid and compositions of the same

#1634
20220281794
2022-09-08

METHOD OF THE ISOLATING CHLOROSESAMONE OR CHLOROSESAMONE-CONTAINING FRACTION FROM ROOTS OF GENUS SESAMUM, AND APPLICATION OF THE FRACTION THEREOF

#1635
20220280531
2022-09-08

Enzymatic process for obtaining 17 alpha-monoesters of cortexolone and/or its 9,11-dehydroderivatives

#1636
20220280496
2022-09-08

PROCESSES OF MAKING AND CRYSTALLINE FORMS OF A MDM2 INHIBITOR

#1637
20220275020
2022-09-01

SALT AND CRYSTAL FORM OF STEROID DERIVATIVE REGULATOR

#1638
20220275011
2022-09-01

Crystalline forms

#1639
20220275004
2022-09-01

MOLECULAR COMPLEXES

#1640
20220274994
2022-09-01

CRYSTALLINE FORM OF (S)-7-(1-ACRYLOYLPIPERIDIN-4-YL)-2-(4-PHENOXYPHENYL)-4,5,6,7-TETRA-HYDROPYRAZOLO[1,5-a]PYRIMIDINE-3-CARBOXAMIDE, PREPARATION, AND USES THEREOF

#1641
20220274977
2022-09-01

NOVEL INHIBITORS

#1642
20220274969
2022-09-01

POLYMORPHS OF (R)-N-(5-(5-ISOPROPYL-1,2,4-OXADIAZOL-3-YL)-2,3-DIHYDRO-1H-INDEN-1-YL)-2-METHYL-2H-TETRAZOLE-5-CARBOXAMIDE

#1643
20220274966
2022-09-01

SURFACTANT SYSTEMS FOR CRYSTALLIZATION OF ORGANIC COMPOUNDS

#1644
20220273663
2022-09-01

Formulations of an AXL/MER inhibitor

#1645
20220267359
2022-08-25

Process for the preparation of the polymorph F of sodium neridronate

#1646
20220267342
2022-08-25

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1647
20220267341
2022-08-25

SOLID FORMS OF TERT-BUTYL (S)-2((2S,3R)-1-AMINO-3-HYDROXY-1-OXOBU TAN-2-YL)-1-OXO-2, 5-DIAZASPIRO [3.4] OCTAN E-5-CARBOXYLATE AND METHODS OF PREPARING THEM

#1648
20220267340
2022-08-25

DOSAGE FORM COMPOSITIONS COMPRISING AN INHIBITOR OF BRUTON'S TYROSINE KINASE

#1649
20220267338
2022-08-25

Hydrates of polymorphs of 6-(1H-indazol-6-yl)-N-(4-morpholinophenyl)-2,3-dihydroimidazo[1,2-a]pyrazin-8-amine bis-mesylate as Syk inhibitors

#1650
20220267334
2022-08-25

CRYSTALLINE FORMS OF AN ORALLY AVAILABLE, SELECTIVE KIT AND PDGFR KINASE INHIBITOR

#1651
20220267326
2022-08-25

CRYSTALLINE FORM OF VALBENAZINE DITOSYLATE, PROCESSES FOR PREPARATION THEREOF AND USE THEREOF

#1652
20220267299
2022-08-25

Crystalline forms of -(3-(2-(2-hydroxyethoxy)-6-morpholinopyridin-4-yl)-4-methvlphenyl)-2 (trifluoromethyl)isonicotinamide as Raf inhibitors for the treatment of cancer

#1653
20220267295
2022-08-25

CRYSTALLINE FORMS OF SOMATOSTATIN MODULATORS

#1654
20220267285
2022-08-25

MANUFACTURING METHODS AND POLYMORPHS OF A THIAZOLINE ANTI-HYPERALGESIC AGENT

#1655
20220267267
2022-08-25

Pharmaceutical composition comprising 5-methoxy-N,N-dimethyltryptamine

#1656
20220267262
2022-08-25

Pharmaceutically acceptable salts of [2-(3-fluoro-5-methane-sulfonylphenoxy)ethyl](propyl)amine and uses thereof

#1657
20220267259
2022-08-25

Crystalline 5-(dimethylamino)-N-(4-(morpholinomethyl) phenyl)naphthalene-1-sulfonamide di-hydrochloride di-hydrate

#1658
20220267257
2022-08-25

Solids of MEK inhibitor N-((R)-2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-benzamide and uses thereof

#1659
20220267248
2022-08-25

Composition of BHET and use thereof

#1660
20220265658
2022-08-25

PHARMACEUTICAL COMPOSITION COMPRISING A TETRAHYDROPYRAZOLOPYRIMIDINONE COMPOUND

#1661
20220265578
2022-08-25

Polymorphic forms of (R)-2-hydroxy-2-methyl-4-(2,4,5-trimethyl-3,6-dioxocyclohexa-1,4-dienyl)butanamide

#1662
20220259627
2022-08-18

Processes for the preparation of (R)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof

#1663
20220259490
2022-08-18

LIGAND-EXCHANGEABLE JANUS NANOPARTICLES AND METHODS OF MAKING THE SAME

#1664
20220259283
2022-08-18

SORCS2 CRYSTAL STRUCTURE AND USES THEREOF

#1665
20220259256
2022-08-18

Crystalline form of vascular leakage blocker compound

#1666
20220259209
2022-08-18

PROCESS FOR THE PREPARATION OF ABROCITINIB

#1667
20220259204
2022-08-18

A PROCESS FOR THE PREPARATION OF VENETOCLAX AND ITS POLYMORPHS THEREOF

#1668
20220259195
2022-08-18

CRYSTALLINE FORMS OF A CYCLIN-DEPENDENT KINASE INHIBITOR

#1669
20220259192
2022-08-18

NOVEL CRYSTALLINE HYDRATE OF TOPRAMEZONE SODIUM SALT AND PREPARATION METHOD THEREFOR

#1670
20220259189
2022-08-18

COCRYSTALS OF POSACONAZOLE, METHODS OF MAKING AND USING SAME

#1671
20220259183
2022-08-18

Crystal form of 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-N-(methyl-d) pyridazine-3-carboxamide

#1672
20220259175
2022-08-18

Crystalline forms of a somatostatin modulator

#1673
20220259162
2022-08-18

SOLID STATE FORMS OF TAFAMIDIS AND SALTS THEREOF

#1674
20220259158
2022-08-18

Solid forms of an N-terminal domain androgen receptor inhibitor and uses thereof

#1675
20220259152
2022-08-18

Crystalline form of compound, method for preparing the same, pharmaceutical composition and use

#1676
20220259147
2022-08-18

Composition comprising a benzoate salt of 5-methoxy-N,N-dimethyltryptamine

#1677
20220259142
2022-08-18

Methods of treating neurofibromatosis with N-((R)-2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-benzamide

#1678
20220259140
2022-08-18

Crystal form and amorphous form of dezocine analogue hydrochloride

#1679
20220257563
2022-08-18

Nitrile-containing antiviral compounds

#1680
20220256879
2022-08-18

CRYO-CRYSTALLISED FAT

#1681
20220256852
2022-08-18

NOVEL CRYSTALLINE FORM OF PYROXASULFONE, METHODS FOR ITS PREPARATION AND USE OF THE SAME

#1682
20220251111
2022-08-11

PROCESS FOR THE PREPARATION OF AMORPHOUS MIDOSTAURIN WITH A LOW CONTENT OF RESIDUAL ORGANIC SOLVENT

#1683
20220251107
2022-08-11

Process for preparing substituted polycyclic pyridone derivative and crystal thereof

#1684
20220251101
2022-08-11

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1685
20220251093
2022-08-11

POTASSIUM SALT CRYSTAL FORM B OF PHOSPHODIESTERASE TYPE 5 INHIBITOR, AND PREPARATION METHOD AND USE THEREFOR

#1686
20220251087
2022-08-11

Substituted imidazo[2,1-f][1,2,4]triazines as PI3K-gamma inhibitors

#1687
20220251078
2022-08-11

Continuous Process for the Preparation of Anticholinergic Drugs

#1688
20220251073
2022-08-11

CRYSTALLINE FORMS OF 7-CHLORO-2-(4-(3-METHOXYAZETIDIN-1-YL)CYCLOHEXYL)-2,4-DIMETHYL-N-((6-METHYL-4-(METHYLTHIO)-2-OXO-1,2-DIHYDROPYRIDIN-3-YL)METHYL)BENZO[D][1,3]DIOXOLE-5-CARBOXAMIDE

#1689
20220251069
2022-08-11

Solid forms of an HIV capsid inhibitor

#1690
20220251063
2022-08-11

COMPOUND FOR ORGANIC ELECTRIC DEVICE, ORGANIC ELECTRIC DEVICE USING THE SAME, AND ELECTRONIC DEVICE THEREOF

#1691
20220251052
2022-08-11

IMPROVED PROCESS FOR THE PREPARATION OF 2-(3,5-DICHLOROPHENYL)-1,3-BENZOXAZOLE-6-CARBOXYLIC ACID OR ITS PHARMACEUTICALLY ACCEPTABLE SALTS AND POLYMORPHS THEREOF

#1692
20220251044
2022-08-11

CRYSTAL FORM OF HYPOXIA-INDUCIBLE FACTOR-PROLYL HYDROXYLASE INHIBITOR

#1693
20220251034
2022-08-11

Preparation Method for Metformin Hydrochloride

#1694
20220251031
2022-08-11

Crystalline Form of y-Aminobutyric Acid Analog

#1695
20220251017
2022-08-11

CRYSTAL FORM I OF CURCUMIN DERIVATIVE, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#1696
20220249976
2022-08-11

Continuous crystallization of cannabinoids in a stirred-tank reactor

#1697
20220243008
2022-08-04

THERMOPLASTIC RESIN, METHOD FOR MANUFACTURING SAME, AND OPTICAL LENS

#1698
20220242897
2022-08-04

CONTINUOUS PROCESS FOR PREPARING THE CRYSTALLINE FORM II OF SOTAGLIFLOZIN

#1699
20220242873
2022-08-04

Method for synthesizing furoimidazopyridine compound, polymorphic substance and polymorphic substance of salt

#1700
20220242860
2022-08-04

Polymorph of latrepirdine dihydrochloride

#1701
20220242851
2022-08-04

CRYSTAL FORM AND SALT OF QUINAZOLINE COMPOUND AND PREPARATION METHOD THEREOF

#1702
20220242836
2022-08-04

Crystalline (2S,4R)-5-(5′-chloro-2′-fluoro-[1,1′-biphenyl]-4-yl)-2-(ethoxymethyl)-4-(3-hydroxyisoxazole-5-carboxamido)-2- methylpentanoic acid and uses thereof

#1703
20220242832
2022-08-04

PROCESS FOR PREPARING XPO1 INHIBITORS AND INTERMEDIATES FOR USE IN THE PREPARATION OF XPO1 INHIBITORS

#1704
20220242829
2022-08-04

PROCESS FOR PREPARATION OF ENZALUTAMIDE

#1705
20220242816
2022-08-04

Methods for making and using endoxifen

#1706
20220242811
2022-08-04

CRYSTAL FORM OF TREPROSTINIL SODIUM SALT AND PREPARATION METHOD THEREFOR

#1707
20220242810
2022-08-04

CRYSTALLINE CANNABIGEROL

#1708
20220241258
2022-08-04

FORMULATIONS OF T-TYPE CALCIUM CHANNEL MODULATORS AND METHODS OF USE THEREOF

#1709
20220235110
2022-07-28

De novo design of potent and selective interleukin mimetics

#1710
20220235085
2022-07-28

PROCESS FOR PREPARING THE CRYSTALLINE FORM II OF SOTAGLIFLOZIN

#1711
20220235079
2022-07-28

Crystalline forms of Tenofovir alafenamide

#1712
20220235063
2022-07-28

MORPHIC FORMS OF MARIZOMIB AND USES THEREOF

#1713
20220235045
2022-07-28

Solid state forms

#1714
20220235039
2022-07-28

CRYSTALLINE SALT FORMS OF 6-(CYCLOPROPANECARBOXAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYLD3) PYRIDAZINE-3-CARBOXAMIDE

#1715
20220235037
2022-07-28

Crystalline forms of a MAGL inhibitor

#1716
20220235030
2022-07-28

SELECTIVE HISTAMINE H3 ANTAGONIST ACID ADDITION SALTS AND PROCESS FOR THE PREPARATION THEREOF

#1717
20220235029
2022-07-28

CRYSTAL FORM OF C-MET/AXL INHIBITOR

#1718
20220235014
2022-07-28

PROCESS FOR THE PREPARATION OF HIGHLY PURE ERLOTINIB HYDROCHLORIDE

#1719
20220234996
2022-07-28

Method for Producing (3S)-3-(4-chloro-3-{[(2S,3R)-2-(4-chlorophenyl)-4,4,4-trifluoro-3-methylbutanoyl]amino}phenyl)-3-cyclo-propylpropanoic Acid and the Crystalline Form Thereof for Use as a Pharmaceutical Ingredient

#1720
20220227784
2022-07-21

SOLID STATE FORMS OF RELUGOLIX

#1721
20220227777
2022-07-21

Synthesis method of furoimidazopyridine compound, crystal form of furoimidazopyridine compound, and crystal form of salt thereof

#1722
20220227770
2022-07-21

Salts of TAM inhibitors

#1723
20220227769
2022-07-21

CRYSTALLINE FORM OF TELMAPITANT OR (5R,8S)-8-[[(1R)-1-[3,5-BIS(TRIFLUOROMETHYL)PHENYL]ETHOXY]METHYL]-8-PHENYL-1,3,7-TRIAZASPIRO[4.5]DECANE-2,4-DIONE

#1724
20220227753
2022-07-21

Methods of preparing heteroaryl-ketone fused azadecalin glucocorticoid receptor modulators

#1725
20220227712
2022-07-21

Cholinesterase inhibitor polymorph and application thereof

#1726
20220226328
2022-07-21

Heterocyclic compounds, preparation methods and uses thereof

#1727
20220220149
2022-07-14

SOLID STATE FORMS OF SAGE-217 AND PROCESSES FOR PREPARATION THEREOF

#1728
20220220146
2022-07-14

MORPHIC FORMS OF 4-AMINO-7-(3,4-DIHYDROXY-5-(HYDROXYMETHYL)TETRAHYDROFURAN-2-YL)-2-METHYL-7H-PYRROLO[2,3-d]PYRIMIDINE-5-CARBOXAMIDE AND USES THEREOF

#1729
20220220123
2022-07-14

AMORPHOUS AND CRYSTALLINE FORMS OF RELUGOLIX

#1730
20220220121
2022-07-14

Solid forms of Alpha-1062 gluconate

#1731
20220220120
2022-07-14

Crystal form of Wee1 inhibitor compound and use thereof

#1732
20220220118
2022-07-14

3-(ethoxydifluoromethyl)-6-(5-fluoro-6-(2,2,2-trifluoroethoxy)pyridin-3-yl)-[1,2,4]triazolo[4,3-a]pyridine as an ion channel modulator

#1733
20220220107
2022-07-14

CRYSTAL FORMS OF ACRYLIC ACID DERIVATIVES, PREPARATION METHOD THEREFOR AND USE THEREOF

#1734
20220220098
2022-07-14

Crystal form of pyrimidine sulfonamide compound and preparation method therefor

#1735
20220220093
2022-07-14

CRYSTALLINE FORMS OF N-(4-(4-(CYCLOPROPYLMETHYL)PIPERAZINE-1-CARBONYL)PHENYL)QUINOLINE-8-SULFONAMIDE

#1736
20220220075
2022-07-14

SOLID FORM OF AROMATIC COMPOUND AND PREPARATION METHOD THEREFOR

#1737
20220220074
2022-07-14

Solid forms of n-tert-butyl-4[[2-(5-chloro-2-hydroxy-phenyl)acetyl]amino]pyridine-2-carboxamide

#1738
20220220059
2022-07-14

PROCESS FOR CRYSTALLIZATION OF HIGH PURITY LUTEIN ESTERS FROM MARIGOLD EXTRACTS

#1739
20220220054
2022-07-14

2,3,5-trimethyl-6-nonylcyclohexa-2,5-diene-1,4-dione for suppressing and treating alpha-synucleinopathies, tauopathies, and other disorders

#1740
20220218706
2022-07-14

Inhalable imatinib formulations, manufacture, and uses thereof

#1741
20220213107
2022-07-07

Tertiary alcohols as PI3K-γ inhibitors

#1742
20220213085
2022-07-07

Compound containing fused ring, use thereof and pharmaceutical composition containing same

#1743
20220213075
2022-07-07

3-ARYLOXY-3-FIVE-MEMBERED HETEROARYL PROPYLAMINE COMPOUND, AND CRYSTAL FORM AND USE THEREOF

#1744
20220213066
2022-07-07

SALTS OF A CLASS OF PYRIMIDINE COMPOUNDS, POLYMORPHS, AND PHARMACEUTICAL COMPOSITIONS THEREOF, PREAPRATION METHODS THEREFOR AND USES THEREOF

#1745
20220213060
2022-07-07

Crystal Form of Quinazolinone Compound and Preparation Method Therefor

#1746
20220213056
2022-07-07

PROCESSES FOR PREPARING 2-(4-CHLOROPHENYL)-N-((2-(2,6-DIOXOPIPERIDIN-3-YL)-1-OXOISOINDOLIN-5-YL)METHYL)-2,2-DIFLUOROACETAMIDE

#1747
20220213051
2022-07-07

NOVEL CRYSTAL FORM OF 3-(4-(BENZYLOXY)PHENYL)HEX-4-INOIC ACID DERIVATIVE

#1748
20220213014
2022-07-07

CRYSTALLINE POLYMORPHS OF 1,6-DIBROMO-1,6-DIDEOXY-DULCITOL

#1749
20220204536
2022-06-30

Crystals

#1750
20220204526
2022-06-30

Hydroxypyridoxazepines as NRF2 activators

#1751
20220204519
2022-06-30

Crystal form of upadacitinib, preparation method therefor, and use thereof

#1752
20220204514
2022-06-30

POLYMORPHS OF 7-CYCLOPENTYL-N,N-DIMETHYL-2-{[5-(PIPERAZIN-1-YL) PYRIDIN-2-YL]-AMINO}-7H-PYRROLO[2,3-D]PYRIMIDINE-6-CARBOXAMIDE AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS AND PROCESS FOR THE PREPARATION THEREOF

#1753
20220204506
2022-06-30

Crystalline salts of a B-RAF kinase inhibitor

#1754
20220204502
2022-06-30

CRYSTAL POLYMORPHISM OF PI3K INHIBITOR AND METHOD FOR PREPARING SAME

#1755
20220204494
2022-06-30

CRYSTAL FORM S4 OF THE PLK4 INHIBITOR (1R,2S)-(E)-2-(3-(4-((CIS-2,6-DIMETHYLMORPHOLINO)METHYL)STYRYL)- 1 H-IMIDAZOL-6- YL)-5'-METHOXYSPIRO[CYCLOPROPANE-1,3'-INDOLIN]-2'-ONE FUMARATE

#1756
20220204493
2022-06-30

CRYSTALLINE FORM OF A BET-INHIBITOR AND MANUFACTURE THEREOF

#1757
20220204480
2022-06-30

Crystalline forms of imidacloprid and methods of use thereof

#1758
20220204475
2022-06-30

SOLID FORM OF DIAMINOPYRIMIDINE COMPOUND OR HYDRATE THEREOF, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#1759
20220204454
2022-06-30

Crystalline salts of a plasma kallikrein inhibitor

#1760
20220204448
2022-06-30

Crystalline forms and methods of producing crystalline forms of a compound

#1761
20220204443
2022-06-30

Metastable crystal modification and method for producing the same (I)

#1762
20220204432
2022-06-30

Honokiol crystal forms, amorphous form and preparation thereof

#1763
20220204431
2022-06-30

METHOD FOR PREPARING CANNABIDIOL COMPOUND

#1764
20220202790
2022-06-30

Salts of selective estrogen receptor degraders

#1765
20220195471
2022-06-23

Method for resolving optical isomer by using supercritical fluid extraction technology

#1766
20220194964
2022-06-23

SOLID FORMS OF AN ORALLY-DELIVERED BETA-LACTAMASE INHIBITOR AND USES THEREOF

#1767
20220194959
2022-06-23

CRYSTAL FORM OF EGFR INHIBITOR AND PREPARATION METHOD THEREOF

#1768
20220194946
2022-06-23

FGFR inhibitors and methods of making and using the same

#1769
20220194936
2022-06-23

CRYSTALLINE FORMS OF N-(5-(5-((1R,2S)-2-FLUOROCYCLOPROPYL)-1,2,4-OXADIAZOL-3-YL)-2-METHYLPHENYL)IMIDAZO[1,2-A]PYRIDINE-3-CARBOXAMIDE

#1770
20220194934
2022-06-23

CRYSTAL FORM OF PHOSPHODIESTERASE INHIBITOR,PREPARATION METHOD THEREFOR AND USE THEREOF

#1771
20220194922
2022-06-23

CYCLOPENTANE COMPOUNDS

#1772
20220194919
2022-06-23

CO-CRYSTALLINE EFINACONAZOLE, AND METHOD FOR PRODUCING SAME

#1773
20220194899
2022-06-23

Highly purified batches of pharmaceutical grade 1-deoxygalactonojirimycin compounds

#1774
20220194898
2022-06-23

Method of preparing a DON prodrug from L-pyroglutamic acid

#1775
20220193057
2022-06-23

Formulations of pimavanserin

#1776
20220185825
2022-06-16

SALT FORM AND CRYSTAL FORM OF A2A RECEPTOR ANTAGONIST AND PREPARATION METHOD THEREFOR

#1777
20220185820
2022-06-16

BRD4 INHIBITOR COMPOUND IN SOLID FORM AND PREPARATION METHOD THEREFOR AND USE THEREOF

#1778
20220185815
2022-06-16

Pyrrolopyrazole derivative

#1779
20220185807
2022-06-16

Crystalline berberine ascorbate salt, methods of preparation and applications thereof

#1780
20220185791
2022-06-16

POLYMORPHS OF A CARDIAC TROPONIN ACTIVATOR

#1781
20220185790
2022-06-16

Polymorphs and cocrystals of a cardiac troponin activator

#1782
20220185781
2022-06-16

BULLEYACONITINE D CRYSTAL AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#1783
20220185780
2022-06-16

PIROCTONE OLAMINE RECRYSTALLIZATION

#1784
20220185776
2022-06-16

Highly purified batches of pharmaceutical grade migalastat and methods of producing the same

#1785
20220185767
2022-06-16

NOVEL TERNARY MOLECULAR COMPLEX OF TAMIBAROTENE FOR CANCER STEM CELLS TREATMENT

#1786
20220184080
2022-06-16

NEBULIZED IMATINIB FORMULATIONS, MANUFACTURE, AND USES THEREOF

#1787
20220184041
2022-06-16

(AZA)Benzothiazolyl Substituted Pyrazole Compounds

#1788
20220177935
2022-06-09

Solid form of (-)-Ambrox formed by a bioconversion of homofarnesol in the presence of a biocatalyst

#1789
20220177531
2022-06-09

Selective and noncovalent inhibitors of oncogenic RAS mutants

#1790
20220177499
2022-06-09

Methods for producing crystalline L-glufosinate ammonium monohydrate

#1791
20220177498
2022-06-09

Crystalline form of L-glufosinate ammonium salt and process for production thereof

#1792
20220177483
2022-06-09

Crystal form of acid addition salt of furopyrimidine compound

#1793
20220177476
2022-06-09

Crystal Forms of (S)-4-(8-amino-3-(1-(but-2-ynoyl)-pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide

#1794
20220177475
2022-06-09

FGFR INHIBITOR COMPOUND IN SOLID FORM AND PREPARATION METHOD THEREFOR

#1795
20220177474
2022-06-09

Purinone derivative hydrochloride

#1796
20220177469
2022-06-09

Solid forms of emetine

#1797
20220177468
2022-06-09

Integrin inhibitor and uses thereof

#1798
20220177463
2022-06-09

Pharmaceutical salts of benzothiazol compounds, polymorphs and methods for preparation thereof

#1799
20220177455
2022-06-09

CRYSTAL FORMS OF A PYRIDAZINONE TRPC INHIBITOR

#1800
20220177453
2022-06-09

CRYSTALLIZATION OF SMAC MIMIC USED AS IAP INHIBITOR AND PREPARATION METHOD THEREOF