ClassID:

90494

C07B2200/13 - page 5 - CPC Classification

Classification description:

Indexing scheme relating to specific properties of organic compounds Crystalline forms, e.g. polymorphs

Recent Application in this class:
#1201
20230151043
2023-05-18

Compounds and methods for treatment of viral infections

#1202
20230151036
2023-05-18

Psilocybin and O-acetylpsilocin, salts and solid state forms thereof

#1203
20230151029
2023-05-18

BORONIC ACID DERIVATIVES AND THERAPEUTIC USES THEREOF

#1204
20230151015
2023-05-18

Crystalline forms of (s)-4-amino-6-((1-(3-chloro-6-phenylimidazo[1,2-b]pyridazine-7-yl)ethyl)amino)pyrimidine-5-carbonitrile as inhibitors of phosphatidylinositol-3-kinase

#1205
20230151010
2023-05-18

CRYSTALLINE FORMS OF (9R, 135S)-13- {4-[5-CHLORO-2-(4-CHLORO-1H,2,3- TRIAZOL- 1 -YL)PHENYL] -6-OXO- 1,6-DIHYDROPYRIMIDIN- 1-YL}-3-(DIFLUOROMETHYL)-9-METHYL-3,4,7,15- TETRAAZATRICYCLO [ 12.3.1.0 2·6] OCTADECA- 1(18), 2(6), 4, 14, 16-PENTAEN-8-ONE

#1206
20230151009
2023-05-18

Polymorphs

#1207
20230151008
2023-05-18

Crystalline imidazo[4,5-b]pyridine compound, pharmaceutical compositions, and their use in treating medical conditions

#1208
20230150994
2023-05-18

METHODS FOR SYNTHESIS OF CHK1 INHIBITORS

#1209
20230150959
2023-05-18

PHARMACEUTICAL COMPOSITION COMPRISING TIZOXANIDE AND PHARMACEUTICAL USE THEREOF

#1210
20230150958
2023-05-18

REFINING METHOD

#1211
20230150957
2023-05-18

REFINING METHOD

#1212
20230150950
2023-05-18

Potassium salt of 2-[(4S)-8-fluoro-2-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[2-methoxy-5-(trifluoromethyl)phenyl]-4H-quinazolin-4-yl]acetic acid

#1213
20230150937
2023-05-18

Crystalline dimethyl tryptamine analogues

#1214
20230150928
2023-05-18

METHOD FOR PRODUCING BENZOPYRANONE COMPOUND AND NOVEL INTERMEDIATE USED THEREIN

#1215
20230150920
2023-05-18

SALTS AND SOLID FORMS OF 4-BROMO-2,5-DIMETHOXYPHENETHYLAMINE

#1216
20230148402
2023-05-11

Boron Containing PDE4 Inhibitors

#1217
20230147959
2023-05-11

COMPOUND FOR ORGANIC OPTOELECTRONIC DEVICE, COMPOSITION FOR ORGANIC OPTOELECTRONIC DEVICE, ORGANIC OPTOELECTRONIC DEVICE AND DISPLAY DEVICE

#1218
20230147756
2023-05-11

CRYSTALLINE FORMS OF A FARNESOID X RECEPTOR AGONIST

#1219
20230147490
2023-05-11

Inhibiting agents for bruton's tyrosine kinase

#1220
20230147121
2023-05-11

Compositions of solid forms of (S)-2-(((S)-6,8-difluoro-1,2,3,4- tetrahydronaphthalen-2-yl)amino)-N-(1-(2-methyl-1-(neopentylamino)propan-2-yl)-1H-imidazol-4-yl)pentanamide

#1221
20230146719
2023-05-11

CRYSTALLINE N-METHYL TRYPTAMINE DERIVATIVES

#1222
20230145648
2023-05-11

Crystalline psilacetin derivatives

#1223
20230144619
2023-05-11

SALT OF ARYLAMINOPURINE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF

#1224
20230144367
2023-05-11

MECHANICAL-BOND-PROTECTED STABLE BISRADICALS

#1225
20230144309
2023-05-11

Crystalline form of L-glufosinate ammonium salt and process for production thereof

#1226
20230144122
2023-05-11

PYRIDONE DERIVATIVE CRYSTAL FORM AND PREPARATION METHOD AND APPLICATION THEREFOR

#1227
20230142424
2023-05-11

A2-73 crystalline polymorph compositions of matter and methods of use thereof

#1228
20230142366
2023-05-11

NOVEL POLYMORPHIC FORMS OF METOPIMAZINE

#1229
20230141887
2023-05-11

CRYSTAL FORM OF DIAZASPIROPYRAN COMPOUND

#1230
20230141783
2023-05-11

DIFFERENT FORMS OF 6-CHLORO-2-ETHYL-N-(4-(4-(4-(TRIFLUOROMETHOXY)PHENYL)PIPERIDINE-1-YL)BENZYL)IMIDAZO[1,2-A]PYRIDINE-3-CARBOXAMIDE

#1231
20230141635
2023-05-11

SALT FORMS OF BEMPEDOIC ACID AND METHODS FOR USING THE SAME

#1232
20230139835
2023-05-04

ALLULOSE IN CRYSTALLINE FORM

#1233
20230139815
2023-05-04

Crystalline forms of a cannabinoid receptor type 1 (CB1) modulator and methods of use and preparation thereof

#1234
20230139741
2023-05-04

LIGHT EMITTING ELEMENT AND POLYCYCLIC COMPOUND FOR THE SAME

#1235
20230139418
2023-05-04

Crystalline salts or co-crystals of 2′,6-difluoro-5′-[3-(1-hydroxy-1-methylethyl)-imidazo[1,2-b][1,2,4]triazin-7-yl]biphenyl-2-carbonitrile with p-toluenesulofonic acid as GABAA positive allosteric modulators

#1236
20230138150
2023-05-04

RADIO-PROTECTIVE AND CHEMO-PROTECTIVE SUBSTITUTED THIOLS

#1237
20230137090
2023-05-04

PROCESSES AND INTERMEDIATE FOR THE LARGE-SCALE PREPARATION OF 2,4,6-TRIFLUORO-N-[6-(1-METHYL-PIPERIDINE-4-CARBONYL)-PYRIDIN-2-YL]-BENZAMIDE HEMISUCCINATE, AND PREPARATION OF 2,4,6-TRIFLUORO-N-[6-(1-METHYL-PIPERIDINE-4-CARBONYL)-PYRIDIN-2-YL]-BENZAMIDE ACETATE

#1238
20230135100
2023-05-04

Process of preparing a peptide epoxyketone immunoproteasome inhibitor, and precursors thereof

#1239
20230134869
2023-05-04

CRYSTAL FORM OF FREE ALKALI OF NITROGEN-CONTAINING AROMATIC DERIVATIVES

#1240
20230133435
2023-05-04

COCRYSTALS DERIVATIVES OF APIXABAN

#1241
20230132370
2023-04-27

Crystal forms of thiazole compound and application thereof

#1242
20230131316
2023-04-27

PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF CARBOPROST AND CARBOPROST TROMETHAMINE, AND CARBOPROST TROMETHAMINE PREPARED THEREFROM

#1243
20230131180
2023-04-27

Processes for producing amide compounds, and their crystalline and salt form

#1244
20230128824
2023-04-27

SPIRO RING-CONTAINING QUINAZOLINE COMPOUND

#1245
20230128162
2023-04-27

TRIAZINE DERIVATIVES HAVING VIRUS REPLICATION INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME

#1246
20230127805
2023-04-27

PROCESS FOR THE PREPARATION OF (R)-4-(1-(6-(4-(TRIFLUOROMETHYL)BENZYL)-6-AZASPIRO[2.5]OCTANE-5-CARBOXAMIDO)-CYCLOPROPYL) BENZOIC ACID OR A SALT THEREOF

#1247
20230127683
2023-04-27

Crystalline bis-miprocin fumarate

#1248
20230126343
2023-04-27

Crystalline 4-hydroxy-N,N-di-n-propyltryptammonium (4-HO-DPT) salts

#1249
20230125950
2023-04-27

METHOD AND DEVICE FOR SEPARATION AND PURIFICATION OF GLYCOLIC ACID BY RECTIFICATION-CRYSTALLIZATION COUPLING PROCESS AND USE

#1250
20230125064
2023-04-20

Crystal form of phosphodiesterase inhibitor, preparation method therefor and use thereof

#1251
20230124801
2023-04-20

Dosing regimens of (S)-1-(4-fluorophenyl)-1-(2-(4-(6-(1-methyl-1H-pyrazol-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl)piperazinyl)-pyrimidin-5-yl)ethan-1-amine for treatment of indolent systemic mastocytosis

#1252
20230124705
2023-04-20

Solid forms, pharmaceutical compositions and preparation of heteroaromatic macrocyclic ether compounds

#1253
20230124137
2023-04-20

Method for treating anxiety disorders, headache disorders, and eating disorders with psilocybin

#1254
20230123250
2023-04-20

Crystalline 5-methoxy-n,n-diallyltryptamine compounds

#1255
20230123104
2023-04-20

CRYSTAL OF TRICYCLIC COMPOUND ACTING ON CRBN PROTEIN AND PREPARATION METHOD THEREFOR

#1256
20230122169
2023-04-20

NOVEL METHOD FOR PREPARING (-)-CIBENZOLINE SUCCINATE

#1257
20230121825
2023-04-20

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#1258
20230121695
2023-04-20

SOLID FORMS OF AN FGFR INHIBITOR AND PROCESSES FOR PREPARING THE SAME

#1259
20230121611
2023-04-20

Monohydrate Salt of Denatonium Acetate

#1260
20230121346
2023-04-20

THE SALTS OF A COMPOUND AND THE CRYSTALLINE FORMS THEREOF

#1261
20230120974
2023-04-20

Compositions for treatment of ocular diseases

#1262
20230120311
2023-04-20

SALTS AND CRYSTALLINE FORMS OF A TAAR1 AGONIST

#1263
20230120254
2023-04-20

Nitrile-Containing Antiviral Compounds

#1264
20230119714
2023-04-20

Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use

#1265
20230119296
2023-04-20

CRYSTAL FORM OF NITROXOLINE PRODRUG, PHARMACEUTICAL COMPOSITION CONTAINING SAME, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#1266
20230118562
2023-04-20

ZIRCONIUM PHOSPHATE

#1267
20230117777
2023-04-20

METHYLATION OF MCL-1 COMPOUNDS

#1268
20230117059
2023-04-20

Solid state forms of Belumosudil and Belumosudil salts

#1269
20230116697
2023-04-13

Complexation of pirfenidone with polyphenolic calixarene or resorcin[4]arenes

#1270
20230115881
2023-04-13

PROCESSES OF MAKING 3-FLUORO-5-(((1S,2aR)-1,3,3,4,4-PENTAFLUORO-2a-HYDROXY-2,2a,3,4-TETRAHYDRO-1H-CYCLOPENTA[CD]INDEN-7-YL)OXY)-BENZONITRILE AND POLYMORPHS THEREOF

#1271
20230115869
2023-04-13

BUDESONIDE 21-PHOSPHATE SALTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME

#1272
20230115817
2023-04-13

CRYSTAL OF PDE3/PDE4 DUAL INHIBITOR AND USE THEREOF

#1273
20230115605
2023-04-13

CRYSTAL FORM OF AROMATIC VINYL DERIVATIVES, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#1274
20230115500
2023-04-13

Process for the preparation of iloprost

#1275
20230113948
2023-04-13

SYNTHETIC PROCESSES AND INTERMEDIATES

#1276
20230112623
2023-04-13

Phosphonium compound, reagent kit for derivatization, mass spectrometric method, and method for producing phosphonium compound

#1277
20230112410
2023-04-13

Crystalline norpsilocin compounds

#1278
20230111912
2023-04-13

Salts of a Pim kinase inhibitor

#1279
20230110129
2023-04-13

Isofagomine salts, methods of use and formulations

#1280
20230109556
2023-04-06

Methods of treating neurofibromatosis type 1 with N-((R))-2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodophenylamino)-benzamide

#1281
20230108971
2023-04-06

Salts and crystal forms of omecamtiv mecarbil

#1282
20230107634
2023-04-06

PROCESSES FOR THE PREPARATION OF GLASDEGIB AND SALT THEREOF AND SOLID STATE FORMS OF GLASDEGIB MALEATE AND PROCESS FOR PREPARATION THEREOF

#1283
20230107185
2023-04-06

(Thio)nicotinamide ribofuranoside salts and compositions, methods of making, and uses thereof

#1284
20230106656
2023-04-06

Crystalline salts of peptide epoxyketone immunoproteasome inhibitor

#1285
20230106142
2023-04-06

CRYSTALS OF ALKYNYL-CONTAINING COMPOUND, SALT AND SOLVATE THEREOF, PREPARATION METHOD, AND APPLICATIONS

#1286
20230106081
2023-04-06

METHODS OF TREATING PARKINSON'S DISEASE

#1287
20230106064
2023-04-06

CRYSTALLINE FORM OF FLUVATINIB OR FLUVATINIB METHANESULFONATE AND PREPARATION METHOD THEREFOR

#1288
20230105412
2023-04-06

5-HT3 RECEPTOR MODULATOR, THE CRYSTALLINE FORM, METHODS OF MAKING, AND USE THEREOF

#1289
20230105181
2023-04-06

SALTS AND POLYMORPHIC FORMS OF 6-CHLORO-7-(4-(4-CHLOROBENZYL)PIPERAZIN-1-YL)-2-(1,3-DIMETHYL-1H-PYRAZOL-4-YL)-3H-IMIDAZO[4,5-B]PYRIDINE

#1290
20230104965
2023-04-06

ENZYMATIC PROCESS FOR OBTAINING 17 ALPHA-MONOESTERS OF CORTEXOLONE AND/OR ITS 9,11-DEHYDRODERIVATIVES

#1291
20230104647
2023-04-06

METHODS AND PROCESSES FOR THE PREPARATION OF KDM1A INHIBITORS

#1292
20230104598
2023-04-06

Solid forms of an N-terminal domain androgen receptor inhibitor and uses thereof

#1293
20230103724
2023-04-06

SOLID STATE FORMS OF AVAPRITINIB AND PROCESS FOR PREPARATION THEREOF

#1294
20230103409
2023-04-06

Crystal form of pyrrolidinyl urea derivative and application thereof

#1295
20230103362
2023-04-06

EBNA1 inhibitor crystalline forms, and methods of preparing and using same

#1296
20230102321
2023-03-30

Method for producing allulose crystals

#1297
20230102273
2023-03-30

Crystalline forms of 2-[(2S)-1-azabicyclo[2.2.2]oct-2-yl]-6-(3-methyl-1H-pyrazol-4-yl)thieno[3,2-d]pyrimidin-4(3H)-one hemihydrate

#1298
20230101987
2023-03-30

Substituted pyridines as DNMT1 inhibitors

#1299
20230101131
2023-03-30

Phenylcarbamate crystalline form and method for manufacturing the same

#1300
20230100647
2023-03-30

COMPOSITION AND METHOD FOR PRODUCING SAME

#1301
20230100211
2023-03-30

PROCESS FOR THE PREPARATION OF SODIUM 4-(2-((1E,3E,5E,7Z)-7-(1,1-DIMETHYL-3-(4-SULFONATOBUTYL)-1H-BENZO[e]INDOL-2(3H)-YLIDENE) HEPTA-1,3,5-TRIENYL)-1,1-DIMETHYL-1H-BENZO[e]INDOLIUM-3-YL) BUTANE-1-SULFONATE (INDOCYANINE GREEN)

#1302
20230099116
2023-03-30

SSTR4 agonist salts

#1303
20230098309
2023-03-30

Crystalline succinate salt of 6-(6-aminopyrazin-2-yl)-N-(4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)imidazo[1,2-a]pyrazin-8-amine as a Syk inhibitor

#1304
20230098234
2023-03-30

Solid state forms of Mitapivat and process for preparation thereof

#1305
20230097470
2023-03-30

PROCESSES AND INTERMEDIATES FOR THE PREPARATIONS OF CARBOPROST AND CARBOPROST TROMETHAMINE, AND CARBOPROST TROMETHAMINE PREPARED THEREFROM

#1306
20230097240
2023-03-30

SOLID STATE FORMS OF ASCIMINIB AND PROCESSES FOR THE PREPARATION THEREOF

#1307
20230096670
2023-03-30

INTERMEDIATE USEFUL FOR SYNTHESIS OF SGLT INHIBITOR AND METHOD FOR PREPARING SGLT INHIBITOR USING SAME

#1308
20230096322
2023-03-30

HYDRATED CRYSTALLINE POLYNUCLEAR METAL COMPLEX, HYDRATED CRYSTALLINE POLYNUCLEAR METAL COMPLEX INCLUDING A GUEST COMPOUND ANALYTE AND ITS USE IN A METHOD FOR DETERMINING MOLECULAR STRUCTURE OF THE GUEST COMPOUND ANALYTE

#1309
20230096245
2023-03-30

Crystalline forms of ALDH2 modulators

#1310
20230095799
2023-03-30

Crystalline forms of 8-(2-fluorobenzyl)-6-(3-(trifluoromethyl)-1H-1,2,4-triazol-5-yl)imidazo[1,2-a]pyrazine as sGC stimulators

#1311
20230094124
2023-03-30

Morphic forms of danicopan

#1312
20230094109
2023-03-30

POLYMORPHS OF ELAFIBRANOR

#1313
20230093755
2023-03-23

COMPOUNDS AND THEIR USE FOR THE TREATMENT OF ALPHA1-ANTITRYPSIN DEFICIENCY

#1314
20230093615
2023-03-23

Crystal forms of 2-[4-[(2,3,4- trimethoxyphenyl)methyl]piperazin-1-yl]ethyl pyridine-3-carboxylate

#1315
20230092495
2023-03-23

SOLID FORMS OF TEZACAFTOR AND PROCESSES FOR THE PREPARATION THEREOF

#1316
20230092359
2023-03-23

GEMFIBROZIL FORMULATION

#1317
20230092143
2023-03-23

Method for the synthesis of 2,4-dimethylpyrimidin-5-ol, intermediates, and method for the synthesis of Lemborexant using the intermediates

#1318
20230092001
2023-03-23

Furaneone glycoside compound, pharmaceutical composition thereof, preparation method therefor, and application thereof

#1319
20230091736
2023-03-23

Crystalline forms of tenofovir alafenamide

#1320
20230091250
2023-03-23

CRYSTALLINE FORM OF JAK INHIBITOR AND APPLICATION THEREOF

#1321
20230089503
2023-03-23

Crystalline forms of N-[4-(chlorodifluoromethoxy)phenyl]-6-[(3R)-3-hydroxypyrrolidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide

#1322
20230089334
2023-03-23

Hydrate of dimethylaminomicheliolide fumarate and preparation method therefor and use thereof

#1323
20230088814
2023-03-23

Fasoracetam crystalline forms

#1324
20230088511
2023-03-23

Polymorphic Form of (-)-Cibenzoline Succinate

#1325
20230087828
2023-03-23

SOLID STATE FORMS OF (S)-2-(((S)-6,8-DIFLUORO-1,2,3,4-TETRAHYDRONAPHTHALEN-2-YL)AMINO)-N-(1-(2-METHYL-1-(NEOPENTYLAMINO)PROPAN-2-YL)-1H-IMIDAZOL-4-YL)PENTANAMIDE AND USES THEREOF

#1326
20230086867
2023-03-23

Polymorphic forms of metopimazine

#1327
20230086578
2023-03-23

Crystalline epinephrine malonate salt

#1328
20230086574
2023-03-23

5-methoxy-N,N-dimethyltryptamine crystalline forms

#1329
20230086230
2023-03-23

Inhalable imatinib formulations, manufacture, and uses thereof

#1330
20230086137
2023-03-23

Crystalline forms of N-[4-[4-(4-morpholinyl)-7H-pyrrolo[2,3-d]pyrimidin-6-yl]phenyl]-4-[[3(r)-[(1-oxo-2-propen-1-yl)amino]-1-piperidinyl]methyl]-2-pyridinecarboxamide as an irreversible inhibitor of menin-MLL interaction

#1331
20230085243
2023-03-16

METHOD FOR IMPROVING THE HUE OF RECYCLED BIS(2-HYDROXYETHYL) TEREPHTHALATE

#1332
20230083960
2023-03-16

Bicyclic 1,4-diazepanones and therapeutic uses thereof

#1333
20230080477
2023-03-16

PROCESS OF SYNTHESIS OF NOVEL CHROMIUM (III) COMPLEXES OF SCHIFF BASE LIGANDS AND THEIR USE THERE OF AS THERAPEUTIC AGENTS

#1334
20230078576
2023-03-16

Compounds and their use

#1335
20230076079
2023-03-09

Polymorphisms of HM30181 mesylate

#1336
20230075170
2023-03-09

NOVEL SALTS OF NILOTINIB AND POLYMORPHIC FORMS THEREOF

#1337
20230074827
2023-03-09

CRYSTALLINE FORMS OF DEUTERIUM-ENRICHED PIOGLITAZONE

#1338
20230074669
2023-03-09

Cycloalkane-1,3-diamine derivative

#1339
20230074179
2023-03-09

POLYMORPH OF EP4 RECEPTOR ANTAGONIST, PREPARATION METHOD THEREFOR AND USE THEREOF

#1340
20230074115
2023-03-09

Synthesis of antibacterial aminoglycoside analogs

#1341
20230074064
2023-03-09

Crystalline forms OF N-[4-(chlorodifluoromethoxy)phenyl]-6-[(3R)-3-hydroxypyrrolidin-1-yl]-5-(1H-pyrazol-5-yl)pyridine-3-carboxamide

#1342
20230072389
2023-03-09

Crystal forms and production methods thereof

#1343
20230071463
2023-03-09

SOLID STATE FORMS OF AVASOPASEM MANGANESE AND PROCESS FOR PREPARATION THEREOF

#1344
20230070611
2023-03-09

Crystal form of thieno[2,3-c]pyridazine-4(1H)-one compound, preparation method therefor and use thereof

#1345
20230068593
2023-03-02

PROCESSES FOR PREPARING TUCATINIB POLYMORPHS

#1346
20230067676
2023-03-02

CO-CRYSTALS AND SALTS OF 8-CHLORO-N-(4-(TRIFLUOROMETHOXY)PHENYL)QUINOLIN-2-AMINE

#1347
20230067666
2023-03-02

METHOD FOR PREPARING COUMARIN COMPOUNDS SUBSTITUTED BY AMIDOALKYL AT 3-POSITION, THE PRODUCTS AND RELATED INTERMEDIATES THEREOF

#1348
20230065420
2023-03-02

COMPOUNDS AND METHODS FOR THE DIAGNOSIS, IMAGING AND TREATMENT OF NEURODEGENERATIVE DISEASES AND DISORDERS

#1349
20230064976
2023-03-02

AMORPHOUS FORM OR CRYSTALLINE FORM OF 2-INDOLINOLINOLOLYLSPIRONONE COMPOUNDS OR THEIR SALTS, SOLVENT COMPLEXES

#1350
20230064948
2023-03-02

HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT OR AMELIORATION OF CANCER

#1351
20230064136
2023-03-02

Citrate salt, pharmaceutical compositions, and methods of making and using the same

#1352
20230063754
2023-03-02

NOVEL METHOD FOR SYNTHESIZING DECURSIN DERIVATIVE

#1353
20230063538
2023-03-02

LARGE SCALE PROCESS

#1354
20230063175
2023-03-02

Crystalline forms of nicotinamide riboside chloride

#1355
20230061806
2023-03-02

Solid forms of 7-[[(1S)-1-[4-[(1S)-2-cyclopropyl-1-(4-prop-2-enoylpiperazin-1-yl)ethyl]phenyl]ethyl]amino]-1-ethyl-4H-pyrimido[4,5-d][1,3]oxazin-2-one

#1356
20230060905
2023-03-02

IRAK4 INHIBITOR CRYSTAL AND PREPARATION METHOD THEREFOR

#1357
20230058425
2023-02-23

Crystal form of pyridopyrimidine derivative and preparation method thereof

#1358
20230058102
2023-02-23

SOLID STATE FORMS OF BLARCAMESINE SALTS

#1359
20230058001
2023-02-23

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1360
20230057884
2023-02-23

CO-CRYSTALS OF TRAMADOL AND COXIBS

#1361
20230057759
2023-02-23

Solid State Form of Pyroxasulfone

#1362
20230057716
2023-02-23

Crystalline form of (S)-7-(1-acryloylpiperidin-4-yl)-2-(4-phenoxyphenyl)-4,5,6,7-tetra-hydropyrazolo[1,5-a]pyrimidine-3-carboxamide, preparation, and uses thereof

#1363
20230057197
2023-02-23

SOLID STATE FORMS OF MAVACAMTEN AND PROCESS FOR PREPARATION THEREOF

#1364
20230057084
2023-02-23

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#1365
20230056721
2023-02-23

INHALABLE IMATINIB FORMULATIONS, MANUFACTURE, AND USES THEREOF

#1366
20230056365
2023-02-23

Crystalline forms of 2-(3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-1-(cyclopropylsulfonyl)azetidin-3-yl)acetonitrile

#1367
20230056273
2023-02-23

CRYSTALLINE AND LIQUID CRYSTALLINE 25-HYDROXY-CHOLEST-5-EN-3-SULFATE SODIUM AND METHODS FOR PREPARING SAME

#1368
20230055908
2023-02-23

MESYLATE SALT OF PARA-TOPOLIN, COMPOSITIONS CONTAINING SAID SALT AND USE THEREOF

#1369
20230054001
2023-02-23

BILE ACID DERIVATIVE SALT, CRYSTAL STRUCTURE THEREOF, PREPARATION METHOD THEREFOR AND USE THEREOF

#1370
20230052703
2023-02-16

Salt Forms of a Kinase Inhibitor

#1371
20230052523
2023-02-16

SALTS/COCRYSTALS OF (R)-N-(4-CHLOROPHENYL)-2-((1S,4S)-4-(6-FLUOROQUINOLIN-4-YL)CYCLOHEXYL)PROPANAMIDE

#1372
20230051259
2023-02-16

Preparation of Trifarotene and intermediates and polymorphs thereof

#1373
20230050777
2023-02-16

Addition salt of S1P1 receptor agonist and crystal form thereof, and pharmaceutical composition

#1374
20230049311
2023-02-16

METHODS OF TREATING DESMOID TUMORS WITH (S)-2-(((S)-6,8-DIFLUORO-1,2,3,4-TETRAHYDRONAPHTHALEN-2-YL)AMINO)-N-(1-(2-METHYL-1-(NEOPENTYLAMINO)PROPAN-2-YL)-1H-IMIDAZOL-4-YL)PENTANAMIDE

#1375
20230049130
2023-02-16

DEUCRAVACITINIB CRYSTAL FORM, PREPARATION METHOD THEREFOR AND USE THEREOF

#1376
20230048512
2023-02-16

COCRYSTALS OF PTEROSTILBENE AND COMPOSITIONS COMPRISING THEM

#1377
20230046859
2023-02-16

Bicyclic compounds and their uses

#1378
20230046329
2023-02-16

MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE

#1379
20230045991
2023-02-16

SALT FORM AND CRYSTAL FORM OF MUTANT IDH1 INHIBITOR AND PREPARATION METHOD THEREFOR

#1380
20230045419
2023-02-09

Solid Forms of 2-((4-((S)-2-(5-Chloropyridin-2-yl)-2-methylbenzo[d][1,3]dioxol-4-yl)piperidin-1-yl)methyl)-1-(((S)-oxetan-2-yl)methyl)-1H-benzo[d]imidazole-6-carboxylic acid, 1,3-Dihydroxy-2-(hydroxymethyl)propan-2-amine Salt

#1381
20230043305
2023-02-09

Morphic forms of G1T38 and methods of manufacture thereof

#1382
20230042479
2023-02-09

NEW CRYSTALLINE FORMS OF A SUCCINATE SALT OF 7-CYCLOPENTYL-2-(5-PIPERAZIN-1-YL-PYRIDIN-2-YLAMINO)-7H-PYRROLO[2,3-D]PYRIMIDINE -6-CARBOXYLIC ACID DIMETHYLAMIDE

#1383
20230041956
2023-02-09

UTIDELONE SEMI-HYDRATED SINGLE CRYSTAL AND PREPARATION METHOD THEREFOR AND USE THEREOF

#1384
20230041504
2023-02-09

METHOD FOR THE INDUSTRIAL PREPARATION OF THE DISODIUM SALT OF ((2S)-3-([1,1'-BIPHENYL]-4-YL)-2-((HYDROXY((1R)-1-(((1-(ISOBUTYRYLOXY)ETHOXY)CARBONYL)AMINO)ETHYL)PHOSPHORYL) METHYL)PROPANOYL)-L-ALANINE

#1385
20230040262
2023-02-09

STEREOSELECTIVE PROCESS FOR PREPARING SUBSTITUTED POLYCYCLIC PYRIDONE DERIVATIVES

#1386
20230039086
2023-02-09

BMS-986165 CRYSTAL FORM, PREPARATION METHOD THEREFOR AND USE THEREOF

#1387
20230036925
2023-02-02

Solvents, methods, and systems for isolating botanical extracts from plants

#1388
20230036336
2023-02-02

CRYSTALLINE FORMS OF SODIUM SALT OF BEMPEDOIC ACID

#1389
20230035586
2023-02-02

Salts of R-ketorolac

#1390
20230035133
2023-02-02

[1,2,4]Triazolo[4,3-B]Pyridazines For Use in the Treatment of Proliferative Diseases

#1391
20230035012
2023-02-02

CRYSTALS AND PRODUCTION METHOD FOR THE SAME

#1392
20230034132
2023-02-02

Crystal form as inhibitor of ACC1 and ACC2, and preparation method therefor and use thereof

#1393
20230032750
2023-02-02

Processes for converting cannabinoids into cannabinoid derivatives and recovering the same

#1394
20230032547
2023-02-02

Processes and systems for converting cannabinoids into cannabinoid derivatives and isolating the same

#1395
20230032403
2023-02-02

Crystalline solids of mek inhibitor n-((r)-2,3-dihydroxypropoxy)-3,4-difluoro-2-(2-fluoro-4-iodo-phenylamino)-benzamide and uses thereof

#1396
20230031980
2023-02-02

METHODS AND COMPOSITIONS FOR TREATING AND DIAGNOSING A SAGE1-RELATED CONDITION

#1397
20230031944
2023-02-02

Pharmaceutical composition comprising 5-methoxy-n,n-dimethyltryptamine

#1398
20230030720
2023-02-02

CYCLOALKANE-1,3-DIAMINE DERIVATIVE

#1399
20230029213
2023-01-26

Crystalline forms and salt forms of a kinase inhibitor

#1400
20230029094
2023-01-26

Selective Inhibitors Of Protein Arginine Methyltransferase 5 (PRMT5)

#1401
20230029066
2023-01-26

CRYSTAL FORMS OF FUSED RING COMPOUND, AND COMPOSITION THEREOF, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#1402
20230028566
2023-01-26

Crystalline Form of a 7H-Benzo[7]Annulene-2-Carboxylic Acid Derivative

#1403
20230028533
2023-01-26

Crystalline forms of piperazine-1,4-diylbis((6-(1H-benzo[d]imidazo-2-yl)pyridin-2yl)methanone)

#1404
20230027952
2023-01-26

NOVEL SALTS OF INDOLEAMINE 2,3-DIOXYGENASE INHIBITORS

#1405
20230027601
2023-01-26

METHOD FOR MANUFACTURING REVAUDIOSIDE-D-CONTAINING CRYSTALLIZED PRODUCT, AND REVAUDIOSIDE-D-CONTAINING CRYSTALLIZED PRODUCT

#1406
20230027502
2023-01-26

METHODS OF TREATING SMALL CELL LUNG CANCER WITH LURBINECTEDIN FORMULATIONS

#1407
20230026869
2023-01-26

CRYSTAL FORM OF NUCLEOPROTEIN INHIBITOR AND USE THEREOF

#1408
20230026095
2023-01-26

PROCESS FOR THE CONTINUOUS MANUFACTURE OF STATINS

#1409
20230025510
2023-01-26

BIARYL ETHER-TYPE QUINAZOLINE DERIVATIVES

#1410
20230025411
2023-01-26

A METHOD FOR PREPARING IVOSIDENIB AND AN INTERMEDIATE THEREOF

#1411
20230025246
2023-01-26

PROCESS FOR PREPARING CHROMAN COMPOUNDS

#1412
20230023953
2023-01-26

HDAC INHIBITOR SOLID STATE FORMS

#1413
20230023780
2023-01-26

PROCESS FOR PURIFICATION OF MALONIC ACID FROM FERMENTATION BROTH

#1414
20230023131
2023-01-26

AMLODIPINE MESYLATE MONOHYDRATE PREPARATION METHOD THEREFOR AND USE THEREOF

#1415
20230023114
2023-01-26

Crystalline forms of trofinetide

#1416
20230023092
2023-01-26

TREATMENT OF DEPRESSION AND OTHER VARIOUS DISORDERS WITH PSILOCYBIN

#1417
20230022803
2023-01-26

NOVEL CRYSTALLINE FORM OF GPR40 AGONIST

#1418
20230022767
2023-01-26

SALTS OF (2R, 6R)-HYDROXYNORKETAMINE, THEIR CRYSTAL FORMS, AND METHODS OF MAKING THE SAME

#1419
20230022196
2023-01-26

ADDITIVE USED IN METHIONINE PREPARATION PROCESS, AND METHIONINE PREPARATION METHOD

#1420
20230022116
2023-01-26

Crystals and production method for the same

#1421
20230022091
2023-01-26

Compound functioning as bromodomain protein inhibitor, and composition

#1422
20230021909
2023-01-26

Crystalline forms of (S, E)-4-(dimethylamino)-N-(3-(4-(2-hydroxy-1-phenylethylamino)-6-phenylfuro[2,3-d]pyrimidin-5-yl)phenyl)but-2- enamide free base

#1423
20230021395
2023-01-26

Salt of an aminopyridine derivative compound, a crystalline form thereof, and a process for preparing the same

#1424
20230020208
2023-01-19

ORGANIC ACID AND THERMAL TREATMENT OF PURIFIED 2,5-FURANDICARBOXYLIC ACID

#1425
20230020197
2023-01-19

CRYSTAL OF INDOCYANINE COMPOUND

#1426
20230019853
2023-01-19

Melanocortin 4 receptor antagonists and uses thereof

#1427
20230019169
2023-01-19

NOVEL PHTHALOCYANINE NANOWIRES AND USES THEREFOR

#1428
20230017378
2023-01-19

GABAA POSITIVE ALLOSTERIC MODULATOR COMPOUNDS, METHODS OF MAKING, AND USES THEREOF

#1429
20230015251
2023-01-19

Solid forms comprising an oxime ether compound and a coformer, compositions and methods of use thereof

#1430
20230014782
2023-01-19

NEW SOLID STATE FORM OF LURBINECTEDIN

#1431
20230014383
2023-01-19

THREE FUSED RING DERIVATIVE-CONTAINING SALT OR CRYSTAL FORM AND PHARMACEUTICAL COMPOSITION THEREOF

#1432
20230013144
2023-01-19

Indazole inhibitors of the Wnt signal pathway and therapeutic uses thereof

#1433
20230012374
2023-01-12

PROCESS FOR PRODUCING HERBICIDE AND INTERMEDIATE THEREOF

#1434
20230012321
2023-01-12

Methods of manufacturing a bifunctional compound, ultrapure forms of the bifunctional compound, and dosage forms comprising the same

#1435
20230010368
2023-01-12

CRYSTALLINE FORM OF ACETYLCHOLINESTERASE INHIBITOR AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#1436
20230002439
2023-01-05

CRYSTALLINE FORMS OF VAMOROLONE

#1437
20230002426
2023-01-05

CHIRAL SYNTHESIS OF A TERTIARY ALCOHOL

#1438
20230002418
2023-01-05

Crystalline bortezomib process

#1439
20230002400
2023-01-05

AMORPHOUS FORM OF NITROGEN-CONTAINING TRICYCLIC COMPOUND AND USE THEREOF

#1440
20230002399
2023-01-05

LONG-ACTING INJECTABLE FORMULATIONS AND CRYSTALLINE FORMS OF BUPRENORPHINE DERIVATIVES

#1441
20230002338
2023-01-05

WATER AND THERMAL TREATMENT OF PURIFIED 2,5-FURANDICARBOXYLIC ACID

#1442
20230002325
2023-01-05

CRYSTAL FORM OF QUINOLINONE COMPOUND AND USE THEREOF

#1443
20230002319
2023-01-05

POLYMORPHS OF PHENYL PYRROLE AMINOGUANDIUM SALTS

#1444
20230002302
2023-01-05

CO-CRYSTAL OF KETOPROFEN AND ITS PREPARATION, PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME AND USES THEREOF

#1445
20230000883
2023-01-05

METHODS FOR TREATING ANXIETY DISORDERS, HEADACHE DISORDERS, AND EATING DISORDERS WITH PSILOCYBIN

#1446
20220411462
2022-12-29

Methods for producing cyclic compounds comprising N-substituted amino acid residues

#1447
20220411439
2022-12-29

POLYMORPHS OF A MACROCYCLIC KINASE INHIBITOR

#1448
20220411386
2022-12-29

Oxazole compound crystal

#1449
20220411380
2022-12-29

ACID ADDITION SALT OF RORy REGULATOR

#1450
20220411376
2022-12-29

Method for preparing nicotinamide mononucleotide cocrystal

#1451
20220411371
2022-12-29

SOLID STATE FORMS OF LUCERASTAT AND PROCESS FOR PREPARATION THEREOF

#1452
20220411368
2022-12-29

NOVEL SALT OF TERPHENYL COMPOUND

#1453
20220409585
2022-12-29

TREATMENT OF AUTOINFLAMMATORY DISORDERS

#1454
20220409548
2022-12-29

AMORPHOUS SOLID DISPERSION OF PYRAZOLE-AMIDE COMPOUND

#1455
20220402961
2022-12-22

NICOTINAMIDE MONONUCLEOTIDE-ISONICOTINE COCRYSTAL AND COMPOSITION THEREOF

#1456
20220402949
2022-12-22

Preparation of psilocybin, different polymorphic forms, intermediates, formulations and their use

#1457
20220402939
2022-12-22

Crystal form of hepatitis B surface antigen inhibitor and application thereof

#1458
20220402937
2022-12-22

Salts, crystal forms, and production methods thereof

#1459
20220402936
2022-12-22

CRYSTALLINE FORM OF A MULTI-TYROSINE KINASE INHIBITOR, METHOD OF PREPARATION, AND USE THEREOF

#1460
20220402906
2022-12-22

Crystal form of lanifibranor, preparation method therefor, and use thereof

#1461
20220402888
2022-12-22

CO-CRYSTAL AND/OR EUTECTIC CRYSTAL OF KOJIC ACID, COMPOSITIONS COMPRISING THE SAME, PROCESS OF PRODUCING THE SAME, AND USES THEREOF

#1462
20220402886
2022-12-22

Process for preparing pitolisant hydrochloride and solid-state forms thereof

#1463
20220402878
2022-12-22

CRYSTAL OF 3-(DIFLUOROMETHYL)-1-METHYL-N-(1,1,3-TRIMETHYL-2,3-DIHYDRO-1H-INDEN-4-YL)-1H-PYRAZOLE-4-CARBOXAMIDE

#1464
20220402874
2022-12-22

SOLID FORMS OF OMECAMTIV MECARBIL DIHYDROCHLORIDE AND PROCESSES THEREOF

#1465
20220402861
2022-12-22

A Crystalline form of (R)-terbutaline Hydrochloride

#1466
20220401422
2022-12-22

Compounds and compositions for inhibiting the activity of HIF2-alpha and their methods of use

#1467
20220396582
2022-12-15

CRYSTALLINE FORMS OF N-(4-(1-(2,6-DIFLUOROBENZYL)-5-((DIMETHYLAMINO)METHYL)-3-(6-METHOXY-3-PYRIDAZINYL)-2,4-DIOXO-1,2,3,4-TETRAHYDROTHIENO[2,3-D]PYRIMIDIN-6-YL)PHENYL)-N'-METHOXYUREA

#1468
20220396573
2022-12-15

Pyrimidine compound as JAK kinase inhibitor

#1469
20220396561
2022-12-15

Crystal of 1,3,5-triazine derivative or solvate thereof and method for producing same

#1470
20220396552
2022-12-15

Composition comprising a benzoate salt of 5-methoxy-N,N-dimethyltryptamine

#1471
20220396543
2022-12-15

Method for Separating Water-Containing Crystals, Method for Producing Methacrylic Acid, and Method for Producing Methacrylic Acid Ester

#1472
20220396540
2022-12-15

METHODS TO SEPARATE CANNABINOIDS FROM IMPURITIES BY CRYSTALLIZATION

#1473
20220395520
2022-12-15

COMPOSITIONS COMPRISING HMOS, THEIR PRODUCTION AND USE FOR THE PREVENTION AND/OR TREATMENT OF VIRAL AND/OR BACTERIAL INFECTIONS

#1474
20220395490
2022-12-15

TREATMENT OF ARTHRITIS

#1475
20220389056
2022-12-08

Polymorph form of (r)-2-[2-amino-3-(indol-3-yl)propionylamino]-2- methylpropionic acid and uses thereof

#1476
20220389024
2022-12-08

CRYSTALLINE FORM OF NITROGEN-CONTAINING TRICYCLIC COMPOUND AND USE THEREOF

#1477
20220389022
2022-12-08

SOLID FORMS OF PONATINIB HYDROCHLORIDE AND PROCESS THEREOF

#1478
20220389017
2022-12-08

NOVEL PURINE DERIVATIVE, INTERMEDIATE AND APPLICATION THEREOF IN PREPARING ANTICANCER MEDICINE

#1479
20220389011
2022-12-08

Crystalline form of Tolebrutinib

#1480
20220389006
2022-12-08

SALTS AND FORMS OF AN ESTROGEN RECEPTOR MODULATOR

#1481
20220388981
2022-12-08

CRYSTALLINE FORMS OF A BIPHENYL COMPOUND

#1482
20220388974
2022-12-08

Synthetic pathway to belzutifan and crystalline phases of synthetic intermediates

#1483
20220388961
2022-12-08

Process for making amino diaryl ethers and amino diaryl ethers hydrochloride salts

#1484
20220388956
2022-12-08

NEW N,N-DIMETHYLTRYPTAMINE SALTS AND CRYSTALLINE SALT FORMS

#1485
20220388948
2022-12-08

Process for the preparation of a metastable crystal modification of n-(aminoiminomethyl)-2-aminoacetic acid (III)

#1486
20220388937
2022-12-08

Methods of making bempedoic acid and compositions of the same

#1487
20220387404
2022-12-08

TREATMENT OF CANCER USING A COMBINATION COMPRISING MULTI-TYROSINE KINASE INHIBITOR AND IMMUNE CHECKPOINT INHIBITOR

#1488
20220387400
2022-12-08

FORMULATIONS OF RBP4 INHIBITORS AND METHODS OF USE

#1489
20220387323
2022-12-08

Amorphous efinaconazole solid dispersion

#1490
20220380363
2022-12-01

Dominant salt forms of pyrimidine derivatives, and crystal forms thereof

#1491
20220380361
2022-12-01

Material for the treatment of gastro-intestinal disorders

#1492
20220380348
2022-12-01

AXL INHIBITOR FORMULATIONS

#1493
20220380344
2022-12-01

Processes for preparing a diaminopyrimidine derivative or acid addition salt thereof

#1494
20220380336
2022-12-01

Salt types, crystal forms, and preparation methods for benzopyrazole compounds as RHO kinase inhibitors

#1495
20220380316
2022-12-01

SOLID STATE FORMS OF ARRY-797 AND PROCESS FOR PREPARATION THEREOF

#1496
20220380315
2022-12-01

Crystalline forms of plasma kallikrein inhibitors

#1497
20220380308
2022-12-01

Crystalline salts of psilocin

#1498
20220380288
2022-12-01

SOLID STATE FORMS OF FEZAGEPRAS AND PROCESS FOR PREPARATION THEREOF

#1499
20220380284
2022-12-01

SOLID FORMS OF DIMETHOXYPILLAR[5]ARENE (DMP5): HYDROCARBON FUEL UPGRADING AND GAS SORPTION

#1500
20220372059
2022-11-24

Crystalline phases of 5,6-dichloro-2-(isopropylamino)-(1 β-L-ribofuranosyl)-1H-benzimidazole