ClassID:

94386

C07D231/56 - page 2 - CPC Classification

Classification description:

Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems Benzopyrazoles; Hydrogenated benzopyrazoles

Recent Application in this class:
#301
20210008046
2021-01-14

Bicyclic compounds and their use in the treatment of cancer

#302
20200399241
2020-12-24

3-arylindazoles as selective MEK4 inhibitors

#303
20200399219
2020-12-24

Dual acting FKBP12 and FKBP52 inhibitors

#304
20200392127
2020-12-17

Indazole derivatives and pharmaceutical composition for preventing, alleviating or treating cancer containing the same

#305
20200392123
2020-12-17

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

#306
20200383988
2020-12-10

Compounds

#307
20200377487
2020-12-03

SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS

#308
20200377462
2020-12-03

Indazole derivatives useful as glucagon receptor antagonists

#309
20200369647
2020-11-26

Methods and intermediates for preparing therapeutic compounds

#310
20200361941
2020-11-19

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#311
20200347070
2020-11-05

Heterocyclic compound, preparation method and use thereof in medicine

#312
20200347025
2020-11-05

Compounds and compositions for inhibition of FASN

#313
20200339591
2020-10-29

COMPOSITIONS AND METHODS OF TREATMENT FOR NEUROLOGICAL DISORDERS COMPRISING A DEMENTIA

#314
20200339586
2020-10-29

Compounds and their use as inhibitors of N-myristoyl transferase

#315
20200339533
2020-10-29

Heterocyclic compounds, compositions comprising heterocyclic compound, and methods of use thereof

#316
20200339522
2020-10-29

Phenoxymethyl derivatives

#317
20200331872
2020-10-22

Methionine metabolic pathway inhibitors

#318
20200317629
2020-10-08

Benzo-fused heterocyclic derivatives useful as agonists of GPR120

#319
20200317615
2020-10-08

Palladium (II)-catalyzed γC(SP)-H alkynylation of amines

#320
20200308173
2020-10-01

Inhibitors of kinase networks and uses thereof

#321
20200299285
2020-09-24

Carboxylic acid, acyl sulfonamide and acyl sulfamide-derivatized bicyclic aza-heteroaromatics as selective Mcl-1 inhibitors and as dual Mcl-1/Bcl-2 inhibitors

#322
20200299272
2020-09-24

Urea derivatives and uses thereof

#323
20200299226
2020-09-24

Mild and efficient preparation method for α-acyloxyenamide compounds and use thereof in synthesis of amide and polypeptide

#324
20200290964
2020-09-17

Sulfonamide derivatives for protein degradation

#325
20200283438
2020-09-10

Bicyclic compounds and their use in the treatment of cancer

#326
20200277276
2020-09-03

Modulators of the cystic fibrosis transmembrane conductance regulator protein and methods of use

#327
20200277275
2020-09-03

Modulators of the cystic fibrosis transmembrane conductance regulator protein and methods of use

#328
20200277274
2020-09-03

Modulators of the cystic fibrosis transmembrane conductance regulator protein and methods of use

#329
20200277273
2020-09-03

Modulators of the cystic fibrosis transmembrane conductance regulator protein and methods of use

#330
20200270223
2020-08-27

Carbamate compounds and methods of making and using same

#331
20200262832
2020-08-20

URAT1 inhibitor for promoting uric acid excretion

#332
20200262793
2020-08-20

Substituted heterocyclyl derivatives as CDK inhibitors

#333
20200255415
2020-08-13

TETRASUBSTITUTED ALKENE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF BREAST CANCER

#334
20200247794
2020-08-06

PHARMACOPHORES, COMPOUNDS AND METHODS HAVING APPLICATION IN THE TREATMENT OF CANCER THROUGH INHIBITION OF CYP17A1 AND CYP19A1

#335
20200247764
2020-08-06

Pharmacophores, compounds and methods having application in the treatment of cancer through inhibition of CYP17A1 and CYP19A1

#336
20200247762
2020-08-06

K-Ras modulators

#337
20200246315
2020-08-06

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#338
20200231579
2020-07-23

Heterocyclic compound

#339
20200223834
2020-07-16

Gamma-diketones as wnt/β-catenin signaling pathway activators

#340
20200216440
2020-07-09

Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response

#341
20200199076
2020-06-25

Therapeutic indazoles

#342
20200196607
2020-06-25

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#343
20200190038
2020-06-18

Method for producing difluoromethylene compound

#344
20200190031
2020-06-18

ARYL ETHERS AND USES THEREOF

#345
20200172521
2020-06-04

Five-membered-fused-six-membered aza-aromatic ring compound, preparation method thereof, pharmaceutical composition and application thereof

#346
20200172492
2020-06-04

Pharmaceutical compound

#347
20200148638
2020-05-14

Mast-cell modulators and uses thereof

#348
20200123113
2020-04-23

Analogs of fexaramine and methods of making and using

#349
20200087281
2020-03-19

Fused bicyclic compounds, compositions and applications thereof

#350
20200071308
2020-03-05

Benzene, Pyridine, and Pyridazine Derivatives

#351
20200069646
2020-03-05

Inhibitors of indoleamine 2,3-dioxygenase and methods of their use

#352
20200055814
2020-02-20

Anti-fibrotic compounds

#353
20200055813
2020-02-20

C7-FLUORO SUBSTITUTED TETRACYCLINE COMPOUNDS

#354
20200039976
2020-02-06

Compounds and methods for inhibiting fascin

#355
20200039941
2020-02-06

CXCR4 CHEMOKINE RECEPTOR MODULATORS

#356
20200039923
2020-02-06

Heat shock protein 90 inhibitors

#357
20200030299
2020-01-30

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#358
20200030290
2020-01-30

INDAZOLE AND INDOLE DERIVATIVES AS INHIBITORS OF RETINOIC ACID RELATED ORPHAN RECEPTOR GAMMA (ROR GAMMA) FOR THE TREATMENT OF IMMUNE-RELATED DISEASES

#359
20200029566
2020-01-30

Pesticial compounds

#360
20200024286
2020-01-23

FUSED DIHYDRO-4H-PYRAZOLO[5,1-C][1,4]OXAZINYL COMPOUNDS AND ANALOGS FOR TREATING CNS DISORDERS

#361
20200017458
2020-01-16

Compounds and compositions for inhibition of FASN

#362
20200010487
2020-01-09

Heterocyclic amide compounds having RORyT inhibitory action

#363
20190382351
2019-12-19

HDAC INHIBITORS

#364
20190375764
2019-12-12

SALTS OF A HETEROCYCLIC COMPOUND AND CRYSTALLINE FORMS, PROCESSES FOR PREPARING, THERAPEUTIC USES, AND PHARMACEUTICAL COMPOSITIONS THEREOF

#365
20190367460
2019-12-05

Heterocyclic compounds as pesticides

#366
20190367459
2019-12-05

Heterocyclic compounds as pesticides

#367
20190367447
2019-12-05

Hydroxamate triterpenoid derivatives

#368
20190365711
2019-12-05

Compound having anti-cancer effect, and preparation method therefor and use thereof

#369
20190359590
2019-11-28

Method for producing indazole compound, and indazole compound

#370
20190350903
2019-11-21

INDOMETHACIN ANALOGS FOR THE TREATMENT OF CASTRATE-RESISTANT PROSTATE CANCER

#371
20190345161
2019-11-14

Toll-like receptor antagonist compounds and methods of use

#372
20190330239
2019-10-31

Indazole derivatives useful as inhibitors of diacylglyceride O-acyltransferase 2

#373
20190328720
2019-10-31

Inhibitors of dihydroceramide desaturase for treating disease

#374
20190322687
2019-10-24

Modulators of ROR-gamma

#375
20190322662
2019-10-24

Activator of TREK (TWIK RElated K channels) channels

#376
20190315712
2019-10-17

Bicyclic carboxamides and methods of use thereof

#377
20190308945
2019-10-10

Substituted bicyclic heteroaryl allosteric modulators of nicotinic acetylcholine receptors

#378
20190300505
2019-10-03

Methods and intermediates for preparing therapeutic compounds

#379
20190300487
2019-10-03

Compounds and methods for IDO and TDO modulation, and indications therefor

#380
20190300480
2019-10-03

Binding Function 3 (BF3) site compounds as therapeutics and methods for their use

#381
20190292155
2019-09-26

THERAPEUTIC INHIBITORY COMPOUNDS

#382
20190292149
2019-09-26

ARYL SUBSTITUTED INDOLES AND THE USE THEREOF

#383
20190284172
2019-09-19

Urea derivatives and uses thereof

#384
20190284135
2019-09-19

PRIMARY CARBOXAMIDES AS BTK INHIBITORS

#385
20190276438
2019-09-12

Substituted indazole compounds as RORgammaT inhibitors and uses thereof

#386
20190270749
2019-09-05

Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain

#387
20190270731
2019-09-05

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

#388
20190270719
2019-09-05

Deoxyuridine triphosphatase inhibitors

#389
20190270712
2019-09-05

Compositions for the treatment of pulmonary fibrosis

#390
20190263775
2019-08-29

Glucosylceramide synthase inhibitors for the treatment of diseases

#391
20190241546
2019-08-08

SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS

#392
20190241533
2019-08-08

Compounds and compositions for inhibition of FASN

#393
20190241532
2019-08-08

Compounds and compositions for inhibition of FASN

#394
20190225596
2019-07-25

Cannabinergic nitrate esters and related analogs

#395
20190218186
2019-07-18

Indazole derivatives useful as glucagon receptor antagonists

#396
20190210973
2019-07-11

COMPOUNDS AND METHODS FOR TREATMENT OF CYSTIC FIBROSIS

#397
20190210957
2019-07-11

Mild and efficient preparation method for α-acyloxyenamide compounds and use thereof in synthesis of amide and polypeptide

#398
20190209580
2019-07-11

Compounds, compositions, and methods for treatment of diseases involving acidic or hypoxic diseased tissues

#399
20190202819
2019-07-04

Indazole sulfonamide derivatives as inverse agonists of retinoid-related orphan receptor gamma (ROR gamma (T))

#400
20190202811
2019-07-04

Aminoacylindazole immunomodulators for treatment of autoimmune diseases

#401
20190194214
2019-06-27

PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS

#402
20190194124
2019-06-27

Compositions and methods for treating cancer

#403
20190185472
2019-06-20

Fused heterocyclic derivatives, their preparation methods thereof and medical uses thereof

#404
20190167644
2019-06-06

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#405
20190161475
2019-05-30

Method for producing indole compound

#406
20190160060
2019-05-30

Substituted benzaldehyde compounds and methods for their use in increasing tissue oxygenation

#407
20190152937
2019-05-23

Benzo-fused heterocyclic derivatives useful as agonists of GPR120

#408
20190144440
2019-05-16

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#409
20190144387
2019-05-16

Selective androgen receptor degrader (SARD) ligands and methods of use thereof

#410
20190142802
2019-05-16

Benzopyrazole compounds and analogues thereof

#411
20190135718
2019-05-09

SMALL MOLECULE INHIBITORS OF NECROPTOSIS

#412
20190134022
2019-05-09

MODULATORS OF CELLULAR ADHESION

#413
20190119214
2019-04-25

Aryl ethers and uses thereof

#414
20190119212
2019-04-25

Versatile ligand for palladium-catalyzed meta-C—H functionalizations of aromatic substrates

#415
20190119210
2019-04-25

Aromatic sulfonamide derivatives

#416
20190112287
2019-04-18

Compounds and uses thereof for the modulation of hemoglobin

#417
20190112275
2019-04-18

Heterocyclic inhibitors of MCT4

#418
20190112270
2019-04-18

Polymorphic form of N-{6-(hydroxypropan-2-yl)-2-[2-(methylsulphonyl)ethyl]-2H-indazol-5-yl}-6-(trifluoromethyl)pyridine-2-carboxamide

#419
20190106407
2019-04-11

Synthesis of indazoles

#420
20190099453
2019-04-04

Medicament for liver regeneration and for treatment of liver failure

#421
20190091265
2019-03-28

MEDICAMENT FOR LIVER REGENERATION AND FOR TREATMENT OF LIVER FAILURE

#422
20190090488
2019-03-28

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#423
20190084939
2019-03-21

Analogs of fexaramine and methods of making and using

#424
20190077784
2019-03-14

Modulators of the cystic fibrosis transmembrane conductance regulator protein and methods of use

#425
20190076401
2019-03-14

Cyanoindazole compounds and uses thereof

#426
20190071433
2019-03-07

Benzimidazole sulfonamide derivatives as inverse agonists of retinoid-related orphan receptor gamma (ROR gamma (T))

#427
20190070173
2019-03-07

Combinations for the treatment of neuroblastoma

#428
20190062328
2019-02-28

Bruton's tyrosine kinase inhibitors

#429
20190062321
2019-02-28

Histone deacetylase inhibitors and compositions and methods of use thereof

#430
20190055227
2019-02-21

γ-diketones as Wnt/β-catenin signaling pathway activators

#431
20190055196
2019-02-21

NUCLEAR RECEPTOR MODULATORS

#432
20190051835
2019-02-14

Organic electroluminescent element and electronic device

#433
20190040016
2019-02-07

INDOLE AND INDAZOLE COMPOUNDS AND THERAPEUTIC USES THEREOF

#434
20190031685
2019-01-31

HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF

#435
20190016680
2019-01-17

MAST-CELL MODULATORS AND USES THEREOF

#436
20190002472
2019-01-03

Immunoregulatory agents

#437
20190002398
2019-01-03

C7-FLUORO SUBSTITUTED TETRACYCLINE COMPOUNDS

#438
20180370974
2018-12-27

Compounds and their use as inhibitors of N-myristoyl transferase

#439
20180370933
2018-12-27

Compounds and compositions for inhibition of FASN

#440
20180362472
2018-12-20

HDAC inhibitors

#441
20180362471
2018-12-20

Substituted heterocyclyl derivatives as CDK inhibitors

#442
20180362451
2018-12-20

Microbiocidal phenylamidine derivatives

#443
20180354908
2018-12-13

Pharmaceutical compound

#444
20180346441
2018-12-06

Substituted benzamides useful as sodium channel blockers

#445
20180346416
2018-12-06

N-SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF

#446
20180334414
2018-11-22

Asymmetric addition reactions

#447
20180327390
2018-11-15

Urea derivatives and uses thereof

#448
20180327389
2018-11-15

Urea derivatives and uses thereof

#449
20180319741
2018-11-08

Sulfonylaminobenzamide compounds as anthelmintics

#450
20180312489
2018-11-01

Substituted indazole compounds as RORgammaT inhibitors and uses thereof

#451
20180305320
2018-10-25

Substituted bicyclic pyrazole compounds as RORgammaT inhibitors and uses thereof

#452
20180297948
2018-10-18

Sodium channel blockers

#453
20180290982
2018-10-11

ARGININE METHYLTRANSFERASE INHIBITORS AND USES THEREOF

#454
20180289672
2018-10-11

Substituted indazole derivatives active as kinase inhibitiors

#455
20180282306
2018-10-04

Kinase inhibitors and method of treating cancer

#456
20180282281
2018-10-04

IMMUNOREGULATORY AGENTS

#457
20180271835
2018-09-27

Indomethacin analogs for the treatment of castrate-resistant prostate cancer

#458
20180265500
2018-09-20

Tetrahydroquinoline sulfonamide derivatives as inverse agonists of retinoid-related orphan receptor gamma (ROR gamma (t))

#459
20180265476
2018-09-20

Condensed ring derivative, and preparation method, intermediate, pharmaceutical composition and use thereof

#460
20180251426
2018-09-06

APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES

#461
20180244627
2018-08-30

Heterocyclic compounds and uses thereof

#462
20180244626
2018-08-30

Aminoindazole derivatives as sodium channel inhibitors

#463
20180244606
2018-08-30

Farnesoid X receptor agonists and uses thereof

#464
20180237450
2018-08-23

Pyrazolo fused heterocyclic compounds as ERK inhibitors

#465
20180230102
2018-08-16

Carboxy substituted (hetero) aromatic ring derivatives and preparation method and uses thereof

#466
20180222919
2018-08-09

N-alkyl-2-phenoxyethanamines, their preparation and use

#467
20180222868
2018-08-09

Indazole Derivatives as Modulators of TNF Activity

#468
20180215757
2018-08-02

Compounds and methods for inhibiting fascin

#469
20180215745
2018-08-02

Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof

#470
20180215716
2018-08-02

Aromatic compound production method

#471
20180208591
2018-07-26

SUBSTITUTED 6,5-FUSED BICYCLIC HETEROARYL COMPOUNDS

#472
20180208568
2018-07-26

CARBAMATE COMPOUNDS AND METHODS OF MAKING AND USING SAME

#473
20180201588
2018-07-19

Phenoxymethyl derivatives

#474
20180201580
2018-07-19

Compounds for treatment of immune inflammatory disorders

#475
20180194767
2018-07-12

5-aromatic alkynyl substituted benzamide compound and preparation method, pharmaceutical composition, and use thereof

#476
20180162822
2018-06-14

Heterocyclic inhibitors of MCT4

#477
20180162807
2018-06-14

Aromatic compounds and uses thereof

#478
20180155359
2018-06-07

SHIP1 MODULATORS AND METHODS RELATED THERETO

#479
20180155319
2018-06-07

Deoxyuridine triphosphatase inhibitors

#480
20180155295
2018-06-07

CXCR4 chemokine receptor modulators

#481
20180155293
2018-06-07

Substituted Heterocyclyl Derivatives as CDK Inhibitors

#482
20180155279
2018-06-07

Aryl ethers and uses thereof

#483
20180153873
2018-06-07

Indazole inhibitors of the WNT signal pathway and therapeutic uses thereof

#484
20180148433
2018-05-31

Pyrazolyl-substituted heteroaryls and their use as medicaments

#485
20180141927
2018-05-24

INHIBITORS OF KRAS G12C MUTANT PROTEINS

#486
20180141913
2018-05-24

TETRASUBSTITUTED ALKENE COMPOUNDS AND THEIR USE

#487
20180127411
2018-05-10

Indazole and azaindazole Btk inhibitors

#488
20180127378
2018-05-10

Tetrasubstituted alkene compounds and their use

#489
20180127377
2018-05-10

5-substituted indazole-3-carboxamides and preparation and use thereof

#490
20180118691
2018-05-03

Heterocyclic derivatives modulating activity of certain protein kinases

#491
20180117040
2018-05-03

Substituted benzaldehyde compounds and methods for their use in increasing tissue oxygenation

#492
20180105497
2018-04-19

ARGININE METHYLTRANSFERASE INHIBITORS AND USES THEREOF

#493
20180099939
2018-04-12

Compounds and methods for IDO and TDO modulation, and indications therefor

#494
20180086716
2018-03-29

Substituted indazoles for treating tendon and/or ligament injuries

#495
20180086697
2018-03-29

Inhibitors of human immunodeficiency virus replication

#496
20180079709
2018-03-22

(Hetero)aryl cyclopropylamine compounds as LSD1 inhibitors

#497
20180078530
2018-03-22

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#498
20180072678
2018-03-15

Condensed ring derivative, and preparation method, intermediate, pharmaceutical composition and use thereof

#499
20180072656
2018-03-15

Sodium channel modulators

#500
20180065955
2018-03-08

Indazole derivatives useful as glucagon receptor antagonists

#501
20180065934
2018-03-08

Indazole derivatives useful as glucagon receptor antagonists

#502
20180050997
2018-02-22

Compounds and compositions for inhibition of FASN

#503
20180030040
2018-02-01

Selective HDAC1 and HDAC2 inhibitors

#504
20180030039
2018-02-01

Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

#505
20180022746
2018-01-25

Indazole and azaindazole substituted compounds as mGluR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction

#506
20180022701
2018-01-25

4-heteroaryl substituted benzoic acid compounds as RORgammaT inhibitors and uses thereof

#507
20180022699
2018-01-25

Aryl substituted indoles and the use thereof

#508
20180016239
2018-01-18

Substituted pyrazole compounds as RORgammaT inhibitors and uses thereof

#509
20180007911
2018-01-11

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#510
20180007907
2018-01-11

Pesticidally active semi-carbazones and thiosemicarbazones derivatives

#511
20180002322
2018-01-04

Bicyclic compound

#512
20180000087
2018-01-04

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#513
20170369428
2017-12-28

Selective histone deactylase 6 inhibitors

#514
20170362250
2017-12-21

SHIP1 modulators and methods related thereto

#515
20170349594
2017-12-07

Biaryl derivative as GPR120 agonist

#516
20170342062
2017-11-30

Indazole sulfonamide derivatives as inverse agonists of retinoid-related orphan receptor gamma (ROR γ (T))

#517
20170342047
2017-11-30

Cancerous cell growth inhibiting compounds

#518
20170340610
2017-11-30

RORgammaT inhibitors

#519
20170340609
2017-11-30

Antimicrobial agents and the method of synthesizing the antimicrobial agents

#520
20170339961
2017-11-30

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#521
20170334948
2017-11-23

LIGANDS FOR ANTIBODY AND FC-FUSION PROTEIN PURIFICATION BY AFFINITY CHROMOTOGRAPHY IV

#522
20170327482
2017-11-16

Compositions and methods for the treatment of mucositis

#523
20170313713
2017-11-02

Aminoindane-, aminotetrahydronaphthalene- and aminobenzocyclobutane-derived PRMT5-inhibitors

#524
20170305915
2017-10-26

Indazole and indole derivatives as inhibitors of retinoic acid related orphan receptor gamma (ROR gamma) for the treatment of immune-related diseases

#525
20170305900
2017-10-26

Histone deacetylase inhibitors and compositions and methods of use thereof

#526
20170305864
2017-10-26

Heterocyclic compounds as pesticides

#527
20170305824
2017-10-26

SMALL MOLECULE INHIBITORS OF NECROPTOSIS

#528
20170298080
2017-10-19

Amino sulfonyl-based compounds, the preparation method therefor and use thereof

#529
20170281621
2017-10-05

Substituted pyridazines as skeletal muscle modulators

#530
20170275301
2017-09-28

Benzenesulfonyl-asymmetric ureas and medical uses thereof

#531
20170275291
2017-09-28

Indazole compounds as FGFR kinase inhibitor, preparation and use thereof

#532
20170275244
2017-09-28

C7-Fluoro Substituted Tetracycline Compounds

#533
20170260176
2017-09-14

γ-diketones as Wnt/β-catenin signaling pathway activators

#534
20170260174
2017-09-14

Benzene, Pyridine, and Pyridazine Derivatives

#535
20170253607
2017-09-07

LONG-ACTING HIV PROTEASE INHIBITOR

#536
20170247389
2017-08-31

SHIP1 MODULATORS AND METHODS RELATED THERETO

#537
20170226053
2017-08-10

Sulfonylaminobenzamide compounds as anthelmintics

#538
20170217910
2017-08-03

INGENOL-3-ACYLATES III AND INGENOL-3-CARBAMATES

#539
20170217882
2017-08-03

Antivirals against molluscum contagiosum virus

#540
20170210728
2017-07-27

Cannabinergic nitrate esters and related analogs

#541
20170204094
2017-07-20

Selective HDAC3 inhibitors

#542
20170197973
2017-07-13

Immunoregulatory agents

#543
20170190714
2017-07-06

Pyrazolo-quinazoline derivatives, process for their preparation and their use as kinase inhibitors

#544
20170190659
2017-07-06

Benzenesulfonamido and related compounds for use as agonists of RORγ and the treatment of disease

#545
20170183313
2017-06-29

BICYCLIC HETEROCYCLES CAPABLE OF MODULATING T-CELL RESPONSES, AND METHODS OF USING SAME

#546
20170166526
2017-06-15

Selective androgen receptor degrader (SARD) ligands and methods of use thereof

#547
20170158702
2017-06-08

MULTIVALENT RAS BINDING COMPOUNDS

#548
20170158692
2017-06-08

Compounds and methods for inhibiting fascin

#549
20170158677
2017-06-08

Substituted indazole derivatives active as kinase inhibitors

#550
20170158642
2017-06-08

Composition for inducing cell reprogramming

#551
20170152288
2017-06-01

LIGANDS FOR ANTIBODY AND Fc-FUSION PROTEIN PURIFICATION BY AFFINITY CHROMATOGRAPHY

#552
20170152230
2017-06-01

Compounds for selective histone deacetylase inhibitors, and pharmaceutical composition comprising the same

#553
20170152228
2017-06-01

Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods

#554
20170137423
2017-05-18

Compounds acting at multiple prostaglandin receptors giving a general anti-inflammatory response

#555
20170101402
2017-04-13

Histone deacetylase inhibitors and compositions and methods of use thereof

#556
20170101380
2017-04-13

Process for the preparation of (E)-3-(4-((E)-2-(2-chloro-4-fluorophenyl)-1-(1H-indazol-5-yl)but-1-en-1-yl)phenyl)acrylic acid

#557
20170096416
2017-04-06

Pyrazole-substituted arylamides as P2Xand P2Xantagonists

#558
20170096400
2017-04-06

Alkynyl indazole derivative and use thereof

#559
20170088549
2017-03-30

ANTIBACTERIAL AGENTS

#560
20170088531
2017-03-30

Benzo-fused heterocyclic derivatives useful as agonists of GPR120

#561
20170081315
2017-03-23

Phenyl and benzodioxinyl substituted indazoles derivatives

#562
20170073333
2017-03-16

Pyrazolyl-substituted heteroaryls and their use as medicaments

#563
20170073320
2017-03-16

Carbamate compounds and methods of making and using same

#564
20170066724
2017-03-09

Analogs of fexaramine and methods of making and using

#565
20170066723
2017-03-09

Naphthylamide compound, preparation method and use thereof

#566
20170065582
2017-03-09

Combinations for the treatment of neuroblastoma

#567
20170065574
2017-03-09

Indazole inhibitors of the Wnt signal pathway and therapeutic uses thereof

#568
20170057956
2017-03-02

Histone deacetylase inhibitors

#569
20170057925
2017-03-02

Indazole derivatives useful as CB-1 inverse agonists

#570
20170049760
2017-02-23

Inhibitors of Rho associated protein kinases (ROCK) and methods of use

#571
20170044158
2017-02-16

Difluoromethylene compound

#572
20170044144
2017-02-16

Selective HDAC1 and HDAC2 inhibitors

#573
20170037044
2017-02-09

Amide derivatives and pharmaceutically acceptable salts thereof, preparation method thereof and medicinal application thereof

#574
20170036969
2017-02-09

NITRIFICATION INHIBITORS

#575
20170029411
2017-02-02

Antibacterial 1-indazole and 1-indole derivatives

#576
20170029372
2017-02-02

Binding function (BF) site compounds as therapeutics and methods for their use

#577
20170029370
2017-02-02

Selective androgen receptor degrader (SARD) ligands and methods of use thereof

#578
20170022198
2017-01-26

Substituted fused heterocycles as GPR119 modulators for the treatment of diabetes, obesity, dyslipidemia and related disorders

#579
20160376240
2016-12-29

6 Phenyl or 6 Pyridin 3 YL Indazole Derivatives and Methods of Use

#580
20160368881
2016-12-22

Therapeutic compounds

#581
20160368857
2016-12-22

(Hetero)aryl cyclopropylamine compounds as LSD1 inhibitors

#582
20160362370
2016-12-15

Nuclear receptor modulators

#583
20160355521
2016-12-08

Bicyclic urea, thiourea, guanidine and cyanoguanidine compounds useful for the treatment of pain

#584
20160355517
2016-12-08

Bicyclic heteroaryl urea, thiourea, guanidine and cyanoguanidine compounds as TrkA kinase inhibitors

#585
20160355511
2016-12-08

NOVEL 1-SUBSTITUTED INDAZOLE DERIVATIVE

#586
20160347717
2016-12-01

Tetrasubstituted alkene compounds and their use

#587
20160347716
2016-12-01

Water-soluble pyrazole derivatives as corrosion inhibitors

#588
20160347708
2016-12-01

Antibacterial agents: Nα-aroyl-N-aryl-phenylalaninamides

#589
20160326170
2016-11-10

Substituted 6,5-fused bicyclic heteroaryl compounds

#590
20160326163
2016-11-10

Bicyclic heteroaryl indole analogues useful as ROR gamma modulators

#591
20160326111
2016-11-10

ARYL SUBSTITUTED INDOLES AND THE USE THEREOF

#592
20160326104
2016-11-10

Cyclohexyl sulfone RORγ modulators

#593
20160318857
2016-11-03

N,N′-diarylurea compounds and N,N′-diarylthiourea compounds as inhibitors of translation initiation

#594
20160317496
2016-11-03

Methods of treating cancer and other disorders

#595
20160311776
2016-10-27

Substituted indazole derivatives active as kinase inhibitiors

#596
20160310465
2016-10-27

Substituted indazole derivatives active as kinase inhibitiors

#597
20160304522
2016-10-20

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#598
20160303082
2016-10-20

Indomethacin analogs for the treatment of castrate-resistant prostate cancer

#599
20160302418
2016-10-20

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#600
20160302417
2016-10-20

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto