ClassID:

94386

C07D231/56 - CPC Classification

Classification description:

Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems Benzopyrazoles; Hydrogenated benzopyrazoles

Recent Application in this class:
#1
20260132130
2026-05-14

INHIBITORS OF NLRP3 INFLAMMASOME

#2
20260125359
2026-05-07

HETEROARYL COMPOUNDS AS MULTI-TARGET PROTEIN KINASE INHIBITORS

#3
20260109665
2026-04-23

C7-FLUORO SUBSTITUTED TETRACYCLINE COMPOUNDS

#4
20260085062
2026-03-26

NOVEL COMPOUNDS AS CK2 INHIBITORS

#5
20260078130
2026-03-19

NAMPT MODULATORS, PREPARATIONS, AND USES THEREOF

#6
20260070902
2026-03-12

SULFONYL DERIVATIVES AS CCR6 INHIBITORS

#7
20260062387
2026-03-05

SALT-INDUCIBLE KINASE INHIBITOR COMPOUND AND PHARMACEUTICAL COMPOSITION INCLUDING THE SAME

#8
20260055063
2026-02-26

COMPOUND CONTAINING BENZENE RING AND APPLICATION THEREOF

#9
20260055062
2026-02-26

HETEROCYCLIC INHIBITORS OF MCT4

#10
20260042753
2026-02-12

INDAZOLYL-ISOXAZOLE DERIVATIVES FOR THE TREATMENT OF DISEASES SUCH AS CANCER

#11
20260015328
2026-01-15

ATM KINASE INHIBITORS

#12
20260015316
2026-01-15

COMPOSITIONS AND METHODS FOR TREATING CANCER

#13
20260008783
2026-01-08

MODULATORS OF FSHR AND USES THEREOF

#14
20250376461
2025-12-11

INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS

#15
20250374822
2025-12-04

AMBIPOLAR MOLECULE, PREPARATION METHOD THEREOF, AND APPLICATION THEREOF

#16
20250359552
2025-11-27

MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO

#17
20250353829
2025-11-20

BICYCLIC CARBOXAMIDES AND METHODS OF USE THEREOF

#18
20250353818
2025-11-20

Compounds

#19
20250333411
2025-10-30

COMPOUNDS AND METHODS FOR INHIBITING FASCIN

#20
20250332156
2025-10-30

PHARMACEUTICAL COMPOSITIONS COMPRISING WRN HELICASE INHIBITORS

#21
20250326757
2025-10-23

SOLID FORMS OF HETEROCYCLYLAMIDES AS IRAK4 INHIBITORS

#22
20250320213
2025-10-16

Nitrogen-Containing Heterocyclic Compounds

#23
20250320186
2025-10-16

HSD17B13 INHIBITORS AND USES THEREOF

#24
20250320184
2025-10-16

SARM1 MODULATORS, PREPARATIONS, AND USES THEREOF

#25
20250304581
2025-10-02

INHIBITORS OF NLRP3 INFLAMMASOME

#26
20250304528
2025-10-02

OLIGO-BENZAMIDE ANALOGS AND THEIR USE IN CANCER TREATMENT

#27
20250296915
2025-09-25

NOVEL AMINO ACID DERIVATIVES

#28
20250296909
2025-09-25

NOVEL BENZENE DERIVATIVE AND IMMUNOSUPPRESSION-RELATED USE THEREOF

#29
20250289815
2025-09-18

MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS AND METHODS

#30
20250289781
2025-09-18

TRIFLUOROMETHANESULFONYLATING AGENT COMPOSITION AND METHOD FOR PRODUCING TRIFLUOROMETHANESULFONYLOXY COMPOUND OR TRIFLUOROMETHANESULFONYL COMPOUND

#31
20250282753
2025-09-11

COMPOUNDS USEFUL FOR REDUCING URIC ACID

#32
20250282735
2025-09-11

BICYCLE COMPOUNDS AS TEAD INHIBITOR

#33
20250276955
2025-09-04

CORONAVIRUS MAIN PROTEASE INHIBITORS AND METHODS USING SAME

#34
20250268868
2025-08-28

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#35
20250250237
2025-08-07

ALKYLAMINE OR HETEROALKYLAMINE DERIVATIVES AS INHIBITORS OF NITRIC OXIDE SYNTHASES (NOS), PHARMACEUTICAL PRODUCTS THEREOF, AND METHODS THEREOF

#36
20250232847
2025-07-17

WORKFLOW FOR GENERATING COMPOUNDS WITH BIOLOGICAL ACTIVITY AGAINST A SPECIFIC BIOLOGICAL TARGET

#37
20250223264
2025-07-10

ESTROGEN RECEPTOR BETA LIGANDS FOR THE PREVENTION AND TREATMENT OF MULTIPLE SCLEROSIS (MS) AND OTHER DEMYELINATING, INFLAMMATORY AND NEURODEGENERATIVE DISEASES

#38
20250214971
2025-07-03

QUATERNARY INDAZOLE GLUCOCORTICOID RECEPTOR ANTAGONISTS

#39
20250214943
2025-07-03

Compounds

#40
20250214942
2025-07-03

INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATMENT OF DISEASE

#41
20250214930
2025-07-03

TETRALIN AND TETRAHYDROQUINOLINE COMPOUNDS AS INHIBITORS OF HIF-2ALPHA

#42
20250206724
2025-06-26

SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS

#43
20250197369
2025-06-19

NOVEL HETEROCYCLIC INHIBITOR FOR HISTONE DEACETYLASE, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME

#44
20250186391
2025-06-12

ORAL COMPLEMENT FACTOR D INHIBITORS

#45
20250179028
2025-06-05

ACRYLAMIDE COMPOUNDS

#46
20250179017
2025-06-05

CARBOXAMIDE COMPOUNDS AS PGE2 RECEPTOR ANTAGONISTS

#47
20250163189
2025-05-22

RAFT AGENT FOR PHOTO-CONTROLLED POLYMERIZATION, PREPARATION METHOD THEREFOR, AND APPLICATIONS THEREOF

#48
20250163044
2025-05-22

COMPOUNDS

#49
20250134105
2025-05-01

MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO

#50
20250122194
2025-04-17

NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS

#51
20250122188
2025-04-17

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#52
20250115598
2025-04-10

BIFUNCTIONAL ARYLSULPHONAMIDE COMPOUNDS

#53
20250115569
2025-04-10

SULFONAMIDE COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL CONDITIONS

#54
20250100999
2025-03-27

METHODS AND INTERMEDIATES FOR PREPARING THERAPEUTIC COMPOUNDS

#55
20250092014
2025-03-20

COMPOUNDS AND METHODS OF ACTIVATING LIPOPROTEIN LIPASE

#56
20250074881
2025-03-06

THERAPEUTIC COMPOUNDS AND METHODS OF USE

#57
20250066389
2025-02-27

HETEROCYCLIC AMIDES AND METHODS OF USING THE SAME

#58
20250059172
2025-02-20

INDAZOLE COMPOUND AND PHARMACEUTICAL

#59
20250042843
2025-02-06

C7-FLUORO SUBSTITUTED TETRACYCLINE COMPOUNDS

#60
20250025443
2025-01-23

COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES

#61
20250011333
2025-01-09

PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS

#62
20250009742
2025-01-09

NOVEL CAPSID ASSEMBLY INHIBITORS

#63
20250008960
2025-01-09

MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO

#64
20240425450
2024-12-26

SMALL MOLECULE INHIBITORS OF BACTERIAL TOXINS

#65
20240409504
2024-12-12

COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER

#66
20240383870
2024-11-21

HETEROCYCLIC ALDEHYDE TRAPPING COMPOUNDS AND USES THEREOF

#67
20240360125
2024-10-31

2-SUBSTITUTED BICYCLO[1.1.1]PENTANES

#68
20240336572
2024-10-10

SUBSTITUTED INDAZOLE PROPIONIC ACID DERIVATIVE COMPOUNDS AND USES THEREOF

#69
20240327334
2024-10-03

Covalent Inhibitors As Antiviral Agents

#70
20240316010
2024-09-26

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#71
20240307409
2024-09-19

ARGININE METHYLTRANSFERASE INHIBITOR AND USE THEREOF

#72
20240306490
2024-09-12

ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE

#73
20240287058
2024-08-29

PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF

#74
20240287003
2024-08-29

ETHACRYNIC ACID DERIVATIVES AS INHIBITORS OF MPRO PROTEASE AND SARS-COV-2 REPLICATION

#75
20240270701
2024-08-15

BETA ADRENERGIC AGONIST AND METHODS OF USING THE SAME

#76
20240262808
2024-08-08

XANTHINE OXIDASE INHIBITOR

#77
20240254089
2024-08-01

MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X4 AND RELATED PRODUCTS AND METHODS

#78
20240254079
2024-08-01

Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2alpha

#79
20240246903
2024-07-25

INDANONE AND TETRALONEKETO OR HYDROXYL OXIMES AS CANCEL THERAPEUTICS

#80
20240246901
2024-07-25

GPX4 INHIBITORS, PHARMACEUTICAL COMPOSITIONS THEREOF, AND THEIR USE FOR TREATING GPX4-MEDIATED DISEASES

#81
20240239752
2024-07-18

BICYCLIC HETEROAROMATIC INHIBITORS OF KLK5

#82
20240228461
2024-07-11

NOVEL METHOD FOR PREPARING SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST

#83
20240228441
2024-07-11

METHOD FOR PREPARING INTERMEDIATE FOR SYNTHESIS OF SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST

#84
20240217935
2024-07-04

METHOD FOR PREPARING INTERMEDIATE FOR SYNTHESIS OF SPHINGOSINE-1-PHOSPHATE RECEPTOR AGONIST

#85
20240208971
2024-06-27

INHIBITORS OF KINASE NETWORKS AND USES THEREOF

#86
20240199554
2024-06-20

Inhibitors of receptor interacting protein kinase I for the treatment of disease

#87
20240190827
2024-06-13

Inhibitors of Rho Associated Coiled-Coil Containing Protein Kinase

#88
20240182478
2024-06-06

TOLL-LIKE RECEPTOR ANTAGONIST COMPOUNDS AND METHODS OF USE

#89
20240174611
2024-05-30

SUBSTITUTED CYCLIC MODULATORS OF PROTEIN PHOSPHATASE 2A (PP2A) AND METHODS USING SAME

#90
20240166652
2024-05-23

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#91
20240166612
2024-05-23

ARYLTHIOETHER ACETAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS

#92
20240166608
2024-05-23

TEAD inhibitors and methods of uses thereof

#93
20240166596
2024-05-23

SULFAMOYL BENZENE DERIVATIVES AND USES THEREOF

#94
20240158355
2024-05-16

BET SUBFAMILY INHIBITORS AND METHODS USING SAME

#95
20240150353
2024-05-09

2-SUBSTITUTED BICYCLO[1.1.1]PENTANES

#96
20240150334
2024-05-09

HSD17B13 INHIBITORS AND/OR DEGRADERS

#97
20240150320
2024-05-09

Quaternary indazole glucocorticoid receptor antagonists

#98
20240150316
2024-05-09

Bicyclic carboxamides and methods of use thereof

#99
20240140940
2024-05-02

CARBOXYLIC ACID, ACYL SULFONAMIDE AND ACYL SULFAMIDE-DERIVATIZED BICYCLIC AZA-HETEROAROMATICS AS SELECTIVE MCL-1 INHIBITORS AND AS DUAL MCL-1/BCL-2 INHIBITORS

#100
20240132480
2024-04-25

INHIBITORS OF MYCOBACTERIUM TUBERCULOSIS LIPOAMIDE DEHYDROGENASE

#101
20240124466
2024-04-18

COMPOUNDS AND USE THEREOF FOR TREATMENT OF NEURODEGENERATIVE, DEGENERATIVE AND METABOLIC DISORDERS

#102
20240124449
2024-04-18

Compounds and methods for inhibiting fascin

#103
20240116933
2024-04-11

INDAZOLE AND PYRAZOLOPYRIDINE COMPOUNDS AS INHIBITORS OF NLRP3 INFLAMMASOME

#104
20240116875
2024-04-11

RATIONAL DESIGN, OPTIMIZATION, AND BIOLOGICAL EVALUATION OF NOVEL MEK4 INHIBITORS AGAINST PANCREATIC ADENOCARCINOMA

#105
20240109847
2024-04-04

HISTONE DEACETYLASE INHIBITORS

#106
20240101533
2024-03-28

Methods and intermediates for preparing therapeutic compounds

#107
20240083903
2024-03-14

ARYL ETHER COMPOUNDS AS TEAD MODULATORS

#108
20240083853
2024-03-14

HSD17B13 INHIBITORS AND USES THEREOF

#109
20240083847
2024-03-14

SULFONAMIDE DERIVATIVES FOR PROTEIN DEGRADATION

#110
20240081145
2024-03-07

Development of material for hole blocking layer with high efficiency and long lifespan, and organic light-emitting device and electronic apparatus utilizing the same

#111
20240067614
2024-02-29

NOVEL COMPOUNDS

#112
20240067610
2024-02-29

Inhibitors of NLRP3 inflammasome

#113
20240059700
2024-02-22

NOVEL DIACYLGLYCERIDE O-ACYLTRANSFERASE 2 INHIBITORS

#114
20240059659
2024-02-22

INHIBITORS OF NLRP3 INFLAMMASOME

#115
20240051923
2024-02-15

INHIBITORS OF NLRP3 INFLAMMASOME

#116
20240043384
2024-02-08

INHIBITORS OF PU.1 FOR THE TREATMENT OF DISEASE

#117
20240034736
2024-02-01

HSD17B13 INHIBITORS AND USES THEREOF

#118
20240034719
2024-02-01

IMIDAZOQUINOLINE OR BENZOINDAZOLONE COMPOUND AND INTERMEDIATE FOR PREPARING SAME

#119
20240025859
2024-01-25

Processes of making 2-((1-benzyl-1H-indazol-3-yl)methoxy)-2-methylpropanoic acid and its derivatives

#120
20240018102
2024-01-18

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH LPA RECEPTOR ACTIVITY

#121
20230399329
2023-12-14

HETEROCYCLIC COMPOUND, ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME, AND COMPOSITION FOR FORMING ORGANIC LAYER

#122
20230391779
2023-12-07

BICYCLIC COMPOUNDS, COMPOSITIONS AND USE THEREOF

#123
20230382871
2023-11-30

CSF1R KINASE INHIBITOR AND USE THEREOF

#124
20230373974
2023-11-23

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR

#125
20230365507
2023-11-16

INHIBITORS OF NLRP3 INFLAMMASOME

#126
20230357161
2023-11-09

Estrogen receptor beta ligands for the prevention and treatment of multiple sclerosis (MS) and other demyelinating, inflammatory and neurodegenerative diseases

#127
20230357139
2023-11-09

SMALL MOLECULE INHIBITORS OF BACTERIAL TOXINS

#128
20230348369
2023-11-02

NAMPT MODULATORS

#129
20230339863
2023-10-26

INDAZOLE DERIVATIVES AS CANNABINOID RECEPTOR PARTIAL AGONISTS

#130
20230331657
2023-10-19

NANOMATERIALS COMPRISING ESTER-LINKED ACETALS

#131
20230322704
2023-10-12

COMPOUNDS AND USES THEREOF FOR THE MODULATION OF HEMOGLOBIN

#132
20230322683
2023-10-12

HETEROCYCLIC COMPOUND

#133
20230321051
2023-10-12

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#134
20230312499
2023-10-05

Carbamate compounds and methods of making and using same

#135
20230312466
2023-10-05

NOVEL COMPOUNDS

#136
20230303567
2023-09-28

Modulators of mas-related G-protein receptor X2 and related products and methods

#137
20230286913
2023-09-14

INHIBITORS OF NITRIC OXIDE SYNTHASES (NOS), PHARMACEUTICAL PRODUCTS THEREOF, AND METHODS THEREOF

#138
20230279010
2023-09-07

PROCESSES FOR PREPARING MODULATORS OF ALPHA-1 ANTITRYPSIN

#139
20230271931
2023-08-31

Carboxylic acid aromatic amides as antagonists of bradykinin B1 receptor

#140
20230255963
2023-08-17

SUBSTITUTED BENZALDEHYDE COMPOUNDS AND METHODS FOR THEIR USE IN INCREASING TISSUE OXYGENATION

#141
20230250086
2023-08-10

METHIONINE METABOLIC PATHWAY INHIBITORS

#142
20230250064
2023-08-10

PREPARATION METHOD FOR FUSED PYRAZOLE-TYPE COMPOUND

#143
20230250062
2023-08-10

Substituted Heterocyclyl Derivatives as CDK Inhibitors

#144
20230242572
2023-08-03

a-CARBONYL ALKENYL ESTER PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#145
20230242529
2023-08-03

Heterocyclic compound

#146
20230242496
2023-08-03

SOX11 INHIBITORS FOR TREATING MANTLE CELL LYMPHOMA

#147
20230219953
2023-07-13

SULFONE DERIVATIVES

#148
20230218578
2023-07-13

BENZOPYRAZOLE COMPOUNDS AND ANALOGUES THEREOF

#149
20230210847
2023-07-06

Substituted Alkynylene Compounds As Anticancer Agents

#150
20230202985
2023-06-29

Indoles, Indazoles, and Related Analogs for Inhibiting YAP/TAZ-TEAD

#151
20230202984
2023-06-29

Pyrazolo compounds and methods of use thereof

#152
20230192623
2023-06-22

Indazole Derivatives

#153
20230183182
2023-06-15

COMPOUND CONTAINING BENZENE RING AND APPLICATION THEREOF

#154
20230180761
2023-06-15

Molecules having pesticidal utility, and intermediates, compositions, and processes, related thereto

#155
20230174470
2023-06-08

COMPOUND AS A UBR BOX DOMAIN LIGAND

#156
20230174465
2023-06-08

COMPOUND AS A UBR BOX DOMAIN LIGAND

#157
20230174460
2023-06-08

AFMT ANALOGS AND THEIR USE IN METHODS OF TREATING PARKINSON'S DISEASE

#158
20230167068
2023-06-01

BENZOPYRAZOLE COMPOUND

#159
20230159466
2023-05-25

Inhibitors of HIF-2α and methods of use thereof

#160
20230159446
2023-05-25

Methods and Compositions for Targeting Tregs using CCR8 Inhibitors

#161
20230150929
2023-05-18

SELECTIVE NON-CYCLIC NUCLEOTIDE ACTIVATORS FOR THE CAMP SENSOR EPAC1

#162
20230122651
2023-04-20

C7-FLUORO SUBSTITUTED TETRACYCLINE COMPOUNDS

#163
20230121086
2023-04-20

RORgT INHIBITOR, PREPARATION METHOD THEREOF AND USE THEREOF

#164
20230117065
2023-04-20

LIGHT EMITTING ELEMENT

#165
20230113085
2023-04-13

Small molecule inhibitors of TEAD transcription factors

#166
20230102879
2023-03-30

TRNA SYNTHETASE INHIBITORS

#167
20230097871
2023-03-30

UREA COMPOUND FOR ANTAGONIZING LPA1 RECEPTOR

#168
20230097420
2023-03-30

INDAZOLE HYDRAZIDE COMPOUND AND APPLICATION THEREOF

#169
20230089368
2023-03-23

POLYAROMATIC UREA DERIVATIVES AND THEIR USE IN THE TREATMENT OF MUSCLE DISEASES

#170
20230086179
2023-03-23

Carboxylic acid aromatic amides as antagonists of bradykinin B1 receptor

#171
20230066771
2023-03-02

NUCLEAR RECEPTOR MODULATORS

#172
20230066268
2023-03-02

INDAZOLE DERIVATIVES AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPES VIRUSES

#173
20230065814
2023-03-02

CONJUGATES OF-ELECTRON-PAIR-DONATING HETEROAROMATIC NITROGEN-COMPRISING COMPOUNDS

#174
20230061429
2023-03-02

Bicyclic compounds

#175
20230053726
2023-02-23

γ-diketones as Wnt/β-catenin signaling pathway activators

#176
20230051130
2023-02-16

Inhibitors of NLRP3 inflammasome

#177
20230046427
2023-02-16

Methods and compounds for restoring mutant p53 function

#178
20230045612
2023-02-09

Bicyclic carboxamides and methods of use thereof

#179
20230043209
2023-02-09

Carboxylic acid aromatic amides

#180
20230041761
2023-02-09

SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF

#181
20230032612
2023-02-02

Quaternary indazole glucocorticoid receptor antagonists

#182
20230024438
2023-01-26

INHIBITORS OF HIF-2ALPHA

#183
20230021476
2023-01-26

Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2alpha

#184
20230019803
2023-01-19

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#185
20230008022
2023-01-12

Substituted piperazine amide compounds as indoleamine 2,3-dioxygenase (IDO) inhibitors

#186
20230000773
2023-01-05

NOVEL HEADGROUP LIPID COMPOUNDS AND COMPOSITIONS FOR INTRACELLULAR DELIVERY OF THERAPEUTIC AGENTS

#187
20220411431
2022-12-29

Novel compounds and their use in therapy

#188
20220396553
2022-12-15

NOVEL HYDRAZONE DERIVATIVE IN WHICH TERMINAL AMINE GROUP IS SUBSTITUTED WITH ARYL GROUP OR HETEROARYL GROUP, AND USE THEREOF

#189
20220395512
2022-12-15

COMPOUNDS

#190
20220388995
2022-12-08

Heterocyclic compound

#191
20220388964
2022-12-08

(AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS

#192
20220380316
2022-12-01

SOLID STATE FORMS OF ARRY-797 AND PROCESS FOR PREPARATION THEREOF

#193
20220378744
2022-12-01

COMPOUNDS FOR TREATING PROLIFERATOR-ACTIVATED RECEPTORS (PPAR) MEDIATED DISEASES OR CONDITIONS

#194
20220371846
2022-11-24

Adaptive sheet caliper control system and apparatus and methods

#195
20220363678
2022-11-17

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#196
20220363646
2022-11-17

Processes of making 2-((1-benzyl-1H-indazol-3-yl)methoxy)-2-methylpropanoic acid and its derivatives

#197
20220348522
2022-11-03

ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE

#198
20220340559
2022-10-27

Modulators of Mas-related G-protein receptor X2 and related products and methods

#199
20220324880
2022-10-13

SMARCA INHIBITORS AND USES THEREOF

#200
20220324812
2022-10-13

Inhibitors of NLRP3 inflammasome

#201
20220324807
2022-10-13

Aromatic sulfonamide derivatives

#202
20220324803
2022-10-13

PROSTAGLANDIN E2 RECEPTOR 4 ANTAGONISTS AND USES THEREOF

#203
20220315534
2022-10-06

BETA ADRENERGIC AGONIST AND METHODS OF USING THE SAME

#204
20220315525
2022-10-06

AROMATIC VINYL OR AROMATIC ETHYL DERIVATIVE, PREPARATION METHOD THEREFOR, INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION

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20220298162
2022-09-22

Toll-like receptor antagonist compounds and methods of use

#206
20220281821
2022-09-08

INDAZOLE COMPOUNDS AND THEIR PHARMACEUTICAL COMPOSITIONS

#207
20220278283
2022-09-01

Organic electroluminescent element and electronic device

#208
20220267260
2022-08-25

COMPOUNDS CONTAINING A SULFONIC GROUP AS KAT INHIBITORS

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20220251047
2022-08-11

HETEROCYCLIC INHIBITORS OF MCT4

#210
20220251028
2022-08-11

TERTIARY AMINE DERIVATIVES AND THEIR USES FOR TREATING A VIRAL INFECTION

#211
20220235010
2022-07-28

Synthesis method for 1-methyl-1H-indazole-6-carboxylic acid

#212
20220204473
2022-06-30

COMPOUND AS IRAK INHIBITOR

#213
20220194939
2022-06-23

Novel compounds and methods of use treating fructose-related disorders or diseases

#214
20220194933
2022-06-23

INHIBITORS OF SARM1

#215
20220194921
2022-06-23

PROCESS FOR PREPARATION OF AXITINIB

#216
20220185785
2022-06-16

INHIBITORS OF CD40-CD154 BINDING

#217
20220169581
2022-06-02

DIRECT AROMATIC CARBON-OXYGEN AND CARBON-HYDROGEN BOND FUNCTIONALIZATION VIA ORGANIC PHOTOREDOX CATALYST

#218
20220144813
2022-05-12

SUBSTITUTED INDAZOLE DERIVATIVES ACTIVE AS KINASE INHIBITORS

#219
20220144781
2022-05-12

Therapeutic indazoles

#220
20220144775
2022-05-12

HYDRAZIDE COMPOUND AND KINASE INHIBITOR

#221
20220135574
2022-05-05

BIARYL DERIVATIVE AS GPR120 AGONIST

#222
20220127254
2022-04-28

INDAZOLYL-ISOXAZOLE DERIVATIVES FOR THE TREATMENT OF DISEASES SUCH AS CANCER

#223
20220125786
2022-04-28

SUBSTITUTED BENZALDEHYDE COMPOUNDS AND METHODS FOR THEIR USE IN INCREASING TISSUE OXYGENATION

#224
20220106265
2022-04-07

Compositions and methods for the treatment of cancer

#225
20220098167
2022-03-31

COMPOUNDS FOR TREATING RESPIRATORY DISEASE

#226
20220098156
2022-03-31

Substituted Heterocyclyl Derivatives as CDK Inhibitors

#227
20220079926
2022-03-17

Inhibitors of dihydroceramide desaturase for treating disease

#228
20220056023
2022-02-24

PREPARATION AND APPLICATION OF CLASS OF N-CONTAINING HETEROCYCLIC COMPOUNDS HAVING IMMUNOREGULATORY FUNCTION

#229
20220041559
2022-02-10

BENZO-AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS

#230
20220017514
2022-01-20

Heterocyclic compound

#231
20220017473
2022-01-20

Indazolylcyanoethylamino compound, compositions of same, method of making, and methods of using thereof

#232
20220017454
2022-01-20

Oligo-benzamide analogs and their use in cancer treatment

#233
20220009904
2022-01-13

Methods and intermediates for preparing therapeutic compounds

#234
20210395203
2021-12-23

DUAL ACTING FKBP12 AND FKBP52 INHIBITORS

#235
20210387985
2021-12-16

Bicyclic compounds and their use in the treatment of cancer

#236
20210379055
2021-12-09

Substituted alkynylene compounds as anticancer agents

#237
20210371420
2021-12-02

Inhibitors of kinase networks and uses thereof

#238
20210371393
2021-12-02

Benzopyrazole compound used as RHO kinase inhibitor

#239
20210363147
2021-11-25

Diacylglyceride O-acyltransferase 2 inhibitors

#240
20210347773
2021-11-11

Activator of TREK (TWIK RElated Kchannels) channels

#241
20210340138
2021-11-04

Compounds and methods for inhibiting fascin

#242
20210317079
2021-10-14

Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2α

#243
20210300942
2021-09-30

FUSED DIHYDRO-4H-PYRAZOLO[5,1-C][1,4]OXAZINYL COMPOUNDS AND ANALOGS FOR TREATING CNS DISORDERS

#244
20210300935
2021-09-30

PYRAZOLO-QUINAZOLINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE AS KINASE INHIBITORS

#245
20210299137
2021-09-30

COMPOUNDS, COMPOSITIONS, AND METHODS FOR TREATMENT OF DISEASES INVOLVING ACIDIC OR HYPOXIC DISEASED TISSUES

#246
20210296592
2021-09-23

Development of material for hole blocking layer with high efficiency and long lifespan, and organic light-emitting device and electronic apparatus utilizing the same

#247
20210290619
2021-09-23

SUBSTITUTED BENZALDEHYDE COMPOUNDS AND METHODS FOR THEIR USE IN INCREASING TISSUE OXYGENATION

#248
20210277030
2021-09-09

Heterocyclic amide compounds having an RORvt inhibitory action

#249
20210261520
2021-08-26

Compounds and uses thereof for the modulation of hemoglobin

#250
20210260035
2021-08-26

Indole compounds and analogues thereof

#251
20210253562
2021-08-19

ACYLSUFONAMIDE COMPOUNDS USEFUL AS EP3 RECEPTOR ANTAGONISTS

#252
20210253548
2021-08-19

SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF

#253
20210253525
2021-08-19

Selective androgen receptor degrader (SARD) ligands and methods of use thereof

#254
20210251960
2021-08-19

Indomethacin analogs for the treatment of castrate-resistant prostate cancer

#255
20210246115
2021-08-12

ANTI-INFECTIVE HETEROCYCLIC COMPOUNDS AND USES THEREOF

#256
20210246100
2021-08-12

Anti-fibrotic compounds

#257
20210238173
2021-08-05

MITOGEN-ACTIVATED PROTEIN KINASE KINASE 7 INHIBITORS

#258
20210238159
2021-08-05

Modulators of the Cystic Fibrosis Transmembrane Conductance Regulator Protein and Methods of Use

#259
20210230121
2021-07-29

Estrogen receptor beta ligands for the prevention and treatment of multiple sclerosis (MS) and other demyelinating, inflammatory and neurodegenerative diseases

#260
20210221810
2021-07-22

COMPOUNDS ACTING AT MULTIPLE PROSTAGLANDIN RECEPTORS GIVING A GENERAL ANTI-INFLAMMATORY RESPONSE

#261
20210220408
2021-07-22

ARYL HYDROCARBON RECEPTOR ANTAGONISTS AND METHODS OF USE

#262
20210214359
2021-07-15

Compounds and Methods for Treating Bacterial Infections

#263
20210214323
2021-07-15

NOVEL COMPOUNDS AND COMPOSITIONS FOR INHIBITION OF FASN

#264
20210205274
2021-07-08

AGENT FOR REDUCING VISCERAL FAT WEIGHT

#265
20210188793
2021-06-24

Carbamate compounds and methods of making and using same

#266
20210188763
2021-06-24

COMPOUNDS AND METHODS FOR HEMATOPOIETIC REGENERATION

#267
20210179614
2021-06-17

Heterocyclic compound

#268
20210179556
2021-06-17

PRIMARY CARBOXAMIDES AS BTK INHIBITORS

#269
20210163454
2021-06-03

Small molecule inhibitors of Ebola and Lassa fever viruses and methods of use

#270
20210163421
2021-06-03

Inhibitors of Rho associated coiled-coil containing protein kinase

#271
20210163408
2021-06-03

METHOD FOR PREPARING A POLYFLUORINATED COMPOUND

#272
20210163403
2021-06-03

COMPOSITIONS AND METHODS FOR TREATING CANCER

#273
20210163402
2021-06-03

Opioid receptor modulators and products and methods related thereto

#274
20210155597
2021-05-27

COMPOSITIONS AND METHODS FOR TREATMENT OF PAIN

#275
20210147365
2021-05-20

Analogs of fexaramine and methods of making and using

#276
20210147343
2021-05-20

OPIOID RECEPTOR MODULATORS AND PRODUCTS AND METHODS RELATED THERETO

#277
20210145824
2021-05-20

MODULATORS OF CELLULAR ADHESION

#278
20210139429
2021-05-13

Compounds for treatment of cardiac arrhythmias and heart failure

#279
20210130301
2021-05-06

Compositions for the treatment of pulmonary fibrosis

#280
20210130293
2021-05-06

NUCLEAR RECEPTOR MODULATORS

#281
20210122710
2021-04-29

Phenylamine compounds

#282
20210122709
2021-04-29

C7-FLUORO SUBSTITUTED TETRACYCLINE COMPOUNDS

#283
20210115061
2021-04-22

Small-Molecule HIV-1 Capsid Protein Inhibitors and Methods Using Same

#284
20210101901
2021-04-08

Preparation of pyrazolo[3,4-B]pyridines as antimalarials

#285
20210094935
2021-04-01

Bicyclic heterocycles as FGFR inhibitors

#286
20210094921
2021-04-01

Inhibitors of receptor interacting protein kinase I for the treatment of disease

#287
20210078970
2021-03-18

PRODRUGS OF THE TYROSINE KINASE INHIBITOR FOR TREATING CANCER

#288
20210070713
2021-03-11

Pesticidal compounds

#289
20210061762
2021-03-04

P300/CBP hat inhibitors

#290
20210061755
2021-03-04

Aromatic vinyl or aromatic ethyl derivative, preparation method therefor, intermediate, pharmaceutical composition, and application

#291
20210057050
2021-02-25

Workflow for generating compounds with biological activity against a specific biological target

#292
20210053997
2021-02-25

TRNA synthetase inhibitors

#293
20210053924
2021-02-25

Heterocyclic compounds as pesticides

#294
20210047278
2021-02-18

E3 UBIQUITIN LIGASE AGONISTS, PHARMACEUTICAL COMPOSITIONS INCLUDING THE E3 UBIQUITIN LIGASE AGONISTS, RELATED METHODS OF USE

#295
20210032239
2021-02-04

Compounds and pharmaceutical compositions for modulating SGK activity, and methods thereof

#296
20210024491
2021-01-28

Bicyclic carboxamides and methods of use thereof

#297
20210024464
2021-01-28

BINDING FUNCTION 3 (BF3) SITE COMPOUNDS AS THERAPEUTICS AND METHODS FOR THEIR USE

#298
20210017136
2021-01-21

Heterocyclic compounds as pesticides

#299
20210009529
2021-01-14

Sulfonyldiazoles and N-(fluorosulfonyl)azoles, and methods of making the same

#300
20210008046
2021-01-14

Bicyclic compounds and their use in the treatment of cancer