ClassID:

94557

C07D243/08 - CPC Classification

Classification description:

Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings

Recent Application in this class:
#1
20260001838
2026-01-01

NANOMATERIALS

#2
20250387490
2025-12-25

IONIZABLE LIPIDS FOR MULTIPLE ORGAN TARGETING

#3
20250296935
2025-09-25

Diamine Derivatives as Inhibitors of Leukotriene A4 Hydrolase

#4
20250205158
2025-06-26

BIODEGRADABLE LIPIDS AND FORMULATIONS FOR DELIVERY OF MRNA

#5
20250170126
2025-05-29

NOVEL B0AT1 INHIBITOR

#6
20250066320
2025-02-27

Active Ingredients with Sialagogue and Tingling/Fizzy Effect, and Preparations Containing Same

#7
20250064938
2025-02-27

IONIZABLE LIPIDS FOR MULTIPLE ORGAN TARGETING

#8
20250043065
2025-02-06

NEW ALIPHATIC POLYAMINES FOR USE AS CURING AGENT FOR EPOXY RESINS

#9
20240417378
2024-12-19

G-PROTEIN-COUPLED RECEPTOR REGULATORS AND METHODS OF USE THEREOF

#10
20240383852
2024-11-21

ANTI-VIRAL COMPOUNDS

#11
20240360083
2024-10-31

THERAPEUTIC COMPOUNDS AND COMPOSITIONS

#12
20230348464
2023-11-02

NOVEL VDAC1 INHIBITORS

#13
20230250104
2023-08-10

Diamine derivatives as inhibitors of leukotriene Ahydrolase

#14
20230174562
2023-06-08

RADIO-AND CHEMO-PROTECTIVE COMPOUNDS

#15
20230159446
2023-05-25

Methods and Compositions for Targeting Tregs using CCR8 Inhibitors

#16
20230138150
2023-05-04

RADIO-PROTECTIVE AND CHEMO-PROTECTIVE SUBSTITUTED THIOLS

#17
20230133132
2023-05-04

NAMPT MODULATORS

#18
20230099139
2023-03-30

Lipid particle, composition comprising lipid particle, and method for delivering activators to cell

#19
20230038589
2023-02-09

Methods and compositions for targeting Tregs using CCR8 inhibitors

#20
20230026611
2023-01-26

ARYL HETEROCYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS

#21
20230015617
2023-01-19

PHTHALAZINONE DERIVATIVES

#22
20220389165
2022-12-08

Diamine Compound, Polyimide Precursor and Polyimide Film Using the Same, and Use Thereof

#23
20220213081
2022-07-07

GEM-DISUBSTITUTED PYRROLIDINES, PIPERAZINES, AND DIAZEPANES, AND COMPOSITIONS AND METHODS OF MAKING THE SAME

#24
20220213034
2022-07-07

Substituted cyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists

#25
20220194923
2022-06-23

Sulfonamideurea compounds

#26
20220177425
2022-06-09

SMALL MOLECULES FOR CANCER THERAPY THAT REDUCE THE EXPRESSION OF TRANSCRIPTION FACTORS KLF5 AND EGR-1

#27
20220119377
2022-04-21

GEM-DISUBSTITUTED PYRROLIDINES, PIPERAZINES, AND DIAZEPANES, AND COMPOSITIONS AND METHODS OF MAKING THE SAME

#28
20210388011
2021-12-16

Radio-protective and chemo-protective substituted thiols

#29
20210292303
2021-09-23

AMINE CATIONIC LIPIDS AND USES THEREOF

#30
20210276966
2021-09-09

Phenyl-Piperazine Derivatives As Serotonin Reuptake Inhibitors

#31
20210230112
2021-07-29

NANOMATERIALS

#32
20210198206
2021-07-01

Therapeutic compounds and compositions

#33
20210069357
2021-03-11

DAZA chelators as ligands in liver imaging

#34
20210009533
2021-01-14

Methods for 1,4-diazo N-heterocycle synthesis

#35
20200308181
2020-10-01

Diamine derivatives as inhibitors of leukotriene A4 hydrolase

#36
20200299297
2020-09-24

Alcoxyamino derivatives for treating pain and pain related conditions

#37
20200290963
2020-09-17

Substituted cyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists

#38
20200277256
2020-09-03

Selective ship inhibitors for treating disease

#39
20200270217
2020-08-27

Biodegradable compound, lipid particle, composition comprising lipid particle, and kit

#40
20200223845
2020-07-16

Viral replication inhibitors

#41
20200199114
2020-06-25

Gem-disubstituted pyrrolidines, piperazines, and diazepanes, and compositions and methods of making the same

#42
20200062781
2020-02-27

Bisaryl heterocycles as NRF2 activators

#43
20200000802
2020-01-02

Phthalazinone derivatives

#44
20190345109
2019-11-14

Therapeutic compounds and compositions

#45
20190276414
2019-09-12

CHIRAL RESOLUTION OF AN INTERMEDIATE OF SUVOREXANT AND COCRYSTALS THEREOF

#46
20190241523
2019-08-08

THERAPEUTIC COMPOUNDS AND COMPOSITIONS

#47
20190218367
2019-07-18

PVC plasticizers and methods for making thereof

#48
20190202783
2019-07-04

Substituted spirocyclohexanes as muscarinic Mreceptor and/or Mreceptor agonists

#49
20190194163
2019-06-27

Dual NAV1.2/5HT2a inhibitors for treating CNS disorders

#50
20190084965
2019-03-21

Amine cationic lipids and uses thereof

#51
20190055205
2019-02-21

Methods for 1,4-diazo n-heterocycle synthesis

#52
20190040052
2019-02-07

Suvorexant intermediate and preparation method thereof

#53
20190040018
2019-02-07

Homopiperazine-based catalysts for neutralization of organophosphorus-based compounds

#54
20190016682
2019-01-17

Azepane derivatives and methods of treating hepatitis B infections

#55
20180327374
2018-11-15

Cyanopyridine derivatives as liver X receptor beta agonists, compositions, and their use

#56
20180305324
2018-10-25

Bis(aminophenylphenol) ligands and transition metal catalysts prepared therefrom

#57
20180273441
2018-09-27

Methods for low temperature fluorine-18 radiolabeling of biomolecules

#58
20180235978
2018-08-23

Method for use of homopiperazinium compounds in the treatment of cancer

#59
20180230159
2018-08-16

DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE

#60
20180185363
2018-07-05

Phthalazinone derivatives

#61
20180148455
2018-05-31

Method of treating Crohn's disease comprising a TLR2 antagonist

#62
20180148425
2018-05-31

N-aralkylcarbonyl-piperazine and -homopiperazine compounds and personal care compositions comprising the same

#63
20180127389
2018-05-10

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#64
20180105491
2018-04-19

Substituted cyclohexanes as muscarinic M1 receptor and/or M4 receptor agonists

#65
20180044300
2018-02-15

Azepane derivatives and methods of treating hepatitis B infections

#66
20180021346
2018-01-25

GLP-1 receptor modulators

#67
20170348324
2017-12-07

DERIVATIVES OF BETULIN

#68
20170313717
2017-11-02

GLP-1 receptor modulators

#69
20170253568
2017-09-07

Homopiperazine-based catalysts for neutralization of organophosphorus-based compounds

#70
20170252356
2017-09-07

Compounds and compositions for treating HIV with derivatives of Betulin

#71
20170226124
2017-08-10

PHTHALAZINONE DERIVATIVES

#72
20170217947
2017-08-03

Route of synthesis for the preparation of suvorexant

#73
20170173040
2017-06-22

Method for use of homopiperazinium compounds in the treatment of cancer

#74
20170137409
2017-05-18

Amine cationic lipids and uses thereof

#75
20170015629
2017-01-19

Azepane derivatives and methods of treating hepatitis B infections

#76
20170001988
2017-01-05

PIPERIDINE AND PIPERAZINE DERIVATIVES AND THEIR USE IN TREATING VIRAL INFECTIONS AND CANCER

#77
20160297810
2016-10-13

Viral replication inhibitors

#78
20160257656
2016-09-08

Heterocyclic compounds and methods for their use

#79
20160228450
2016-08-11

GLP-1 receptor modulators

#80
20160214993
2016-07-28

GLP-1 receptor modulators

#81
20160137620
2016-05-19

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#82
20160046587
2016-02-18

Preparation and method for use in the treatment of respiratory diseases

#83
20160024066
2016-01-28

Method of treating Ebola

#84
20160024024
2016-01-28

Choline kinase inhibitors

#85
20150315159
2015-11-05

Azepane derivatives and methods of treating hepatitis B infections

#86
20150225355
2015-08-13

Azepane derivatives and methods of treating hepatitis B infections

#87
20150197533
2015-07-16

Azepane derivatives and methods of treating hepatitis B infections

#88
20150158833
2015-06-11

Sulfonamide derivative having PGD2 receptor antagonistic activity

#89
20150087824
2015-03-26

Production method for isoquinoline derivatives and salts thereof

#90
20150087823
2015-03-26

Trans-2-decenoic acid derivative and drug containing same

#91
20150087645
2015-03-26

Therapeutic piperazines

#92
20150080382
2015-03-19

Diamine derivatives as inhibitors of leukotriene A4 hydrolase

#93
20150038493
2015-02-05

COMPOUNDS THAT TRAP ALPHA-OXOALDEHYDES AND ALPHA-BETA-UNSATURATED ALDEHYDES, META-COMPOUNDS CONTAINING SUCH COMPOUNDS, AND USE OF SAID COMPOUNDS IN TREATING ILLNESSES RELATED TO THE ACCUMULATION OF AGES AND ALES

#94
20150038416
2015-02-05

GLP-1 receptor modulators

#95
20150037261
2015-02-05

Class of diazepine derivative chelating agents and complexes with paramagnetic metals thereof as MRI contrast agents

#96
20150011527
2015-01-08

GLP-1 receptor modulators

#97
20140349986
2014-11-27

Substituted aminoindanes and analogs thereof, and the pharmaceutical use thereof

#98
20140163043
2014-06-12

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#99
20140128380
2014-05-08

METHODS OF MODULATING THE ACTIVITY OF THE MC1 RECEPTOR AND TREATMENT OF CONDITIONS RELATED TO THIS RECEPTOR

#100
20140128361
2014-05-08

Cyclic amide BACE-1 inhibitors having a benzamide substituent

#101
20140038979
2014-02-06

Sulfonyl-derivatives as novel inhibitors of histone deacetylase

#102
20140038945
2014-02-06

PIPERAZINE PDE4 INHIBITORS AND USES THEREOF

#103
20140005176
2014-01-02

2-phenoxy- and 2-phenylsulfonamide derivatives with CCR3 antagonistic activity for the treatment of inflammatory or immunological disorders

#104
20130296551
2013-11-07

7-MEMBERED RING COMPOUND AND METHOD OF PRODUCTION AND PHARMACEUTICAL APPLICATION THEREOF

#105
20130237529
2013-09-12

Compound that can inhibit UBC13-UEV interactions, pharmaceutical compositions and therapeutic uses

#106
20130231476
2013-09-05

Transamination of nitrogen-containing compounds to make cyclic and cyclic/acyclic polyamine mixtures

#107
20130231332
2013-09-05

Small molecule inhibitors of ebola and lassa fever viruses and methods of use

#108
20130225565
2013-08-29

2,5-disubstituted arylsulfonamide CCR3 antagonists

#109
20130225563
2013-08-29

Methods of modulating the activity of the MC5 receptor and treatment of conditions related to this receptor

#110
20130184263
2013-07-18

Derivatives of betulin

#111
20130178420
2013-07-11

GLP-1 receptor modulators

#112
20130144054
2013-06-06

Production method for isoquinoline derivatives and salts thereof

#113
20130131034
2013-05-23

DERIVATIVES OF AMINOINDANES, THEIR PREPARATION AND THEIR APPLICATION IN THERAPEUTICS

#114
20130123243
2013-05-16

DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE

#115
20130035329
2013-02-07

THERAPEUTICALLY ACTIVE COMPOSITIONS AND THEIR METHODS OF USE

#116
20130018047
2013-01-17

N-PHENYL-(PIPERAZINYL OR HOMOPIPERAZINYL)-BENZENESULFONAMIDE OR BENZENESULFONYL-PHENYL-(PIPERAZINE OR HOMOPIPERAZINE) COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE SEROTONIN 5-HT6 RECEPTOR

#117
20130004518
2013-01-03

Cyclic amine BACE-1 inhibitors having a benzamide substituent

#118
20120302553
2012-11-29

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#119
20120283247
2012-11-08

Diazepane acetamide derivatives as selective 11B-HSD1 inhibitors

#120
20120259111
2012-10-11

Seven-membered ring compound and pharmaceutical use therefor

#121
20120238749
2012-09-20

INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME

#122
20120195985
2012-08-02

Glycine transporter-1 inhibitors

#123
20120142674
2012-06-07

N-phenyl-(homo)piperazinyl-benzenesulfonyl or benzenesulfonamide compounds suitable for treating disorders that respond to the modulation of the serotonin 5-HTreceptor

#124
20120141392
2012-06-07

METHODS OF MODULATING THE ACTIVITY OF THE MC1 RECEPTOR AND TREATMENT OF CONDITIONS RELATED TO THIS RECEPTOR

#125
20120115850
2012-05-10

Substituted arylamine compounds and methods of treatment

#126
20120108573
2012-05-03

Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them

#127
20120088754
2012-04-12

Sulfonyl-derivatives as novel inhibitors of histone deacetylase

#128
20120065193
2012-03-15

Cyclopropyl amide derivatives

#129
20120046198
2012-02-23

Ligand libraries for screening GPCRs

#130
20120040969
2012-02-16

N-phenyl-(piperazinyl or homopiperazinyl)-benzenesulfonamide or benzenesulfonyl-phenyl-(piperazine or homopiperazine) compounds suitable for treating disorders that respond to modulation of the serotonin 5-HT6 receptor

#131
20120022049
2012-01-26

Nicotinic receptor agonists for the treatment of inflammatory diseases

#132
20120010204
2012-01-12

Phthalazinone derivatives

#133
20120004315
2012-01-05

Selective estrogen receptor modulator

#134
20110288057
2011-11-24

SALICYLIC ACID DERIVATIVES BEING FARNESYL PYROPHOSPHATE SYNTHASE ACTIVITY INHIBITORS

#135
20110269747
2011-11-03

Polyarylcarboxamides useful as lipid lowering agents

#136
20110263572
2011-10-27

3-aminoalkyl-1,4-diazepan-2-one melanocortin-5-receptor antagonists

#137
20110256067
2011-10-20

Contrast agents endowed with high relaxivity

#138
20110201590
2011-08-18

Substituted aminoindanes and analogs thereof, and the pharmaceutical use thereof

#139
20110166342
2011-07-07

7-membered ring compound and method of production and pharmaceutical application thereof

#140
20110160189
2011-06-30

Compound that can inhibit UBC13-UEV interactions, pharmaceutical compositions and therapeutic uses

#141
20110136787
2011-06-09

DIPHENYL AZEPANE, DIAZEPANE AND OXAZEPANE DERIVATIVES AND USES THEREOF

#142
20110130387
2011-06-02

Sirtuin modulating compounds

#143
20110129542
2011-06-02

SUBSTITUTED AZEPINE- AND DIAZEPINE-SULFONAMIDES USEFUL TO INHIBIT 11BETA-HYDROXYSTEROID DEHYDROGENASE TYPE-1

#144
20110098282
2011-04-28

Compounds

#145
20110092698
2011-04-21

Heterocyclyl compounds

#146
20110082295
2011-04-07

Therapeutic agent for Alzheimer's disease

#147
20110082280
2011-04-07

Methods Of Coupling Multidentate AZA Ligands To Targeting Molecules

#148
20110077231
2011-03-31

COMPOUNDS

#149
20110065691
2011-03-17

Therapeutic piperazines

#150
20110065689
2011-03-17

Piperazine PDE4 inhibitors and uses thereof

#151
20110065688
2011-03-17

Therapeutic piperazines

#152
20110059952
2011-03-10

3-substituted-1,4-diazepan-2-one melanocortin-5 receptor antagonists

#153
20110039835
2011-02-17

Substituted arylamide diazepinopyrimidone derivatives

#154
20110039833
2011-02-17

1-benzoyl substituted diazepine derivatives as selective histamine H3 receptor agonists

#155
20110039714
2011-02-17

Probes, Systems, and Methods for Drug Discovery

#156
20110015371
2011-01-20

Inhibitors of interleukin-1 beta converting enzyme

#157
20110009641
2011-01-13

Amine-containing lipids and uses thereof

#158
20110009423
2011-01-13

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#159
20110003784
2011-01-06

Opsin-binding ligands, compositions and methods of use

#160
20100331307
2010-12-30

Therapeutic compounds and compositions

#161
20100311699
2010-12-09

Carboxylic acid 4-phenylazo-phenyl ester derivatives and their use as monoamine neurotransmitter re-uptake inhibitors

#162
20100292221
2010-11-18

Benzenesulfonanilide compounds suitable for treating disorders that respond to modulation of the serotonin 5-HTreceptor

#163
20100292220
2010-11-18

Benzenesulfonanilide compounds suitable for treating disorders that respond to modulation of the serotonin 5-HTreceptor

#164
20100286109
2010-11-11

Amide derivatives as positive allosteric modulators and methods of use thereof

#165
20100280014
2010-11-04

N-phenyl- (piperazinyl or homopiperazinyl)-benzenesulfonamide or benzenesulfonyl-phenl-(piperazine or homopiperazine) compounds suitable for treating disorders that respond to modulation of the serotonin 5-HTreceptor

#166
20100279997
2010-11-04

ANALGESIC THAT BINDS FILAMIN A

#167
20100279986
2010-11-04

HETEROCYCLIC DERIVED METALLOPROTEASE INHIBITORS

#168
20100273782
2010-10-28

2,5-disubstituted arylsulfonamide CCR3 antagonists

#169
20100256122
2010-10-07

BUTYL AND BUTYNYL BENZYL AMINE COMPOUNDS

#170
20100240640
2010-09-23

(THIO) Carbamoyl-Cyclohexane Derivatives as D3/D2 Receptor Antagonists

#171
20100240639
2010-09-23

Sulfonyl-derivatives as novel or histone deacetylase

#172
20100222330
2010-09-02

New Compounds

#173
20100210630
2010-08-19

Diamine derivatives as inhibitors of leukotriene A4 hydrolase

#174
20100210474
2010-08-19

HETEROCYCLIC SCAFFOLDS USEFUL FOR PREPARATION OF COMBINATORIAL LIBRARIES, LIBRARIES AND METHODS FOR PREPARATION THEREOF

#175
20100204213
2010-08-12

Arylsulfonamide derivatives for use as CCR3 antagonists in the treatment of inflammatory and immunological disorders

#176
20100197668
2010-08-05

1,2,3,4-TETRAHYDROPYRROLO[1,2-A]PYRAZINE-6-CARBOXAMIDE AND 2,3,4,5-TETRAHYDROPYRROLO[1,2-a][1,4]-DIAZEPINE-7-CARBOXAMIDE DERIVATIVES, PREPARATION AND THERAPEUTIC USE THEREOF

#177
20100152138
2010-06-17

Cyclic amine BACE-1 inhibitors having a benzamide substituent

#178
20100144708
2010-06-10

HETEROCYCLIC COMPOUNDS CONTAINING NITROGEN ATOMS OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF, PROCESS FOR THE PREPARATION THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME FOR TREATMENT OF CANCER

#179
20100120769
2010-05-13

CYCLOHEXYL PIPERAZINYL METHANONE DERIVATIVES

#180
20100105894
2010-04-29

Cyclopropane compounds and pharmaceutical use thereof

#181
20100104629
2010-04-29

CATIONIC LIPIDS AND USES THEREOF

#182
20100099676
2010-04-22

SULFONYLUREA DERIVATIVE CAPABLE OF SELECTIVELY INHIBITING MMP-13

#183
20100087423
2010-04-08

Benzamide derivatives as bradykinin antagonists

#184
20100075978
2010-03-25

SULFONAMIDE DERIVATIVES AS BRADYKININ ANTAGONISTS

#185
20100075953
2010-03-25

SUBSTITUTED PIPERAZINES, (1,4) DIAZEPINES, AND 2,5-DIAZABICYCLO (2.2.1) HEPTANES AS HISTAMINE H1 AND/OR H3 ANTAGONISTS OR HISTAMINE H3 REVERSE ANTAGONISTS

#186
20100069638
2010-03-18

Sulfonamide derivative having PGD2 receptor antagonistic activity

#187
20100069628
2010-03-18

Multidentate AZA ligands able to complex metal ions and the use thereof in diagnostics and therapy

#188
20100069365
2010-03-18

Diazepane-acetamide derivatives as selective 11β-HSD1 inhibitors

#189
20100063040
2010-03-11

Sulfonamide derivative having PGD2 receptor antagonistic activity

#190
20100029621
2010-02-04

Hexafluoroisopropanol derivatives

#191
20100022518
2010-01-28

Heterocyclyl compounds

#192
20100016282
2010-01-21

Heterocyclyl compounds

#193
20090325930
2009-12-31

Selective estrogen receptor modulator

#194
20090286771
2009-11-19

2-Phenoxy- and 2-Phenylsulfonamide Derivatives with CCR3 Antagonistic Activity for the Treatment of Inflammatory or Immunological Disorders

#195
20090285849
2009-11-19

Thiosemicarbazones as anti-virals and immunopotentiators

#196
20090275727
2009-11-05

Peptide turn mimetics

#197
20090264416
2009-10-22

N-benzyl,N'-arylcarbonylpiperazine derivatives

#198
20090263407
2009-10-22

Cationic Lipids and Uses Thereof

#199
20090253908
2009-10-08

NOVEL M3 MUSCARINIC ACETYLCHOINE RECEPTOR ANTAGONISTS

#200
20090253683
2009-10-08

7-membered ring compound and method of production and pharmaceutical application thereof

#201
20090253670
2009-10-08

Amide derivatives as positive allosteric modulators and methods of use thereof

#202
20090227595
2009-09-10

Glycine transporter-1 inhibitors

#203
20090221558
2009-09-03

Methods of modulating the activity of the MC5 receptor and treatment of conditions related to this receptor

#204
20090221557
2009-09-03

3-aminoalkyl-1,4-diazepan-2-one melanocortin-5 receptor antagonists

#205
20090181951
2009-07-16

PARP INHIBITORS

#206
20090176768
2009-07-09

Diaza heterocyclic amide compounds and their uses

#207
20090143365
2009-06-04

Derivatives of alkylpiperazine- and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors

#208
20090124601
2009-05-14

Tartaric Acid Salts of a Dipeptidyl Peptidase-IV Inhibitor

#209
20090118303
2009-05-07

SEROTONIN 5-HT3 RECEPTOR AGONIST

#210
20090111796
2009-04-30

7-membered ring compound and method of production and pharmaceutical application thereof

#211
20090111793
2009-04-30

HYDROXYALKANOYLAMINOLACTAMS AND RELATED STRUCTURES AS INHIBITORS OF A BETA PROTEIN PRODUCTION

#212
20090093463
2009-04-09

NOVEL COMPOUNDS OF SUBSTITUTED AND UNSUBTITUTED ADAMANTYL AMIDES

#213
20090076030
2009-03-19

Piperazine compounds

#214
20090076020
2009-03-19

Cyclopropyl amide derivatives

#215
20090075982
2009-03-19

Piperazine compounds

#216
20090069304
2009-03-12

MMP-13 SELECTIVE INHIBITOR

#217
20090069302
2009-03-12

CHEMICAL COMPOUNDS

#218
20090054460
2009-02-26

Piperazine derivatives and methods of use

#219
20080306258
2008-12-11

Cyclopropane compounds and pharmaceutical use thereof

#220
20080300237
2008-12-04

Pharmaceutically Active Diazepanes

#221
20080280883
2008-11-13

Muscarinic Receptor Antagonists

#222
20080279917
2008-11-13

Bisbenzamidines for the Treatment of Pneumonia

#223
20080275028
2008-11-06

Modulators or Alpha7 Nicotinic Acetylcholine Receptors and Therapeutic Uses Thereof

#224
20080261994
2008-10-23

CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF

#225
20080261948
2008-10-23

Ligands for G-Protein Coupled Receptors

#226
20080234247
2008-09-25

Heterocyclic analgesic compounds and methods of use thereof

#227
20080227784
2008-09-18

N-(3,4-disubstituted phenyl) salicylamide derivatives

#228
20080200469
2008-08-21

Phthalazinone derivatives

#229
20080194520
2008-08-14

Sulfonyl amino cyclic derivatives and use thereof

#230
20080167347
2008-07-10

Ctgf Expression Inhibitor

#231
20080161292
2008-07-03

Pyrroloquinoxalinone inhibitors of poly(ADP-ribose)polymerase

#232
20080161281
2008-07-03

Amino-substituted tricyclic derivatives and methods of use

#233
20080153826
2008-06-26

Substituted aryl cycloalkanoyl derivatives and methods of their use

#234
20080132489
2008-06-05

Alkyl substituted homopiperazine derivatives and their use as monoamine neurotransmitter re-uptake inhibitors

#235
20080132482
2008-06-05

Hydroxyalkanoylaminolactams and related structures as inhibitors of aβ protein production

#236
20080125412
2008-05-29

POLYARYLCARBOXAMIDES USEFUL AS LIPID LOWERING AGENTS

#237
20080114000
2008-05-15

Suppressor of excess accumulation of intracellular sodium ions

#238
20080113968
2008-05-15

Substituted piperazines and diazepanes

#239
20080108601
2008-05-08

Sulfonyl-derivatives as novel inhibitors or histone deacetylase

#240
20080103129
2008-05-01

Heterocyclic derived metalloprotease inhibitors

#241
20080096936
2008-04-24

Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them

#242
20080096873
2008-04-24

Aryl sulfonamide compounds for treating obesity

#243
20080096869
2008-04-24

Adamantyl acetamides as 11-β hydroxysteroid dehydrogenase inhibitors

#244
20080070953
2008-03-20

Inhibitors of interleukin-1β converting enzyme

#245
20080045508
2008-02-21

SUBSTITUTED AMINOMETHYL BENZAMIDE COMPOUNDS

#246
20080045505
2008-02-21

1-benzoyl substituted diazepine derivatives as selective histamine H3 receptor agonists

#247
20080004289
2008-01-03

Glycine transporter-1 inhibitors

#248
20080004258
2008-01-03

Butyl and butynyl benzyl amine compounds

#249
20070265277
2007-11-15

Serotonin 5-HT3 receptor agonist

#250
20070258905
2007-11-08

Contrast agents endowed with high relaxivity for use in magnetic resonance imaging (MRI) which contain a chelating moiety with polyhydroxylated substituents

#251
20070254865
2007-11-01

Aminocyclohexanes as dipeptidyl peptidase-IV inhibitors for the treatment or prevention of diabetes

#252
20070249626
2007-10-25

Diaza heterocyclic amide compounds and their uses

#253
20070244087
2007-10-18

2-alkoxy-3,4,5-trihydroxy-alkylamides, preparation thereof, compositions containing them and use thereof

#254
20070219176
2007-09-20

Viral polymerase inhibitors

#255
20070213316
2007-09-13

N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives

#256
20070203124
2007-08-30

Therapeutic piperazines

#257
20070173494
2007-07-26

Diaza heterocyclic sulfonamide derivatives and their uses

#258
20070167436
2007-07-19

Cyclohexyl piperazinyl methanone derivatives

#259
20070155727
2007-07-05

Amide inhibitors of leukotriene A4 hydrolase

#260
20070155726
2007-07-05

Diamine derivatives as inhibitors of leukotriene Ahydrolase

#261
20070155725
2007-07-05

2-phenoxy- and 2-phenylsulfonamide derivatives with CCR3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders

#262
20070142393
2007-06-21

Sulfonyl-derivatives as novel inhibitors of histone deacetylase

#263
20070135414
2007-06-14

Tachykinin Antagonists

#264
20070082888
2007-04-12

Polyarylcarboxamides useful as lipid lowering agents

#265
20070066600
2007-03-22

Substituted naphthalene sulfonamides

#266
20070066599
2007-03-22

New compounds

#267
20070066598
2007-03-22

Compounds

#268
20070060624
2007-03-15

Bioisosteres of actinonin

#269
20070060574
2007-03-15

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#270
20070049571
2007-03-01

Dipiperazinyl ketones and related analogues

#271
20070037810
2007-02-15

Sirtuin modulating compounds

#272
20070037809
2007-02-15

Sirtuin modulating compounds

#273
20070027141
2007-02-01

Derivatives of alkylpiperazine and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors

#274
20070027132
2007-02-01

Hydroxyalkanoylaminolactams and related structures as inhibitors of Aβ protein production

#275
20060287293
2006-12-21

Heterocyclylakylamines as muscarinic receptor antagonists

#276
20060276465
2006-12-07

1,2-di(cyclic) substituted benzene compounds

#277
20060241113
2006-10-26

Polyarylcarboxamides useful as lipid lowering agents

#278
20060229318
2006-10-12

Piperazine compounds

#279
20060229298
2006-10-12

Melanin concentrating hormone receptor ligands: substituted 1-benzyl-4-aryl piperazine analogues

#280
20060229297
2006-10-12

(Thio) carbamoyl-cyclohexane derivatives as D3/D2 receptor antagonists

#281
20060205737
2006-09-14

Substituted arylamine compounds and methods of treatment

#282
20060199826
2006-09-07

Cyclopropane compounds and pharmaceutical use thereof

#283
20060178366
2006-08-10

Compounds for the treatment of inflammatory disorders

#284
20060167247
2006-07-27

Urea inhibitors of MAP kinases

#285
20060167013
2006-07-27

Inhibitors for excessive accumulation of sodium ion in cells

#286
20060160821
2006-07-20

Ureas as factor Xa inhibitors

#287
20060148821
2006-07-06

N,N-disubstituted diazocycloalkanes

#288
20060148780
2006-07-06

Diazepanes derivatives useful as IFA inhibitors

#289
20060123565
2006-06-15

Para-phenylenediamine derivatives comprising a cyclic diaza group substituted with a cationic radical, and use of these derivatives for dyeing keratin fibers

#290
20060116364
2006-06-01

Selective estrogen receptor modulator

#291
20060089368
2006-04-27

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#292
20060084662
2006-04-20

Phenyl-piperazine derivatives as serotonin reuptake inhibitors

#293
20060084658
2006-04-20

Nitrogen-containing cyclic compound and pharmaceutical composition containing the compound

#294
20060084641
2006-04-20

IL-8 receptor antagonists

#295
20060079506
2006-04-13

Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors

#296
20060052597
2006-03-09

Aryloxyalkylamine derivatives as h3 receptor ligands

#297
20060052396
2006-03-09

Arylamines for the treatment of conditions associated with gsk-3

#298
20060052363
2006-03-09

Haloperidol analogs

#299
20060034773
2006-02-16

Multidentate AZA ligands able to complex metal ions and the use thereof in diagnostics and therapy

#300
20060025404
2006-02-02

Substituted piperazines,(1,4) diazepines, and 2,5-diazabicyclo (2.2.1)iieptanes as histamine H1 and/or H3 antagonists or histamine H3 reverse antagonists