ClassID:

94766

C07D277/48 - CPC Classification

Classification description:

Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms; Nitrogen atoms; Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines

Recent Application in this class:
#1
20250276953
2025-09-04

SMALL MOLECULE SIRTUIN INHIBITORS AND USES THEREOF

#2
20250011315
2025-01-09

ARYL HYDROCARBON RECEPTOR (AHR) AGONISTS AND USES THEREOF

#3
20250009693
2025-01-09

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#4
20240270735
2024-08-15

CDK19-Selective Inhibitors, and Methods of Use Thereof

#5
20230404954
2023-12-21

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#6
20230348450
2023-11-02

CARBOXYLIC ACID-CONTAINING COMPOUNDS AS MODULATORS OF BIS-PHOSPHOGLYCERATE MUTASE FOR THE TREATMENT OF SICKLE CELL DISEASE

#7
20230295147
2023-09-21

Aryl hydrocarbon receptor (AHR) agonists and uses thereof

#8
20230121825
2023-04-20

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#9
20210276963
2021-09-09

Pesticidal compositions and methods

#10
20210230153
2021-07-29

Aryl hydrocarbon receptor (AHR) agonists and uses thereof

#11
20200375930
2020-12-03

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#12
20200308156
2020-10-01

Biguanide derivatives and their rearrangement products for use in the treatment of cancer

#13
20200199067
2020-06-25

Hydrogen sulfide donor in organic salt form and preparation method therefor

#14
20180238863
2018-08-23

CHEMICAL SYNTHESIS

#15
20180120306
2018-05-03

Haptens, hapten conjugates, compositions thereof and method for their preparation and use

#16
20170360730
2017-12-21

Modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

#17
20170037016
2017-02-09

GUANIDINE COMPOUNDS AND USE THEREOF AS BINDING PARTNERS FOR 5-HT5 RECEPTORS

#18
20160318886
2016-11-03

Compound, organic cation transporter 3 detection agent, and organic cation transporter 3 activity inhibitor

#19
20160229804
2016-08-11

TrkA kinase inhibitors, compositions and methods thereof

#20
20150038483
2015-02-05

Aromatic 5-membered heterocyclic derivative having TRPV4-Inhibiting activity

#21
20140349848
2014-11-27

Fungicidal 4-substituted-3-{phenyl[(heterocyclylmethoxy)imino]methyl}-1,2,4-oxadizol-5(4H)-one derivatives

#22
20140275189
2014-09-18

Methods for modulating bacterial virulence and related compounds

#23
20140228388
2014-08-14

Phenyl-guanidine derivatives

#24
20140155597
2014-06-05

Amidine compound or salt thereof

#25
20140121250
2014-05-01

Alkylamidothiazoles, cosmetic or dermatological preparations containing said alkylamidothiazoles, and use thereof to combat or prevent undesired pigmentation of the skin

#26
20130324537
2013-12-05

Guanidine compounds, and use thereof as binding partners for 5-HT5 receptors

#27
20130281708
2013-10-24

Process for the Production of 2-Amino-5-Fluorothiazole

#28
20130217706
2013-08-22

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#29
20130040993
2013-02-14

Fungicide hydroximoyl-heterocycles derivatives

#30
20130039870
2013-02-14

Cosmetic or dermatological preparations with a content of one or more thiazole derivates

#31
20120322761
2012-12-20

Heterocyclic CETP inhibitors

#32
20120283255
2012-11-08

UREA DERIVATIVES, METHODS FOR THEIR MANUFACTURE, AND USES THEREFOR

#33
20120252759
2012-10-04

Thiazole derivatives for the treatment of diseases such as cancer

#34
20120165375
2012-06-28

Urea glucokinase activators

#35
20120122920
2012-05-17

LIBRARIES OF N-SUBSTITUTED-N-PHENYLETHYLSULFONAMIDES FOR DRUG DISCOVERY

#36
20120122710
2012-05-17

LIBRARIES OF N-SUBSTITUTED-N-PHENYLETHYLSULFONAMIDES FOR THE IDENTIFICATION OF BIOLOGICAL AND PHARMACOLOGICAL ACTIVITY

#37
20120071475
2012-03-22

UREA DERIVATIVES HAVING PI3K-INHIBITING ACTIVITY

#38
20120015990
2012-01-19

TASPASE1 inhibitors and their uses

#39
20120015941
2012-01-19

Antibacterial amide and sulfonamide substituted heterocyclic urea compounds

#40
20120003229
2012-01-05

MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN ALPHAVBETA3 RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY

#41
20110301158
2011-12-08

ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS

#42
20110237589
2011-09-29

Guanidine compounds, and use thereof as binding partners for 5-HT5 receptors

#43
20110124693
2011-05-26

5-PHENYL-4-METHYL-THIAZOL-2-YL-AMINE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL 3 KINASE ENZYMES (PI3) FOR THE TREATMENT OF INFLAMMATORY DISEASES

#44
20110124624
2011-05-26

5-PHENYL-4-METHYL-THIAZOL-2-YL-AMINE DERIVATIVES AS INHIBITORS OF PHOSPHATIDYLINOSITOL 3 KINASE ENZYMES (PI3) FOR THE TREATMENT OF INFLAMMATORY DISEASES

#45
20110118470
2011-05-19

Nitrogen-containing aromatic derivatives

#46
20110118126
2011-05-19

Methods of chemotype evolution

#47
20110086855
2011-04-14

Compounds as cannabinoid receptor ligands and uses thereof

#48
20110077234
2011-03-31

Urea glucokinase activators

#49
20110060019
2011-03-10

Heteroaryl-ureas and their use as glucokinase activators

#50
20110053958
2011-03-03

Modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto

#51
20100298340
2010-11-25

Thiazol-Guanidine Derivatives Useful As A (Beta)-Related Pathologies

#52
20100297725
2010-11-25

Haptens, hapten conjugates, compositions thereof and method for their preparation and use

#53
20100286169
2010-11-11

Antibacterial sulfone and sulfoxide substituted heterocyclic urea compounds

#54
20100267669
2010-10-21

Heterocyclic CETP inhibitors

#55
20100247468
2010-09-30

Compounds that modulate PPARγ-type receptors and cosmetic/pharmaceutical compositions comprising said compounds

#56
20100240890
2010-09-23

Benzamidine derivatives, process for the preparation thereof and pharmaceutical composition comprising the same

#57
20100240889
2010-09-23

Urea derivatives methods for their manufacture and uses thereof

#58
20100204288
2010-08-12

Heteroaryl-ureas and their use as glucokinase activators

#59
20100197911
2010-08-05

Nitrogen-containing aromatic derivatives

#60
20100184087
2010-07-22

Haptens, hapten conjugates, compositions thereof and method for their preparation and use

#61
20100152188
2010-06-17

Novel Heterocyclic Compounds

#62
20100137315
2010-06-03

Sphingosine Kinase Inhibitors and Methods of Their Use

#63
20100105900
2010-04-29

Inhibitors of carnitine palmitoyltransferase and treating cancer

#64
20100105683
2010-04-29

COMPOUNDS USEFUL FOR INHIBITING CHK1

#65
20100099689
2010-04-22

Methods of modulating PPAR gamma-type receptors

#66
20100093814
2010-04-15

Compounds as cannabinoid receptor ligands and uses thereof

#67
20100093690
2010-04-15

5-phenylthiazole derivatives and use as PI3 kinase inhibitors

#68
20100041711
2010-02-18

Urea glucokinase activators

#69
20100016383
2010-01-21

4-(3,3-DIHALO-ALLYLOXY)PHENOL DERIVATIVES HAVING PESTICIDAL PROPERTIES

#70
20100016259
2010-01-21

Malonyl-CoA decarboxylase inhibitors useful as metabolic modulators

#71
20100010057
2010-01-14

THIAZOLE DERIVATIVES AS INHIBITORS OF P13 KINASE

#72
20100009989
2010-01-14

Urea glucokinase activators

#73
20090311266
2009-12-17

Inhibitors of the endothelin signalling pathway and alphavbeta3 integrin receptor antagonists for combination therapy

#74
20090234132
2009-09-17

5-phenyl-thiazol-2-yl-urea derivatives and use as PI3 kinase inhibitors

#75
20090216013
2009-08-27

Heteroaryl-ureas and their use as glucokinase activators

#76
20090137420
2009-05-28

Methods, compounds and compositions with genotype selective anticancer activity

#77
20090118501
2009-05-07

Dicycloalkyl urea glucokinase activators

#78
20090105482
2009-04-23

Ureido-thiazole glucokinase activators

#79
20090069395
2009-03-12

DEUTERIUM-ENRICHED FAMOTIDINE

#80
20080319033
2008-12-25

Organic compounds

#81
20080306067
2008-12-11

Modulators of Chemokine Receptor Activity

#82
20080280871
2008-11-13

5-phenyl-4-methyl-thiazol-2-yl-amine derivatives as inhibitors of phosphatidylin ositol 3 kinase enzymes (PI13) for treatment of inflammatory diseases

#83
20080268462
2008-10-30

Haptens, hapten conjugates, compositions thereof and method for their preparation and use

#84
20080227783
2008-09-18

5-Substituted Thiazol-2-Yl Amino Compounds and Compositions as Protein Kinase Inhibitors

#85
20080207764
2008-08-28

Benzamidine derivatives having anti-inflammatory and immunosuppressive activity

#86
20080207703
2008-08-28

Antibacteriall heterocyclic ureas

#87
20080188531
2008-08-07

Thiazole derivatives and use thereof

#88
20080132546
2008-06-05

Alkyl urea substituted pyridines

#89
20080125424
2008-05-29

Derivatives of urea and related diamines, methods for their manufacture, and uses therefor

#90
20080119455
2008-05-22

Aryl carbonyl derivatives as therapeutic agents

#91
20080119454
2008-05-22

Aryl carbonyl derivatives as therapeutic agents

#92
20080096869
2008-04-24

Adamantyl acetamides as 11-β hydroxysteroid dehydrogenase inhibitors

#93
20080064699
2008-03-13

Compounds as cannabinoid receptor ligands and uses thereof

#94
20080058335
2008-03-06

Compounds as cannabinoid receptor ligands and uses thereof

#95
20070299074
2007-12-27

Guanidine compounds, and use thereof as binding partners for 5-HT5 receptors

#96
20070281979
2007-12-06

FBPase inhibitors for diabetes

#97
20070213301
2007-09-13

Substituted Aminothiazole Derivatives With Anti-HCV Activity

#98
20070173504
2007-07-26

Calcium channel antagonists

#99
20070135631
2007-06-14

Heterocyclic CETP inhibitors

#100
20070135523
2007-06-14

Novel benzamidine derivatives having anti-inflammatory and immunosuppressive activity

#101
20070060584
2007-03-15

Biaryl substituted thiazoles, oxazoles and imidazoles as sodium channel blockers

#102
20070054909
2007-03-08

VLA-4 inhibitor compounds

#103
20070054897
2007-03-08

Heteroaryl-ureas and their use as glucokinase activators

#104
20070032531
2007-02-08

SPHINGOSINE KINASE INHIBITORS AND METHODS OF THEIR USE

#105
20070027147
2007-02-01

Biarylurea derivatives

#106
20070004788
2007-01-04

Nitrosated and nitrosylated Hreceptor antagonist compounds, compositions and methods of use

#107
20060276521
2006-12-07

Thiazole derivatives

#108
20060247259
2006-11-02

Nitrogen-containing aromatic derivatives

#109
20060194854
2006-08-31

New 2-substituted - 1,3-thiazole compounds

#110
20060183783
2006-08-17

Aryl carbonyl derivatives as therapeutic agents

#111
20060167247
2006-07-27

Urea inhibitors of MAP kinases

#112
20060166866
2006-07-27

Cell adhesion inhibitors

#113
20060160856
2006-07-20

Diarylurea derivatives and their use as chloride channel blockers

#114
20060160832
2006-07-20

Nitrogen-containing aromatic derivatives

#115
20060159678
2006-07-20

Modulators of cytokine mediated signaling pathways and integrin alphabeta3 receptor antagonists for combination therapy

#116
20060148862
2006-07-06

Compounds that modulate PPARγ type receptors and cosmetic/pharmaceutical compositions comprised thereof

#117
20060128770
2006-06-15

Thiazole derivatives

#118
20060100232
2006-05-11

Inhibitors of HIV-1 capsid formation: substituted aryl aminomethyl thiazole ureas and analogues thereof

#119
20060079506
2006-04-13

Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors

#120
20060074110
2006-04-06

Multicyclic compounds which inhibit leukocyte adhesion mediated by VLA-4

#121
20060069139
2006-03-30

Thiazole-based nitric oxide donors capable of releasing two or more nitric oxide molecules and uses thereof

#122
20050288186
2005-12-29

4-(3,3-dihalo-allyloxy) phenol derivatives having pesticidal properties

#123
20050250816
2005-11-10

Positive allosteric modulators of the nicotinic acetylcholine receptor

#124
20050250758
2005-11-10

Nitrosated and nitrosylated Hreceptor antagonist compounds, compositions and methods of use

#125
20050245525
2005-11-03

Urea or thiourea substituted 1,4-pyrazine compounds useful as anti-cancer agents and for inhibiting Chk1

#126
20050176719
2005-08-11

Pyrazinone derivatives

#127
20050153970
2005-07-14

N-ureidoalkyl-amino compounds as modulators of chemokine receptor activity

#128
20050131042
2005-06-16

HIV protease inhibiting compounds

#129
20050119321
2005-06-02

2-substituted-1,3-thiazole compounds

#130
20050119320
2005-06-02

5-phenylthiazole derivatives and use as Pi3 kinase inhibitors

#131
20050101642
2005-05-12

Chemical complex comprising a pyridine carboxy derivative and an H2 histamine receptor antagonist

#132
20050038035
2005-02-17

Heterocyclic amide compounds as apolipoprotein b inhibitors