Novel nitrogen-containing heteroaryl compounds and methods of use thereof

Trisubstituted aryl and heteroaryl derivatives as modulators of metabolism and the prophylaxis and treatment of disorders related thereto

5,6-trimethylenepyrimidin-4-one compounds

Substituted bis-amide metalloprotease inhibitors

Aminoindazole derivatives as medicaments and pharmaceutical compositions including them

Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents

Diamine derivatives as inhibitors of leukotriene Ahydrolase

2-phenoxy- and 2-phenylsulfonamide derivatives with CCR3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders

Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof

Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof

Pyrrolidine melanocortin-specific compounds

N-sulfonyldicarboximide containing tethering compounds

Methods of preparing a crystalline form of 7-(4-chlorobutoxy)-3,4-dihydro-2(1h)-quinolinone and the use thereof in the synthesis of Aripiprazole

Process for producing phenylacetic acid derivative

Substituted pyrrole derivatives as hmg-coa reductase inhibitors

Pyrrole derivatives, their preparation and their therapeutic use

5-aminoalkylpyrazole derivatives as pesticidal agents

5-phenylpyrimidines, their preparation, compositions comprising them and their use

Substituted arylpyrazoles

4-Anilino-quinazoline derivatives as antiproliferative agents

Imidazole compounds

Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors

Inhibitors of Akt activity

Imidazoyl-benzamide anti-cancer agents

Plant growth regulation

1-Alkyl-3-thio-substituted indole-2-alkynoic acids useful for the treatment of alzheimer's disease and related conditions

Azabicyclo (3.1.0.) hexane derivatives useful as modulators of dopamine Dreceptors

N-linked aryl heteroaryl inhibitors of LTA4H for treating inflammation

Pyrazole derivatives as inhibitors of receptor tyrosone kinases

Sulfonyl-derivatives as novel inhibitors of histone deacetylase

Piperazine-2-carboxamide derivatives

Substituted pyrazole compounds

4,5-Dihydro-(1H)-pyrazole derivatives as cannabinoid CB1 receptor modulators

Benzamide inhibitors of the P2Xreceptor

N-substituted tricyclic 1-aminopyrazoles as inhibitors for the treatment of cell proliferative disorders

Inhibitors of hepatitis C virus NS3 protease

Antibacterial compounds having a (pyrrole carboxamide)-(benzamide)-(imidazole carboxamide) motif

Prolinyl derivatives for the treatment of thrombosis

HETEROCYCLIC COMPOUNDS AND METHODS OF USE

Heterocyclic CETP inhibitors

LACTAM CONTAINING CYCLIC DIAMINES AND DERIVATIVES AS FACTOR XA INHIBITORS

Lactam-containing compounds and derivatives thereof as factor Xa inhibitors

Substituted propenyl piperazine derivatives as novel inhibitors of histone deacetylase

Short-acting benzodiazepines

Short-acting benzodiazepines

Short-acting benzodiazepines

Compositions and methods for inhibiting the proliferation of cells

Azetidine ring compounds and drugs comprising the same

Thrombopoietin activity modulating compounds and methods

Hexahydro-cyclooctyl pyrazole cannabinoid modulators

Maleate salts of a quinazoline derivative useful as an antiangiogenic agent

HIV INTEGRASE INHIBITORS

Sbstituted chroman derivatives, processes for their preparation and their use as antiinflammatory agents

Pyrimidine derivatives useful for the treatment of diseases mediated by CRTH2

Melanocortin receptor agonists

Thrombopoietin mimetics

Hexahydro-cycloheptapyrazole cannabinoid modulators

Pyrimidine compounds

4-Bromo-5-(2-chloro-benzoylamino)-1h-pyrazole-3-carboxylic acid (phenyl) amide derivatives and related compounds as bradykinin b1 receptor antagonists for the treatment of inflammatory diseases

1,1-dioxo-thiomorpholinyl indolyl methanone derivatives

N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase

Inhibitors of cathepsin S

1,5-substituted indol-2-yl amide derivatives

PYRROLO-NAPHTHYL ACIDS AND METHODS FOR USING THEM

Medical devices employing triazine compounds and compositions thereof

4-aminopyrimidine-5-thione derivatives

Pyrimidine derivatives for treatment of hyperproliferative disorders

Methods and compositions of novel triazine compounds

2-(benzimidazol-1-yl)-acetamide bisaryl derivatives

Carbocyclic fused cyclic amines

Heterocyclic compounds as pSTAT3/IL-6 inhibitors

4-Phenyl-6-substituted-pyrimidine-2-carbonitrile derivatives

Carboxamide spirohydantoin CGRP receptor antagonists

Synthesis of substituted heterocyclic compounds

Cyclohexanecarboxylic acid compound

Cyclic guanidines, compositions containing such compounds and methods of use

Indol-containing beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions

Amino substituted pyrazine derivatives for the treatment of pain

RETINOIC ACID MIMETIC ANILIDES

2, 4-Di (phenylamino) pyrimidines useful in the treatment of proliferative disorders

Inhibitors of serine proteases

Prodrugs of compounds that inhibit TRPV1 receptor

Indazolo-tetrahydropyrimidine-carboxamide derivative kinase inhibitors

Substituted pyrrolones as allosteric modulators of glucokinase

Dihydroisoindolones as allosteric modulators of glucokinase

Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4

N-(2-ARYLETHYL)BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR

1-amino-phthalazine derivatives, the preparation and the therapeutic use thereof

Methods and compositions of novel triazine compounds

Methods for the treatment of cancer

Benzamidazoles, compositions containing such compounds and methods of use

Benzimidazole carboxamides as raf kinase inhibitors

Aminoindazole derivatives as medicaments and pharmaceutical compositions including them

Short-acting benzodiazepines

1-[(4-Ethynylphenyl)]-2-[(phenyl)]-pyrrolidine-1,2-dicarboxamide derivatives as inhibitors of coagulation factors Xa and VIIa for the treatment of thrombosis

Acyl indoles, compositions containing such compounds and methods of use

Novel amidine compounds for treating microbial infections

N-[4-(heteroarylmethyl)phenyl]-heteroarylamines

INDOLINONES AND THEIR USE AS ANTIPROLIFERATIVE AGENTS

Quinazoline derivatives as antitumor agents

Fluorinated 4-azasteroid derivatives as androgen receptor modulators

CB1 antagonist compounds

Dihydroxypyrimidine carboxamide inhibitors of HIV integrase

Quinazoline derivatives as antitumor agents

Pyrrole compounds for the treatment of prostaglandine mediated diseases

Benzotriazepine derivatives and their use as gastrin and cholecystokinin receptor ligands

BIARYL SUBSTITUTED HETEROCYCLE INHIBITORS OF LTA4H FOR TREATING INFLAMMATION

Substituted heteroaryl CB1 antagonists

Heterocyclic sulfonamides as modulators of cardiac sarcomeres

Enzyme modulators and treatments

4-Substituted Pyrazoline Compounds, their Preparation and Use as Medicaments

Androgen modulators

2-(3,4-dimethylphenyl)-4-{[2-hydroxy-3′-(1h-tetrazol-5-yl)biphenyl-3-yl]-hydrazono}-5-methyl-2,4-dihydropyrazol-3-one choline

PPAR active compounds

Quinolin-isoquinolin-and quinazolin-oxyalkylamides and their use as fungicides

Bis-aryl amide compounds and methods of use

Apoptosis promoters

Benzimidazole derivatives compositions containing them, preparation thereof and uses thereof

Heterocyclic aspartyl protease inhibitors

Selected CGRP antagonists, processes for preparing them and their use as pharmaceutical compositions

Biaryl substituted heterocycle inhibitors of LTA4H for treating inflammation

Benzimidazoles

Quinazoline compounds

Imidazole compounds for the treatment of neurological disorders

Aniline derivatives

ARYL PHENYLHETEROCYCLYL SULFIDE DERIVATIVES AND THEIR USE AS CELL ADHESION-INHIBITING ANTI-INFLAMMATORY AND IMMUNE-SUPPRESSIVE AGENTS

Pyrrole and pyrazole derivatives as potentiators of glutamate receptors

Imidazole derivatives, their preparation and their use as medicaments

Large conductance calcium-activated k channel opener

Acid secretion inhibitor

Methods for treating, preventing and managing chronic lymphocytic leukemia with indazole compounds

Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds

Chemokine receptor binding heterocyclic compounds

Inhibitors of protein arginine methyl transferases

Acyltryptophanols

Sulfopyrroles

Indolyl derivatives which are L-CPT1 inhibitors

Benzazepine derivatives as histamine h3 antagonists

3-Azabicyclo[3.1.0]hexane derivatives

c-Met modulators and methods of use

Aryl nitrogen-containing bicyclic compounds and methods of use

Use of GALR3 receptor antagonists for the treatment of depression and/or anxiety and compounds useful in such methods

Azinyl-3-sulfonylindazole derivatives as 5-hydroxytryptamine-6 ligands

2-Phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents

Bis-aryl urea compounds and methods of use

Amino-tetrazoles analogues and methods of use

Compounds as inhibitors of hepatitis C virus NS3 serine protease

Diaminopyrimidines as P2Xand P2Xmodulators

Amide derivatives

Methods and compositions of novel triazine compounds

Sirtuin modulating compounds

Compositions of novel opioid compounds and method of use thereof

Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use

Phenyl pyrrolidine ether tachykinin receptor antagonists

1,3 Disubstituted azetidine derivatives for use as ccr-3 receptor antagonists in the treatment of inflammatory and allergic diseases

Quinazoline derivatives

Inhibitors of P2X

PROCESS FOR DESILYLATION OF CARBAPENEM INTERMEDIATES

Sirtuin modulating compounds

Substituted imidazole compounds as KSP inhibitors

MCH receptor antagonists

Azinone and diazinone V3 inhibitors for depression and stress disorders

Substituted piperazines as metabotropic glutamate receptor antagonists

Anti-inflammatory medicaments

Benzimidazole derivatives

Substituted-3-sulfonylindazole derivatives as 5-hydroxytryptamine-6 ligands

Fluoro substituted 2-oxo-azepan derivatives

Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use

Inhibitors of cancer cell, T-cell and keratinocyte proliferation

Therapeutic applications of pro-apoptotic benzodiazepines

Imidazolyl derivatives

Cyclic derivatives as modulators of chemokine receptor activity

Nitric oxide enhancing angiotensin II antagonist compounds, compositions and methods of use

Cyclic derivatives as modulators of chemokine receptor activity

Diphenylmethyl compounds useful as muscarinic receptor antagonists

2,4-diamino-pyrimidines as aurora inhibitors

Quinazoline derivatives

Quinazoline derivatives useful in cancer treatment

Fused-ring compounds and use thereof as drugs

Thyroid hormone analogs

Cytokine inhibitors

Kinase inhibitors

Novel compounds useful for bradykinin B1 receptor antagonism

Compounds as inhibitors of hepatitis C virus NS3 serine protease

Triazine derivatives as universal peptide isotope tag reagents (U-PIT)

Quinoline derivatives and quinazoline derivatives

Novel ligands and methods for preparing same

Indol-3-y-carbonyl-piperidin and piperazin-derivatives

High affinity small molecule C5a receptor modulators

2-Amino-quinazolin-5-ones

N-heteroaryl indole carboxamides and analogues thereof, for use as glucokinase activators in the treatment of diabetes

Heterocyclic compounds which inhibit leukocyte adhesion mediated by αintegrins

Transition-state Inhibitors of Pin1, alpha-Ketoamide-containing peptidomimetics, and synthesis thereof

Compounds, methods, complexes, apparatuses and uses relating to stabile forms of NAD/NADH

(4-phenylpiperazin-1-yl)acylpiperidine derivatives, preparation thereof and application of same in therapeutics

1,5,7-trisubstituted benzimidazole derivatives and their use for modulating the GABAreceptor complex

Substituted triazole compounds

Pyrazole derivatives and use thereof as orexin receptor antagonists

Aminobenzimidazole derivatives

Pyrimidine derivatives for the prevention of hiv infection

Substituted pyrazoline compounds, their preparation and use as medicaments

Azole derivatives and fused bicyclic azole derivatives as therapeutic agents

Histone deacetylase inhibitors

Apoptosis promoters

Quinazoline derivatives useful in cancer treatment

Substituted benzylamino quinolines as cholesterol ester-transfer protein inhibitors

Pyrimidineamines as angiogenesis modulators

Indol kinase inhibitors

Benzimidazolone and dihydroindolone derivatives and uses thereof

Quinazoline derivatives as antitumor agents

Methods and apparatus for treating back pain

Optically active 3,3'-dithiobis(2-amino-2methylpropionic acid) derivative and process for producing optically active 2-amino-3-mercapto-2-methylpropionic acid derivative

Pyrimidine compounds

Pyrrole substituted 2-indolinone protein kinase inhibitors

Indole derivatives for use as chemical uncoupler

Fused pyramidine derivative and use thereof

Cycloamine ccr5 receptor antagonists

3,6-disubstituted azabicyclo [3.1.0] hexane derivatives useful as muscarinic receptor antagonists

Nitrogen-containing aromatic derivatives

Indoline derivatives substituted in the 6-position, their preparation and their use as medicaments

Methods and compositions of novel triazine compounds

Hydroxypyridinone derivatives, metal complexes thereof and the use thereof for preparing conjugates with biomolecules

5-Chloro-4-alkyl-3,4-dihydro-quinazolin-2-ylamine derivatives

Sulfonylquinoxalone derivatives and related compounds as bradykinin antagonists

Pyrimidine compounds

Phenylpiperazines

Compositions and methods for inhibition of the JAK pathway

Indole, azaindole and related heterocyclic pyrrolidine derivatives

Diarylmethyl and related compounds

Substituted arylpyrazoles

Melanocortin receptor-specific piperazine and keto-piperazine compounds

Melanocortin receptor-specific piperazine compounds with diamine groups

Substituted melanocortin receptor-specific single acyl piperazine compounds

Pyrazinedicarboxamides and their use

Mitotic kinesin inhibitors

Heterocyclylakylamines as muscarinic receptor antagonists

Benzofuran compounds

Aadenosine receptor antagonists

Resolution of enantiomeric mixtures of beta-lactams

Pyrimidine derivatives for the treatment of abnormal cell growth

4-bromo-5-(2-chloro-benzoylamino)-1H-pyrazole-3-carboxylic acid amide derivatives and related compounds as bradykinin Breceptor antagonists for the treatment of inflammatory diseases

Pyrimidine compounds

IL-12 modulatory compounds

Novel carboxylic acid derivatives, their preparation and use

2,5-Dioxoimidazolidin-4-yl acetamides and analogues as inhibitors of metalloproteinase MMP12

Tripeptidyl peptidase inhibitors

N-heterocyclic inhibitors of TNF-α expression

Compounds useful for DPP-IV enzyme inhibition

Carboxylic acid derivatives that inhibit the binding of integrins to their receptors

Carboxylic acid derivatives, their preparation and use

Urea derivatives and their use as vanilloid receptor antagonists in the treatment of pain

Dipeptidyl peptidase-IV inhibitors

Chemical compounds

Anti-cancer agents and uses thereof

Hydrazono-malonitriles

Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them

Methods of synthesizing 6-alkylaminoquinoline derivatives

Quinoxaline derivatives as neutrophil elastase inhibitors and their use

Substituted pyrimidines useful as protein kinase inhibitors

N-substituted heterocyclic sulfonamides

Ring-substituted diphenylazetidinones, process for their preparation, medicaments comprising these compounds, and their use

Heterocyclic hydrazones as novel anti-cancer agents

INHIBITORS OF FACTOR Xa AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION CASCADE

Indole acetic acid derivatives and their use as pharmaceutical agents

P38 inhibitors and methods of use thereof

Pyrazole derivative

Substituted pyrazoles

Hepatitis C inhibitor peptide analogs

Compounds for the treatment of inflammatory diseases

N-substituted hydroxypyrimidinone carboxamide inhibitors of HIV integrase

1,5-Disubstituted imidazolidin-2-one derivatives for use as ep4 receptor agonists in the treatment of eye and bone diseases

Neurotherapeutic azole compounds

Indole derivatives

Triazole compounds useful as protein kinase inhibitors

Apoptosis promoters

Methods and compositions of novel triazine compounds

Chemical process

Androgen modulators

Substituted benzimidazoles and imidazo-[4,5]-pyridines

Compounds for the treatment of inflammatory disorders

HIV inhibiting pyrimidines derivatives

Cinnoline compounds

Substituted 4,5-dihydro-1,2,4-triazin-6-ones, 1,2,4-triazin-6-ones, and their use as fungicides

Imino acid derivatives as inhibitors of matrix metalloproteinases

N-(4-(imidazo[1,2A]pyridin-YL)phenethyl)benzamide inhibitors of the mitotic kinesin CENP-E for treating certain cellular proliferation diseases

Substituted heterocyclic compounds and methods of use

2,4 Di (hetero) -arylamino-pyrimidine derivatives as ZAP-70 and/or syk inhibitors

Quinoxalinones and their use especially in the treatment of cardiovascular diseases

Pesticidal compositions

Melanocortin receptor ligands

Vanilloid receptor ligands and their use in treatments

Nitrogen-containing 5-membered ring compound

Triazole compounds and the therapeutic use thereof

Heteroaryloxy-substituted phenylaminopyrimidines as rho-kinase inhibitors

Pyrimidinone derivatives and their use in the treatment of atherosclerosis

Substituted piperazines as CB1 antagonists

Compounds and methods of use

Pesticidal 1-aryl-3-amidoxime-pyrazole derivatives

Benzamide modulators of metabotropic glutamate receptors

Vanilloid receptor ligands and their use in treatments