ClassID:

95252

C07D403/12 - page 3 - CPC Classification

Classification description:

Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links

Recent Application in this class:
#601
20240132470
2024-04-25

Antibacterial Compounds

#602
20240132464
2024-04-25

HETEROCYCLIC COMPOUNDS AS E3 LIGASE INHIBITORS

#603
20240124466
2024-04-18

COMPOUNDS AND USE THEREOF FOR TREATMENT OF NEURODEGENERATIVE, DEGENERATIVE AND METABOLIC DISORDERS

#604
20240124449
2024-04-18

Compounds and methods for inhibiting fascin

#605
20240124448
2024-04-18

TYK2 inhibitors and compositions and methods thereof

#606
20240124426
2024-04-18

Polo like kinase 4 inhibitors

#607
20240124425
2024-04-18

Solid state forms of Belumosudil and Belumosudil salts

#608
20240122951
2024-04-18

METHOD TO TREAT LIPID DYSREGULATION BY MODULATING ACTIVITY OF PROPROTEIN CONVERTASE SUBTILISIN/KEXIN TYPE 9 (PCSK9) PROTEIN WITH SMALL MOLECULE LIGANDS

#609
20240122936
2024-04-18

Method of synthesizing thyroid hormone analogs and polymorphs thereof

#610
20240116926
2024-04-11

HETEROAROMATIC COMPOUNDS

#611
20240116902
2024-04-11

ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4

#612
20240116898
2024-04-11

NOVEL GLUTAMINYL CYCLASE INHIBITORS AND THE USE THEREOF IN TREATMENT OF VARIOUS DISEASES

#613
20240116897
2024-04-11

BENZOTHIAZOLE AND BENZIMIDAZOLE DERIVATIVES, PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT

#614
20240116894
2024-04-11

PROTEASOME ACTIVITY ENHANCING COMPOUNDS

#615
20240116878
2024-04-11

2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-METHYL PYRAZINES AS ALLOSTERIC SHP2 INHIBITORS

#616
20240116877
2024-04-11

KIT KINASE INHIBITORS AND METHODS OF USE THEREOF

#617
20240116871
2024-04-11

MATERIALS FOR ORGANIC ELECTROLUMINESCENT DEVICES

#618
20240114908
2024-04-11

2,6-DIOXO-3,6-DIHYDROPYRIMIDINE COMPOUND, AGRICULTURAL AND HORTICULTURAL BACTERICIDE, NEMATICIDE, AND MEDICAL AND VETERINARY ANTIFUNGAL AGENT

#619
20240109905
2024-04-04

4-ALKOXY-6-OXO-PYRIDAZINE DERIVATIVES MODULATING NLRP3

#620
20240109896
2024-04-04

FGFR KINASE INHIBITOR AND USE THEREOF

#621
20240109871
2024-04-04

Anti-viral compounds

#622
20240109870
2024-04-04

COVALENT IMMUNE RECRUITER COMPOUNDS FOR IMMUNE CELL RECOGNITION AND ASSOCIATED USES

#623
20240109862
2024-04-04

SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH

#624
20240109842
2024-04-04

ACRYLAMIDE COMPOUNDS

#625
20240103005
2024-03-28

N-ACRYLOYLINDOLES AND METHODS OF USE

#626
20240101532
2024-03-28

Heteroaryl carboxamide compound

#627
20240100199
2024-03-28

COMPOSITIONS, METHODS, AND SYSTEMS FOR THE SYNTHESIS AND USE OF IMAGING AGENTS

#628
20240092788
2024-03-21

MASP-2 INHIBITORS AND METHODS OF USE

#629
20240092773
2024-03-21

DIHYDRO-CYCLOPENTA-ISOQUINOLINE SULFONAMIDES DERIVATIVES

#630
20240092770
2024-03-21

Heterocycle RMB39 Modulators

#631
20240092766
2024-03-21

MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS

#632
20240092763
2024-03-21

ISOINDOLINONE AMINOPYRIMIDINE COMPOUNDS AS INHIBITORS OF NUAK KINASES, COMPOSITIONS AND USES THEREOF

#633
20240092757
2024-03-21

HETEROARYL DIAMIDE IRE1/XBP1s ACTIVATORS

#634
20240092755
2024-03-21

Spiroheptanyl hydantoins as ROCK inhibitors

#635
20240092745
2024-03-21

DRUGS AND COMPOSITIONS FOR THE TREATMENT OF OCULAR DISORDERS

#636
20240083882
2024-03-14

Benzethers and anilines of pyrazolyl-amino-pyrimidinyl derivatives, and compositions and methods thereof

#637
20240083881
2024-03-14

Benzamides of pyrazolyl-amino-pyrimidinyl derivatives, and compositions and methods thereof

#638
20240083872
2024-03-14

CYCLIC AMINE DERIVATIVES HAVING SEROTONIN RECEPTOR BINDING ACTIVITY

#639
20240083871
2024-03-14

DIPHENYLPYRAZOLE COMPOUND, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#640
20240083860
2024-03-14

AROMATIC COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#641
20240083857
2024-03-14

2-Methyl-Quinazolines

#642
20240083854
2024-03-14

TEAD INHIBITORS AND USES THEREOF

#643
20240083847
2024-03-14

SULFONAMIDE DERIVATIVES FOR PROTEIN DEGRADATION

#644
20240076291
2024-03-07

MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS

#645
20240076287
2024-03-07

SOLID FORMS OF A CDK2 INHIBITOR

#646
20240067639
2024-02-29

SMALL MOLECULES THAT TARGET THE RNA THAT CAUSES ALS

#647
20240067631
2024-02-29

PYRAZOLE DERIVATIVES USEFUL AS NAMPT MODULATORS

#648
20240067615
2024-02-29

HERBICIDAL TETRAZOLE COMPOUNDS

#649
20240067610
2024-02-29

Inhibitors of NLRP3 inflammasome

#650
20240065096
2024-02-22

COMPOSITION FOR ORGANIC OPTOELECTRONIC DEVICE, ORGANIC OPTOELECTRONIC DEVICE, AND DISPLAY DEVICE

#651
20240059688
2024-02-22

CONOLIDINE ANALOGUES AS SELECTIVE ACKR3 MODULATORS FOR THE TREATMENT OF CANCER

#652
20240059682
2024-02-22

THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS

#653
20240059678
2024-02-22

Synthesis Method for Aminopyrimidine FAK Inhibitor Compound

#654
20240059677
2024-02-22

SUBSTITUTED PYRIMIDINE DERIVATIVES AS NICOTINIC ACETYLCHOLINESTERASE RECEPTOR ALPHA 6 MODULATOR

#655
20240059659
2024-02-22

INHIBITORS OF NLRP3 INFLAMMASOME

#656
20240059647
2024-02-22

Linkers for antibody drug conjugates

#657
20240051970
2024-02-15

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#658
20240051952
2024-02-15

HMOX1 inducers

#659
20240051945
2024-02-15

PYRIMIDINE COMPOUNDS, COMPOSITIONS, AND MEDICINAL APPLICATIONS THEREOF

#660
20240051923
2024-02-15

INHIBITORS OF NLRP3 INFLAMMASOME

#661
20240043417
2024-02-08

COMPOUNDS FOR THE TREATMENT OF SARS

#662
20240043408
2024-02-08

CRYSTAL FORM OF FIBROBLAST GROWTH FACTOR RECEPTOR INHIBITOR AND PREPARATION METHOD THEREFOR

#663
20240043404
2024-02-08

APOPTOSIS INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES

#664
20240043403
2024-02-08

HETEROARYL CARBOXAMIDE COMPOUND

#665
20240043371
2024-02-08

NOVEL SPIROFLUORENE COMPOUND AND ORGANIC LIGHTEMITTING DEVICE INCLUDING SAME

#666
20240042052
2024-02-08

PROCESS FOR THE PREPARATION OF DRUG LINKER COMPOUNDS

#667
20240034733
2024-02-01

KRAS G12D INHIBITORS

#668
20240034726
2024-02-01

MAP KINASE KINASE (MKK7) INHIBITORS AND USES THEREOF

#669
20240032541
2024-02-01

HERBICIDAL COMPOUNDS

#670
20240025892
2024-01-25

SALT INDUCIBLE KINASE INHIBITORS

#671
20240025890
2024-01-25

HEPATITIS B CORE PROTEIN MODULATORS

#672
20240025883
2024-01-25

PYRIMIDIN-2-YL SULFONAMIDE DERIVATIVES

#673
20240025882
2024-01-25

Benzamides of pyrazolylamino-pyrimidinyl derivatives, and compositions and methods thereof

#674
20240025881
2024-01-25

Belumosudil metabolites and uses thereof in the treatment of chronic graft-versus-host disease

#675
20240025880
2024-01-25

AMINO QUINAZOLINE DERIVATIVES AS P2X3 INHIBITORS

#676
20240025875
2024-01-25

A COMPOUND AS A THYROID HORMONE BETA RECEPTOR AGONIST AND USE THEREOF

#677
20240025862
2024-01-25

SUBSTITUTED N-PHENYLURACILS AND SALTS THEREOF, AND USE THEREOF AS HERBICIDAL ACTIVE SUBSTANCES

#678
20240025849
2024-01-25

INHIBITORS OF NO PRODUCTION

#679
20240018130
2024-01-18

Pyrimidine Derivative, Method For Preparing Same And Use Thereof In Medicine

#680
20240018126
2024-01-18

ANTI-VIRAL COMPOUNDS

#681
20240018125
2024-01-18

CYCLIC ISOTHIOUREA DERIVATIVES AS CXCR4 MODULATORS

#682
20240010657
2024-01-11

BIOTIN DERIVATIVES

#683
20240010634
2024-01-11

PYRIMIDINYL SULFONAMIDES AS INHIBITORS OF ACK1/TNK2 TYROSINE KINASE

#684
20240002388
2024-01-04

PYRIMIDINONE COMPOUNDS AND USES THEREOF

#685
20240002371
2024-01-04

PHTHALAZINE DERIVATIVES AS P2X3 INHIBITORS

#686
20240002369
2024-01-04

NOVEL TREATMENTS OF ATTENTION DEFICIT/HYPERACTIVITY DISORDER

#687
20240002368
2024-01-04

STING ANTAGONISTS AND USES THEREOF

#688
20240002361
2024-01-04

COMPOSITIONS AND METHODS FOR BLOCKING NEUROPILIN RECEPTOR 1 FOR THE TREATMENT OF PAIN AND PREVENTION OF VIRAL ENTRY

#689
20240002351
2024-01-04

QUINAZOLIN-4-ONE AND THIENO[2,3-D]PYRIMIDIN-4-ONE INHIBITORS OF ERBB4 (HER4) FOR USE IN THE TREATMENT OF CANCER

#690
20240002350
2024-01-04

PROTEIN AND LIPID THERAPEUTIC TARGETS

#691
20240002339
2024-01-04

THERAPEUTIC COMPOUNDS AND METHODS

#692
20240000964
2024-01-04

COMPOUND OR SALT THEREOF, AND ANTIBODY OBTAINED BY USING THE SAME

#693
20240000790
2024-01-04

THERAPEUTIC COMPOSITIONS, COMBINATIONS, AND METHODS OF USE

#694
20230416263
2023-12-28

CARM1 INHIBITORS AND USES THEREOF

#695
20230416262
2023-12-28

TRPML MODULATORS

#696
20230416239
2023-12-28

COMPOUNDS AND METHODS FOR TREATING A CYTOKINE-MEDIATED DISEASE

#697
20230416236
2023-12-28

INHIBITING ATAXIA TELANGIECTASIA AND RAD3-RELATED PROTEIN (ATR)

#698
20230416235
2023-12-28

Benzamides of pyrazolylamino-pyrimidinyl derivatives, and compositions and methods thereof

#699
20230416234
2023-12-28

CRYSTAL FORM OF RESMETIROM, PREPARATION METHOD THEREFOR, AND USE THEREOF

#700
20230416233
2023-12-28

(AZA)QUINOLINE 4-AMINES DERIVATIVES AS P2X3 INHIBITORS

#701
20230416232
2023-12-28

PYRIMIDINE COMPOUNDS, COMPOSITIONS, AND MEDICINAL APPLICATIONS THEREOF

#702
20230416225
2023-12-28

DIAMINOPYRIMIDINE CARBOXAMIDE INHIBITORS OF HPK1

#703
20230407285
2023-12-21

PCSK9 INHIBITORS AND METHODS OF USE THEREOF

#704
20230406845
2023-12-21

Potassium channel inhibitors

#705
20230406838
2023-12-21

MUTANT SELECTIVE EGFR INHIBITORS AND METHODS OF USE THEREOF

#706
20230406822
2023-12-21

SILICON COMPOUND AND METHOD OF MANUFACTURING INTEGRATED CIRCUIT DEVICE USING THE SAME

#707
20230399320
2023-12-14

NOVEL CAPSID ASSEMBLY INHIBITOR

#708
20230399316
2023-12-14

CRYSTAL FORMS OF 5-FLUORO-1-(4-FLUORO-3-(4-(PYRIMIDIN-2-YL)PIPERAZINE-1-CARBONYL)BENZYL)QUINAZOLINE-2,4(1H,3H)-DIONE AND PREPARATION THEREOF

#709
20230391757
2023-12-07

Crystalline forms of a 4-pyrimidinesulfamide derivative aprocitentan

#710
20230391756
2023-12-07

NEW COMPOUND

#711
20230391755
2023-12-07

Solid state forms of Belumosudil and Belumosudil salts

#712
20230391754
2023-12-07

CRYSTALLINE FORM OF SELINEXOR

#713
20230391753
2023-12-07

THIOBENZIMIDAZOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND USE THEREOF

#714
20230391751
2023-12-07

SUBSTITUTED 1,2,4-TRIAZOLES AS INTERMEDIATES IN THE SYNTHESIS OF TYK2 INHIBITORS

#715
20230391730
2023-12-07

INHIBITORS OF THE BROMODOMAIN PHD FINGER TRANSCRIPTION FACTOR (BPTF) AS ANTI-CANCER AGENTS

#716
20230390242
2023-12-07

PYRROLE COMPOUNDS

#717
20230382857
2023-11-30

HEPTAMETHINE CYANINES FOR USE AS FLUORESCENT MARKERS OF THE BILIARY AND RENAL SYSTEMS

#718
20230374024
2023-11-23

Compounds for the treatment of kinase-dependent disorders

#719
20230373974
2023-11-23

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR

#720
20230373935
2023-11-23

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR

#721
20230373930
2023-11-23

AMINOIMIDAZOLE FPR2 AGONISTS

#722
20230372297
2023-11-23

MEDICAMENTS FOR THE TREATMENT OR PREVENTION OF FIBROTIC DISEASES

#723
20230365534
2023-11-16

MODULATORS OF NLRP3 INFLAMMASOME AND RELATED PRODUCTS AND METHODS

#724
20230365533
2023-11-16

BICYCLOHEPTANE PYRROLIDINE OREXIN RECEPTOR AGONISTS

#725
20230365524
2023-11-16

2,4,5-TRISUBSTITUTED 1,2,4-TRIAZOLONES USEFUL AS INHIBITORS OF DHODH

#726
20230365509
2023-11-16

BENZO[H]QUINAZOLIN-4-AMINE AND THIENO[3,2-H]QUINAZOLIN-4-AMINE DERIVATIVES FOR THE TREATMENT OF CANCER

#727
20230365507
2023-11-16

INHIBITORS OF NLRP3 INFLAMMASOME

#728
20230357261
2023-11-09

ARYL HYDROCARBON RECEPTOR LIGANDS AND THEIR ANALOGUES FOR THE PREVENTION AND TREATMENT OF INFLAMMATORY DISORDERS

#729
20230357259
2023-11-09

BIOACTIVE CONJUGATE, PREPARATION METHOD THEREFOR AND USE THEREOF

#730
20230357218
2023-11-09

N-FORMAMIDOPYRAZOLINE DERIVATIVE AS P2X3 RECEPTOR ANTAGONIST AND USE THEREOF

#731
20230357208
2023-11-09

MYST FAMILY HISTONE ACETYLTRANSFERASE INHIBITORS

#732
20230357188
2023-11-09

PHENANTHRENE ORGANIC COMPOUND AND USE THEREOF

#733
20230357185
2023-11-09

C4-carboxylic acid-substituted tryptamine derivatives and methods of using

#734
20230357179
2023-11-09

RAF KINASE INHIBITORS AND METHODS OF USE THEREOF

#735
20230357162
2023-11-09

COMPOUNDS, COMPOSITIONS AND METHODS

#736
20230357145
2023-11-09

C4-carboxylic acid-substituted tryptamine derivatives and methods of using

#737
20230354812
2023-11-09

3-(PYRIDAZIN-4-YL)-5,6-DIHYDRO-4H-1,2,4-OXADIAZINE DERIVATIVES AS FUNGICIDES FOR CROP PROTECTION

#738
20230348501
2023-11-02

Heteroaryl inhibitors of PDE4

#739
20230348438
2023-11-02

PYRAZOLE COMPOUND AND PHARMACEUTICAL USE THEREOF

#740
20230348437
2023-11-02

COMPOUNDS, COMPOSITIONS AND METHODS

#741
20230348436
2023-11-02

COMPOUNDS FOR TREATING TUBERCULOSIS

#742
20230348401
2023-11-02

Inhibitors of Glucose-6-phosphate Dehydrogenase and Uses Thereof

#743
20230348369
2023-11-02

NAMPT MODULATORS

#744
20230346748
2023-11-02

PHARMACEUTICAL COMBINATION, COMPOSITION AND COMPOUND PREPARATION CONTAINING GLUCOKINASE ACTIVATOR AND K-ATP CHANNEL BLOCKER, PREPARATION METHOD THEREFOR AND USE THEREOF

#745
20230339960
2023-10-26

Bicyclic-fused heteroaryl or aryl compounds

#746
20230339911
2023-10-26

PYRIDAZINONE COMPOUNDS

#747
20230339910
2023-10-26

RAS INHIBITORS AND METHODS OF USING THE SAME

#748
20230339886
2023-10-26

REV-ERB AGONISTS FOR THE TREATMENT OF TH17-MEDIATED INFLAMMATORY DISORDERS

#749
20230339866
2023-10-26

Quinazoline compounds and the use thereof in the treatment of cancer

#750
20230339865
2023-10-26

QUINAZOLINE-DERIVED HCK INHIBITORS FOR USE IN THE TREATMENT OF MYD88 MUTATED DISEASES

#751
20230338376
2023-10-26

AMINOPYRIMIDINE AMIDE AUTOPHAGY INHIBITORS AND METHODS OF USE THEREOF

#752
20230331707
2023-10-19

PROGRAMMED CELL NECROSIS INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF

#753
20230331705
2023-10-19

Fused Imidazole Derivatives as AHR Antagonists

#754
20230329106
2023-10-12

ORGANIC LIGHT EMITTING ELEMENT

#755
20230322738
2023-10-12

Prodrug of pyrrolidone derivatives as glucokinase activator

#756
20230322737
2023-10-12

Stable salt and crystal forms of 2-[3-({1-[2-(dimethylamino)ethyl]-2-(2,2-dimethylpropyl)-1H-1,3-benzodiazol-5-yl}sulfonyl)azetidin-1-yl]ethan-1-ol

#757
20230322732
2023-10-12

RIP1 Inhibitory Compounds and Methods for Making and Using the Same

#758
20230322726
2023-10-12

QUINAZOLINES AS POTASSIUM ION CHANNEL INHIBITORS

#759
20230322672
2023-10-12

COMPOUNDS AND FORMULATIONS FOR TREATING OPHTHALMIC DISEASES

#760
20230322668
2023-10-12

Protease inhibitors as antivirals

#761
20230322667
2023-10-12

DIHYDROFOLATE SYNTHASE (DHFS) INHIBITING AGENTS AND METHODS OF MAKING AND USING SAME

#762
20230321040
2023-10-12

C-carbonothioate-substituted tryptamine derivatives and methods of using

#763
20230312571
2023-10-05

Ring-modified proline short peptide compound and use thereof

#764
20230312567
2023-10-05

Capsid inhibitors for the treatment of HIV

#765
20230312539
2023-10-05

METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION

#766
20230312536
2023-10-05

3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF

#767
20230312529
2023-10-05

Pyrimidine small-molecule compound and application thereof

#768
20230312528
2023-10-05

2-OXO-IMIDAZOLIDINE-4-CARBOXAMIDES AS NAV1.8 INHIBITORS

#769
20230312527
2023-10-05

CYANOTRIAZINE DERIVATIVE, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#770
20230312525
2023-10-05

AZIRIDINYL FUNCTIONAL COMPOUND

#771
20230312483
2023-10-05

Amino Pyrimidine Derivatives

#772
20230312481
2023-10-05

SUBSTITUTED (PHTHALAZIN-1-YLMETHYL)UREAS, SUBSTITUTED N-(PHTHALAZIN-1-YLMETHYL)AMIDES, AND ANALOGUES THEREOF

#773
20230312466
2023-10-05

NOVEL COMPOUNDS

#774
20230310428
2023-10-05

EGFR INHIBITOR AND PREPARATION METHOD AND USE THEREOF

#775
20230310423
2023-10-05

CHECKPOINT KINASE 1 (CHK1) INHIBITORS AND USES THEREOF

#776
20230310373
2023-10-05

METHODS FOR TREATING PULMONARY EMPHYSEMA USING SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C

#777
20230303566
2023-09-28

Inhibtors of Raf kinases

#778
20230303544
2023-09-28

LMO2 PROTEIN INHIBITORS

#779
20230303540
2023-09-28

2-AMINOQUINAZOLINES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF

#780
20230303531
2023-09-28

5-MEMBERED AZA-HETEROCYCLIC CONTAINING DELTA-OPIOID RECEPTOR MODULATING COMPOUNDS, METHODS OF USING AND MAKING THE SAME

#781
20230303530
2023-09-28

Compounds as nuclear transport modulators and uses thereof

#782
20230303522
2023-09-28

ARYLTETRAHYDROPYRIDAZINE DERIVATIVE OR SALT THEREOF, INSECTICIDAL AGENT CONTAINING THE COMPOUND, AND METHOD OF USE THEREOF

#783
20230303502
2023-09-28

HETEROARYL AND HETEROCYCLYL COMPOUNDS

#784
20230303499
2023-09-28

INHIBITORS OF ACK1/TNK2 TYROSINE KINASE

#785
20230295145
2023-09-21

PYRROLIDINE DERIVATIVES AND METHODS OF USE

#786
20230295129
2023-09-21

INHIBITORS OF ACK1/TNK2 TYROSINE KINASE

#787
20230295087
2023-09-21

AGONISTS OF ROR GAMMAt

#788
20230293535
2023-09-21

ErbB/BTK inhibitors

#789
20230286957
2023-09-14

HERBICIDAL COMPOUNDS

#790
20230286948
2023-09-14

HALOALKYLPYRIDYL TRIAZOLE MLL1-WDR5 PROTEIN-PROTEIN INTERACTION INHIBITOR

#791
20230286942
2023-09-14

NEW PqsR INVERSE AGONISTS

#792
20230286925
2023-09-14

PHENYL TRIAZOLE MLL1-WDR5 PROTEIN-PROTEIN INTERACTION INHIBITOR

#793
20230286923
2023-09-14

QUINAZOLINONE HSD17B13 INHIBITORS AND USES THEREOF

#794
20230286913
2023-09-14

INHIBITORS OF NITRIC OXIDE SYNTHASES (NOS), PHARMACEUTICAL PRODUCTS THEREOF, AND METHODS THEREOF

#795
20230279020
2023-09-07

Carm1 inhibitors and uses thereof

#796
20230278994
2023-09-07

HETEROCYCLYL PYRIMIDINES AND TRIAZINES AS NOVEL FUNGICIDES

#797
20230278988
2023-09-07

THRB RECEPTOR AGONIST COMPOUND AND PREPARATION METHOD AND USE THEREOF

#798
20230278987
2023-09-07

Antimicrobial Compounds and Methods

#799
20230278958
2023-09-07

TRICYCLIC HETEROCYCLES

#800
20230277547
2023-09-07

Substituted quinoxalines and benzo[c][1,2,5]oxadiazoles as DNA-PK inhibitors

#801
20230271983
2023-08-31

FUNCTIONALIZED ISONITRILES AND PRODUCTS, PREPARATION AND USES THEREOF

#802
20230271975
2023-08-31

Imidazole-containing inhibitors of ALK2 kinase

#803
20230271951
2023-08-31

DIFLUOROCYCLOHEXYL DERIVATIVES AS IL-17 MODULATORS

#804
20230271946
2023-08-31

PROCESS FOR THE PREPARATION OF 6-(CYCLOPROPANEAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE

#805
20230271945
2023-08-31

Inhibitors of APOL1 and methods of using same

#806
20230271941
2023-08-31

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#807
20230271936
2023-08-31

EFGR INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#808
20230271926
2023-08-31

INHIBITION OF OLIG2 ACTIVITY

#809
20230265098
2023-08-24

ALKYNE QUINAZOLINE DERIVATIVES AS INHIBITORS OF ERBB2

#810
20230265085
2023-08-24

RET kinase inhibitors

#811
20230257367
2023-08-17

NOVEL THYROID HORMONE BETA RECEPTOR AGONIST

#812
20230257354
2023-08-17

NOVEL HETEROCYCLIC COMPOUNDS

#813
20230257352
2023-08-17

RAF kinase inhibitors and methods of use thereof

#814
20230257349
2023-08-17

SUBSTITUTED (1,2,3,4-TETRAHYDROCYCLOPENTA[b]INDOL-3-YL)ACETIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS

#815
20230250106
2023-08-10

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#816
20230250104
2023-08-10

Diamine derivatives as inhibitors of leukotriene Ahydrolase

#817
20230250089
2023-08-10

MAP4K3 SMALL MOLECULE DRUG INHIBITORS AND METHODS OF USE THEREOF

#818
20230250088
2023-08-10

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#819
20230250087
2023-08-10

SOLID FORMS OF APOL1 INHIBITOR AND METHODS OF USING SAME

#820
20230250086
2023-08-10

METHIONINE METABOLIC PATHWAY INHIBITORS

#821
20230250079
2023-08-10

SMALL MOLECULE MODULATORS OF IL-17

#822
20230250062
2023-08-10

Substituted Heterocyclyl Derivatives as CDK Inhibitors

#823
20230250060
2023-08-10

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#824
20230248841
2023-08-10

REVERSIBLE LINKERS AND USE THEREOF

#825
20230242544
2023-08-03

QUINAZOLINE COMPOUNDS, PREPARATION METHODS AND USES THEREOF

#826
20230242529
2023-08-03

Heterocyclic compound

#827
20230242523
2023-08-03

Compound, tautomer of compound or salt of compound or tautomer, method for producing same, coloring composition, dyeing method, and dyed article

#828
20230242518
2023-08-03

ORGANIC ELECTROLUMINESCENT COMPOUND AND ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING THE SAME

#829
20230242517
2023-08-03

Polymorphs of selinexor

#830
20230242516
2023-08-03

Polymorphs of Selinexor

#831
20230242515
2023-08-03

Crystalline form of 6-(cyclopropanecarboxamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-n-(methyl-D3) pyridazine-3-carboxamide

#832
20230242507
2023-08-03

INDAZOLE-FUSED CYCLIC COMPOUND

#833
20230234943
2023-07-27

TREX1 INHIBITORS AND USES THEREOF

#834
20230234935
2023-07-27

KINASE INHIBITOR COMPOUNDS AND COMPOSITIONS AND METHODS OF USE

#835
20230233560
2023-07-27

Modulators of cystic fibrosis transmembrane conductance regulator

#836
20230227695
2023-07-20

COMPOUND, CMP SLURRY COMPOSITION INCLUDING THE SAME AND POLISHING METHOD USING THE SAME

#837
20230227484
2023-07-20

PYRIMIDINE COMPOUND AS AXL INHIBITOR

#838
20230227447
2023-07-20

BENZYLAMINE DERIVATIVES AS DDRS INHIBITORS

#839
20230227439
2023-07-20

SPAK/OSR INHIBITORS AND METHODS OF USING SAME

#840
20230227436
2023-07-20

Compounds, compositions, and methods

#841
20230227435
2023-07-20

SMALL MOLECULE MODULATORS OF IL-17

#842
20230227429
2023-07-20

SULPHONAMIDE COMPOUNDS

#843
20230227428
2023-07-20

AMIDO COMPOUNDS

#844
20230227427
2023-07-20

IL-17A MODULATORS

#845
20230219986
2023-07-13

NOVEL AMINOPYRIMIDINE EGFR INHIBITOR

#846
20230219904
2023-07-13

HERBICIDAL COMPOUNDS

#847
20230219897
2023-07-13

Pyrazole MAGL inhibitors

#848
20230219896
2023-07-13

Cannabinoid receptor mediating compounds

#849
20230218612
2023-07-13

NITROGEN-CONTAINING HETEROCYCLIC COMPOUND HAVING INHIBITORY EFFECT ON PRODUCTION OF KYNURENINE

#850
20230218578
2023-07-13

BENZOPYRAZOLE COMPOUNDS AND ANALOGUES THEREOF

#851
20230212186
2023-07-06

Cyano cyclobutyl compounds for Cbl-b inhibition and uses thereof

#852
20230212157
2023-07-06

PYRAZOLE DERIVATIVES FOR THE TREATMENT OF CYSTIC FIBROSIS

#853
20230212153
2023-07-06

Lactams as CBL-B inhibitors selective over C-CBL

#854
20230212152
2023-07-06

INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF

#855
20230212147
2023-07-06

ALKENYL PYRIMIDINE COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#856
20230212143
2023-07-06

PRMT5 INHIBITOR COMPOUNDS

#857
20230212142
2023-07-06

Substituted 5-Cyclopropyl-1H-pyrazole-3-yl-amine Derivatives as Selective CDK12/13 Inhibitors

#858
20230212116
2023-07-06

SARS-COV-2 MAIN PROTEASE INHIBITORS

#859
20230203016
2023-06-29

DICARBOXYLIC ACID BISAMIDE DERIVATIVES, USE THEREOF, PHARMACEUTICAL COMPOSITION BASED THEREON AND METHODS FOR PRODUCING DICARBOXYLIC ACID BISAMIDE DERIVATIVES

#860
20230203015
2023-06-29

MAP KINASE KINASE (MKK7) INHIBITORS AND USES THEREOF

#861
20230203005
2023-06-29

COMPOUNDS WITH TUBULIN POLYMERISATION INHIBITORY ACTIVITY AND IMMUNOMODULATORY PROPERTIES

#862
20230203002
2023-06-29

6-MEMBERED AZA-HETEROCYCLIC CONTAINING DELTA-OPIOID RECEPTOR MODULATING COMPOUNDS, METHODS OF USING AND MAKING THE SAME

#863
20230202989
2023-06-29

COMPOUNDS

#864
20230202985
2023-06-29

Indoles, Indazoles, and Related Analogs for Inhibiting YAP/TAZ-TEAD

#865
20230202983
2023-06-29

CANNABINOID RECEPTOR MEDIATING COMPOUNDS

#866
20230201200
2023-06-29

Methods for Treating Huntington’s Disease

#867
20230193057
2023-06-22

WATERBORNE CROSSLINKER COMPOSITION

#868
20230192683
2023-06-22

FUSED RING COMPOUNDS, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF

#869
20230192677
2023-06-22

CYP11A1 INHIBITORS

#870
20230192673
2023-06-22

Compounds

#871
20230192663
2023-06-22

INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF

#872
20230192662
2023-06-22

Receptor-Interacting Protein 1 Inhibitors Including Piperazine Heterocyclic Amide Ureas

#873
20230192661
2023-06-22

1, 4, 5, 6-TETRAHYDROPYRIMIDINE-2-AMINE DERIVATIVE

#874
20230192660
2023-06-22

Protease Inhibitors for Treatment or Prevention of Coronavirus Disease

#875
20230192659
2023-06-22

N-(HETEROCYCLYL AND HETEROCYCLYLALKYL)-3-BENZYLPYRIDIN-2-AMINE DERIVATIVES AS SSTR4 AGONISTS

#876
20230192645
2023-06-22

INDOLE CARBOXAMIDE COMPOUNDS

#877
20230192628
2023-06-22

MICROBIOCIDAL DERIVATIVES

#878
20230192626
2023-06-22

NOVEL SOLUBLE EPOXIDE HYDROLASE INHIBITORS AND METHOD OF USE THEREOF

#879
20230192617
2023-06-22

AZABICYCLIC(THIO)AMIDES AS FUNGICIDAL COMPOUNDS

#880
20230189638
2023-06-15

Organic compound and electronic device and electronic apparatus thereof

#881
20230183219
2023-06-15

CONDENSED SUBSTITUTED HYDROPYRROLES AS ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4

#882
20230183218
2023-06-15

CONDENSED SUBSTITUTED HYDROPYRROLES AS ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4

#883
20230183217
2023-06-15

Inhibitors of LRRK2 kinase

#884
20230183216
2023-06-15

PYRIDIZIN-3(2H)-ONE DERIVATIVES

#885
20230183215
2023-06-15

Notch Inhibitors and Uses Thereof

#886
20230183197
2023-06-15

INHIBITORS OF MLH1 AND/OR PMS2 FOR CANCER TREATMENT

#887
20230183184
2023-06-15

3-(Carboxyethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives

#888
20230180757
2023-06-15

SUBSTITUTED ISOPHTHALIC ACID DIAMIDES AND THEIR USE AS HERBICIDES

#889
20230180756
2023-06-15

TRIAZINE AND PYRIMIDINE (THIO)AMIDES AS FUNGICIDAL COMPOUNDS

#890
20230174540
2023-06-08

3-(Carboxymethyl)-8-Amino-2-Oxo-1,3-Diaza-Spiro-[4.5]-Decane Derivatives

#891
20230174518
2023-06-08

KRAS G12D PROTEIN INHIBITORS

#892
20230174517
2023-06-08

METHOD FOR THE PREPARATION OF ANDROGEN RECEPTOR ANTAGONISTS AND INTERMEDIATES THEREOF

#893
20230174515
2023-06-08

Apoptosis signal-regulating kinase 1 inhibitors and methods of use thereof

#894
20230174488
2023-06-08

SARS-COV-2 INHIBITORS HAVING COVALENT MODIFICATIONS FOR TREATING CORONAVIRUS INFECTIONS

#895
20230174485
2023-06-08

LIPOXYGENASE INHIBITORS

#896
20230167092
2023-06-01

SUBSTITUTED N-(METHYL-D3)PYRIDAZINE-3-CARBOXAMIDE OR N-(METHYL-D3)-NICOTINAMIDE COMPOUNDS AS IL-12, IL-23 AND/OR IFNALPHA MODULATORS

#897
20230167091
2023-06-01

Substituted pyridazinone compound and use thereof

#898
20230167090
2023-06-01

SOLID STATE FORMS OF APROCITENTAN AND PROCESS FOR PREPARATION THEREOF

#899
20230167082
2023-06-01

PRODRUGS IN THE MODULATION OF INTERLEUKIN

#900
20230167073
2023-06-01

ARYL OR HETEROARYL DERIVATIVE