ClassID:

95252

C07D403/12 - page 4 - CPC Classification

Classification description:

Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links

Recent Application in this class:
#901
20230167057
2023-06-01

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#902
20230165860
2023-06-01

PYRIMIDINEDIONE COMPOUNDS

#903
20230165859
2023-06-01

N-SUBSTITUTED INDOLE DERIVATIVES

#904
20230165857
2023-06-01

AXL KINASE INHIBITORS AND USE OF THE SAME

#905
20230165848
2023-06-01

CHEMICAL COMPOUNDS

#906
20230159520
2023-05-25

TYK-2 INHIBITOR

#907
20230159508
2023-05-25

INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATMENT OF DISEASE

#908
20230159502
2023-05-25

INDOLE DERIVATIVES AS ALPHA-1-ANTITRYPSIN MODULATORS FOR TREATING ALPHA-1-ANTITRYPSIN DEFICIENCY (AATD)

#909
20230159491
2023-05-25

Antimicrobial Compounds and Methods

#910
20230159469
2023-05-25

NOVEL PHTHALAZINE DERIVATIVE HAVING ECTONUCLOEOTIDE PYROPHOSPHATASE/PHOSPHODIESTE RASE INHIBITORY ACTIVITY, AND USE THEREOF

#911
20230159465
2023-05-25

IMMUNOMODULATOR

#912
20230159453
2023-05-25

INHIBITORS OF NOROVIRUS AND CORONAVIRUS REPLICATION

#913
20230151018
2023-05-18

Inhibitors of protein arginine deiminases

#914
20230150991
2023-05-18

Substituted benzyl-triazole compounds for Cbl-b inhibition, and further uses thereof

#915
20230150986
2023-05-18

ANTAGONISTS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4

#916
20230150981
2023-05-18

N-HETEROARYLALKYL-2-(HETEROCYCLYL AND HETEROCYCLYLMETHYL) ACETAMIDE DERIVATIVES AS SSTR4 AGONISTS

#917
20230150980
2023-05-18

COLLAGEN 1 TRANSLATION INHIBITORS AND METHODS OF USE THEREOF

#918
20230150979
2023-05-18

AMIDE-DISUBSTITUTED PYRIDINE OR PYRIDAZINE COMPOUNDS

#919
20230150972
2023-05-18

PYRIDINYL DERIVATIVES AS SODIUM CHANNEL ACTIVATORS

#920
20230150948
2023-05-18

Aurora kinase and janus kinase inhibitors for prevention of graft versus host disease

#921
20230150947
2023-05-18

PYRIMIDINE-2,4-DIAMINE COMPOUND AND PREPAREATION METHOD AND APPLICATION THEREOF

#922
20230147603
2023-05-11

Host-targeted pan-respiratory antiviral small molecule therapeutics

#923
20230147507
2023-05-11

Indoline compounds for inhibiting KIF18A

#924
20230147428
2023-05-11

BENZIMIDAZOLONE-BASED CINNAMAMIDE DERIVATIVE AS TRPV1 ANTAGONIST AND PHARMACEUTICAL COMPOSITION FOR TREATMENT OR PREVENTION OF PAIN CONTAINING SAME AS ACTIVE INGREDIENT

#925
20230145481
2023-05-11

SUBSTITUTED BENZENECARBOXAMIDES AS IL-17A MODULATORS

#926
20230145071
2023-05-11

MASP-2 inhibitors and methods of use

#927
20230145050
2023-05-11

Sulphonyl urea derivatives as NLRP3 inflammasome modulators

#928
20230143532
2023-05-11

Apoptosis inducing agents for the treatment of cancer and immune and autoimmune diseases

#929
20230142910
2023-05-11

LANTHIONINE SYNTHETASE C-LIKE 2-BASED THERAPEUTICS

#930
20230142839
2023-05-11

N4-phenyl-quinazoline-4-amine derivatives and related compounds as ErbB type I receptor tyrosine kinase inhibitors for the treatment of hyperproliferative diseases

#931
20230142654
2023-05-11

NOVEL COMPOUND, PREPARATION METHOD THEREOF, AND USE THEREOF

#932
20230142274
2023-05-11

SUBSTITUTED ARYL COMPOUND

#933
20230142119
2023-05-11

TETRACYCLIC COMPOUND

#934
20230141212
2023-05-11

SUBSTITUTED BENZENECARBOXAMIDES AS IL-17A MODULATORS

#935
20230140764
2023-05-04

AZIRIDINE FUNCTIONAL COMPOUND

#936
20230140216
2023-05-04

COMBINATION THERAPY FOR TREATING MPS1

#937
20230140210
2023-05-04

Inhibitors of platelet function and methods for use of the same

#938
20230138310
2023-05-04

PHARMACEUTICAL USE OF ALDEHYDE-BASED COMPOUND

#939
20230138225
2023-05-04

PYRAZOLE CARBOXYLATE ESTER COMPOUND AND USE THEREOF

#940
20230137585
2023-05-04

6-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING DISEASES AND CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY

#941
20230136495
2023-05-04

Multi-aziridine compound

#942
20230134821
2023-05-04

Myc-Max inhibitor compound therapeutics for cancer treatment, methods and uses associated therewith

#943
20230133581
2023-05-04

Novel 3,5-Diaminobenzoic Acid Compound, and PIN1 Inhibitor and Therapeutic Agent for Inflammatory Diseases Using Same

#944
20230133465
2023-05-04

Compositions and methods for treating and preventing neurodegenerative disorders

#945
20230131830
2023-04-27

PYRIMIDINE COMPOUNDS AND THEIR PHARMACEUTICAL USES

#946
20230128765
2023-04-27

Small Molecule Activators of Parkin Enzyme Function

#947
20230127839
2023-04-27

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#948
20230127655
2023-04-27

MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS

#949
20230127229
2023-04-27

Multi-aziridine compound

#950
20230127046
2023-04-27

G9a INHIBITOR

#951
20230126280
2023-04-27

Hydantoin containing deoxyuridine triphosphatase inhibitors

#952
20230126252
2023-04-27

Fused pyrrolines which act as ubiquitin-specific protease 30 (USP30) inhibitors

#953
20230124361
2023-04-20

SMALL MOLECULE STING ANTAGONISTS

#954
20230122912
2023-04-20

Methods and compositions of 4-substituted benzoylpiperazine-1-substituted carbonyls as β-catenin/B-cell lymphoma 9 inhibitors

#955
20230122028
2023-04-20

COATING COMPOSITION

#956
20230122024
2023-04-20

OX2R compounds

#957
20230121818
2023-04-20

BTK INHIBITORS

#958
20230121721
2023-04-20

MONOACYLGLYCEROL LIPASE INHIBITORS

#959
20230121497
2023-04-20

COMPOUNDS AND USES THEREOF

#960
20230121086
2023-04-20

RORgT INHIBITOR, PREPARATION METHOD THEREOF AND USE THEREOF

#961
20230120254
2023-04-20

Nitrile-Containing Antiviral Compounds

#962
20230119665
2023-04-20

Cardiac sarcomere inhibitors

#963
20230119479
2023-04-20

A HISTONE DEACETYLASE INHIBITOR HAVING A NITROGEN-CONTAINING AROMATIC HETEROCYCLYL GROUP

#964
20230119149
2023-04-20

Method and apparatus for sorting heterogeneous material

#965
20230117592
2023-04-20

LIPOXYGENASE INHIBITORS

#966
20230117295
2023-04-20

NITROGEN CONTAINING HETEROCYCLES AS CDK12 INHIBITORS

#967
20230117059
2023-04-20

Solid state forms of Belumosudil and Belumosudil salts

#968
20230116770
2023-04-13

Small molecule activators of nicotinamide phosphoribosyltransferase (NAMPT) and uses thereof

#969
20230116686
2023-04-13

THERAPEUTIC COMPOUNDS AND USES THEREOF

#970
20230116201
2023-04-13

COLLAGEN 1 TRANSLATION INHIBITORS AND METHODS OF USE THEREOF

#971
20230116093
2023-04-13

Substituted diaminocarboxamide and diaminocarbonitrile pyrimidines, compositions thereof, and methods of treatment therewith

#972
20230115865
2023-04-13

Novel Substituted 6,7-Dihydro-5H-Benzo[7]Annulene Compounds, Processes for Their Preparation and Therapeutic Uses Thereof

#973
20230115335
2023-04-13

Pyrazole derivatives with anticancer activity

#974
20230115275
2023-04-13

Amide compounds and method for making and using

#975
20230115176
2023-04-13

Complement Modulators and Related Methods

#976
20230113598
2023-04-13

HETEROCYCLIC COMPOUNDS USEFUL AS PDK1 INHIBITORS

#977
20230113588
2023-04-13

METABOTROPIC GLUTAMATE RECEPTOR NEGATIVE ALLOSTERIC MODULATORS (NAMS) AND USES THEREOF

#978
20230112865
2023-04-13

RIP1 INHIBITORY COMPOUNDS AND METHODS FOR MAKING AND USING THE SAME

#979
20230111252
2023-04-13

THIOSEMICARBAZATES AND USES THEREOF

#980
20230111132
2023-04-13

STABILIZATION OF MHC COMPLEXES

#981
20230110928
2023-04-13

Methods and compositions useful in treating cancer and reducing Wnt mediated effects in a cell

#982
20230109670
2023-04-06

Substituted bicyclic compounds as farnesoid X receptor modulators

#983
20230109505
2023-04-06

SMALL MOLECULE INHIBITORS OF SCL15A4 WITH ANTI-INFLAMMATORY ACTIVITY

#984
20230109134
2023-04-06

PYRIDAZINONE OR PYRIDAZINE COMPOUND AND DERIVATIVE AND PHARMACEUTICAL COMPOSITION THEREOF

#985
20230107941
2023-04-06

HEPATITIS B CAPSID ASSEMBLY MODULATORS

#986
20230106420
2023-04-06

ARYL-N-ARYL DERIVATIVES FOR TREATING A RNA VIRUS INFECTION

#987
20230104740
2023-04-06

Inhibitors of glycogen synthase 1 (GYS1) and methods of use thereof

#988
20230104283
2023-04-06

JNK INHIBITOR, AND PHARMACEUTICAL COMPOSITION AND USE THEREOF

#989
20230101819
2023-03-30

SMYD Inhibitors

#990
20230100975
2023-03-30

DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 ANTAGONISTS

#991
20230100634
2023-03-30

MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS

#992
20230100082
2023-03-30

Human plasma kallikrein inhibitors

#993
20230098888
2023-03-30

DRG-MDM2-6 FOR USE AS A NOVEL MOUSE DOUBLE MINUTE 2 (MDM2) INHIBITOR

#994
20230098031
2023-03-30

METHODS FOR CELL IMAGING

#995
20230097964
2023-03-30

1,2-diaminobenzimidazole derivative

#996
20230097706
2023-03-30

MULTI-AZIRIDINE COMPOUND

#997
20230097700
2023-03-30

AZETIDINE SULFONAMIDE COMPOUND

#998
20230096600
2023-03-30

WATERBORNE CROSSLINKER COMPOSITION

#999
20230096380
2023-03-30

COMPOUNDS, COMPOSITIONS, METHODS FOR TREATING DISEASES AND NERVE DAMAGE, AND METHODS FOR PREPARING COMPOUNDS

#1000
20230095835
2023-03-30

2,4-DIAMINO-PYRIMIDINE COMPOUNDS AND METHOD FOR MAKING AND USING THE COMPOUNDS

#1001
20230094305
2023-03-30

Human plasma kallikrein inhibitors

#1002
20230093302
2023-03-23

A NOVEL MAO-B INHIBITOR DRG-MAOB-1 FOR USE IN TREATMENT OF NEURODEGENERATIVE DISEASES

#1003
20230093249
2023-03-23

Anti-viral compounds

#1004
20230092892
2023-03-23

AMINO QUINAZOLINE DERIVATIVES AS P2X3 INHIBITORS

#1005
20230092163
2023-03-23

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#1006
20230091225
2023-03-23

Bifunctional chimeric heterocyclic compounds for targeted degradation of androgen receptors and use thereof

#1007
20230090742
2023-03-23

AMINOPYRIMIDINYLAMINOBENZONITRILE DERIVATIVES AS NEK2 INHIBITORS

#1008
20230089582
2023-03-23

1,2,4-TRIAZINE-3,5-DIONE COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#1009
20230089374
2023-03-23

GLYCOLATE OXIDASE INHIBITORS FOR THE TREATMENT OF DISEASE

#1010
20230088611
2023-03-23

A NOVEL SELECTIVE MAO-B INHIBITOR DRG-MAOB-2 FOR USE IN TREATMENT OF NEURODEGENERATIVE DISEASES

#1011
20230088214
2023-03-23

GLYCOLATE OXIDASE INHIBITORS FOR THE TREATMENT OF DISEASE

#1012
20230086064
2023-03-23

CBL-B MODULATORS AND USES THEREOF

#1013
20230084752
2023-03-16

ACSS2 INHIBITORS AND METHODS OF USE THEREOF

#1014
20230080054
2023-03-16

INHIBITORS OF ANOCTAMIN 6 PROTEIN AND USES THEREOF

#1015
20230079913
2023-03-16

GLYCOLATE OXIDASE INHIBITORS FOR THE TREATMENT OF DISEASE

#1016
20230077268
2023-03-09

INDAZOLES AND AZAINDAZOLES AS LRRK2 INHIBITORS

#1017
20230076435
2023-03-09

MODIFIER OF FOUR-MEMBERED RING DERIVATIVE, PREPARATION METHOD AND APPLICATION THEREOF

#1018
20230075198
2023-03-09

Substituted indoles and methods of use thereof

#1019
20230074669
2023-03-09

Cycloalkane-1,3-diamine derivative

#1020
20230071340
2023-03-09

DRG-MDM2-4 FOR USE AS A NOVEL MOUSE DOUBLE MINUTE 2 (MDM2) INHIBITOR

#1021
20230069886
2023-03-09

AROMATIC SULPHONAMIDES DERIVATIVES THAT INHIBITS PDI A3, THEIR SYNTHESIS AND USE

#1022
20230069357
2023-03-02

TWO-COMPONENT COATING SYSTEM

#1023
20230063230
2023-03-02

NURR1 RECEPTOR MODULATORS

#1024
20230062975
2023-03-02

HEPATITIS B CAPSID ASSEMBLY MODULATORS

#1025
20230061118
2023-03-02

NEW FYN AND VEGFR2 KINASE INHIBITORS

#1026
20230060011
2023-02-23

Antibacterial compounds

#1027
20230060004
2023-02-23

Diacylglycerol kinase modulating compounds

#1028
20230057341
2023-02-23

HETEROCYCLIC RIP1 KINASE INHIBITORS

#1029
20230056538
2023-02-23

Human plasma kallikrein inhibitors

#1030
20230056202
2023-02-23

Anti-malarial agents

#1031
20230056135
2023-02-23

MONOMER AND MULTIMERIC ANTI-HBV AGENTS

#1032
20230054883
2023-02-23

MTA-Cooperative PRMT5 Inhibitors

#1033
20230054196
2023-02-23

MULTI-AZIRIDINE COMPOUND

#1034
20230054028
2023-02-23

PD-L1 ANTAGONIST COMPOUND

#1035
20230053746
2023-02-23

IL-17 ligands and uses thereof

#1036
20230052528
2023-02-16

TASPASE1 INHIBITORS AND USES THEREOF

#1037
20230052191
2023-02-16

Compounds

#1038
20230051130
2023-02-16

Inhibitors of NLRP3 inflammasome

#1039
20230049402
2023-02-16

NOVEL PHENOL COMPOUND OR SALT THEREOF

#1040
20230049130
2023-02-16

DEUCRAVACITINIB CRYSTAL FORM, PREPARATION METHOD THEREFOR AND USE THEREOF

#1041
20230047905
2023-02-16

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#1042
20230044941
2023-02-09

TRIARYL COMPOUNDS FOR TREATMENT OF PD-L1 DISEASES

#1043
20230044112
2023-02-09

Hepatitis b core protein modulators

#1044
20230043970
2023-02-09

Certain chemical entities, compositions, and methods

#1045
20230043400
2023-02-09

Compounds, Compositions and Methods

#1046
20230043159
2023-02-09

MATRIPTASE 2 INHIBITORS AND USES THEREOF

#1047
20230043136
2023-02-09

Quinazoline Compounds

#1048
20230041761
2023-02-09

SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF

#1049
20230041576
2023-02-09

METHODS AND MATERIALS FOR INHIBITING NF-kB ACTIVITY

#1050
20230039836
2023-02-09

AROMATIC SULPHONAMIDES DERIVATIVES THAT INHIBITS PDI A3, THEIR SYNTHESIS AND USE

#1051
20230039586
2023-02-09

Bicyclic compounds as androgen receptor modulators

#1052
20230039309
2023-02-09

Substituted indole Mcl-1 inhibitors

#1053
20230039086
2023-02-09

BMS-986165 CRYSTAL FORM, PREPARATION METHOD THEREFOR AND USE THEREOF

#1054
20230038823
2023-02-09

Capsid inhibitors for the treatment of HIV

#1055
20230037883
2023-02-09

Alkene-containing amide compound and application thereof

#1056
20230033285
2023-02-02

Protease Inhibitors for Treatment of Coronavirus Infections

#1057
20230032612
2023-02-02

Quaternary indazole glucocorticoid receptor antagonists

#1058
20230031213
2023-02-02

Methods and compositions for targeting PD-L1

#1059
20230030720
2023-02-02

CYCLOALKANE-1,3-DIAMINE DERIVATIVE

#1060
20230030414
2023-02-02

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

#1061
20230028700
2023-01-26

CHIRAL GUANIDINES, SALTS THEREOF, METHODS OF MAKING CHIRAL GUANIDINES AND SALTS THEREOF, AND USES OF CHIRAL GUANIDINES AND SALTS THEREOF IN THE PREPARATION OF ENANTIOMERICALLY PURE AMINO ACIDS

#1062
20230027985
2023-01-26

SUBSTITUTED HYDANTOINAMIDES AS ADAMTS7 ANTAGONISTS

#1063
20230027929
2023-01-26

MrgprX2 Antagonists and Uses Thereof

#1064
20230027716
2023-01-26

NOVEL PYRIDINYLTRIAZINE DERIVATIVE HAVING PROTEIN KINASE INHIBITORY ACTIVITY, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING, AMELIORATING, OR TREATING CANCER COMPRISING SAME

#1065
20230027295
2023-01-26

FXIA INHIBITORS AND PREPARATION METHOD THEREFOR AND PHARMACEUTICAL USE THEREOF

#1066
20230027055
2023-01-26

HIV inhibitor compounds

#1067
20230026696
2023-01-26

TRPV4 RECEPTOR LIGANDS

#1068
20230026611
2023-01-26

ARYL HETEROCYCLIC COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS

#1069
20230026438
2023-01-26

Protease inhibitors as antivirals

#1070
20230026348
2023-01-26

NITROXYLATED PROTEINS AND METHODS FOR THE USE THEREOF

#1071
20230026313
2023-01-26

Checkpoint kinase 1 (CHK1) inhibitors and uses thereof

#1072
20230025656
2023-01-26

TRIARYLAMINE DERIVATIVE AND ORGANIC ELECTROLUMINESCENT DEVICE THEREOF

#1073
20230025025
2023-01-26

Substituted pyrazole amides

#1074
20230024438
2023-01-26

INHIBITORS OF HIF-2ALPHA

#1075
20230024240
2023-01-26

Heteroaryl inhibitors of PDE4

#1076
20230024012
2023-01-26

Protease inhibitors for treatment of coronavirus infections

#1077
20230023761
2023-01-26

Substituted pyridazines as TYK2 inhibitors

#1078
20230023066
2023-01-26

N-(HETEROARYL) QUINAZOLIN-2-AMINE DERIVATIVES AS LRRK2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF

#1079
20230022304
2023-01-26

WDR5-MYC INHIBITORS

#1080
20230021916
2023-01-26

Modulators of Rho-associated protein kinase

#1081
20230021834
2023-01-26

Piperidinyl-3-(aryloxy)propanamides and propanoates

#1082
20230021705
2023-01-26

GLP-1R MODULATING COMPOUNDS

#1083
20230021554
2023-01-26

Substituted 1,2,4-triazoles as intermediates in the synthesis of TYK2 inhibitors

#1084
20230021448
2023-01-26

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#1085
20230021177
2023-01-19

1,2,4-triazine-4-amine derivatives

#1086
20230020663
2023-01-19

SULFONAMIDE INHIBITORS AS CTPS1 INHIBITORS

#1087
20230020273
2023-01-19

Amide-substituted heterocyclic compounds for the treatment of conditions related to the modulation of IL-12, IL-23 and/or IFN-alpha

#1088
20230019129
2023-01-19

HEPATITIS B CORE PROTEIN ALLOSTERIC MODULATORS

#1089
20230018702
2023-01-19

Quinazolinones as PARP14 inhibitors

#1090
20230018460
2023-01-19

1-AMINOSULFONYL-2-CARBOXYPYRROLE DERIVATIVES AS METALLO-BETA-LACTAMASE INHIBITORS

#1091
20230015617
2023-01-19

PHTHALAZINONE DERIVATIVES

#1092
20230014907
2023-01-19

INHIBITORS OF APOL1 AND METHODS OF USING SAME

#1093
20230014173
2023-01-19

Antibacterial compounds

#1094
20230013778
2023-01-19

SUBSTITUTED TRICYCLIC COMPOUNDS

#1095
20230012560
2023-01-19

HEPATITIS B ANTIVIRAL AGENTS

#1096
20230012449
2023-01-12

COMPOUNDS FOR THE TREATMENT OF HIV

#1097
20230012073
2023-01-12

Selective octahydro-cyclopenta[c]pyrrole negative modulators of NR2B

#1098
20230011118
2023-01-12

Inhibitors of APOL1 and methods of using same

#1099
20230010562
2023-01-12

4,9-dioxo-4,9-dihydronaphtho[2,3-B]furan-3-carboxamide derivatives and uses thereof for treating proliferative diseases and infectious diseases

#1100
20230010108
2023-01-12

A CONJUGATION LINKER CONTAINING 2,3-DIAMINOSUCCINYL GROUP

#1101
20230009626
2023-01-12

INDOLINONE COMPOUNDS FOR USE AS MAP4K1 INHIBITORS

#1102
20230009122
2023-01-12

3-PHOSPHOGLYCERATE DEHYDROGENASE INHIBITORS AND USES THEREOF

#1103
20230008022
2023-01-12

Substituted piperazine amide compounds as indoleamine 2,3-dioxygenase (IDO) inhibitors

#1104
20230002362
2023-01-05

BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF

#1105
20230002357
2023-01-05

7-PYRIMIDINE-2-YL-OXY-INDAZOLE DERIVATIVES AND THEIR USE AS HERBICIDES

#1106
20230002356
2023-01-05

COMPOUNDS AND USES THEREOF

#1107
20230002352
2023-01-05

SULFONAMIDE DERIVATIVES AS CTPS1 INHIBITORS

#1108
20230002345
2023-01-05

Fused ring compounds

#1109
20220411440
2022-12-29

Glycosidase inhibitors

#1110
20220411433
2022-12-29

Modulators of eukaryotic initiation factor 2B, compositions and methods

#1111
20220411431
2022-12-29

Novel compounds and their use in therapy

#1112
20220411418
2022-12-29

CDGSH iron sulfur domain 2 activators and use thereof

#1113
20220411410
2022-12-29

Modulators of ATP-binding cassette transporters

#1114
20220411408
2022-12-29

Small Molecule Compound

#1115
20220411383
2022-12-29

AMINOPYRAZINE DERIVATIVES AS PI3K-y INHIBITORS

#1116
20220409629
2022-12-29

BENZODIAZEPINE DERIVATIVES FOR TREATING A RESPIRATORY SYNCYTIAL VIRUS (RSV) INFECTION

#1117
20220409589
2022-12-29

CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY

#1118
20220409523
2022-12-29

COMPOSITIONS IN THE FORM OF AN INJECTABLE AQUEOUS SOLUTION COMPRISING AMYLIN, AN AMYLIN RECEPTOR AGONIST OR AN AMYLIN ANALOG AND A CO-POLYAMINO ACID

#1119
20220407026
2022-12-22

ORGANIC ELECTROLUMINESCENT DEVICE

#1120
20220402915
2022-12-22

BCL-2 inhibitors

#1121
20220402899
2022-12-22

COMPOUNDS FOR THE TREATMENT OF HUMAN IMMUNODEFICIENCY VIRUS

#1122
20220402896
2022-12-22

INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF

#1123
20220402895
2022-12-22

Method and System for Synthesising Compounds

#1124
20220402891
2022-12-22

TRIAZACYCLODODECANSULFONAMIDE (TCD)-BASED PROTEIN SECRETION INHIBITORS

#1125
20220402881
2022-12-22

SMALL MOLECULE PROSTAGLADIN TRANSPORT INHIBITORS

#1126
20220402879
2022-12-22

Hydantoin containing deoxyuridine triphosphatase inhibitors

#1127
20220402875
2022-12-22

S1P3 Antagonists

#1128
20220400676
2022-12-22

HERBICIDAL COMPOUNDS

#1129
20220396583
2022-12-15

COMPOUNDS AS MODULATORS OF TLR2 SIGNALING

#1130
20220396573
2022-12-15

Pyrimidine compound as JAK kinase inhibitor

#1131
20220396565
2022-12-15

NOVEL HETEROCYCLIC COMPOUNDS

#1132
20220395501
2022-12-15

TREATMENT OF GVHD

#1133
20220389028
2022-12-08

BAX INHIBITORS AND USES THEREOF

#1134
20220388968
2022-12-08

INHIBITORS OF ERYTHROCYTE BAND 3 TYROSINE PHOSPHORYLATION AND USES THEREOF

#1135
20220388967
2022-12-08

Phenyl Amino Pyrimidine Compounds and Uses Thereof

#1136
20220388964
2022-12-08

(AZA)INDAZOLYL-ARYL SULFONAMIDE AND RELATED COMPOUNDS AND THEIR USE IN TREATING MEDICAL CONDITIONS

#1137
20220388957
2022-12-08

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#1138
20220387428
2022-12-08

1,4-DISUBSTITUTED PYRIDAZINE ANALOGS THERE OF AND METHODS FOR TREATING SMN-DEFICIENCY-RELATED CONDITIONS

#1139
20220387395
2022-12-08

UREA, AMIDE, AND SUBSTITUTED HETEROARYL COMPOUNDS FOR CBL-B INHIBITION

#1140
20220380378
2022-12-01

ANDROGEN RECEPTOR MODULATORS AND METHODS FOR THEIR USE

#1141
20220380349
2022-12-01

PHARMACEUTICAL COMPOUNDS

#1142
20220380348
2022-12-01

AXL INHIBITOR FORMULATIONS

#1143
20220380347
2022-12-01

INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF

#1144
20220380322
2022-12-01

P2X4 receptor antagonist

#1145
20220380319
2022-12-01

SUBSTITUTED BENZIMIDAZOLE CARBOXAMIDES AND THEIR USE IN THE TREATMENT OF MEDICAL DISORDERS

#1146
20220378745
2022-12-01

CHK1/2 INHIBITORS FOR USE IN THE TREATMENT OF NEUROBLASTOMAS AND/OR SOFT TISSUE SARCOMAS

#1147
20220378744
2022-12-01

COMPOUNDS FOR TREATING PROLIFERATOR-ACTIVATED RECEPTORS (PPAR) MEDIATED DISEASES OR CONDITIONS

#1148
20220372038
2022-11-24

Heterocyclic compounds and uses thereof

#1149
20220372022
2022-11-24

COMPOUNDS FOR USE IN SYNTHESIS OF PEPTIDOMIMETICS

#1150
20220372021
2022-11-24

RESMETIROM CRYSTAL, PREPARATION METHOD FOR SAME, AND USES THEREOF

#1151
20220372005
2022-11-24

Cycloolefin substituted heteroaromatic compounds and their use

#1152
20220370469
2022-11-24

Theramutein modulators

#1153
20220363667
2022-11-17

T-TYPE CALCIUM CHANNEL BLOCKER

#1154
20220363648
2022-11-17

Glucose uptake inhibitors

#1155
20220363645
2022-11-17

Beta-amino acid derivative, kinase inhibitor and pharmaceutical composition containing the same, and method for performing an in vivo related application that benefits from the inhibition of a kinase

#1156
20220363639
2022-11-17

Small molecules that sensitize HIV-1 infected cells to antibody dependent cellular cytotoxicity

#1157
20220362257
2022-11-17

Theramutein modulators

#1158
20220356182
2022-11-10

INHIBITORS OF HEPATITIS C VIRUS REPLICATION

#1159
20220356181
2022-11-10

3,5-DISUBSTITUTED PYRAZOLE COMPOUNDS AS KINASE INHIBITORS AND USES THEREOF

#1160
20220356180
2022-11-10

AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFN ALPHA RESPONSES

#1161
20220356179
2022-11-10

5-membered and bicyclic heterocyclic amides as inhibitors of ROCK

#1162
20220356176
2022-11-10

Kv11.1-3.1 INHIBITING METHODS AND COMPOSITIONS

#1163
20220356175
2022-11-10

Aryl-n-aryl derivatives for treating a RNA virus infection

#1164
20220356171
2022-11-10

ISOINDOLINE DERIVATIVES

#1165
20220356167
2022-11-10

Apoptosis signal-regulating kinase 1 inhibitors and methods of use thereof

#1166
20220356148
2022-11-10

ANTIVIRAL COMPOUNDS

#1167
20220354864
2022-11-10

Substituted quinazolines for inhibiting kinase activity

#1168
20220348588
2022-11-03

7-membered aza-heterocyclic containing delta-opioid receptor modulating compounds, methods of using and making the same

#1169
20220348587
2022-11-03

Benzoimidazole Derivatives As Anticancer Agents

#1170
20220348561
2022-11-03

THYROID HORMONE RECEPTOR BETA AGONIST COMPOUNDS

#1171
20220348560
2022-11-03

N-(1H-IMIDAZOL-2-YL)BENZAMIDE COMPOUND AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME AS ACTIVE INGREDIENT

#1172
20220348559
2022-11-03

Bicyclic lactams and methods of use thereof

#1173
20220340553
2022-10-27

2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE

#1174
20220340546
2022-10-27

INHIBITORS OF SARM1

#1175
20220340523
2022-10-27

Inhibitors of APOL1 and methods of using same

#1176
20220334031
2022-10-20

REVERSIBLE FIXING REAGENTS AND METHODS OF USE THEREOF

#1177
20220332723
2022-10-20

Imidazole-containing inhibitors of ALK2 kinase

#1178
20220332711
2022-10-20

N2-phenylpyrimidine-2,4-diamine compounds, and preparation methods and methods of use thereof

#1179
20220332708
2022-10-20

SULFONAMIDE COMPOUNDS AS CARDIAC SARCOMERE ACTIVATORS

#1180
20220332707
2022-10-20

Halogen-substituted phenylate compound and applications thereof

#1181
20220332706
2022-10-20

CRYSTALLINE FORMS OF A JAK2 INHIBITOR

#1182
20220332705
2022-10-20

Biaryl inhibitors of Bruton's tyrosine kinase

#1183
20220332686
2022-10-20

ONIUM SALT OF NITROGEN-CONTAINING HETEROARYL COMPOUND AND PEST CONTROL AGENT

#1184
20220324851
2022-10-13

AMINE-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS EHMT2 INHIBITORS, SALTS THEREOF, AND METHODS OF SYNTHESIS THEREOF

#1185
20220324845
2022-10-13

Inhibitors of LRRK2 kinase

#1186
20220324844
2022-10-13

INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF

#1187
20220324843
2022-10-13

DICARBOXYLIC ACID BISAMIDE DERIVATIVES, USE THEREOF, PHARMACEUTICAL COMPOSITION BASED THEREON AND METHODS FOR PRODUCING DICARBOXYLIC ACID BISAMIDE DERIVATIVES

#1188
20220324842
2022-10-13

CANCER TREATMENTS TARGETING CANCER STEM CELLS

#1189
20220324836
2022-10-13

QUINAZOLINES AS POTASSIUM ION CHANNEL INHIBITORS

#1190
20220324835
2022-10-13

INHIBITORS OF CBL-B AND METHODS OF USE THEREOF

#1191
20220324812
2022-10-13

Inhibitors of NLRP3 inflammasome

#1192
20220324800
2022-10-13

SARS-3CL PROTEASE INHIBITORS

#1193
20220323460
2022-10-13

Combination pharmaceutical agents as RSV inhibitors

#1194
20220315564
2022-10-06

Methods and compounds for restoring mutant p53 function

#1195
20220315563
2022-10-06

ALK-5 inhibitors and uses thereof

#1196
20220315562
2022-10-06

Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders

#1197
20220315555
2022-10-06

APOPTOSIS INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES

#1198
20220315537
2022-10-06

MACROMOLECULE-SUPPORTED AMINOBENZAZEPINE COMPOUNDS

#1199
20220306640
2022-09-29

HYDANTOIN DERIVATIVE

#1200
20220306610
2022-09-29

COMPOUNDS USEFUL FOR TREATING GASTROINTESTINAL TRACT DISORDERS