ClassID:

95252

C07D403/12 - page 7 - CPC Classification

Classification description:

Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links

Recent Application in this class:
#1801
20200353101
2020-11-12

DNA-PK inhibitors

#1802
20200352946
2020-11-12

COMPOUNDS FOR THE PREVENTION AND TREATMENT OF CARDIOVASCULAR DISEASES

#1803
20200352941
2020-11-12

Carbazole EHop-016 derivatives as anticancer and anti-migratory agents

#1804
20200352925
2020-11-12

Amide derivatives useful in the treatment of HBV infection or HBV-induced diseases

#1805
20200347075
2020-11-05

Bioactive molecule conjugate, preparation method and use thereof

#1806
20200347068
2020-11-05

Small molecule myristate inhibitors of Bcr-abl and methods of use

#1807
20200347035
2020-11-05

Substituted pyridazinone compound

#1808
20200347034
2020-11-05

Compounds and their use for reducing uric acid levels

#1809
20200347033
2020-11-05

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#1810
20200347022
2020-11-05

Azole derivatives as apelin receptor agonist

#1811
20200347021
2020-11-05

Metabotropic glutamate receptor negative allosteric modulators (NAMs) and uses thereof

#1812
20200347012
2020-11-05

Compositions and methods for treating and preventing neurodegenerative disorders

#1813
20200347010
2020-11-05

Compounds with antimicrobial activity

#1814
20200345735
2020-11-05

HYDROXYLATED AND METHOXYLATED PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORS

#1815
20200345732
2020-11-05

1,4-disubstituted pyridazine analogs thereof and methods for treating SMN-deficiency-related conditions

#1816
20200339586
2020-10-29

Compounds and their use as inhibitors of N-myristoyl transferase

#1817
20200339570
2020-10-29

BICYCLIC DERIVATIVES

#1818
20200339554
2020-10-29

Substituted imidazoles for the treatment of cancer

#1819
20200339548
2020-10-29

PYRIMIDINE DERIVATIVES AND THEIR USE FOR THE TREATMENT OF CANCER

#1820
20200339545
2020-10-29

Compounds and their use for reducing uric acid levels

#1821
20200339537
2020-10-29

NOVEL COMPOUND AS INHIBITOR AGAINST BINDING OF PF34 PROTEIN TO NEDD4-1 PROTEIN AND USE THEREOF

#1822
20200339534
2020-10-29

BENZAMIDE DERIVATIVE COMPOUND, METHOD FOR PREPARING SAME, AND PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING INFLAMMATORY DISEASE CONTAINING SAME AS ACTIVE INGREDIENT

#1823
20200339522
2020-10-29

Phenoxymethyl derivatives

#1824
20200339521
2020-10-29

Hydrazide containing nuclear transport modulators and uses thereof

#1825
20200339518
2020-10-29

Inhibitors of protein arginine deiminases (PADs) and methods of preparation and use thereof

#1826
20200331895
2020-10-22

Optical brightener for whitening paper

#1827
20200331894
2020-10-22

D-amino acid oxidase inhibitors and therapeutic uses thereof

#1828
20200331893
2020-10-22

DIMERIC CONTRAST AGENTS

#1829
20200331890
2020-10-22

Apoptosis signal-regulating kinase 1 inhibitors and methods of use thereof

#1830
20200331872
2020-10-22

Methionine metabolic pathway inhibitors

#1831
20200331861
2020-10-22

Cannabinoid receptor mediating compounds

#1832
20200331860
2020-10-22

C-Met Modulators and Methods of Use

#1833
20200330471
2020-10-22

Therapeutic compositions, combinations, and methods of use

#1834
20200330435
2020-10-22

MEDICAMENTS FOR THE TREATMENT OR PREVENTION OF FIBROTIC DISEASES

#1835
20200325148
2020-10-15

COMPOSITIONS AND METHODS OF TREATMENT FOR NEUROLOGICAL DISORDERS COMPRISING MOTOR NEURON DISEASES

#1836
20200325126
2020-10-15

Heterocyclic amides useful as protein modulators

#1837
20200325120
2020-10-15

Quinazoline derivative or its salt and pharmaceutical composition comprising the same

#1838
20200323854
2020-10-15

Therapeutic compounds and uses thereof

#1839
20200323850
2020-10-15

Pyrimidine derivative kinase inhibitors

#1840
20200323821
2020-10-15

Pyrrole compounds

#1841
20200317700
2020-10-08

Sulfonyldiazoles and N-(fluorosulfonyl)azoles, and methods of making the same

#1842
20200317691
2020-10-08

Compounds, Compositions and Methods

#1843
20200317645
2020-10-08

Crystalline FGFR4 inhibitor compound and uses thereof

#1844
20200317644
2020-10-08

PYRAZOLE COMPOUND AND PHARMACEUTICAL USE THEREOF

#1845
20200317642
2020-10-08

AMINE-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS EHMT2 INHIBITORS AND DERIVATIVES THEREOF

#1846
20200317624
2020-10-08

BICYCLIC QUINAZOLINONE DERIVATIVES

#1847
20200317623
2020-10-08

Carboxylic acid compounds

#1848
20200316231
2020-10-08

Compositions And Methods For Imaging Immune Cells

#1849
20200316079
2020-10-08

ErbB/BTK inhibitors

#1850
20200316068
2020-10-08

Methods for Treating MS Using Pyrimidine and Pyridine Compounds with BTK Inhibitory Activity

#1851
20200308181
2020-10-01

Diamine derivatives as inhibitors of leukotriene A4 hydrolase

#1852
20200308169
2020-10-01

HETEROCYCLIC COMPOUNDS AS ANTIBACTERIALS

#1853
20200308156
2020-10-01

Biguanide derivatives and their rearrangement products for use in the treatment of cancer

#1854
20200308142
2020-10-01

Substituted pyrazole derivatives as selective CDK12/13 inhibitors

#1855
20200308109
2020-10-01

FLUORENE COMPOUND AND PHARMACEUTICAL USE THEREOF

#1856
20200306259
2020-10-01

Substituted quinazolines for inhibiting kinase activity

#1857
20200300843
2020-09-24

Clozapine Immunoassay

#1858
20200299307
2020-09-24

Androgen receptor modulating compounds

#1859
20200299285
2020-09-24

Carboxylic acid, acyl sulfonamide and acyl sulfamide-derivatized bicyclic aza-heteroaromatics as selective Mcl-1 inhibitors and as dual Mcl-1/Bcl-2 inhibitors

#1860
20200299284
2020-09-24

Sulfonylureas and related compounds and use of same

#1861
20200299276
2020-09-24

2,4-diamino-pyrimidine compounds and method for making and using the compounds

#1862
20200299275
2020-09-24

Synthesis of 2-indolinone derivatives

#1863
20200299274
2020-09-24

Organic electroluminescent compound and organic electroluminescent device comprising the same

#1864
20200299273
2020-09-24

Pyrrolidine derivative

#1865
20200299261
2020-09-24

WNT signaling pathway inhibitors for treatments of disease

#1866
20200297726
2020-09-24

PYRIMIDINEDIONE COMPOUNDS

#1867
20200297725
2020-09-24

ALLOSTERIC BCR-ABL PROTEOLYSIS TARGETING CHIMERIC COMPOUNDS

#1868
20200297721
2020-09-24

Type II raf kinase inhibitors

#1869
20200297710
2020-09-24

Chemical compounds

#1870
20200297700
2020-09-24

BICYCLIC COMPOUND, PRODUCTION AND USE THEREOF

#1871
20200291032
2020-09-17

Pyrimidine derivatives

#1872
20200291007
2020-09-17

Benzimidazole derivatives, and pharmaceutical compositions and methods of use thereof

#1873
20200291000
2020-09-17

Dopamine D3 receptor selective antagonists/partial agonists; method of making; and use thereof

#1874
20200290977
2020-09-17

Inhibitors of low molecular weight protein tyrosine phosphatase and uses thereof

#1875
20200290973
2020-09-17

Farnesoid X receptor agonists and uses thereof

#1876
20200290964
2020-09-17

Sulfonamide derivatives for protein degradation

#1877
20200289507
2020-09-17

N-substituted indole derivatives as PGE2 receptor modulators

#1878
20200288710
2020-09-17

SUBSTITUTED SULPHONAMIDES FOR CONTROLLING ANIMAL PESTS

#1879
20200283419
2020-09-10

Polymorphs of selinexor

#1880
20200283418
2020-09-10

N-(2,2-difluoroethyl)-N-[(pyrimidinylamino)propanyl]arylcarboxamides

#1881
20200283407
2020-09-10

Heteroaromatic compounds and their use as dopamine D1 ligands

#1882
20200283397
2020-09-10

KDM1A inhibitors for the treatment of disease

#1883
20200283383
2020-09-10

MEK inhibitors and methods of their use

#1884
20200277281
2020-09-03

Antibacterial compound and uses of same

#1885
20200270247
2020-08-27

Therapeutic compounds as inhibitors of the orexin-1 receptor

#1886
20200270238
2020-08-27

Pyrimidinyloxy benzene derivatives as herbicides

#1887
20200268757
2020-08-27

Compounds and their use for reducing uric acid levels

#1888
20200268730
2020-08-27

Amide derivatives useful in the treatment of HBV infection or HBV-induced diseases

#1889
20200264530
2020-08-20

Photoresponsive low-molecular weight material, adhesive, toner, and image forming method

#1890
20200262850
2020-08-20

SUBSTITUTED ASYMMETRIC UREAS AS MODULATORS OF GHRELIN RECEPTOR ACTIVITY

#1891
20200262844
2020-08-20

Substituted isoquinolines as rock kinase inhibitors

#1892
20200262838
2020-08-20

1-cyano-pyrrolidine derivatives as inhibitors of USP30

#1893
20200262836
2020-08-20

Inhibitors of hepatitis C virus replication

#1894
20200262821
2020-08-20

Process for the preparation of Pazopanib or a pharmaceutically acceptable salt thereof

#1895
20200262820
2020-08-20

Process for the preparation of pazopanib or a pharmaceutically acceptable salt thereof

#1896
20200262818
2020-08-20

Aryl, heteroaryl, and heterocyclic compounds for treatment of immune and inflammatory disorders

#1897
20200262796
2020-08-20

6-membered heterocyclic derivatives and pharmaceutical composition comprising the same

#1898
20200262793
2020-08-20

Substituted heterocyclyl derivatives as CDK inhibitors

#1899
20200261447
2020-08-20

Lanthionine synthetase C-like 2-based therapeutics

#1900
20200261421
2020-08-20

HETEROCYCLIC COMPOUNDS AS HIV PROTEASE INHIBITORS

#1901
20200261411
2020-08-20

TRPV4 antagonists

#1902
20200255409
2020-08-13

Potassium channel inhibitors

#1903
20200255407
2020-08-13

Quinazolines as potassium ion channel inhibitors

#1904
20200255403
2020-08-13

5-alkyl pyrrolidine orexin receptor agonists

#1905
20200255385
2020-08-13

Hydantoin containing deoxyuridine triphosphatase inhibitors

#1906
20200255377
2020-08-13

Carbazole derivatives

#1907
20200255375
2020-08-13

Phenylpyrrolidinone formyl peptide 2 receptor agonists

#1908
20200253995
2020-08-13

Method to treat lipid dysregulation by modulation of proprotein convertase subtilisin/kexin type 9 (PCSK9) protein activity with small molecule ligands

#1909
20200253974
2020-08-13

Quinazoline compounds as modulators of Ras signaling

#1910
20200247814
2020-08-06

Hetero-halo inhibitors of histone deacetylase

#1911
20200247796
2020-08-06

Pyrrole derivatives as PLK1 inhibitors

#1912
20200247790
2020-08-06

AMINE-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS EHMT2 INHIBITORS, SALTS THEREOF, AND METHODS OF SYNTHESIS THEREOF

#1913
20200247789
2020-08-06

ISOINDOLINONE INHIBITORS OF THE MDM2-P53 INTERACTION HAVING ANTICANCER ACTIVITY

#1914
20200247788
2020-08-06

Quinazolinones as PARP14 inhibitors

#1915
20200247785
2020-08-06

IL-17 ligands and uses thereof

#1916
20200247784
2020-08-06

CDK2 inhibitors

#1917
20200247755
2020-08-06

ETHERS, SECONDARY AMINES AND DERIVATIVES THEREOF AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#1918
20200239458
2020-07-30

Inhibitors of protein kinases

#1919
20200239452
2020-07-30

IDO/TDO inhibitor

#1920
20200239451
2020-07-30

Substituted pyrazole-pyrimidines, variants thereof, and uses therefore

#1921
20200239450
2020-07-30

Crystal forms of an androgen receptor antagonist, preparation method and use thereof

#1922
20200239449
2020-07-30

CRYSTAL FORM OF 6-(CYCLOPROPANECARBOXAMIDO)-4-((2-METHOXY-3-(1-METHYL-1H-1,2,4-TRIAZOL-3-YL)PHENYL)AMINO)-N-(METHYL-D3) PYRIDAZINE-3-CARBOXAMIDE

#1923
20200239442
2020-07-30

Bis(pentahydroxyhexyl)amino substituted 2-{[(3-amino-pyrazin-2-yl)formamido]methyl}-1H-1,3-benzodiazol-3-ium derivatives as ENaC inhibitors for treating respiratory diseases

#1924
20200239434
2020-07-30

Antibacterial compounds

#1925
20200239433
2020-07-30

Pyrrole and pyrazole compounds and methods of use thereof

#1926
20200239421
2020-07-30

Pyrimidines and variants thereof, and uses therefor

#1927
20200239415
2020-07-30

EBNA1 inhibitors and methods using same

#1928
20200237763
2020-07-30

3-hydroxy-quinazoline-2,4-dione derivatives and their use as nuclease modulators

#1929
20200237757
2020-07-30

3-oxo-2,6-diphenyl-2,3-dihydropyridazine-4-carboxamides

#1930
20200231584
2020-07-23

PCSK9 inhibitors and methods of use thereof

#1931
20200231577
2020-07-23

Aryl substituted pyrimidines for use in influenza virus infection

#1932
20200231575
2020-07-23

N-[(pyrimidinylamino)propanyl]-,n-[pyridylamino)propanyl]- and n-[(pyrazinylaminol)propanyl]arylcarboxamides

#1933
20200231574
2020-07-23

Halogen complexes of compounds comprising at least one ether, thioether, and/or imine moiety and at least two lactam moieties

#1934
20200231573
2020-07-23

Fluorene derivative or pharmaceutically acceptable salt thereof, preparation method therefor, and pharmaceutical composition comprising same as effective ingredient for preventing or treating HCV-related disease

#1935
20200231572
2020-07-23

Bis-cyclic guanidines as antibacterial agents

#1936
20200231571
2020-07-23

Substituted phenylpyrrolecarboxamides with therapeutic activity in HIV

#1937
20200231568
2020-07-23

Lysophosphatidic acid receptor 1 (LPAR1) inhibitor compounds

#1938
20200231566
2020-07-23

APOPTOSIS INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES

#1939
20200231564
2020-07-23

6-membered aza-heterocyclic containing delta-opioid receptor modulating compounds, methods of using and making the same

#1940
20200231549
2020-07-23

Inhibitors of lysine specific demethylase-1

#1941
20200230264
2020-07-23

Compositions, methods, and systems for the synthesis and use of imaging agents

#1942
20200230110
2020-07-23

Nuclear transport modulators and uses thereof

#1943
20200223845
2020-07-16

Viral replication inhibitors

#1944
20200223830
2020-07-16

Bisamide sarcomere activating compounds and uses thereof

#1945
20200223829
2020-07-16

Bisamide sarcomere activating compounds and uses thereof

#1946
20200223828
2020-07-16

Phenoxyquinazoline compounds and their use in treating cancer

#1947
20200223826
2020-07-16

Glucose-6-Phosphate Dehydrogenase (G6PD)-Modulating Agents And Methods Of Treating G6PD Deficiency

#1948
20200223806
2020-07-16

P2X4 receptor antagonist

#1949
20200223803
2020-07-16

Compositions and methods for treating toxoplasmosis, cryptosporidiosis, and other apicomplexan protozoan related diseases

#1950
20200216486
2020-07-09

MARKERS, CONJUGATES, COMPOSITIONS AND METHODS FOR HYPOXIA IMAGING, MAPPING, AND THERAPY

#1951
20200216476
2020-07-09

PROCESS OF MAKING CENICRIVIROC AND RELATED ANALOGS

#1952
20200216469
2020-07-09

Activators of autophagic flux and phospholipase d and clearance of protein aggregates including tau and treatment of proteinopathies

#1953
20200216431
2020-07-09

COMPOSITIONS AND METHODS FOR INHIBITION OF THE JAK PATHWAY

#1954
20200216423
2020-07-09

Pyrazolo and triazolo bicyclic compounds as JAK kinase inhibitors

#1955
20200216422
2020-07-09

ODM-201 crystalline form, preparation method therefor, and pharmaceutical composition thereof

#1956
20200207769
2020-07-02

DIAZASPIROCYCLOALKANE AND AZASPIROCYCLOALKANE

#1957
20200207745
2020-07-02

Pyrimidine derivative, method for preparing same and use thereof in medicine

#1958
20200207721
2020-07-02

Inhibitors of alpha-amino-beta-carboxymuconic acid semialdehyde decarboxylase

#1959
20200207720
2020-07-02

Benzimidazole derivatives as adenosine receptor antagonists

#1960
20200207711
2020-07-02

Combination of isoindolinone derivatives with SGI-110

#1961
20200199175
2020-06-25

Method for synthesis of protein amphiphiles

#1962
20200199168
2020-06-25

Class A GPCR-binding compound modifier

#1963
20200199126
2020-06-25

Cyanopyrrolidine derivatives with activity as inhibitors of USP30

#1964
20200199113
2020-06-25

Cyclopropyl urea formyl peptide 2 receptor and formyl peptide 1 receptor agonists

#1965
20200199108
2020-06-25

Reactive oxygen species scavengers and use for treating diseases

#1966
20200199098
2020-06-25

Diarylhydantoin compounds and methods of use thereof

#1967
20200199085
2020-06-25

Functionalized 1,2,4,5-tetrazine compounds for use in bioorthogonal coupling reactions

#1968
20200199078
2020-06-25

Compounds for treating proliferative diseases

#1969
20200197393
2020-06-25

Compounds and their use for reducing uric acid levels

#1970
20200197382
2020-06-25

Bacterial efflux pump inhibitors

#1971
20200196602
2020-06-25

Heteroarylphenylaminoquinolines and analogues

#1972
20200190092
2020-06-18

Substituted pyrazolo[3,4-d]pyrimidines as kinase inhibitors

#1973
20200190091
2020-06-18

Nitrogenous heterocyclic compound, preparation method, intermediate, composition, and application

#1974
20200190073
2020-06-18

SUBSTITUTED SUCCINIMIDE DERIVATIVES AS PESTICIDES

#1975
20200190066
2020-06-18

Compound used as autophagy regulator, and preparation method therefor and uses thereof

#1976
20200190064
2020-06-18

THRβ receptor agonist compound and preparation method and use thereof

#1977
20200188540
2020-06-18

CONFORMATIONALLY STRAINED TRANS-CYCLOALKENES FOR RADIOLABELING

#1978
20200181130
2020-06-11

Compositions and methods for inhibition of the JAK pathway

#1979
20200181122
2020-06-11

Degradable imidazolium oligomer and polymer for antimicrobial applications

#1980
20200181117
2020-06-11

SUBSTITUTED 3-HETEROARYLOXY-1H-PYRAZOLES AND SALTS THEREOF AND THEIR USE AS HERBICIDAL ACTIVE SUBSTANCES

#1981
20200181086
2020-06-11

1-cyano-pyrrolidine compounds as USP30 inhibitors

#1982
20200179376
2020-06-11

NITROGEN-CONTAINING HETEROCYCLIC COMPOUND HAVING INHIBITORY EFFECT ON PRODUCTION OF KYNURENINE

#1983
20200172533
2020-06-04

HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS

#1984
20200172525
2020-06-04

Compounds and pharmaceutical compositions containing at least one of the compounds

#1985
20200172519
2020-06-04

Substituted cyanopyrrolidines with activity as DUB inhibitors

#1986
20200172518
2020-06-04

Sulfonamide-substituted cyanopyrrolidines with activity as DUB inhibitors

#1987
20200172517
2020-06-04

Pyridazinone compound or its salt, and herbicide containing it

#1988
20200172516
2020-06-04

Compounds

#1989
20200172510
2020-06-04

Substituted amino six-membered nitric heterocyclic ring compound and preparation and use thereof

#1990
20200172506
2020-06-04

Inhibitors of lysine specific demethylase-1

#1991
20200172495
2020-06-04

Certain chemical entities, compositions, and methods

#1992
20200172492
2020-06-04

Pharmaceutical compound

#1993
20200165262
2020-05-28

Quinazoline and indole compounds to treat medical disorders

#1994
20200165257
2020-05-28

INHIBITORS OF PHOSPHOINOSITIDE 3-KINASE AND HISTONE DEACETYLASE FOR TREATMENT OF CANCER

#1995
20200165231
2020-05-28

KRAS G12C inhibitors and methods of using the same

#1996
20200165230
2020-05-28

3,4,5-trisubstituted-1,2,4-triazoles and 3,4,5-trisubstituted-3-thio-1,2,4-triazoles and uses thereof

#1997
20200165229
2020-05-28

Polyfluoro-substituted aromatic heterocyclic derivative, pharmaceutical composition containing same, and applications thereof

#1998
20200165222
2020-05-28

INDOLE CARBOXAMIDE COMPOUNDS

#1999
20200165206
2020-05-28

Inhibitors of Rho associated coiled-coil containing protein kinase

#2000
20200163935
2020-05-28

Substituted phenylpyrrolecarboxamides with therapeutic activity in HIV

#2001
20200157081
2020-05-21

COMPOUNDS, COMPOSITIONS AND METHODS

#2002
20200157052
2020-05-21

S1P3 antagonists

#2003
20200155531
2020-05-21

Fumarate analogs and uses thereof

#2004
20200147083
2020-05-14

Small molecule modulators of human sting

#2005
20200140460
2020-05-07

ANTIBACTERIAL THERAPEUTICS AND PROPHYLACTICS

#2006
20200140447
2020-05-07

Substituted indole Mcl-1 inhibitors

#2007
20200140436
2020-05-07

LACTAM-CONTAINING COMPOUNDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS

#2008
20200140430
2020-05-07

Pyrimidine compound as JAK kinase inhibitor

#2009
20200140415
2020-05-07

Salt and polymorph of benzopyrimidinone compound and pharmaceutical composition and use thereof

#2010
20200140412
2020-05-07

Substituted isoquinolines and phthalazines as rock kinase inhibitors

#2011
20200140396
2020-05-07

Process for preparing 4-amino-pyridazines

#2012
20200140393
2020-05-07

Bacterial efflux pump inhibitors

#2013
20200138780
2020-05-07

METHODS FOR TREATING PULMONARY EMPHYSEMA USING SUBSTITUTED 2-AZA-BICYCLO[2.2.1]HEPTANE-3-CARBOXYLIC ACID (BENZYL-CYANO-METHYL)-AMIDES INHIBITORS OF CATHEPSIN C

#2014
20200131168
2020-04-30

Hepatitis B core protein modulators

#2015
20200131157
2020-04-30

Pyrazole derivatives for the treatment of cystic fibrosis

#2016
20200131156
2020-04-30

ARYLSULFONYLPYROLECARBOXAMIDE DERIVATIVES AS Kv3 POTASSIUM CHANNEL ACTIVATORS

#2017
20200131151
2020-04-30

Pyridazines

#2018
20200131134
2020-04-30

Farnesoid X receptor agonists and uses thereof

#2019
20200129512
2020-04-30

NOVEL ANTI-INFLAMMATORY AGENTS

#2020
20200123129
2020-04-23

2,4,5-trisubstituted 1,2,4-triazolones useful as inhibitors of DHODH

#2021
20200123115
2020-04-23

COMPOUNDS HAVING MULTIMODAL ACTIVITY AGAINST PAIN

#2022
20200123105
2020-04-23

Hepatitis B capsid assembly modulators

#2023
20200123103
2020-04-23

METHOD FOR THE SYNTHESIS OF AN N-ACYL COMPOUND WITHOUT THE USE OF ORGANIC SOLVENT OR ACID CHLORIDE

#2024
20200121647
2020-04-23

Substituted indoline derivatives as dengue viral replication inhibitors

#2025
20200115366
2020-04-16

Modulators of ATP-binding cassette transporters

#2026
20200115362
2020-04-16

Thyroid hormone receptor beta agonist compounds

#2027
20200115354
2020-04-16

THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF

#2028
20200115347
2020-04-16

DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 ANTAGONISTS

#2029
20200115343
2020-04-16

FUSED-BICYCLIC ARYL QUINOLINONE DERIVATIVES AS MUTANT-ISOCITRATE DEHYDROGENASE INHIBITORS

#2030
20200115339
2020-04-16

EFFLUX-PUMP INHIBITORS AND THERAPEUTIC USES THEREOF

#2031
20200115338
2020-04-16

2,3-dihydroisoindole-1-carboxamides useful as ROR-gamma modulators

#2032
20200115326
2020-04-16

Linkers for antibody drug conjugates

#2033
20200113904
2020-04-16

Methods for treating Huntington's disease

#2034
20200113900
2020-04-16

Benzathine analogs

#2035
20200109134
2020-04-09

Process for the preparation of 6-(cyclopropaneamido)-4-((2-methoxy-3-(1-methyl-1H-1,2,4-triazol-3-yl)phenyl)amino)-N-(methyl-d3)pyridazine-3-carboxamide

#2036
20200109130
2020-04-09

DNA-PK inhibitors

#2037
20200109127
2020-04-09

Inhibitors of the fibroblast growth factor receptor

#2038
20200109120
2020-04-09

PKM2 modulators and methods for their use

#2039
20200109115
2020-04-09

Carbon monoxide releasing norbornenone compounds

#2040
20200108070
2020-04-09

INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF

#2041
20200108054
2020-04-09

SUBSTITUTED BENZAMIDES AND METHODS OF USE THEREOF

#2042
20200108052
2020-04-09

Inhibitors of lysine specific demethylase-1

#2043
20200101047
2020-04-02

Inhibitors of integrated stress response pathway

#2044
20200095252
2020-03-26

Fused pyrimidine compounds as BRD4 and JAK2 dual inhibitors and methods for use thereof

#2045
20200095237
2020-03-26

Substituted phenazines and methods of treating cancer and bacterial diseases

#2046
20200095233
2020-03-26

4,9-dioxo-4,9-dihydronaphtho[2,3-b]furan-3-carboxamide derivatives and uses thereof for treating proliferative diseases and infectious diseases

#2047
20200095231
2020-03-26

Inhibitors of indoleamine 2,3-dioxygenase and methods of their use

#2048
20200095230
2020-03-26

SYNTHETIC ROUTE TO ANTI-VIRAL AGENTS

#2049
20200095229
2020-03-26

Purified cenicriviroc and purified intermediates for making cenicriviroc

#2050
20200087313
2020-03-19

NUCLEAR TRANSPORT MODULATORS AND USES THEREOF

#2051
20200087297
2020-03-19

Quaternary amine compounds and antibody-drug conjugates thereof

#2052
20200087285
2020-03-19

Glutaminyl cyclase inhibitors and the use thereof in treatment of various diseases

#2053
20200087264
2020-03-19

Selective ligand for dopamine D3 receptor, preparation method therefor, and pharmaceutical application thereof

#2054
20200085824
2020-03-19

Small molecule regulators of steroid receptor coactivators and methods of use thereof

#2055
20200085820
2020-03-19

2,4-pyrimidinediamine compounds and their uses

#2056
20200079763
2020-03-12

(R)-8-(1-((3-fluorophenyl)amino)ethyl)-N-(2-hydroxyethyl)-2-morpholinoquinoxaline-6-carboxamide for inhibiting phosphoinositide-3-kinase activity

#2057
20200079761
2020-03-12

Isoindolinone inhibitors of the MDM2-p53 interaction having anticancer activity

#2058
20200079756
2020-03-12

Positive allosteric modulators of the muscarinic acetylcholine receptor M

#2059
20200079754
2020-03-12

INHIBITORS OF BRUTONS TYROSINE KINASE

#2060
20200079753
2020-03-12

Hetroarylamine compounds for modulating the hedgehog pathway and preparing method and uses thereof

#2061
20200077658
2020-03-12

Pesticidal Compounds

#2062
20200071315
2020-03-05

Amide-substituted heterocyclic compounds useful as modulators of IL-12, IL-23 and/or IFN alpha responses

#2063
20200071308
2020-03-05

Benzene, Pyridine, and Pyridazine Derivatives

#2064
20200071305
2020-03-05

Biaryl piperidine amide compounds and methods of use thereof

#2065
20200071303
2020-03-05

Diphenylaminopyrimidine compound for inhibiting kinase activity

#2066
20200071295
2020-03-05

Method for producing benzimidazole derivative

#2067
20200071277
2020-03-05

Photoreactive ligands and uses thereof

#2068
20200069686
2020-03-05

N-SUBSTITUTED INDOLE DERIVATIVES

#2069
20200069646
2020-03-05

Inhibitors of indoleamine 2,3-dioxygenase and methods of their use

#2070
20200062790
2020-02-27

Aryl, heteroaryl, and heterocyclic compounds for treatment of complement mediated disorders

#2071
20200062738
2020-02-27

ANTI-CANCER STEMNESS DRUGS

#2072
20200062735
2020-02-27

HETEROCYCLIC AMIDES AS KINASE INHIBITORS

#2073
20200062732
2020-02-27

DNA-PK inhibitors

#2074
20200061062
2020-02-27

Inhibitors of human phosphatidylinositol 3-kinase delta

#2075
20200061061
2020-02-27

Combinations of a 4-pyrimidinesulfamide derivative with active ingredients for the treatment of endothelin related diseases

#2076
20200061059
2020-02-27

Pyrimidine derivatives for the treatment of viral infections

#2077
20200061041
2020-02-27

Piperidinyl-3-(aryloxy)propanamides and propanoates

#2078
20200055838
2020-02-20

O-aminoheteroaryl alkynyl-containing compound, preparation method therefor, and use thereof

#2079
20200055826
2020-02-20

Pyrimidinyloxy benzo-fused compounds as herbicides

#2080
20200055817
2020-02-20

SPIRO-COMPOUNDS AS SIP MODULATORS

#2081
20200048227
2020-02-13

Compositions and methods for modulating protease activity

#2082
20200048225
2020-02-13

Methods for preparing Nintedanib and intermediates thereof

#2083
20200048224
2020-02-13

Polymorph of pazopanib hydrochloride and preparation process thereof

#2084
20200048223
2020-02-13

WNT SIGNALING PATHWAY INHIBITORS AND THERAPEUTIC APPLICATIONS THEREOF

#2085
20200048221
2020-02-13

Substituted 2-(het)arylimidazolylcarboxyamides as pesticides

#2086
20200048205
2020-02-13

PYRAZOLE DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#2087
20200048197
2020-02-13

Substituted heterocyclic sulfonamide compounds useful as TRPA1 modulators

#2088
20200048195
2020-02-13

SUBSTITUTED PYRROLIDINE CARBOXAMIDE COMPOUNDS

#2089
20200048194
2020-02-13

SUBSTITUTED BENZAMIDES

#2090
20200046718
2020-02-13

Theramutein modulators

#2091
20200046694
2020-02-13

Lanthionine synthetase C-like 2-based therapeutics

#2092
20200044164
2020-02-06

Organic electroluminescent element, display device, lighting device, π-conjugated compound, and light-emitting thin film

#2093
20200039998
2020-02-06

AMINE-SUBSTITUTED HETEROCYCLIC COMPOUNDS AS EHMT2 INHIBITORS AND METHODS OF USE THEREOF

#2094
20200039976
2020-02-06

Compounds and methods for inhibiting fascin

#2095
20200039966
2020-02-06

Uracil containing compounds

#2096
20200039962
2020-02-06

Flame retardants

#2097
20200039961
2020-02-06

SUBSTITUTED FUSED BI- OR TRI- HETEROCYCLIC COMPOUNDS AS EHMT2 INHIBITORS

#2098
20200039958
2020-02-06

Benzimidazole compounds as c-Kit inhibitors

#2099
20200039943
2020-02-06

Compounds, devices, and uses thereof

#2100
20200039941
2020-02-06

CXCR4 CHEMOKINE RECEPTOR MODULATORS