95260 ⎘
Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
2,6-substituted-4-monosubstitutedamino-pyrimidine as prostaglandin D2 receptor antagonists
#72025-amido-indole-2-carboxamide derivatives
#7203Hydroxamic acid esters and pharmaceutical use thereof
#7204COMPOUNDS AND THERAPEUTICAL USE THEREOF
#7205COMPOUNDS AND THERAPEUTICAL USE THEREOF
#7206Novel Compounds Having an Anti-Bacterial Activity
#72073-Phenyl-Pyrazole Derivatives as Modulators of the 5-Ht2A Serotonin Receptor Useful for the Treatment of Disorders Related Thereto
#7208Substituted benzoyl derivatives as herbicides
#7209CB 1 receptor inverse agonists
#7210Nitrosated And Nitrosylated Cardiovascular Compounds, Compositions And Methods Of Use
#7211Compounds
#7212INHIBITORS OF MACROPHAGE MIGRATION INHIBITORY FACTOR AND METHODS FOR IDENTIFYING THE SAME
#72133,4-diamino-3-cyclobutene-1,2-dione derivatives as potassium channel openers
#7214Indole compounds having sphingosine-1-phosphate (S1P) receptor antagonist
#72152-Imino-benzimidazoles
#7216N-phenylbenzotriazolyl c-kit inhibitors
#7217Chromen-2-one derivatives and their use as monoamine neurotransmitter re-uptake inhibitors
#7218Hedgehog pathway antagonists
#7219Sulfoximine-substituted pyrimidines, processes for production thereof and use thereof as drugs
#7220Small molecule toll-like receptor (TLR) antagonists
#7221Piperazine derivatives of dialkyl oxindoles
#7222Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
#7223Compounds that are ERK inhibitors
#7224Inhibitors of soluble adenylate cyclase
#7225Phenyl-substituted pyrimidine derivatives as mGluR antagonists
#7226Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis C viral infections and associated diseases
#7227Ultra-sensitive chemiluminescent substrates for enzymes and their conjugates
#7228Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
#7229Phenyl Compounds And Their Use In The Treatment Of Conditions Mediated By The Action Of Pge2 At The Ep1 Receptor
#7230Bicycloheteroaryl compounds as P2Xmodulators and uses thereof
#7231Substituted 4-phenyltetrahydroisoquinolines, pharmaceutical compositions thereof, methods for their preparation and therapeutic use
#72322,4-pyrimidinediamine compounds and their uses
#7233Pyrazole Compounds Useful In The Treatment Of Inflammation
#7234Arylalkylamine compound and process for preparing the same
#7235Therapeutic Compounds: Pyridine as Scaffold
#7236Substituted Arylpyrazines
#7237Inhibitors of soluble adenylate cyclase
#7238Substituted gamma lactams as therapeutic agents
#7239Therapeutic Compounds: Pyridine N-Oxide Scaffold
#7240Dual NK2/NK3-antagonists, pharmaceutical compositions comprising them, and processes for their preparation
#7241Pyridyl alkene and pyridyl alkine- acid amides as cytostatics and immuno-suppressives
#7242ALKYLAMINE-SUBSTITUTED BICYCLIC ARYL COMPOUNDS USEFUL AS MODULATORS OF PPAR
#7243Triazole derivatives useful as Axl inhibitors
#7244Substituted 2, 6-diamino-3, 5-dicyano-4-arylpyridines and their use as adenosine-receptor-selective ligands
#7245NOVEL NON-PSYCHOTROPIC CANNABINOIDS
#7246Substituted 3-cyanoquinolines as MEK inhibitors
#7247Azole derivatives and fused bicyclic azole derivatives as therapeutic agents
#7248Substituted arylalkanoic acid derivatives and use thereof
#7249Modulators of hepatocyte growth factor/c-Met activity
#7250N,N′-substituted-1,3-diamino-2-hydroxypropane derivatives
#7251Modulators of muscarinic receptors
#7252Dibenzyl amine compounds and derivatives
#7253Methods of labeling nucleic acids with energy transfer dyes
#7254Amino methyl imidazoles and related compounds as C5a receptor modulators
#7255Biphenyl derivatives
#7256Process for Preparing Cephalosporin Intermediates Using Alpha-Iodo-1-Azetidineacetic Acid Esters and Trialkylphosphites
#7257Tao Kinase Modulators And Method Of Use
#7258Piperidinyl derivatives as modulators of chemokine receptor activity
#7259Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
#7260Aryl imidazoles and related compounds as C5a receptor modulators
#7261COMPOUNDS AND THERAPEUTICAL USE THEREOF
#7262HIV inhibiting 5-carbo- or heterocyclic substituted pyrimidines
#7263Vasculostatic agents and methods of use thereof
#7264Substituted sulfonamides and ureas useful for inhibiting kinase activity
#7265Indol-1-yl-acetic acid derivatives
#72663-phenyl-pyrazole derivatives as modulators of the 5-HTserotonin receptor useful for the treatment of disorders related thereto
#7267Substituted N-aryl heterocycles, process for their preparation and their use as medicaments
#7268Carboxylic acid derivatives, their preparation and use
#7269Substituted gamma lactams as therapeutic agents
#7270Phosphodiesterase 4 inhibitors
#7271Novel Indolin-2-one Derivatives, Their Preparation and the Pharmaceutical Compositions Comprising Them
#7272Diaryl piperidines as CB1 modulators
#7273COMPOSITIONS AND METHODS FOR INHIBITION OF THE JAK PATHWAY
#72742-pyridone derivatives as neutrophil elastase inhibitors and their use
#7275SUBSTITUTED INDOLE COMPOUNDS, THEIR PREPARATION AND USE IN MEDICAMENTS
#7276Sulfonyl substituted 1H-indoles as ligands for the 5-hydroxytryptamine receptors
#7277Pyrazolyl-substituted heterocycles and their use as phytosanitary products
#7278Methods For Detecting Substances Which Bind To The Amyloid Precursor Protein Or Beta Amyloid Fragments, And Binding Compounds
#7279Coumarin derivative
#7280Aminocyclohexyl ether compounds and uses thereof
#7281Cannabinoid receptor modulators
#7282Acylated amino acid amidyl pyrazoles and related compounds
#7283Substituted hydantoins
#7284Heterocyclic substituted 4-(aminomethyl)-piperidine benzamides as 5HT-antagonists
#7285Benzenesulfonyl-chromane, thiochromane, tetrahydronaphthalene and related gamma secretase inhibitors
#7286Compositions and methods to treat diseases characterized by cellular proliferation and angiogenesis
#7287Inhibitors of macrophage migration inhibitory factor and methods for identifying the same
#7288N-{'4-substituted piperazine-1-sulfonylmethylalkyl}-n-hydroxyfomamide compounds as metalloproteinase inhibitors
#7289Amido compounds and their use as pharmaceuticals
#7290Compositions and methods for modulating gated ion channels
#7291Herbicidal pyrimidines
#7292Unsaturated tetracyclic tetrahydrofuran derivatives
#7293Novel process for the preparation of 1-(9h-carbazol-4-yloxy)-3-[[2-(-methoxyphenoxy)-ethyl] amino]-propan-2-ol
#7294Deuterated benzo[][1,3]-dioxol derivatives
#7295Derivatives of 3-aminocarbonylquinoline, pharmaceutical compositions containing them and processes and intermediates for their preparation
#7296Kinase inhibitors
#7297Bi-aryl meta-pyrimidine inhibitors of kinases
#7298Urotensin II receptor antagonists
#7299AMINOPIPERIDINE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF
#7300Substituted sulfonamides and ureas useful for inhibiting kinase activity
#73013-Cyano-quinoline derivatives
#73023-((Hetero)arylsulfonyl)-8-'(aminoalkyl)oxyquinolines as 5-ht6 receptor antagonists for the treatment of cns disorders
#7303Pharmaceutically active 4,6-disubstituted aminopyrimidine derivatives as modulators of protein kinases
#7304N-substituted benzene sulfonamides
#7305Anti-inflammatory medicaments
#7306Amino cyclopropane carboxamide derivatives as bradykinin antagonists
#73072-Mercapto-4,5-Diarylimidazole Derivatives and the use thereof as Cyclooxygenase Inhibitors
#7308Beta-secretase modulators and methods of use
#7309Heteroaryl and benzyl amide compounds
#7310Beta-Secretase modulators and methods of use
#7311Bicyclic Heterocycles, Pharmaceutical Compositions Containing These Compounds, Their Use and Processes for Preparing Them
#7312Benzazepine derivatives for the treatment of neurological and psychiatric disorders
#7313M3 muscarinic acetylchoine receptor antagonists
#7314Pyrimidine derivatives
#7315Novel m3 muscarinic acetylcholine receptor antagonists
#7316INHIBITORS OF MACROPHAGE MIGRATION INHIBITORY FACTOR AND METHODS FOR IDENTIFYING THE SAME
#7317Novel M3 Muscarinic Acetylcholine Receptor Antagonists
#7318Opioid receptor antagonists
#7319Hydroxyl compounds and compositions for cholesterol management and related uses
#7320Assays for detection of bioactive compounds that interact with heat shock protein 90
#73214-(2-Phenylsulfanyl-phenyl)-1,2,3,6- tetrahydropyridine derivatives as serotonin reuptake inhibitors
#7322Beta-secretase modulators and methods of use
#7323Melanin concentrating hormone antagonist
#7324Azetidinecarboxamide derivatives and their use in the treatment of cb1 receptor mediated disordrs
#7325Detection of markers in nascent proteins
#7326Novel herbicides
#7327Processes for making pioglitazone and compounds of the processes
#7328SUBSTITUTED PYRIMIDINONES
#73294-Carbox pyrazole derivatives useful as anti-viral agents
#7330Substituted imidazoles
#7331Biaryl linked hydroxamates: preparation and pharmaceutical applications
#7332Carboxylic acid compounds
#7333Therapeutic compounds
#7334Phenylalanine enamide derivatives
#7335Substituted quinazoline compounds useful as p38 kinase inhibitors
#7336Nitrogen-containing heterocyclic compounds and medicinal use thereof
#7337Mercaptoimidazoles as ccr2 receptor antagonists
#7338Therapeutic amide derivatives
#7339Benzamide derivative or salt thereof
#7340Xanthones, thioxanthones and acridinones as DNA-PK inhibitors
#7341Pyrrolidine compound and a process for preparing the same
#7342Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
#73433,4,5-Substituted piperidines as therapeutic compounds
#7344Compounds for the treatment of inflammatory disorders and microbial diseases
#7345Process for the preparation of terazosin hydrocloride dihydrate
#7346Hydrazide type compounds and the use thereof in pharmaceutical compositions for the treatment of cardiovascular diseases
#7347Heterocyclic CETP inhibitors
#7348ETHER DERIVATIVES USEFUL AS INHIBITORS OF PDE4 ISOZYMES
#73493,5-dibenzoyl-4-phenyl-piperidine anti-cancer compounds
#7350Erastin analogs and uses thereof
#7351Substituted indazoles, compositions containing the same, and the preparation and use thereof
#7352Tethered dimers and trimers of 1,4-diphenylazetidin-2-ones
#7353Regents labeled with energy transfer dyes
#7354PPAR active compounds
#7355Hsp90 family protein inhibitors
#73564-(5-aminomethyl)-indole-1-ylmethyl)-benzamide derivatives and related compounds as opioid receptor antagonists for the treatment of obesity
#7357Peptide deformylase inhibitors
#7358Meta-benzamidine derivatives as serine protease inhibitors
#7359Quinoline inhibitors of cGMP phosphodiesterase
#7360Substituted cyclohexyl and piperidinyl derivates as melanocortin-4 receptor modulators
#7361Quinoline Inhibitors of cGMP Phosphodiesterase
#7362INHIBITORS OF FATTY ACID AMIDE HYDROLASE
#7363Aminoindazole derivatives as medicaments and pharmaceutical compositions including them
#7364Diamine derivatives as inhibitors of leukotriene Ahydrolase
#7365Chemokine receptor antagonists
#7366Platelet ADP receptor inhibitors
#7367Substituted azetidinone compounds, processes for preparing the same, formulations and uses thereof
#7368ENERGY TRANSFER DYES WITH ENHANCED FLUORESCENCE
#7369Oligonucleotides and analogs labeled with energy transfer dyes
#7370Fumagillol derivative and the medical use thereof
#7371PPAR active compounds
#7372Pyrrole derivatives, their preparation and their therapeutic use
#7373Piperidine derivative and use thereof
#7374Acidic quinoline derivatives and their use for the prevention and/or treatment of hyperglycaemia-related pathologies
#7375Benzo-fused 5-membered heterocyclic compounds, their production and use
#7376Substituted arylpyrazoles
#7377Diarylamine-containing compounds and compositions, and their use as modulators of c-kit receptors
#7378Bicyclic compounds with kinase inhibitory activity
#73793-aminocyclopentanecrboxamides as modulators of chemokine receptors
#7380Amino heterocyclic modulators of chemokine receptor activity
#7381Plant growth regulation
#7382Detection of disease related genes
#7383Conjugates of mycophenolic acid
#7384Chromane substituted benzimidazole derivatives
#7385Pyrimidinyl amide compounds which inhibit leukocyte adhesion mediated by VLA-4
#7386Piperazine-2-carboxamide derivatives
#7387Calcium receptor modulating agents
#7388Pyridyl Alkene and Pyridyl Alkine-Acid Amides as Cytostatics and Immunosuppressives
#7389Quinoline derivatives as phosphodiesterase inhibitors
#7390Compounds and uses thereof
#7391N-substituted tricyclic 1-aminopyrazoles as inhibitors for the treatment of cell proliferative disorders
#7392Inhibitors of hepatitis C virus NS3 protease
#7393Aralkyl ester soft drugs
#7394HETEROCYCLIC COMPOUNDS AND METHODS OF USE
#7395Fab I inhibitor and process for preparing same
#7396Chroman compounds
#7397INHIBITORS OF HISTONE DEACETYLASE FOR THE TREATMENT OF DISEASE
#7398Nitrogen-containing bicycle heterocycles for use as antibacterials
#7399Azetidine ring compounds and drugs comprising the same
#7400Anti-hypercholesterolemic compounds
#7401Prodrugs of CC-1065 analogs
#7402Aminodibenzodioxin derivative and organic electroluminescent using the same
#7403New pyrrolidinium derivatives
#7404Carbamate compounds which inhibit leukocyte adhesion mediated by VLA-4
#7405N-type calcium channel antagonists for the treatment of pain
#7406LACTAM-CONTAINING DIAMINOALKYL, Beta-AMINOACIDS, Alpha-AMINOACIDS AND DERIVATIVES THEREOF AS FACTOR XA INHIBITORS
#7407Sbstituted chroman derivatives, processes for their preparation and their use as antiinflammatory agents
#7408Pyrimidine derivatives useful for the treatment of diseases mediated by CRTH2
#7409Melanocortin receptor agonists
#7410Novel 4-amino-2(5H)-furanones
#7411EPreceptor antagonists
#7412Phosphodiesterase 4 inhibitors, including aminoindazole and aminobenzofuran analogs
#7413Inhibitors of cathepsin S
#7414PAR2-modulating compounds and their use
#7415Medical devices employing triazine compounds and compositions thereof
#74162-Pyridinylethylcarboxamide derivatives and their use as fungicides
#7417Quinoline inhibitors of cGMP phosphodiesterase
#7418NAPTHALIMIDE DERIVATIVES, METHODS FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS THEREFROM
#7419Anthranilamides and methods of their use
#7420Alkylamino, arylamino, and sulfonamido cyclopentyl amide modulators of chemokine receptor activity
#7421Methods and compositions of novel triazine compounds
#74223-(2-hydroxy-phenyl)-1H-pyrazole-4-carboxylic acid amide derivatives as HSP90 inhibitors for the treatment of cancer
#7423Benzopyran derivatives, method of production and use thereof
#7424Amino nicotinate derivatives as glucokinase (GLK) modulators
#7425Substituted phenylpiperidines with serotoninergic activity and enhanced therapeutic properties
#7426Heterocyclic compounds as pSTAT3/IL-6 inhibitors
#7427Dibenzo[b,f]oxepine-10-carboxamides and pharmaceutical uses thereof
#7428Vitamin D receptor modulators
#7429Alkynyl aryl carboxamides
#7430Indol-containing beta-agonists, methods for the preparation thereof and their use as pharmaceutical compositions
#7431PROCESS FOR THE PREPARATION OF ALFUZOSIN
#7432Heat-shock protein binders
#7433Biphenylcarboxylic amide derivatives as p38 kinase inhibitors
#7434RETINOIC ACID MIMETIC ANILIDES
#7435Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders
#7436Heterocyclic compounds useful for the treatment of inflammatory and allergic disorders: process for their preparation and pharmaceutical compositions containing them
#74372-'4-(Hydroxymethyl-phenylamino)-piperidine-1-yl!-n-(9h-carbazol-3-yl) - acetamine derivatives and related compounds as neuropeptide y5 (npy5) ligands for the treatment of obesity
#74381,3-Dioxane derivatives and analogues thereof useful in the treatment of i.a. obesity and diabetes
#7439Prodrugs of muscarinic agonists and methods of treatment of neuropsychiatric disorders
#7440Modulators of ATP-binding cassette transporters
#7441T1r hetero-oligomeric taste receptors, cell lines that express said receptors, and taste compounds
#7442Crystalline alfuzosin base
#7443Substituted piperazines and piperidines as modulators of the neuropeptide Y2 receptor
#7444LXR receptor modulators
#7445Prodrugs of compounds that inhibit TRPV1 receptor
#7446HIF-1 inhibitors
#7447N-aryl piperidine substituted biphenylcarboxamides as inhibitors of apolipoprotein b
#7448Indole derivatives as serotonin reuptake inhibitors
#7449Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4
#7450Composition and synthesis of new reagents for inhibition of HIV replication
#7451N-(2-ARYLETHYL)BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR
#7452Methods and compositions of novel triazine compounds
#7453Vinyl phenyl derivatives as GLK activators
#74544-Amino-piperidine derivatives as monoamine uptake inhibitors
#7455Tetrahydroisoquinoline LXR Modulators
#7456Aminoindazole derivatives as medicaments and pharmaceutical compositions including them
#7457Mycobacterial inhibitors
#7458Pyrimidines and pyrazines useful as modulators of ion channels
#7459Modulators of calcitonin and amylin activity
#7460Novel amidine compounds for treating microbial infections
#7461Biphenyl derivatives
#7462Fluorinated 4-azasteroid derivatives as androgen receptor modulators
#7463Diaryl Substituted Pyridinones
#7464CB1 antagonist compounds
#7465Conjugates of antioxidants with metal chelating ligands for use in diagnostic and therapeutic applications
#7466Dihydroxypyrimidine carboxamide inhibitors of HIV integrase
#7467Pyrrole compounds for the treatment of prostaglandine mediated diseases
#7468Pyrazine-based tubulin inhibitors
#7469HIV protease inhibitors
#7470BIARYL SUBSTITUTED HETEROCYCLE INHIBITORS OF LTA4H FOR TREATING INFLAMMATION
#7471α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
#7472PYRIDINE CARBOXYLIC ACID DERIVATIVES AS GLUCOKINASE MODULATORS
#7473Phosphodiesterase 4 inhibitors
#7474Substituted heteroaryl CB1 antagonists
#7475Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related thereto
#7476Enzyme modulators and treatments
#7477Cyclic amine derivatives, processes for their preparation, and pharmaceutical compositions containing them
#7478Androgen modulators
#7479PPAR active compounds
#74801-Amino-isoquinoline derivatives for the treatment of diseases associated with inappropriate alk5
#7481P-glycoprotein inhibitor, method for preparing the same and pharmaceutical composition comprising the same
#7482Bis-aryl amide compounds and methods of use
#7483Apoptosis promoters
#7484Diaryl and arylheteroaryl urea derivatives as modulators of the 5-HT2A serotonin receptor useful for the prophylaxis and treatment of disorders related thereto
#7485Survivin inhibitors
#7486Benzopyran derivatives as potassium channel openers
#7487Quaternary salt derivatives of 1,4-diphenylazetidin-2-ones
#7488PREPARATION OF ALFUZOSIN
#7489Biaryl substituted heterocycle inhibitors of LTA4H for treating inflammation
#7490HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THE SAME, THEIR PHARMACEUTICAL USES, MATERIALS FOR THEIR SYNTHESIS
#74913-aminopiperidines and 3-aminoquinuclidines as inhibitors of monoamine uptake
#7492Entry inhibitors of the HIV virus
#7493Imidazole compounds for the treatment of neurological disorders
#7494Acylhydrazones as kinase modulators
#7495Quinoline-2-one derivatives for the treatment of airways diseases
#7496Amido compounds and their use as pharmaceuticals
#7497Imidazole derivatives, their preparation and their use as medicaments
#7498Compounds with mixed pde-inhibitory and beta-adrenergic antagonist or partial agonist activity for treatment of heart failure
#7499Bioisosteres of actinonin
#7500Nicotinamide-based kinase inhibitors