95260 ⎘
Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Spirocyclic piperidines as MCH1 antagonists and uses thereof
#7802Heterocyclic amides, method for the production thereof, substances containing said heterocyclic amides, and use thereof as pesticides
#7803Quinazolines useful as modulators of ion channels
#7804Compounds for inflammation and immune-related uses
#7805Aminoalkoxyphenyl indolone derivatives
#7806Azetidine compounds
#7807Methods and compositions of novel triazine compounds
#7808Sulfonamide inhibitors of aspartyl protease
#7809Compounds and methods for the inhibition of compounds cruzi
#7810Stereoisomerically enriched 3-aminocarbonyl bicycloheptene pyrimidinediamine compounds and their uses
#7811Substituted benzodioxepines
#7812Non-nucleoside reverse transcriptase inhibitors
#7813Tetrahydroquinoline derivatives and their use as FSH receptor modulators
#7814Tricyclic amino alcohols, processes for synthesis of same and use of same as anti-inflammatory drugs
#7815Aminobenzophenone compounds
#7816Pyrrolydin-2-one derivatives as inhibitors of thrombin and factor xa
#7817Cell adhesion inhibitors
#7818Substituted tetracycline compounds
#7819Cell adhesion inhibitors
#7820Antidepressant cycloalkylamine derivatives of 2,3-dihydro-1,4-benzodioxan
#7821Bicyclic heterocycles as cannabinoid receptor modulators
#7822Heteroaryl fused aminoalkyl imidazole derivatives: selective modulators of GABAreceptors
#7823Nitrogen-containing aromatic derivatives
#7824Indole derivatives as serotonin reuptake inhibitors
#7825Ureas as factor Xa inhibitors
#7826Ion channel modulators and methods of use
#7827Carboxylic acid derivatives, their preparation and their use
#7828Cinnamide and hydrocinnamide derivatives with kinase inhibitory activity
#7829Pyrimidinone derivatives as therapeutic agents against acute and chronic inflammatory, ischaemic and remodelling processes
#7830Transcription factor modulating compounds and methods of use thereof
#7831Thioureas as factor Xa inhibitors
#7832Adenosine receptor selective modulators
#7833Fungicidal 1,2,3 triazole derivatives
#7834Phosphodiesterase 4 inhibitors
#7835Quinazolines useful as modulators of ion channels
#7836Isophthalic acid derivatives
#7837Hemiasterlin derivatives and uses thereof
#7838Phthalazinone derivatives
#7839Antidepressant cycloalkylamine derivatives of 2,3-dihydro-1,4-benzodioxan
#7840Coumarin-amide derivatives and its preparation, said drug composition and its use
#7841Protein kinase inhibitors
#7842Pyrazole compounds
#7843Therapeutic agents useful for treating pain
#7844Pyrimidines as PLK inhibitors
#7845Hetero substituted sodium channel blockers
#7846Benzofuran compounds and their use as antidepressants and anxiolytics
#7847Delta 1-pyrrolines used as pesticides
#7848Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
#7849Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidine derivatives
#7850Hydroxycarbonylphenyl substituted 4-(aminomethyl)-piperidine benzamides as 5HTantagonists
#7851Aminosulfonyl substituted 4-(aminomethyl)-piperidine benzamides as 5HT-antagonists
#7852Piperidine derivative and use thereof
#7853Tetrahydroquinoline derivatives
#78545-HT7 receptor antagonists
#7855Sodium channel blockers
#7856Phthalazinone derivatives
#7857Process for the preparation N-(3,5-dichloropyrid-4-yl)-4-difluoromethoxy-8-methane sulfonamido-dibenzo[b,d]furan-1-carboxamide
#78581h-Indazole-3-carboxamide compounds as cyclin dependent kinase (cdk) inhibitors
#78592-acylamino-4-phenylthiazole derivatives, preparation thereof and therapeutic application thereof
#78602,4-Pyrimidinediamine compounds and their uses
#7861Phosphodiesterase 4 inhibitors
#7862Platelet adenosine diphosphate receptor antagonists
#78635-ARYLTETRAZOLE COMPOUNDS AND COMPOSITIONS THEREOF
#7864Chemical compounds containing tocopherol and at least one additional pharmaceutical active substrate
#7865Piperazine derivatives and their use as anti-inflammatory agents
#7866Antibacterial agents
#7867Tyrosine kinase inhibitors
#7868Flavaxate derivatives as muscarinic receptor antagonists
#7869Triazole substituted aminobenzophenone compounds
#7870Biaryl compounds having anti-infective activity
#7871Androgen receptor agonists
#7872Indoles useful in the treatment of androgen-receptor related diseases
#7873Chromanylurea compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor and uses thereof
#7874Heterocyclic compounds having inhibitory activity against HIV integrase
#78759-ketospinosyn derivatives
#78763-cyclopropyl-4-(3-amino-2-methylbenzoyl)pyrazoles and their use as herbicides
#7877Computer program code size partitioning method for multiple memory multi-processing systems
#7878Tri-substituted 2-benzhydryl-5-benzlamino-tetrahydro-pyran-4-ol and 6-benzhydryl-4-benzylamino-tetrahydro-pyran-3-ol analogues, and novel 3,6-disubstituted pyran derivatives
#7879Quinoline and quinoxaline compounds
#7880Substituted amino carboxylic acids
#7881Heterocycle substituted carboxylic acids
#7882Fused heteroaryl derivatives for use as P38 kinase inhibitors
#7883Uracil-thioether
#7884N-(indolethyl-)cycloamine compounds
#7885Platelet adenosine diphosphate receptor antagonists
#7886Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
#7887Medicinal composition containing triazole compound
#78885-substituted quinoline and isoquinoline derivatives, a process for their production and their use as anti-inflammatory agents
#7889Fab I inhibitors
#7890Hepatitis c virus inhibitors
#78911-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
#7892Integrin antagonists useful as anticancer agents
#7893Selective estrogen receptor modulator
#7894Amides useful as monoamine re-uptake inhibitors
#7895Fused indazole compounds
#78962-Amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
#7897Substituted 5-carboxyamide pyrazoles and [1,2,4]triazoles as antiviral agents
#7898Sulfur-containing naphthalimide derivatives
#7899Cathepsin cysteine protease inhibitors and their use
#7900Gonadotropin releasing hormone receptor antagonists
#7901Aryl sulfonamides
#7902Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient
#7903Benzimidazole acetic acids exhibiting CRTH2 receptor antagonism and uses thereof
#7904Chemical compounds
#7905Aminopyridine derivatives having Aurora A selective inhibitory action
#7906Mitotic kinesin inhibitors
#7907Furan or thiophene derivative and medicinal use thereof
#7908Substituted biphenyl-4-carboxylic acid arylamide analogues
#79094-(2-phenylsulfanyl-phenyl)-piperidine derivatives as serotonin reuptake inhibitors
#79102-Thiopyrimidinones as therapeutic agents
#7911Heteroaryl guanidines; inhibitors of viral replication
#7912Quinazoline derivatives and pharmaceutical compositions containing them
#7913Bradykinin-B1 antagonists, process for their preparation and their use as medicaments
#7914Pyrimidine derivatives
#7915Class of arylamide compounds useful as inhibitors of c-fms kinase
#7916Mitotic kinesin inhibitors
#79173-Aryl-3-hydroxy-2-methylenepropionic acid esters as fungicides
#7918Novel uracil derivatives and medicinal use thereof
#7919Inhibitors of macrophase migration inhibitory factor and methods for identifying the same
#7920N-heterocyclic derivatives as NOS inhibitors
#7921NK1 antagonists
#79225-Ht4 receptor antagonists for the treatment of heart failure
#79232-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents
#7924Adsorbing pathogen-inactivating compounds with porous particles immobilized in a matrix
#7925Substituted 3-cyanoquinolines as MEK inhibitors
#7926Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
#7927Inhibitors of glycogen synthase kinase 3
#7928Substituted imidazoles as cannabinoid receptor modulators
#7929Substituted (thioxo)carbonylaminophenyluracils
#7930Isoindoline compounds and methods of making and using the same
#7931Benzofuran oxyethylamines as antidepressants and anxiolytics
#7932Aromatic sulfone hydroxamic acid metalloprotease inhibitor
#7933Substituted alkyl amido piperidines
#7934Small molecule inhibitors of anti-apoptotic BCL-2 family members and the uses thereof
#7935Pyrimidine compounds, process for their preparation and compositions containing them
#7936Pyridine compounds, process for their preparation and compositions containing them
#7937Radio-labeled compounds, compositions, and methods of making the same
#7938Inhibitors of monomine uptake
#7939Piperazine derivatives having SST1 antagonistic activity
#7940Spiroindoline modulators of muscarinic receptors
#7941Production of polyketides and other natural products
#7942Hydroxamic acid and amide compounds and their use as protease inhibitors
#7943Asymmetric process for the preparation of diarylethylpiperazines derivatives and novel asymmetric diarylmethylamines as intermediates
#7944Cyclic AMP-specific phosphodiesterase inhibitors
#7945Aminoindazole derivatives as medicaments and pharmaceutical compositions including them
#7946N-aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF receptor tyrosine kinase inhibitors
#7947Inhibitors of soluble adenylate cyclase
#7948Modulators of ATP-binding cassette transporters
#7949Substituted arylamides
#7950Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
#7951Indazolone derivatives useful as 11b-HSD1 inhibitors
#7952Ophthalmic compositions for treating ocular hypertension
#795317β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
#7954Triazine compounds
#7955Histamine-3 receptor antagonists
#7956Receptor-type kinase modulators and methods of use
#7957Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
#7958Inhibitors of 15-lipoxygenase
#7959Indole inhibitors of 15-lipoxygenase
#79604-arylspirocycloalkyl-2-aminopyrimidine carboxamide KCNQ potassium channel modulators
#79613-Hetero arylmethoxy ! pyridines and their analogues as p38 map kinase inhibitors
#7962Sodium channel blockers
#7963Pyridyl inhibitors of hedgehog signalling
#7964Use of aryl- and heteroaryl-substituted tetrahydroisoquinolines to block reuptake of norepinephrine, dopamine, and serotonin
#7965Indole, indazole, and benzazole derivative
#7966Paroxetine cholate or cholic acid derivative salts, and composition comprising paroxetine and cholic acid or derivative thereof
#79672-substituted heteroaryl compounds
#7968Novel bicyclic hydroxamates as inhibitors of histone deacetylase
#7969N-Benzodioxolyl, n-benzodioxanyl and n-benzodioxepinyl arylcarboxamide derivatives and pharmaceutical compositions comprising them
#7970Benzofuran derivatives, process for their preparation and intermediates thereof
#7971Vanilloid receptor ligands and their use in treatments
#7972Benzamide, heteroarylamide and reverse amides
#79732,4-pyrimidinediamine compounds and their uses
#7974Hydrazone compound, electrophotographic photoreceptor comprising the hydrazone compound, and image forming apparatus equipped with the electrophotographic photoreceptor
#7975Aryloxyalkylamine derivatives as h3 receptor ligands
#7976Conjugation agent
#7977Pyridone derivatives having a binding activity to the cannabinoid type 2 receptor
#7978Cyclopropyl compounds as ccr5 antagonists
#7979Aryl piperidine derivatives as inducers of ldl-receptor expression for the treatment of hypercholesterolemia
#7980Pyridazin-3(2)-one derivatives as PDE4 inhibitors
#7981Aryl- and heteroaryl-substituted tetrahydroisoquinolines and use thereof to block reuptake of norepinephrine, dopamine, and serotonin
#7982Amino-tetrazole analogues and methods of use
#7983Pyridine derivatives as fungicidal compounds
#7984Protease inhibitors
#7985Modulators of ATP-binding cassette transporters
#7986Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
#7987Aromatic heterocyclic-based charge transport materials having two amino groups
#7988Methods of crystal precipitation
#7989Monocyclic aroylpyridinones as antiinflammatory agents
#7990Cytokine inhibitors
#7991Prodrugs containing novel bio-cleavable linkers
#7992Substituted alkyl amido piperidines
#7993Process for producing paroxetine hydrochloride hydrate
#7994Novel triazolo pyrimidine compounds
#7995Substituted amide beta secretase inhibitors
#7996Cox-2 inhibiting pyridine derivatives
#7997Thiobenzimidazole derivatives
#7998Substituted aryl-amine derivatives and methods of use
#7999Substituted pyridinecarboxamides for the treatment of cancer
#80004-pyrimidineamine compounds and their uses as anti-proliferative agents
#8001Compounds with anti-bacterial activity
#8002Benzodiazepine derivatives and pharmaceutical compositions containing them
#8003Piperazine urea derivatives as melanocortin-4 receptor agonists
#8004Substituted indole compounds, their preparation and use in medicaments
#8005Benzopyran derivatives substituted with secondary amines including tetrazole, method for the preparation thereof and pharmaceutical compositions containing them
#80062,4-pyrimidinediamine compounds and their uses
#8007Cycloalkyl substituted pyrimidinediamine compounds and their uses
#8008Lipid-rich plaque regressing agents
#8009D-xylopyranosyl-phenyl-substituted cycles, medicaments containing such compounds, their use and process for their manufacture
#8010N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation
#8011Vanilloid receptor ligands and their use in treatments
#8012Anilinopyrimidine derivatives as IKK inhibitors and compositions and methods related thereto
#8013Amide derivatives and nociceptin antagonists
#8014Glucocorticoid mimetics, methods of making them, pharmaceutical formulations, and uses thereof
#8015Substituted pyridines having antiangiogenic activity
#8016Cell adhesion inhibitors
#8017Triazole derivative
#8018Hydroxyethylamine derivatives for the treatment of Alzheimer's disease
#8019Isoindoline compounds and methods of their use
#8020Pyrimidyl sulphone amide derivatives as chemokine receptor modulators
#8021N-pyrazinyl-phenylsulphonamides and their use in the treatment of chemokine mediated diseases
#8022Compositions useful as inhibitors of voltage-gated sodium channels
#8023Peptide deformylase inhibitors
#80242,4-pyrimidinediamine compounds and their uses
#80251,2,3,4-tetrahydropyrazin-2-yl acetamides and methods of use
#8026D-xylopyranosyl-phenyl-substituted cycles, medicaments containing such compounds, their use and process for their manufacture
#8027Detection of markers in nascent proteins
#8028Bioavailable diacylhydrazine ligands for modulating the expression of exogenous genes via an ecdysone receptor complex
#8029Coumarin derivatives useful as TNFα inhibitors
#80303-aminocyclopentanecarboxamides as modulators of chemokine receptors
#8031Processes and intermediates
#8032Pyrazole derivatives
#8033Compounds, compositions and methods
#8034Biphenyloxy-acids
#8035Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
#80364-amino-quinazolines
#8037Therapeutic chromone compounds
#8038Bicyclic and tricyclic amines as modulators of chemokine receptor activity
#8039Substituted aryl thioureas and related compounds; inhibitors of viral replication
#80403-(Cyclopenten-1-yl)-benzyl-or 3-(cyclopenten-1-yl)-heteroarylmethyl-amine derivatives and use thereof as medicines for treating schizophrenia
#8041Heterocyclo inhibitors of potassium channel function
#8042Phenyl-piperidin-4-ylidene-methyl-benzamide derivatives for the treatment of pain or gastrointestinal disorders
#8043BICYCLIC, SUBSTITUTED TRIAZOLES AS MODULATORS OF PPAR AND METHODS OF THEIR PREPARATION
#8044Nicotinamide derivatives useful as PDE4 inhibitors
#8045Methods for the use of inhibitors of cytosolic phospholipase A2
#804617 β-hydroxysteroid dehydrogenase type 3 inhibitors for the treatment of androgen dependent diseases
#8047Peptidyl prodrugs and linkers and stabilizers useful therefor
#8048N-(2-Arylethyl) benzylamines as antagonists of the 5-HTreceptor
#8049Novel tetrahydropyridine derivatives as renin inhibitors
#8050Indolinone hydrazides as c-Met inhibitors
#8051Substituted imidazole derivatives
#8052Prodrugs of CC-1065 analogs
#8053Substituted aryl amides as IP antagonists
#8054Inhibitors of HCV NS5B polymerase
#8055N-substituted piperidines and their use as pharmaceuticals
#80564-, 5-, 6- and 7-indole derivatives useful for the treatment of CNS disorders
#80573-aminocyclopentanecarboxamides as modulators of chemokine receptors
#8058Quinazoline derivatives as angiogenesis inhibitors
#8059Cinnamide compound
#8060Triazines derivatives as cell adhesion inhibitors
#80613-amino-2-phenylpyrrolidine derivatives
#8062PPAR active compounds
#8063Bicyclic androgen and progesterone receptor modulator compounds and methods
#8064Certain triazole-based compounds, compositions, and uses thereof
#8065Triamide-substituted heterobicyclic compounds
#8066Dual molecules containing a peroxide derivative, synthesis and therapeutic applications thereof
#80672,4-diaminoquinazolines for spinal muscular atrophy
#8068Method for screening an agent that modulates activity of macrophage migration inhibitory factor
#8069Novel ligands and libraries of ligands
#8070Non nucleoside reverse transcriptase inhibitors
#8071Pyrrolidinium derivatives
#8072Cannabinoid receptor ligands
#80733-Cyano-quinoline derivatives
#8074Substituted pyrimidines as selective cyclooxygenase-2 inhibitors
#8075Thio-substituted tricyclic and bicyclic aromatic methanesulfinyl derivatives
#8076Vasculostatic agents and methods of use thereof
#8077Oxindole derivatives
#8078Heteroaryl-hydrazone compounds
#8079Benzofuran derivative
#8080Phenantridine analogues and uses thereof
#8081Method for screening an agent that modulates activity of macrophage migration inhibitory factor
#8082Preparation of paroxetine involving novel intermediates
#8083Novel tetrahydroquinoline derivatives
#8084Substituted tricyclic compounds as protein kinase inhibitors
#80854,5-disubstituted-2-aryl pyrimidines
#8086Vanilloid receptor ligands and their use in treatments
#8087Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor
#8088Vanilloid receptor ligands and their use in treatments
#8089Vanilloid receptor ligands and their use in treatments
#8090Phosphodiesterase 4 inhibitors
#8091Disulfide prodrugs and linkers and stabilizers useful therefor
#8092Biphenyl carboxamides
#8093Small molecule inhibitors of rotamase enzyme activity
#8094Vanilloid receptor ligands and their use in treatments
#8095Diaminopyrimidinecarboxamide derivative
#8096Leptomycin compounds
#8097Hydrazonopyrazole derivatives and their use as therapeutics
#8098Production of polyketides and other natural products
#8099Chromanol derivatives, a process for their production and their use as anti-inflammatory agents
#8100Benzopyran derivatives substituted with secondary amines including imidazole, their preparation and pharmaceutical compositions containing them