1,2,4-triazole derivatives, compositions, process of making and methods of use

Urea derivatives as FLT-3 modulators

α- and β-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors

Vanilloid receptor ligands and their use in treatments

Benzimidazole and imidazopyridine derivatives and use thereof as a medicament

Ansamycins having improved pharmacological and biological properties

Urea antagonists of P2Yreceptor useful in the treatment of thrombotic conditions

Propane-1, 3-dione derivative

Modulators of cellular adhesion

3- or 4-monosubtituted phenol and thiophenol derivatives useful as H3 ligands

Inhibitors of hepatitis C virus NS3 protease

Pyrrolidine and thiazolidine compounds

Tyrosine kinase inhibitors

Anthranilamides and their use as pharmaceutical agents

2-(Bicyclo)alkylamino-derivatives as mediatores of chronic pain and inflammation

Novel 2-amino-4-quinazolinones and 2-amino-4-oxoquinazolones as LXR nuclear receptor binding compounds with partial agonistic properties

Substituted 3-carboxamido isoxazoles as kinase modulators

Process for preparing 3,3-dimethylindolines

Substituted heteroaryl derivatives, compositions, and methods of use

Compounds which inhibit leukocyte adhesion mediated by VLA-4

Aminotriazole compounds useful as inhibitors of protein kinases

Spiro and dispiro 1,2,4-trioxolane antimalarials

Substituted pyrazolyl compounds for the treatment of inflammation

EP2 receptor agonists

NK1 and NK3 antagonists

β-alanine derivatives and the use thereof

Substituted pyridazinones

Protease inhibitors

Protease inhibitors

Protease inhibitors

Fredericamycin derivatives

Quinoxalin-2-one derivatives, compositions which protect useful plants and comprise these derivatives, and processes for their preparation and their use

Non-peptide GnRH agents, pharmaceutical compositions and methods for their use

Ortho substituted aryl or heteroaryl amide compounds

Fab I inhibitors

Quinzoline derivatives for use in the treatment of cancer

Substituted piperidine compounds useful as modulators of chemokine receptor activity

Hydroxamic acid derivatives as metalloprotease inhibitors

Pyridine compounds

HIV protease inhibitors, compositions containing the same, their pharmaceutical uses and materials for their synthesis

Anomeric derivatives of monosaccharides

Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin K inhibitors for the treatment of bone loss

2,5-dioxoimidazolidin-4-yl acetamines and analogues as inhibitors of metalloproteinase mmp12

Naphthyl ether compounds and their use

Tri-substituted ureas as cytokine inhibitors

Amide derivatives

Compounds and methods of use

Urea or thiourea substituted 1,4-pyrazine compounds useful as anti-cancer agents and for inhibiting Chk1

Therapeutic heterocycles

Succinoylamino lactams as inhibitors of A-β protein production

Pyrazole derivatives as herbicidal compositions containing them

Non-nucleoside reverse transcriptase inhibitors

New compounds

Substituted hydroxyethylamine aspartyl protease inhibitors

Piperidine compounds

Alkyne compounds with MCH antagonistic activity and medicaments comprising these compounds

Tri-substituted ureas as cytokine inhibitors

Novel compounds

Substituted tricyclic compounds as protein kinase inhibitors

Substituted tricyclic compound as protein kinase inhibitors

Substituted hydroxyethylamine aspartyl protease inhibitors

Quinazoline derivatives and pharmaceutical compositions containing them

Triazoles as farnesyl transferase inhibitors

Gonadotropin-releasing hormone receptor antagonists and methods relating thereto

1-phenylpiperidin-3-one derivatives and processes for the preparation thereof

Methods of treating or preventing autoimmune diseases with 2, 4-pyrimidinediamine compounds

N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones

Cyclic amine derivatives and methods of use

Organic compounds

Substituted 1-benzazepines and derivatives thereof

Amino-substituted tricyclic derivatives and methods of use

Caspase inhibitors and uses thereof

Platelet ADP receptor inhibitors

Chemical compounds

Substituted benzofurans and benzothiophenes, methods of making and methods of use as integrin antagonists

Substituted tricyclic compounds as protein kinase inhibitors

Vanilloid receptor ligands and their use in treatments

Heterocyclic amides with anti-tuberculosis activity

Chroman derivatives

Pyrazole-amine compounds for the treatment of neurodegenerative disorders

Inhibitors of GSK-3 and uses thereof

3,4-diarylpyrazoles and their use in the therapy of cancer

Phosphodiesterase 4 inhibitors, including N-substituted diarylamine analogs

Nitrogen heterocycle biaryls for osteoporosis and other diseases

Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same

Use of pyrimidine—or triazine—2 carbonitiles for treating diseases associated with cysteine prostease activity and novel pyrimidine-2-carbonitile derivatives

Benzenesulfonamide derivatives as antipsychotic agents

Azetidine derivatives as CCR-3 receptor antagonists

O-cyclopropyl-carboxanilides and their use as fungicides

Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds

Method for the purification of Piribedil

Pharmaceutical compositions as inhibitors of dipeptidyl peptidase-IV (DPP-IV)

2-phenyl-1-[4-(2-aminoethoxy)-benzyl]-indoles as estrogenic agents

Substituted indoles and their use as hcv inhibitors

Imidazole compounds for the treatment of neurodegenerative disorders

2,6-Substituted chroman derivatives useful as beta-3 adrenoreceptor agonists

Inhibitors of glutaminyl cyclase

Pharmaceutical dosage forms and compositions

Substituted arylpyrazines

Melanin concentrating hormone receptor antagonist

Polymer compounds containing oxetane and maleimide functionality

Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents

Compounds and compositions as protein kinase inhibitors

Benzimidazoles useful as modulators of ion channels

Piperidinyl- and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors

Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor

Metabotropic glutamate receptor antagonists

Diaminopyrimidines as P2Xand P2Xantagonists

Process for preparing N-aryl-piperazine derivatives

Compositions and methods for inducing cardiomyogenesis

5-Fluoro-4N-phenyl-4-pyrimidineamine compounds

Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds

Quinoline compound

Methods for monitoring IL-18

Process for the preparation of benazepril hydrochloride

PI-3 kinase inhibitor prodrugs

Ion channel modulators

6-alkylamino-2,2′-disubstituted-7,8-disubstituted-2H-1-benzopyran derivatives as 5-lipoxygenase inhibitor

Process for the preparation of paroxetine substantially free of alkoxy impurities

Biphenyl compounds useful as muscarinic receptor antagonists

Bicyclic amides

Heteroaryl, heterocyclic and aryl compounds which inhibit leukocyte adhesion mediated by VLA-4

Biphenyl compounds useful as muscarinic receptor antagonists

Urea derivatives as PDGFR modulators

Amide compounds as ion channel ligands and uses thereof

Novel quinoline, tetrahydroquinazoline, and pyrimidine derivatives and methods of treatment related to the use thereof

Ink jet recording material

Triazine compounds, polymers comprising triazine structural units, and method

Urea derivatives as C-kit modulators

Quinazolinone compounds with reduced bioaccumulation

Heteroarylaminopyrazole derivatives useful for the treatment of diabetes

Amide compounds as ion channel ligands and uses thereof

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity

Substituted benzazoles and methods of their use as inhibitors of Raf kinase

Ligands of melanocortin receptors and compositions and methods related thereto

Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor

Aminotetralin-derived urea modulators of vanilloid VR1 receptor

Integrin receptor inhibitors

Triazoles as oxytocin antagonists

Phosphodiesterase iv inhibitor containing pyridylacrylamide derivative

Hydroxamates as therapeutic agents

Tricyclic modulators of the glucocorticoid receptor, AP-1, and/or NF-κB activity and use thereof

Nitrosated and nitrosylated alpha-adrenergic receptor antagonist compounds

Compositions useful as inhibitors of voltage-gated ion channels

Extended tethering approach for rapid identification of ligands

Naphthofluorescein-based metal sensors, and methods of making and using the same

Derivatives of dioxane-2-alkyl carbamates, preparation thereof and application thereof in therapeutics

C10 carbamoyloxy substituted taxane compositions

Phthalimide compounds useful as protein kinase inhibitors

Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases

Therapeutic heterocyclic compounds

5-substituted-alkylaminopyrazole derivatives as pesticides

Bicyclic heterocyclic compounds, pharmaceutical compositions containing these compounds, their use and process for preparing them

Nicotinamide derivatives useful as p38 inhibitors.

Pyrrolidine derivatives as prostaglandin modulators

Substituted pyridinones

2-cyano-4-fluoropyrrolidine derivative or its salt

3-Thia-4-arylquinolin-2-one potassium channel modulators

Chk-1 inhibitors

Vanilloid receptor ligands and their use in treatments

Piperidine and piperazine derivatives possessing affinity at 5ht-1 type receptors

Pyrazinone derivatives

Amide derivatives as glycogen synthase kinase 3-β inhibitors

Integrin expression inhibitor

Inhibitors of hepatitis C virus RNA-dependent RNA polymerase, and compositions and treatments using the same

Piperidinylaminomethyl trifluoromethyl cyclic ether compounds as substance P antagonists

2-furancarboxylic acid hydrazides and pharmaceutical compositions containing the same

Broadspectrum substituted benzimidazole sulfonamide hiv protease inhibitors

Amide derivatives as PDGFR modulators

Amide derivatives as FLT-3 modulators

5-substituted-alkylaminopyrazole derivatives as pesticides

Prodrugs of potassium channel inhibitors

Piperidylcarboxamide derivatives and their use in the treatment of tachykinin-mediated diseases

Aryl and heteroaryl compounds, compositions, and methods of use

Non-peptidic BRS-3 agonists

Diaminopyrimidine derivatives as selective growth hormone secrectgogue receptor (GHS-R) antagonists

Diaminopyrimidine derivatives as growth hormone secrectgogue receptor (GHS-R) antagonists

MCH antagonists and their use in the treatment of obesity

Amide derivatives as C-KIT modulators

Quinoline and isoquinoline derivatives, a process for their production and their use as inflammation inhibitors

Vanilloid receptor ligands and their use in treatments

Vanilloid receptor ligands and their use in treatments

Substituted benzofurans and benzothiophenes, methods of making and methods of use as integrin antagonists

Urea derivatives as ABL modulators

Vanilloid receptor ligands and their use in treatments

Isoxazolyl urea derivatives as kinase modulators

Polycyclic aryl and heteroaryl substituted 4-pyrones useful for selective inhibition of the coagulation cascade

Retinoic acid mimetic anilides

Benzimidazoles and analogs thereof as antivirals

N-substituted benzene sulfonamides

3-substituted oxindole β3 agonists

5-Aryltetrazole compounds and uses thereof

Indole derivatives

Pharmaceutical agents

5-Aryltetrazoles compounds and compositions thereof

Compounds, compositions and methods

Pyrrolidinyl, piperidinyl or homopiperidinyl substituted (benzodioxan, benzofuran or benzopyran) derivatives

Methods and compositions related to tagging of membrane surface proteins

5-Sulphanyl-4h-1,2,4-triazole derivatives and their use as medicine

Compounds that modulate PPAR activity and methods for their preparation

Vanilloid receptor ligands and their use in treatments

Substituted indoles

Triazole compounds

Substituted arylamine derivatives and methods of use

β2-adrenoceptor agonists

Benzopyran compounds useful for treating inflammatory conditions

Antidepressant

Dicationic triaryl analogs as anti-protozoan agents

2-guanidinylimidazolidinedione compounds and methods of making and using thereof

3-imino-2-indolones for the treatment of depression and/or anxiety

Amino heterocyclyl inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1

Benzopyran compounds for use in the treatment and prevention of inflammation related conditions

HIV protease inhibiting compounds

Amide derivatives as ABL modulators

LFA-1 antagonist compounds

Quinoxalinones

Imidazole compositions useful as inhibitors of protein kinases

Sulphonamide derivatives as prodrugs of aspartyl protease inhibitors

Fluorescent sensor for phosphate ion and phosphorylated peptide

C10 heterosubstituted acetate taxane compositions

Taxanes having a C7 heterosubstituted acetate substituent

Inhibitors of interleukin-1beta converting enzyme

Calcium receptor modulating agents

Biaryl sulfonamides and methods for using same

4-aminopyrimidines and their use for the antimicrobial treatment of surfaces

Benzodioxole derivatives

Methods for ligand discovery

Absorbing pathogen-inactivating compounds with porous particles immobilized in a matrix

Quinoline derivatives

Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor

Histone deacetylase inhibitors

Benzyl sulfonamide derivatives

4-arylamino-quinazolines and analogs as activators of caspases and inducers of apoptosis and the use thereof

hPPARs activators

Substituted n-aryl amidines as selective D dopamine receptor antagonists for the treatment of obesity and CNS disorders

Anthranilamides with heteroarylsulfonyl side chain, process of preparation, and use

Medical devices employing triazine compounds and compositions thereof

Aryl sulfonamides

Compositions useful as inhibitors of voltage-gated sodium channels

Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor

Optical interleaver

(Oxime)carbamoyl fatty acid amide hydrolase inhibitors

c-fms kinase inhibitors

Acetylene derivatives as inhibitors of histone deacetylase

Quinolines and pharmaceutical compositions thereof

N-arylheteroaromatic products compositions containing them and use thereof

Inhibitors of cathepsin S

Assay for entactogens

Assay for entactogens

Ecstasy haptens and immunogens

Substituted cyclic compounds

Indole compounds

N-phenylarylsulfonamide compound, pharmaceutical composition comprising the compound as active ingredient, synthetic intermediate for the compound and process for its preparation

Benzylcycloalkyl amines as modulators of chemokine receptor activity

Urea thiadiazole inhibitors of plasminogen activator inhibior-1

Compounds and methods of use

Process for preparing chiral diol sulfones and dihydroxy acid HMG CoA reductase inhibitors

Pyrimidine derivatives useful as inhibitors of PKC-theta

Benzimidazoles and analogs thereof as antivirals

Piperazine derivatives and their use as modulators of nuclear hormone receptor function

Medical devices employing triazine compounds and compositions thereof

3,4-Dihydroisoquinolin-1-one derivatives as inducers of apoptosis

5-Substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists

8-azaprostaglandin derivative compounds and drugs containing the compounds as the active ingredient

Mitotic kinesin inhibitors

Small molecule toll-like receptor (TLR) antagonists

Phenylpyrimidine amines as ige inhibitors

Phosphodiesterase 4 inhibitors, including N-substituted aniline and diphenylamine analogs

Inhibitors of C-FMS kinase

Compounds that modulate PPAR activity and methods for their preparation

Piperidin-4-yl urea derivatives and related compounds as chemokine receptor inhibitors for the treatment of inflammatory diseases

2,4-pyrimidinediamine compounds and uses as anti-proliferative agents

Sodium channel blockers

Sodium channel blockers

Sodium channel blockers

Quinoline inhibitors of cGMP phosphodiesterase

Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases

Medical devices employing triazine compounds and compositions thereof

Indazole compounds and compositions thereof as JNK inhibitors and for the treatment of diseases associated therewith

Benzyl urea and thiourea derivatives

Pyridinyl-methyl-ethyl cyclohexanecarboxamides as serotonergic agents

Heteroaromatic urea derivatives as VR-1 receptor modulators for treating pain

Pyrrole derivatives as antimycobacterial compounds

Eponemycin and epoxomicin analogs and uses thereof

Phenylalanine derivatives

Benzylether amine compounds useful as CCR-5 antagonists

Aromatic sulfone hydroxamic acids and their use as protease inhibitors

4-Substituted quinolines as antitumor agents

Antipruritics

STAT modulators

Fluorescent probes for use in protein kinase inhibitor binding assay

Aminoalkyl substituted (benzodioxan, benzofuran or benzopyran) derivatives

Bicyclic [3.1.0] derivatives as glycine transporter inhibitors

Substituted biaryl amides as C5A receptor modulators

3-Thia-4-arylquinolin-2-one derivatives as smooth muscle relaxants

N-ureidoalkyl-piperidines as modulators of chemokine receptor activity

Therapeutic quinolone compounds with 5-ht-antagonistic properties

Aminoalcohol derivatives as beta-3 adrenergic receptor agonists

Aspartic protease inhibitors

Methods of reducing risk of infection from pathogens