ClassID:

95260

C07D405/12 - page 9 - CPC Classification

Classification description:

Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Recent Application in this class:
#2401
20180327361
2018-11-15

Phenyl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#2402
20180327358
2018-11-15

Piperidinone formyl peptide 2 receptor and formyl peptide 1 receptor agonists

#2403
20180327350
2018-11-15

Neprilysin inhibitors

#2404
20180325112
2018-11-15

Insecticidal compositions and methods

#2405
20180319818
2018-11-08

Activators of autophagic flux and phospholipase D and clearance of protein aggregates including tau and treatment of proteinopathies

#2406
20180319812
2018-11-08

HETEROCYCLIC COMPOUND

#2407
20180319779
2018-11-08

Substituted benzofuranyl and benzoxazolyl compounds and uses thereof

#2408
20180319764
2018-11-08

Tricyclic spiro compound

#2409
20180319761
2018-11-08

Pyrone based compounds for treating bacterial infections

#2410
20180319748
2018-11-08

Kinase inhibitors

#2411
20180318309
2018-11-08

Aryl-or heteroaryl-substituted benzene compounds

#2412
20180318308
2018-11-08

Pyrazolone derivatives as nitroxyl donors

#2413
20180318274
2018-11-08

Cyclohexene derivative, preparation method thereof, and pharmaceutical composition for preventing or treating metabolic disease comprising the same as active ingredient

#2414
20180318255
2018-11-08

Pro-Neurogenic Compounds

#2415
20180312633
2018-11-01

Lipid derivative in which hydrophilic polymer is bound through cyclic benzylidene acetal linker

#2416
20180312527
2018-11-01

Activators of autophagic flux and phospholipase D and clearance of protein aggregates including tau and treatment of proteinopathies

#2417
20180312526
2018-11-01

Activators of autophagic flux and phospholipase D and clearance of protein aggregates including tau and treatment of proteinopathies

#2418
20180312524
2018-11-01

Benzopiperazine compositions as BET bromodomain inhibitors

#2419
20180312507
2018-11-01

Fused indazole pyridone compounds as antivirals

#2420
20180312503
2018-11-01

Nitrogen-containing aromatic heterocyclic compound

#2421
20180312494
2018-11-01

Polymorphic forms of Afatinib free base and Afatinib dimaleate

#2422
20180312489
2018-11-01

Substituted indazole compounds as RORgammaT inhibitors and uses thereof

#2423
20180312485
2018-11-01

Substituted benzofuran, benzothiophene and indole Mcl-1 inhibitors

#2424
20180312470
2018-11-01

Derivatives of halo quinabactin

#2425
20180311254
2018-11-01

DNA-PK INHIBITORS

#2426
20180311242
2018-11-01

PYRIMIDINEDIONE COMPOUNDS

#2427
20180311222
2018-11-01

Opioid receptor ligands and methods of using and making same

#2428
20180305403
2018-10-25

PPAR agonists and methods of use thereof

#2429
20180305383
2018-10-25

Kinase inhibitors

#2430
20180305345
2018-10-25

COMPOSITIONS AND METHODS FOR ENHANCING ONCOLYTIC VIRUS EFFICACY

#2431
20180305328
2018-10-25

Compounds for treating mitochondrial disease

#2432
20180305326
2018-10-25

Disubstituted 1, 2, 4-triazine compound

#2433
20180305322
2018-10-25

Substituted diaminocarboxamide and diaminocarbonitrile pyrimidines, compositions thereof, and methods of treatment therewith

#2434
20180305317
2018-10-25

Alkynyl pyridine prolyl hydroxylase inhibitor, and preparation method and medical use thereof

#2435
20180305313
2018-10-25

COLORED PHOTOSENSITIVE RESIN COMPOSITION AND LIGHT SHIELDING SPACER PREPARED THEREFROM

#2436
20180305312
2018-10-25

EBNA1 inhibitors and methods using same

#2437
20180305304
2018-10-25

N-hydroxylsulfonamide derivatives as nitroxyl donors

#2438
20180303822
2018-10-25

PRMT5 inhibitors and uses therof

#2439
20180298043
2018-10-18

Alkyne Compounds for Treatment of Complement Mediated Disorders

#2440
20180298020
2018-10-18

Piperidine derivative and preparation method and pharmaceutical use thereof

#2441
20180298010
2018-10-18

PRMT5 INHIBITORS AND USES THEREOF

#2442
20180297989
2018-10-18

Process for the preparation of N-[4-[(3-chloro-4-fluoro phenyl) amino]-7-[[(3s-tetrahydro-3-furanyl]oxy]-6-quinazolinyl]-4-(dimethyl amino)-(2E)-2-butenamide (2Z)-2-butenedioate (1:2) and its polymorphs thereof

#2443
20180297959
2018-10-18

Benzimidazole derivatives, preparation method therefor, and applications thereof

#2444
20180297939
2018-10-18

Alpha-cinnamide compounds and compositions as HDAC8 inhibitors

#2445
20180291047
2018-10-11

ALKYNE COMPOUNDS FOR TREATMENT OF COMPLEMENT MEDIATED DISORDERS

#2446
20180291046
2018-10-11

ALKYNE COMPOUNDS FOR TREATMENT OF COMPLEMENT MEDIATED DISORDERS

#2447
20180291035
2018-10-11

MYC MODULATORS AND USES THEREOF

#2448
20180290999
2018-10-11

Processes for making triazolo[4,5D] pyramidine derivatives and intermediates thereof

#2449
20180290984
2018-10-11

BRD4-kinase inhibitors as cancer therapeutics

#2450
20180290982
2018-10-11

ARGININE METHYLTRANSFERASE INHIBITORS AND USES THEREOF

#2451
20180290978
2018-10-11

Monocarboxylate transport modulators and uses thereof

#2452
20180290974
2018-10-11

Urea derivative or pharmacologically acceptable salt thereof

#2453
20180289704
2018-10-11

Compounds useful as modulators of TRPM8

#2454
20180289700
2018-10-11

CRMP2 SUMOylation inhibitors and uses thereof

#2455
20180289677
2018-10-11

Covalent small molecule DCN1 inhibitors and therapeutic methods using the same

#2456
20180289672
2018-10-11

Substituted indazole derivatives active as kinase inhibitiors

#2457
20180289664
2018-10-11

Benzhydrol derivatives for the management of conditions related to hypoxia inducible factors

#2458
20180287068
2018-10-04

Compound and organic light emitting diode comprising same

#2459
20180282343
2018-10-04

CARM1 inhibitors and uses thereof

#2460
20180282341
2018-10-04

3-(CARBOXYMETHYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES

#2461
20180282326
2018-10-04

Fused tricyclic urea compounds as Raf kinase and/or Raf kinase dimer inhibitors

#2462
20180282313
2018-10-04

1,3-benzodioxole derivative

#2463
20180282312
2018-10-04

Hydrochloride salt form for EZH2 inhibition

#2464
20180282311
2018-10-04

MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS

#2465
20180282301
2018-10-04

Pyridinone dicarboxamide for use as bromodomain inhibitors

#2466
20180282287
2018-10-04

Azolylacryloyl derivatives as therapeutic agents for sickle cell disease

#2467
20180282276
2018-10-04

Compound for organic electric element, organic electric element comprising the same and electronic device thereof

#2468
20180279614
2018-10-04

Pyridone compounds and agricultural and horticultural fungicides containing said compounds as active ingredient

#2469
20180277767
2018-09-27

Compound and organic electronic device comprising same

#2470
20180273547
2018-09-27

Bromodomain inhibitors

#2471
20180273519
2018-09-27

HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS

#2472
20180273491
2018-09-27

3-(CARBOXYETHYL)-8-AMINO-2-OXO-1,3-DIAZA-SPIRO-[4.5]-DECANE DERIVATIVES

#2473
20180273476
2018-09-27

AMINE DERIVATIVES AS POTASSIUM CHANNEL BLOCKERS

#2474
20180273475
2018-09-27

Hydrophilic fentanyl derivatives

#2475
20180269400
2018-09-20

Materials for organic electroluminescent devices

#2476
20180265524
2018-09-20

SMALL MOLECULES FOR THE MODULATION OF MCL-1 AND METHODS OF MODULATING CELL DEATH, CELL DIVISION, CELL DIFFERENTIATION AND METHODS OF TREATING DISORDERS

#2477
20180265518
2018-09-20

Apelin receptor (APJ) agonists and uses thereof

#2478
20180265501
2018-09-20

Cyclopropanecarboxamide modulators of cystic fibrosis transmembrane conductance regulator

#2479
20180265500
2018-09-20

Tetrahydroquinoline sulfonamide derivatives as inverse agonists of retinoid-related orphan receptor gamma (ROR gamma (t))

#2480
20180265489
2018-09-20

Anticancer agent

#2481
20180265444
2018-09-20

Small molecule stimulators of steroid receptor coactivator proteins and their use in the treatment of cancer

#2482
20180258134
2018-09-13

PSMA imaging agents

#2483
20180258099
2018-09-13

Labeled chemically reactive and biologically active conjugates, and methods and compositions thereof

#2484
20180258098
2018-09-13

Bicyclic derivatives, a process for their preparation and pharmaceutical compositions containing them

#2485
20180258052
2018-09-13

5-[(piperazin-1-yl)-3-oxo-propyl]-imidazolidine-2,4-dione derivatives as ADAMTS inhibitors for the treatment of osteoarthritis

#2486
20180258049
2018-09-13

Human plasma kallikrein inhibitors

#2487
20180258046
2018-09-13

Oxy-cyanoquinolinone PDE9 inhibitors

#2488
20180258043
2018-09-13

PYRIDYL INHIBITORS OF HEDGEHOG SIGNALLING

#2489
20180258038
2018-09-13

N,N-SUBSTITUTED 3-AMINOPYRROLIDINE COMPOUNDS USEFUL AS MONOAMINES REUPTAKE INHIBITORS

#2490
20180256575
2018-09-13

Pyrimidinone amide compounds as PDE2 inhibitors

#2491
20180256558
2018-09-13

Methods and compositions of inhibiting DCN1-UBC12 interaction

#2492
20180251473
2018-09-06

Compound for organic electronic element, organic electronic element using same, and electronic device comprising same

#2493
20180251458
2018-09-06

Histone demethylase inhibitors

#2494
20180251454
2018-09-06

DNA binding agents with a minor groove binding tail

#2495
20180251443
2018-09-06

METHOD OF TREATING OR PREVENTING RAS-MEDIATED DISEASES

#2496
20180251441
2018-09-06

Ion-activated photolabile compounds

#2497
20180251432
2018-09-06

Amino pyrimidine derivatives

#2498
20180251429
2018-09-06

Farnesoid X receptor agonists and uses thereof

#2499
20180251426
2018-09-06

APOPTOSIS-INDUCING AGENTS FOR THE TREATMENT OF CANCER AND IMMUNE AND AUTOIMMUNE DISEASES

#2500
20180250307
2018-09-06

Inhibitors of peptidyl arginine deiminase (PAD) enzymes and uses thereof

#2501
20180250277
2018-09-06

POSITIVE ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTOR

#2502
20180248124
2018-08-30

Materials for electronic devices

#2503
20180244683
2018-08-30

ANTIVIRAL COMPOUNDS

#2504
20180244666
2018-08-30

Dual mechanism inhibitors for the treatment of disease

#2505
20180244643
2018-08-30

HIGHLY SENSITIVE DETECTION OF BIOMOLECULES USING PROXIMITY INDUCED BIOORTHOGONAL REACTIONS

#2506
20180244640
2018-08-30

Modulators of the cystic fibrosis transmembrane conductance regulator protein and methods of use

#2507
20180244632
2018-08-30

HIV replication inhibiting pyrimidines

#2508
20180244631
2018-08-30

INHIBITION OF OLIG2 ACTIVITY

#2509
20180244627
2018-08-30

Heterocyclic compounds and uses thereof

#2510
20180243316
2018-08-30

Salt form of a human histone methyltransferase EZH2 inhibitor

#2511
20180243315
2018-08-30

INHIBITORS OF HUMAN EZH2, AND METHODS OF USE THEREOF

#2512
20180242583
2018-08-30

SYNERGISTIC FUNGICIDAL MIXTURES FOR FUNGAL CONTROL IN CEREALS

#2513
20180242582
2018-08-30

MACROCYCLIC PICOLINAMIDES AS FUNGICIDES

#2514
20180238912
2018-08-23

Fluorogenic pH sensitive dyes and their method of use

#2515
20180237427
2018-08-23

Inhibitors of β-hydroxylase for treatment of cancer

#2516
20180237423
2018-08-23

Neprilysin inhibitors

#2517
20180237398
2018-08-23

Urea derivative and use therefor

#2518
20180237397
2018-08-23

PYRAZOLE DERIVATIVES AS ARGININE METHYLTRANSFERASE INHIBITORS AND USES THEREOF

#2519
20180230159
2018-08-16

DIAMINE DERIVATIVES AS INHIBITORS OF LEUKOTRIENE A4 HYDROLASE

#2520
20180230136
2018-08-16

Crystal form of 3-(6-(1-(2,2-difluorobenzo[d][1,3]dioxole-5-yl)cyclopropane formamido)-3-methylpyridine-2-yl)benzoic acid and preparation method thereof

#2521
20180230109
2018-08-16

Triazole compounds as T-type calcium channel blockers

#2522
20180230108
2018-08-16

Heterocyclic compounds for the inhibition of PASK

#2523
20180228159
2018-08-16

Picolinamide compounds with fungicidal activity

#2524
20180226579
2018-08-09

Amine-based compound and organic light-emitting device including the same

#2525
20180222894
2018-08-09

N-acylethanolamine hydrolyzing acid amidase (NAAA) inhibitors and their use thereof

#2526
20180222883
2018-08-09

Heterocyclic compounds useful as modulators of TNF alpha

#2527
20180222862
2018-08-09

3-indol substituted derivatives, pharmaceutical compositions and methods for use

#2528
20180222838
2018-08-09

Kynurenine-3-monooxygenase inhibitors, pharmaceutical compositions, and methods of use thereof

#2529
20180221367
2018-08-09

Compounds and their use as BACE inhibitors

#2530
20180221279
2018-08-09

MODIFIED DRUGS FOR USE IN LIPOSOMAL NANOPARTICLES

#2531
20180220650
2018-08-09

PLANT GROWTH REGULATOR COMPOUNDS

#2532
20180219157
2018-08-02

COMPOUND, MATERIAL FOR ORGANIC ELECTROLUMINESCENCE ELEMENTS, ORGANIC ELECTROLUMINESCENCE ELEMENT, AND ELECTRONIC DEVICE

#2533
20180215757
2018-08-02

Compounds and methods for inhibiting fascin

#2534
20180215749
2018-08-02

Dual mechanism inhibitors for the treatment of disease

#2535
20180215741
2018-08-02

1-(arylmethyl)quinazoline-2,4(1H,3H)-diones as PARP inhibitors and the use thereof

#2536
20180215739
2018-08-02

2-(1-heteroarylpiperazin-4-yl)methyl-1,4-benzodioxane derivatives as alpha2C antagonists

#2537
20180215738
2018-08-02

Inhibitors of ACK1/TNK2 tyrosine kinase

#2538
20180215727
2018-08-02

LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF

#2539
20180214444
2018-08-02

Piperazine-Substituted Benzothiophenes For Treatment of Mental Disorders

#2540
20180214439
2018-08-02

Substituted quinolinones as PDE9 inhibitors

#2541
20180213780
2018-08-02

Substituted furano-/thienocycloalkylamino-2-pyrimidine derivatives and use thereof for controlling undesired plant growth

#2542
20180208586
2018-07-26

Substituted oxazoles for the treatment of cancer

#2543
20180208573
2018-07-26

Indenyl compounds, pharmaceutical compositions, and medical uses thereof

#2544
20180207155
2018-07-26

Pyrimidine derivatives for the treatment of viral infections

#2545
20180206497
2018-07-26

Aryloxypyrimidinyl ethers as herbicides

#2546
20180206491
2018-07-26

SUBSTITUTED CYCLIC ARYL AND HETEROARYL CARBOXYLIC ACID HYDRAZIDES OR SALTS THEREOF AND USE THEREOF TO INCREASE STRESS TOLERANCE IN PLANTS

#2547
20180201607
2018-07-19

Heterocycle derivatives having TrkA inhibitory activity

#2548
20180201587
2018-07-19

P2X4 receptor antagonist

#2549
20180200238
2018-07-19

Agent for treating and/or preventing adult T cell leukemia/lymphoma

#2550
20180200229
2018-07-19

Triazolone compounds as MPGES-1 inhibitors

#2551
20180194780
2018-07-12

Bridged bicyclic kallikrein inhibitors

#2552
20180194776
2018-07-12

Neprilysin inhibitors

#2553
20180194773
2018-07-12

Bicyclic heterocyclic amide derivative

#2554
20180194769
2018-07-12

HETERO-HALO INHIBITORS OF HISTONE DEACETYLASE

#2555
20180194768
2018-07-12

Substrate selective inhibitors of insulin-degrading enzyme (IDE) and uses thereof

#2556
20180194757
2018-07-12

NEPRILYSIN INHIBITORS

#2557
20180194754
2018-07-12

Polymorphs and process for the preparation of quinazolinyl derivatives

#2558
20180194746
2018-07-12

Compounds for the treatment of HIV

#2559
20180194739
2018-07-12

Methods to treat lymphoplasmacytic lymphoma

#2560
20180194736
2018-07-12

Hydantoin containing deoxyuridine triphosphatase inhibitors

#2561
20180194731
2018-07-12

THERAPEUTIC COMPOUNDS

#2562
20180193338
2018-07-12

NEPRILYSIN INHIBITORS

#2563
20180190904
2018-07-05

Compound, material for organic electroluminescent element, organic electroluminescent element, and electronic device

#2564
20180186806
2018-07-05

ANTIVIRAL COMPOUNDS

#2565
20180186798
2018-07-05

PRMT5 INHIBITORS AND USES THEREOF

#2566
20180186783
2018-07-05

Inhibitors of protein kinases

#2567
20180186779
2018-07-05

G protein-coupled receptor kinase inhibitors and methods for use of the same

#2568
20180186777
2018-07-05

Sulfonamide compounds as voltage-gated sodium channel modulators

#2569
20180186776
2018-07-05

Hesperetin aza-cinnamic acid derivatives with anti-tumor activities and a method of preparing the same

#2570
20180186755
2018-07-05

LYSYL OXIDASE-LIKE 2 INHIBITORS AND USES THEREOF

#2571
20180186746
2018-07-05

6-aminoisoquinoline compounds

#2572
20180186745
2018-07-05

Histone methyltransferase inhibitors

#2573
20180186744
2018-07-05

Compounds for inhibiting c-myc/max/DNA complex formation

#2574
20180186739
2018-07-05

Spiro[cyclobutane-1,3′-indolin]-2′-one derivatives as bromodomain inhibitors

#2575
20180186737
2018-07-05

Hydantoin containing deoxyuridine triphosphatase inhibitors

#2576
20180185363
2018-07-05

Phthalazinone derivatives

#2577
20180182974
2018-06-28

Compound, material for organic electroluminescence devices, organic electroluminescence device, and electronic device

#2578
20180182972
2018-06-28

Compound for organic electric element, organic electric element comprising the same and electronic device thereof

#2579
20180179193
2018-06-28

N-sulfonyl homoserine lactone derivatives, preparation method and use thereof

#2580
20180179166
2018-06-28

SMALL MOLECULE INHIBITORS OF GP120-MEDIATED HIV INFECTION AND METHODS OF USE

#2581
20180179160
2018-06-28

C5aR antagonists

#2582
20180179159
2018-06-28

1,4-substituted piperidine derivatives

#2583
20180179158
2018-06-28

Efflux-pump inhibitors and therapeutic uses thereof

#2584
20180177750
2018-06-28

Compounds and methods for the targeted degradation of enhancer of zeste homolog 2 polypeptide

#2585
20180170943
2018-06-21

Piperidine derivative and preparation method and pharmaceutical use thereof

#2586
20180170929
2018-06-21

Pyrimidine-2,4-diamine derivatives for treatment of cancer

#2587
20180170922
2018-06-21

Substituted pyrazines as ATR kinase inhibitors

#2588
20180170917
2018-06-21

Compounds and compositions as RAF kinase inhibitors

#2589
20180170916
2018-06-21

Inhibitors of CXCR2

#2590
20180170898
2018-06-21

Beta- and gamma-amino-isoquinoline amide compounds and substituted benzamide compounds

#2591
20180170895
2018-06-21

Substituted β-lapachones for treating cancer

#2592
20180170883
2018-06-21

Hsp70 modulators and methods for making and using the same

#2593
20180170857
2018-06-21

PPAR agonists

#2594
20180169099
2018-06-21

HYDROXYLATED AND METHOXYLATED PYRIMIDYL CYCLOPENTANES AS AKT PROTEIN KINASE INHIBITORS

#2595
20180169070
2018-06-21

DIARYL AND ARYLHETEROARYL UREA DERIVATIVES AS MODULATORS OF THE 5-HT2A SEROTONIN RECEPTOR USEFUL FOR THE PROPHYLAXIS AND TREATMENT OF DISORDERS RELATED THERETO

#2596
20180168154
2018-06-21

PLANT GROWTH REGULATING COMPOUNDS

#2597
20180162885
2018-06-14

Compounds useful in the synthesis of halichondrin B analogs

#2598
20180162847
2018-06-14

PRMT5 INHIBITORS CONTAINING A DIHYDRO- OR TETRAHYDROISOQUINOLINE AND USES THEREOF

#2599
20180162844
2018-06-14

CYCLOPROPANE DERIVATIVE AND DRUG CONTAINING SAME

#2600
20180162842
2018-06-14

Modulators of ATP-binding cassette transporters

#2601
20180162823
2018-06-14

Phthalazinones and isoquinolinones as rock inhibitors

#2602
20180161336
2018-06-14

DNA-PK inhibitors

#2603
20180161324
2018-06-14

SHIP1 modulators and methods related thereto

#2604
20180155310
2018-06-07

Inhibitors of LecB

#2605
20180155297
2018-06-07

Inhibitors of ACK1/TNK2 tyrosine kinase

#2606
20180155295
2018-06-07

CXCR4 chemokine receptor modulators

#2607
20180155289
2018-06-07

Mixed disulfide conjugates of thienopyridine compounds and uses thereof

#2608
20180153882
2018-06-07

Aza spiro alkane derivatives as inhibitors of metalloproteases

#2609
20180153873
2018-06-07

Indazole inhibitors of the WNT signal pathway and therapeutic uses thereof

#2610
20180153857
2018-06-07

N-phenyl-carboxamide derivatives and the use thereof as medicaments for the treatment of hepatitis B

#2611
20180148419
2018-05-31

Benzoimidazol-1,2-yl amides as Kv7 channel activators

#2612
20180148418
2018-05-31

AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES

#2613
20180148411
2018-05-31

Indanylaminopyridylcyclopropanecarboxylic acids, pharmaceutical compositions and uses thereof

#2614
20180148408
2018-05-31

Direct inhibitors of Keap1-Nrf2 interaction as antioxidant inflammation modulators

#2615
20180141934
2018-05-24

Modulators of chemokine receptors

#2616
20180141923
2018-05-24

Substituted piperazines as selective HDAC1,2 inhibitors

#2617
20180141919
2018-05-24

DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 ANTAGONISTS

#2618
20180141910
2018-05-24

Fused-bicyclic aryl quinolinone derivatives as mutant-isocitrate dehydrogenase inhibitors

#2619
20180141909
2018-05-24

ROR gamma (RORγ) modulators

#2620
20180141906
2018-05-24

INDOLE AND AZAINDOLE DERIVATIVE HAVING AMPK-ACTIVATING ACTIVITY

#2621
20180141905
2018-05-24

Sulphamoylpyrrolamide derivatives and the use thereof as medicaments for the treatment of hepatitis B

#2622
20180141902
2018-05-24

Cannabinoid receptor CB2 ligand 4-(aminomethyl)-N,N-dialkylanilines

#2623
20180134727
2018-05-17

Inhibitors of RAD52 recombination protein and methods using same

#2624
20180134659
2018-05-17

Oxindole compounds and pharmaceutical compositions thereof

#2625
20180134658
2018-05-17

Salts and prodrugs of 1-methyl-D-tryptophan

#2626
20180133225
2018-05-17

Therapeutic compounds and uses thereof

#2627
20180127432
2018-05-10

Bicyclic-fused heteroaryl or aryl compounds

#2628
20180127420
2018-05-10

Condensed-ring pyrimidylamino derivative, preparation method therefor, and intermediate, pharmaceutical composition and applications thereof

#2629
20180127398
2018-05-10

Solid forms of 3-(6-(1-(2,2-difluorobenzo[D][1,3]dioxol-5-yl)cyclopropanecarboxamido)-3-methylpyridin-2-yl) benzoic acid

#2630
20180127377
2018-05-10

5-substituted indazole-3-carboxamides and preparation and use thereof

#2631
20180127368
2018-05-10

Tricyclic sulfones as ROR gamma modulators

#2632
20180127367
2018-05-10

Pro-Neurogenic Compounds

#2633
20180125985
2018-05-10

Lipids and compositions for the delivery of therapeutics

#2634
20180125855
2018-05-10

Substituted quinazolines for inhibiting kinase activity

#2635
20180125848
2018-05-10

PREPARATION AND METHODS OF USE FOR ORTHO-ARYL 5-MEMBERED HETEROARYL-CARBOXAMIDE CONTAINING MULTI-TARGETED KINASE INHIBITORS

#2636
20180123043
2018-05-03

AROMATIC AMINE DERIVATIVE, AND ORGANIC ELECTROLUMINESCENT ELEMENT USING SAME

#2637
20180118748
2018-05-03

Compounds for improving mRNA splicing

#2638
20180118724
2018-05-03

Solid dosage formulations of substituted quinazoline receptor-type kinase modulators and methods of use thereof

#2639
20180118715
2018-05-03

P-toluenesulfonate for MEK kinase inhibitor, and crystal form thereof and preparation method therefor

#2640
20180118705
2018-05-03

Process for preparing 4-amino-5-biphenyl-4-yl-2-hydroxymethyl-2-methyl-pentanoic acid compound

#2641
20180118704
2018-05-03

Compounds for treating parasitic infections

#2642
20180118694
2018-05-03

6-membered heterocyclic derivatives and pharmaceutical composition comprising the same

#2643
20180118691
2018-05-03

Heterocyclic derivatives modulating activity of certain protein kinases

#2644
20180118683
2018-05-03

Indolone compounds and their use as AMPA receptor modulators

#2645
20180112190
2018-04-26

Compositions and methods for viral sensitization

#2646
20180111920
2018-04-26

Deuterated CFTR modulators

#2647
20180111914
2018-04-26

Substituted naphtho[2,3-b]furans as water-soluble prodrugs for preventing and/or treating cancer

#2648
20180105509
2018-04-19

Amino-substituted heterocyclic derivatives as sodium channel inhibitors

#2649
20180105497
2018-04-19

ARGININE METHYLTRANSFERASE INHIBITORS AND USES THEREOF

#2650
20180105496
2018-04-19

Pyrazole compounds and their use as T-type calcium channel blockers

#2651
20180102479
2018-04-12

Phenanthrene compounds for organic electronic devices

#2652
20180099977
2018-04-12

Inhibitors of histone deacetylase

#2653
20180099976
2018-04-12

Compounds as rearranged during transfection (RET) inhibitors

#2654
20180099953
2018-04-12

Benzofurans substituted with secondary benzamide as HCV inhibitors

#2655
20180098987
2018-04-12

PRMT5 Inhibitors and Uses Thereof

#2656
20180098968
2018-04-12

Anesthetic compounds and related methods of use

#2657
20180097184
2018-04-05

Organic compound, and organic light emitting diode and organic light emitting display device including the same

#2658
20180093997
2018-04-05

Use of physiological cooling active ingredients, and agents containing such active ingredients

#2659
20180093981
2018-04-05

2-Acylaminopropoanol-Type Glucosylceramide Synthase Inhibitors

#2660
20180093976
2018-04-05

Pyridazinone compounds and methods for the treatment of cystic fibrosis

#2661
20180093955
2018-04-05

Quinoline derivatives as inhibitors of heat shock factor 1 pathway activity

#2662
20180092971
2018-04-05

Lipids and compositions for the delivery of therapeutics

#2663
20180092924
2018-04-05

Quinazolinones as bromodomain inhibitors

#2664
20180092880
2018-04-05

Somatostatin receptor subtype 4 (SSTR4) agonists

#2665
20180086744
2018-03-29

COMBINATION TREATMENT OF CANCER COMPRISING EGFR/HER2 INHIBITORS

#2666
20180086716
2018-03-29

Substituted indazoles for treating tendon and/or ligament injuries

#2667
20180086713
2018-03-29

CGAS in systemic lupus erythematosus (SLE)

#2668
20180086707
2018-03-29

Disubstituted piperidines as butyrylcholinesterase inhibitors

#2669
20180086693
2018-03-29

Nitrobenzyl derivatives of anti-cancer agents

#2670
20180085365
2018-03-29

Amino-quinolines as kinase inhibitors

#2671
20180085348
2018-03-29

Methods for treating cancer with RORγ inhibitors

#2672
20180079746
2018-03-22

Heterocyclic modulators of lipid synthesis

#2673
20180079727
2018-03-22

9-membered fused ring derivative

#2674
20180079720
2018-03-22

Substituted 6,7-dihydro-5H-benzo[7]annulene compounds, processes for their preparation and therapeutic uses thereof

#2675
20180079712
2018-03-22

Inhibitors of indoleamine-2,3-dioxygenase for the treatment of cancer

#2676
20180076392
2018-03-15

Condensed-cyclic compound and organic light-emitting device comprising the same

#2677
20180072762
2018-03-15

ALKYNE COMPOUNDS FOR TREATMENT OF COMPLEMENT MEDIATED DISORDERS

#2678
20180072756
2018-03-15

Methods of treating or preventing autoimmune diseases with 2,4-pyrimidinediamine compounds

#2679
20180072674
2018-03-15

4,5-substituted picolinamide and picolinonitrile metabotropic glutamate receptor 2 negative allosteric modulators

#2680
20180072667
2018-03-15

Selective FKBP51 ligands for treatment of psychiatric disorders

#2681
20180072660
2018-03-15

Inhibitors of indoleamine-2,3-dioxygenase for the treatment of cancer

#2682
20180071306
2018-03-15

Carbazole-containing sulfonamides as cryptochrome modulators

#2683
20180066081
2018-03-08

SUBSTITUTED CYCLIC ETHER POLYMERS AND CONJUGATES AND USES THEREOF

#2684
20180065954
2018-03-08

SUBSTITUTED 6,5-FUSED BICYCLIC HETEROARYL COMPOUNDS

#2685
20180065943
2018-03-08

1,1,1-trifluoro-3-hydroxypropan-2-yl carbamate derivatives and 1,1,1-trifluoro-4-hydroxybutan-2-yl carbamate derivatives as MAGL inhibitors

#2686
20180065932
2018-03-08

ANTIVIRAL COMPOUNDS

#2687
20180065929
2018-03-08

Carboxamide derivatives and the use thereof as medicaments for the treatment of hepatitis B

#2688
20180057486
2018-03-01

HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS

#2689
20180057478
2018-03-01

AMPK-activating heterocyclic compounds and methods for using the same

#2690
20180057455
2018-03-01

Compounds useful as immunomodulators

#2691
20180055049
2018-03-01

USE OF PRO-FUNGICIDES OF UK-2A FOR CONTROL OF BROWN ROT DIESEASE ON STONE AND POME FRUITS

#2692
20180051011
2018-02-22

Amide compounds as 5-HT4 receptor agonists

#2693
20180050997
2018-02-22

Compounds and compositions for inhibition of FASN

#2694
20180050052
2018-02-22

Neprilysin inhibitors

#2695
20180049437
2018-02-22

Substituted cyclic amides as herbicides

#2696
20180044334
2018-02-15

Histone demethylase inhibitors

#2697
20180044331
2018-02-15

Piperazine derivatives for treating disorders

#2698
20180044330
2018-02-15

Phthalazinone compounds and methods for the treatment of cystic fibrosis

#2699
20180044328
2018-02-15

Peptidyl nitril compounds as dipeptidyl peptidase I inhibitors

#2700
20180044314
2018-02-15

Method of treating or preventing Ras-mediated diseases