ClassID:

95301

C07D417/12 - CPC Classification

Classification description:

Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links

Recent Application in this class:
#1
20260146041
2026-05-28

PANNEXIN-1 MODULATORS AND METHODS OF TREATING DISORDERS IN WHICH PANNEXIN-1 IS IMPLICATED

#2
20260146037
2026-05-28

PEPTIDYL NITRILE COMPOUND AND USE THEREOF

#3
20260146034
2026-05-28

1H-CYCLOPENTA[B]BENZOFURAN DERIVATIVES FOR THE PREVENTION AND TREATMENT OF VIRUS DISEASES

#4
20260138984
2026-05-21

1-(5-(2-CYANOPYRIDIN-4-YL)OXAZOLE-2-CARBONYL)-4-METHYLHEXAHYDROPYRROLO[3,4-B]PYR ROLE-5(1H)-CARBONITRILE ASUSP30 INHIBITOR FOR USE IN THE TREATMENT OF MITOCHONDRIAL DYSFUNCTION, CANCER AND FIBROSIS

#5
20260138966
2026-05-21

WNT SIGNALING PATHWAY INHIBITORS FOR TREATMENTS OF DISEASE

#6
20260138959
2026-05-21

QUINAZOLINE DERIVATIVE COMPOUND AND USE THEREOF

#7
20260137680
2026-05-21

NOVEL COMPOUNDS

#8
20260137669
2026-05-21

NOVEL ENANTIOMERS OF A SERIES OF ANTIVIRAL COMPOUNDS

#9
20260132126
2026-05-14

IMIDAZOLE DERIVATIVES

#10
20260132121
2026-05-14

INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF

#11
20260132109
2026-05-14

COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY

#12
20260130902
2026-05-14

HIPK4 Degraders as Non-Hormonal Male Contraceptives

#13
20260125359
2026-05-07

HETEROARYL COMPOUNDS AS MULTI-TARGET PROTEIN KINASE INHIBITORS

#14
20260124213
2026-05-07

STAPHYLOCOCCUS AUREUS PBP4 INHIBITORS AND METHOD OF USE

#15
20260124205
2026-05-07

MODULATORS OF BETA CATENIN AND USES THEREOF

#16
20260123278
2026-04-30

COMPOUND FOR ORGANIC ELECTRONIC DEVICE, ORGANIC ELECTRONIC DEVICE USING THE SAME, AND ELECTRONIC DEVICE THEREOF

#17
20260116874
2026-04-30

HETEROAROMATIC INDOLESULFONAMIDES

#18
20260116872
2026-04-30

THIOPHENE BASED APYRASE INHIBITORS

#19
20260116866
2026-04-30

METHOD FOR PREPARING DITHIOCYCLOPENTENONE DERIVATIVE AND APPLICATION THEREOF

#20
20260109713
2026-04-23

SIRTUIN MODULATING COMPOUNDS, INCLUDING SIRTUIN ACTIVATING COMPOUNDS, AND APPLICATIONS THEREOF

#21
20260109709
2026-04-23

2-AMINO IMIDAZOLE DERIVATIVES AS PRMT5 INHIBITORS

#22
20260109694
2026-04-23

HETEROCYCLIC COMPOUNDS AND USES THEREOF

#23
20260103444
2026-04-16

8-HYDROXYQUINOLINE COMPOUND AND USE THEREOF

#24
20260098030
2026-04-09

NEGATIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR 2

#25
20260098018
2026-04-09

BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF

#26
20260097047
2026-04-09

Small molecule inhibitors of the ribosome biogenesis factor NVL2

#27
20260097046
2026-04-09

PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS

#28
20260092061
2026-04-02

COMPOUNDS FOR TARGETED PROTEIN DEGRADATION

#29
20260092057
2026-04-02

BCL-XL/BCL-2 DEGRADERS AND USES THEREOF

#30
20260091024
2026-04-02

PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE

#31
20260085074
2026-03-26

COMPOSITIONS AND METHODS FOR TREATING CANCER

#32
20260085068
2026-03-26

A NOVEL CRYSTALLINE FORM OF PRITELIVIR

#33
20260085064
2026-03-26

SUBSTITUTED BENZOFURANYL AND BENZOXAZOLYL COMPOUNDS AND USES THEREOF

#34
20260085048
2026-03-26

ACSS2 INHIBITORS AND METHODS OF USE THEREOF

#35
20260078091
2026-03-19

Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer

#36
20260076975
2026-03-19

TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES

#37
20260070900
2026-03-12

A NOVEL CRYSTALLINE FORM OF PRITELIVIR

#38
20260070899
2026-03-12

N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-QUINOLINE-4-CARBOXAMIDES

#39
20260070896
2026-03-12

HETEROCYCLE DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS

#40
20260070878
2026-03-12

TNKS2 INHIBITORS

#41
20260062420
2026-03-05

NOVEL DPP1 INHIBITORS AND USES THEREOF

#42
20260062416
2026-03-05

INHIBITORS OF KIF18A AND USES THEREOF

#43
20260062407
2026-03-05

PEROXIREDOXIN 3 INHIBITORS AND METHODS OF USE FOR TREATING CANCER

#44
20260062402
2026-03-05

KCC2 POTENTIATORS AND USES THEREOF

#45
20260062393
2026-03-05

Compounds

#46
20260055098
2026-02-26

TOLFENPYRAD DERIVATIVES EXHIBIT POTENT FRANCISELLA-SPECIFIC ANTIBACTERIAL ACTIVITY WITHOUT TOXICITY TO MAMMALIAN CELLS IN VITRO

#47
20260055096
2026-02-26

AZOLE PESTICIDAL COMPOUNDS

#48
20260055067
2026-02-26

CERTAIN (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES AS DIPEPTIDYL PEPTIDASE 1 INHIBITORS

#49
20260049074
2026-02-19

THIADIAZOLYL DERIVATIVES

#50
20260049062
2026-02-19

SARS-COV-2 INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS

#51
20260049061
2026-02-19

SMALL MOLECULES AS KCNQ2/3 (KV7.2/3) CHANNEL ACTIVATORS AND THEIR MEDICAL USE THEREOF

#52
20260048068
2026-02-19

PHENYLUREA DERIVATIVES AND THEIR PHARMACEUTICAL USES

#53
20260042747
2026-02-12

KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF

#54
20260041673
2026-02-12

PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE

#55
20260035360
2026-02-05

INHIBITORS OF MYC AND USES THEREOF

#56
20260034113
2026-02-05

THIADIAZOLONE DERIVATIVES, COMPOSITIONS AND USES THEREOF

#57
20260034105
2026-02-05

Generative AI-Assisted Identification of Novel PI3K-alpha Inhibitors

#58
20260028335
2026-01-29

NOVEL ISOTHIAZOL-3-YL AND ISOXAZOL-3-YL SULFONAMIDE COMPOUNDS

#59
20260022117
2026-01-22

COMPOUNDS AND METHODS FOR THE ENHANCED DEGRADATION OF TARGETED PROTEINS

#60
20260022114
2026-01-22

N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (1,3-THIAZOLYL)](SUBSTITUTED)CARBOXAMIDE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING THE AMIDE COMPOUNDS AND OF THEIR USE

#61
20260021107
2026-01-22

STIMULATOR OF INTERFERON GENES AGONISTS

#62
20260015360
2026-01-15

BIARYL DERIVATIVES AND RELATED USES

#63
20260015325
2026-01-15

ALKOXY HETEROARYL- CARBOXAMIDE OR THIOAMIDE COMPOUNDS

#64
20260008777
2026-01-08

INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE, COMPOSITIONS, AND METHODS OF USE

#65
20260008758
2026-01-08

LINEAR DIPEPTIDYL PEPTIDASE 1 INHIBITORS AND USES THEREOF

#66
20260001873
2026-01-01

NOVEL INHIBITORS

#67
20260001872
2026-01-01

BENZISOTHIAZOLE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF

#68
20260001871
2026-01-01

TRIAZOLE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR D

#69
20260001870
2026-01-01

INHIBITOR COMPOUNDS

#70
20260001861
2026-01-01

PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8

#71
20260001846
2026-01-01

SPIROCYCLOHEXANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS ANTI-APOPTOTIC INHIBITORS

#72
20250388601
2025-12-25

Compounds, Compositions and Methods

#73
20250388584
2025-12-25

TPK AGONIST AND METHOD FOR TREATING NEURODEGENERATIVE DISEASES USING SAME

#74
20250388573
2025-12-25

FUSED BICYCLIC EGFR INHIBITORS AND METHODS OF USE THEREOF

#75
20250388551
2025-12-25

COMPOUNDS INDUCING PRODUCTION OF PROTEINS BY IMMUNE CELLS

#76
20250388536
2025-12-25

3-ALKYNYL CARBOXAMIDES AS AEP MODULATORS

#77
20250382298
2025-12-18

NITROGEN-CONTAINING COMPOUND AND USE THEREOF

#78
20250382273
2025-12-18

BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS

#79
20250382269
2025-12-18

METHODS AND COMPOSITIONS FOR SELECTIVELY INHIBITING PATHOGENIC MICROBES

#80
20250382268
2025-12-18

METHODS AND COMPOSITIONS FOR SELECTIVELY INHIBITING PATHOGENIC MICROBES

#81
20250380697
2025-12-18

ISOXAZOLINE DERIVATIVE COMPOUND AND INSECTICIDAL COMPOSITION COMPRISING SAME

#82
20250376461
2025-12-11

INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS

#83
20250376452
2025-12-11

17-Beta-Hydroxysteroid Dehydrogenase Type 13 Inhibitors and Methods of Use Thereof

#84
20250376443
2025-12-11

MASP-2 INHIBITORS AND METHODS OF USE

#85
20250368637
2025-12-04

SOLID-STATE FORMS OF N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-6-MORPHOLINOQUINOLINE-4-CARBOXAMIDE

#86
20250368605
2025-12-04

Novel Substituted 6,7-Dihydro-5H-Benzo[7]Annulene Compounds, Processes for their Preparation and Therapeutic Uses Thereof

#87
20250368604
2025-12-04

MASP-2 INHIBITORS AND METHODS OF USE

#88
20250367209
2025-12-04

IDENTIFICATION OF NOVEL BENZOTHIAZONES AS TAU-SH3 INTERACTION INHIBITORS FOR THE TREATMENT OF ALZHEIMER’S DISEASE

#89
20250361213
2025-11-27

1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF

#90
20250360145
2025-11-27

CSF-1R INHIBITORS AND USES THEREOF

#91
20250353853
2025-11-20

FLAVIVIRUS INHIBITORS

#92
20250353821
2025-11-20

BENZENE SULFONAMIDE THIAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCERS

#93
20250346943
2025-11-13

DEGRADER COMPOUNDS OF QSOX1 mRNA

#94
20250346588
2025-11-13

IMIDAZOPYRIDINE AND OXAZOLOPYRIDINE DERIVATIVES AND ANALOGS THEREOF, METHODS OF PREPARATION THEREOF, METHODS OF HIF-1/2A PATHWAY INHIBITION, AND INDUCTION OF FERROPTOSIS

#95
20250346583
2025-11-13

NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS

#96
20250346573
2025-11-13

AZAQUINOLINONE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF

#97
20250346569
2025-11-13

NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS

#98
20250340886
2025-11-06

INTRACELLULAR KINASE ASSOCIATED WITH RESISTANCE AGAINST ANTI-TUMOUR IMMUNE RESPONSES, AND USES THEREOF

#99
20250340543
2025-11-06

GPR84 ANTAGONISTS AND USES THEREOF

#100
20250333423
2025-10-30

SMALL MOLECULE MODULATORS OF GP130 SIGNALING PATHWAYS

#101
20250333417
2025-10-30

IRAK DEGRADERS AND USES THEREOF

#102
20250333411
2025-10-30

COMPOUNDS AND METHODS FOR INHIBITING FASCIN

#103
20250333404
2025-10-30

DEUTERATED COMPOUNDS

#104
20250333400
2025-10-30

CERTAIN PLADIENOLIDE COMPOUNDS AND METHODS OF USE

#105
20250332161
2025-10-30

PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY

#106
20250332148
2025-10-30

RILUZOLE PRODRUGS AND THEIR USE

#107
20250326746
2025-10-23

EIF4E INHIBITORS AND USES THEREOF

#108
20250326744
2025-10-23

PIPERAZINE DERIVATIVE OR SALT THEREOF, AND PHARMACEUTICAL COMPOSITION

#109
20250326732
2025-10-23

CHROMEN-2-ONE MODULATORS OF POLRMT

#110
20250326725
2025-10-23

PI4-Kinase Inhibitors and Methods of Using the Same

#111
20250326713
2025-10-23

INHIBITORS OF MsbA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF

#112
20250325552
2025-10-23

SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS

#113
20250324971
2025-10-23

HERBICIDAL DERIVATIVES

#114
20250320186
2025-10-16

HSD17B13 INHIBITORS AND USES THEREOF

#115
20250320184
2025-10-16

SARM1 MODULATORS, PREPARATIONS, AND USES THEREOF

#116
20250313574
2025-10-09

SIALIC ACID DERIVATIVES AND METHODS OF USING SAME

#117
20250313555
2025-10-09

2-SUBSTITUTED THIAZOLE AND BENZOTHIAZOLE COMPOSITIONS AND METHODS AS DUX4 INHIBITORS

#118
20250313554
2025-10-09

PTPN2 INHIBITORS

#119
20250313535
2025-10-09

ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF

#120
20250304600
2025-10-02

PHARMACEUTICAL COMPOUNDS AND COMPOSITIONS AS c-KIT KINASE INHIBITORS

#121
20250304574
2025-10-02

3,4,6,7-TETRAHYDRO-2,7-NAPHTHYRIDINE-2(1H)-CARBOXAMIDE DERIVATIVES AS GPR65 INHIBITORS FOR THE TREATMENT OF CANCER AND AUTOIMMUNE DISEASES

#122
20250304571
2025-10-02

BIOLOGICALLY ACTIVE COMPOUNDS AND METHODS THEREOF

#123
20250304542
2025-10-02

Fused Heterobicyclic Antiviral Agents

#124
20250296928
2025-09-25

A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF

#125
20250296927
2025-09-25

HETEROCYCLIC COMPOUNDS AND USES THEREOF

#126
20250296926
2025-09-25

SELECTIVE LIGANDS FOR MODULATION OF GIRK CHANNELS

#127
20250296920
2025-09-25

FORMULATIONS COMPRISING N-SUBSTITUTED-DIOXOCYCLOBUTENYLAMINO-3-HYDROXY-PICOLINAMIDE COMPOUNDS AND USES THEREOF

#128
20250295789
2025-09-25

TREATMENT OR PROPHYLAXIS OF PROLIFERATIVE CONDITIONS

#129
20250295652
2025-09-25

Inhibitors of Molluscum Contagiosum Infection and Methods Using the Same

#130
20250289811
2025-09-18

HETEROCYCLIC DERIVATIVES AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITORS

#131
20250289789
2025-09-18

REVERSIBLE LYSINE COVALENT MODIFIERS OF CDK2 AND USES THEREOF

#132
20250289785
2025-09-18

INDOLE DERIVATIVE, METHOD FOR PREPARING SAME, AND USE THEREOF

#133
20250282792
2025-09-11

GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO

#134
20250282760
2025-09-11

OREXIN RECEPTOR AGONISTS

#135
20250282740
2025-09-11

COMPOSITIONS FOR TREATING AND/OR PREVENTING CELL OR TISSUE NECROSIS SPECIFICALLY TARGETING CATHEPSIN C AND/OR CELA1 AND/OR CELA3A AND/OR STRUCTURALLY RELATED ENZYMES THERETO

#136
20250276952
2025-09-04

4-AMINOPHENYL-THIAZOLE DERIVATIVES AND METHODS OF USE THEREOF

#137
20250275952
2025-09-04

4-METHYLSULFONYL-SUBSTITUTED PIPERIDINE UREA COMPOUNDS

#138
20250270194
2025-08-28

PYRAZOLE-SUBSTITUTED CYCLOPENTANOL ESTER DERIVATIVE AND USE THEREOF

#139
20250270171
2025-08-28

HUMAN PLASMA KALLIKREIN INHIBITORS

#140
20250268879
2025-08-28

METHODS OF TREATING NEUROLOGICAL, METABOLIC, AND OTHER DISORDERS USING ENANTIOPURE DEUTERIUM-ENRICHED PIOGLITAZONE

#141
20250263407
2025-08-21

Compounds

#142
20250263406
2025-08-21

DEUTERATED DERIVATIVES OF LANIFIBRANOR

#143
20250257042
2025-08-14

NOVEL DRP-1 INHIBITORS AS THERAPEUTIC AGENTS

#144
20250257040
2025-08-14

HUMAN PLASMA KALLIKREIN INHIBITORS

#145
20250257035
2025-08-14

1,4-Substituted Piperidine Derivatives

#146
20250250265
2025-08-07

BENZOTHIAZOLE-PHENYLSULFONYL-PIPERIDINE ANALOGS AS ACTIVATORS OF NACYLPHOSPHATIDYLETHANOLAMINE HYDROLYZING PHOSPHOLIPASE D

#147
20250250259
2025-08-07

METHODS FOR TREATING CANCER

#148
20250243193
2025-07-31

AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFN ALPHA RESPONSES

#149
20250243192
2025-07-31

CRYSTALLINE FORM OF LANIFIBRANOR

#150
20250236590
2025-07-24

A METHOD FOR THE PREPARATION OF INDOLE-3-CARBOXYLIC ACID DERIVATIVES

#151
20250230153
2025-07-17

2,3-DIHYDROBENZO[B][1,4]DIOXIN-6-YL CONTAINING COMPOUNDS USEFUL AS IMMUNOMODULATORS

#152
20250230144
2025-07-17

QUINAZOLINES AS POTASSIUM ION CHANNEL INHIBITORS

#153
20250223280
2025-07-10

POTENT ASGPR-BINDING COMPOUNDS FOR THE DEGRADATION OF IMMUNOGLOBULINS AND OTHER PROTEINS

#154
20250223267
2025-07-10

CYCLOOLEFIN SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE

#155
20250223265
2025-07-10

COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR

#156
20250221411
2025-07-10

SUBSTITUTED BENZAMIDES AS HERBICIDES

#157
20250214987
2025-07-03

THIOBENZIMIDAZOLE DERIVATIVE PREPARATION METHOD AND NOVEL INTERMEDIATE THEREFOR

#158
20250214986
2025-07-03

P2X3 INHIBITOR COMPOUND, SALT THEREOF, POLYMORPH THEREOF AND USE THEREOF

#159
20250214980
2025-07-03

MULTICYCLIC COMPOUNDS

#160
20250214963
2025-07-03

SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH

#161
20250214947
2025-07-03

3,4-DIHYDROQUINOXALINE-2-CARBOXIMIDE DERIVATIVE COMPOUND AND PHARMACEUTICAL COMPOSITION COMPRISING SAME FOR PREVENTING OR TREATING CANCER DISEASE

#162
20250214945
2025-07-03

THIOBENZIMIDAZOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND USE THEREOF

#163
20250214940
2025-07-03

HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHOLOGICAL DISORDERS

#164
20250206755
2025-06-26

ANTIMICROBIAL AGENTS

#165
20250206731
2025-06-26

COMPOUND, POLYMERIZABLE COMPOSITION, POLYMER, HOLOGRAPHIC RECORDING MEDIUM, OPTICAL MATERIAL, AND OPTICAL COMPONENT

#166
20250206730
2025-06-26

THIAZOLE DERIVATIVE COMPOUND AND USES THEREOF

#167
20250206709
2025-06-26

METHOD FOR FORMING AMINOTHIAZOLE DERIVATIVES WITH SUPER-PARAMAGNETIC NANOPARTICLE CATALYST

#168
20250205232
2025-06-26

MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR

#169
20250205204
2025-06-26

Transcription Factor Brn2 Inhibitory Compounds for Use as Therapeutics

#170
20250197387
2025-06-19

BCL-XL DEGRADERS AND USES THEREOF

#171
20250197385
2025-06-19

COMPOUNDS, SALTS THEREOF AND METHODS FOR TREATMENT OF DISEASES

#172
20250197379
2025-06-19

NOVEL RAS INHIBITORS

#173
20250197368
2025-06-19

2-OXO-DIHYDROQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS GABA TYPE A RECEPTOR MODULATORS

#174
20250197363
2025-06-19

THIADIAZOLE COMPOUND, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING INFLAMMATORY DISEASES, INCLUDING SAME

#175
20250197353
2025-06-19

METHOD OF FORMING BOND BY COUPLING REACTION

#176
20250195485
2025-06-19

PROPIONIC ACID DERIVATIVE AND MEDICAL USE THEREOF

#177
20250188072
2025-06-12

COMPOUNDS FOR TREATMENT OF CANCER

#178
20250188057
2025-06-12

NON-AROMATIC CYCLIC-PYRIMIDINE ANALOGS AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS

#179
20250179122
2025-06-05

Telomerase Reverse Transcriptase (TERT) Expression Enhancing Compounds and Methods for Using the Same

#180
20250179061
2025-06-05

RIP1 MODULATORS, PREPARATIONS, AND USES THEREOF

#181
20250179039
2025-06-05

ELECTRON ACCEPTOR, AND REAGENT LAYER AND SENSOR EACH USING SAME

#182
20250179033
2025-06-05

NEW ANTIVIRAL TRIAZOLE DERIVATIVES, THEIR SYNTHESIS AND THEIR USE FOR TREATMENT OF MAMMALIAN VIRAL INFECTIONS

#183
20250179013
2025-06-05

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PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS

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2025-05-29

METHOD FOR FORMING A SCHIFF BASE WITH CATALYTIC SUPER-PARAMAGNETIC IRON OXIDE NANOPARTICLES

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2025-05-29

PYRROLIDINE COMPOUNDS

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2025-05-29

MRGPRX2 MODULATORS AND RELATED METHODS OF TREATMENT

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2025-05-29

ARYL-OR HETEROARYL-SUBSTITUTED BENZENE COMPOUNDS

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2025-05-29

MODULATORS OF ACKR3 AND USES THEREOF

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A METHOD FOR TREATING ROSAH SYNDROME

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2025-05-22

SUBSTITUTED 1,2,4-TRIAZOLES AND METHODS OF USE

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MCL-1 INHIBITORS

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2025-05-15

1,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF

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2025-05-08

PROTEIN DEGRADERS AND USES THEREOF

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2025-05-08

THIAZOLE COMPOUNDS AND METHODS OF USE THEREOF

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2025-05-08

MODULATORS OF THE INTEGRATED STRESS PATHWAY

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2025-05-08

CATHEPSIN K INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#198
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2025-05-08

THIOSTREPTON-INSPIRED COMPOUNDS FOR TREATMENT OF CANCER AND PREPARATION THEREOF

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RAD51 INHIBITORS

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2025-05-01

THIADIAZOLONE DERIVATIVES USEFUL AS AMPK ACTIVATOR

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SMO MODULATOR COMPOUNDS

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MASP-2 INHIBITORS AND METHODS OF USE

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MYST Inhibitors

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PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF

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KAT6 Inhibitors

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2025-04-10

SULFOXIMINE GLYCOSIDASE INHIBITORS

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cGAS ANTAGONIST COMPOUNDS

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PYRIDAZINE DERIVATIVES AND RELATED USES

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BICYCLIC-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS

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COMPOSITIONS AND METHODS FOR TREATING CANCER

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PEPTIDYL NITRILE COMPOUND AND USE THEREOF

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NOVEL KALIRIN INHIBITORS FOR REGULATION OF SYNAPTIC PLASTICITY AND NEUROPATHIC PAIN TREATMENT

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SPIROCYCLIC CAV2.3 ANTAGONISTS

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2025-03-27

MEK INHIBITORS AND METHODS OF THEIR USE

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COMPOSITIONS AND METHODS FOR TREATING CANCER

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2025-03-20

RIPK3 INHIBITORS AND METHODS OF USE

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2025-03-20

ENHANCERS OF PARTICULATE GUANYLYL CYCLASE RECEPTOR A

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COMPOUNDS AND METHODS OF ACTIVATING LIPOPROTEIN LIPASE

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NOVEL DRP-1 INHIBITORS AS THERAPEUTIC AGENTS

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COMPOSITIONS AND METHODS FOR MAKING AND USING SMALL MOLECULES FOR TUBULIN-TARGETED THERAPY IN THE TREATMENT OF CANCERS AND RELATED CONDITIONS

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SMALL MOLECULE PROTEIN SYNTHESIS MODULATORS

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SUBSTITUTED HETEROCYCLES AS HSET INHIBITORS

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PYRAZOLE-SUBSTITUTED CYCLOPENTANOL ESTER DERIVATIVE AND USE THEREOF

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PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF

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4-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES

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NSD2-TARGETED CHECMICAL DEGRADERTS AND COMPOSITIONS AND METHODS OF USE THEREOF

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PYRIDAZINONES AS PARP7 INHIBITORS

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Novel Aminobenzene Derivative Having Cancer Cell Growth Inhibitory Effect, and Preventive or Therapeutic Pharmaceutical Composition Containing Same as Active Ingredient

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SUBSTITUTED (1,2,3,4-TETRAHYDROCYCLOPENTA[b]INDOL-3-YL)ACETIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS

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SOLID FORMS OF A BENZTHIAZOLE-PIPERAZINYL-OXAZOLE COMPOUND AND METHODS OF USE THEREOF

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COMPOSITIONS AND METHODS OF USE TO TREAT 12-LIPOXYGENASE (12-LOX) MEDIATED DISEASES

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BENZOTHIAZOLE, BENZOISOXAZOLE, AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS

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DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 ANTAGONISTS

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THIADIAZINE DERIVATIVES

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Anti-inflammatory Compounds, Pharmaceutical Compositions, and Treatment Methods

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Pharmaceutical Compounds and Compositions as C-Kit Kinase Inhibitors

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CARDIAC SARCOMERE INHIBITORS

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TLR MODULATOR AND USE THEREOF

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MODULATORS OF MYOCYTE LIPID ACCUMULATION AND INSULIN RESISTANCE AND METHODS OF USE THEREOF

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SMALL MOLECULE INHIBITORS OF PR3 AND HNE AND USES THEREOF

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THERAPEUTIC COMPOUNDS AND METHODS

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CRYSTALLINE FORMS OF A DEOXYCYTIDINE KINASE INHIBITOR AND USES THEREOF

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2025-02-06

N-[5-(aminosulfonyl)-4-methyl-1,3-thiazol-2-yl]-N-methyl-2-[4-(2-pyridinyl)-phenyl]-acetamide free base hemihydrate, methods of manufacture and uses thereof

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PREPARATION OF INDOLONE-3YL-HYDRAZONO-SUBSTITUTED 1,3-THIAZOLIDINONE DERIVATIVES AND APPLICATION THEREOF

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2025-01-30

CHROMOBOX PROTEIN INHIBITORS AND USES THEREOF

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2025-01-30

QUINOLINE DERIVATIVES

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EGFR INHIBITORS AND METHODS OF USE THEREOF

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2025-01-23

TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS

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N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (THIAZOLYL)])(SUBSTITUTED)CARBOXAMIDE COMPOUNDS AND USE THEREOF FOR INHIBITING HUMAN POLYMERASE THETA

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ENHANCERS OF PARTICULATE GUANYLYL CYCLASE RECEPTOR A

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QUINAZOLINONE DIONE COMPOUNDS AND USES THEREOF

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ARYL OR HETEROARYL DERIVATIVE, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF KINASE-RELATED DISEASES

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SELECTIVE PEPTIDOMIMETIC MODULATORS OF CAV2.2 (N-TYPE) VOLTAGE-GATED CALCIUM CHANNELS AND USES THEREOF

#261
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PEROXIREDOXIN 3 INHIBITORS AND METHODS OF USE FOR TREATING CANCER

#262
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ARYL HYDROCARBON RECEPTOR (AHR) AGONISTS AND USES THEREOF

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LONG-CHAIN COMPOUND THAT ACTS ON ACLY, PREPARATION METHOD THEREFOR AND USE THEREOF

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HETEROCYCLIC COMPOUNDS AND USES THEREOF

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FUSED BICYCLIC SUBSTITUTED N-(1H-INDOL-7-YL)BENZENESULFONAMIDES AND USES THEREOF

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NOVEL PYRIDINE DERIVATIVE COMPOUND AS RON INHIBITOR

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FLUORINE-CONTAINING PYRAZOLE COMPOUND AND PRODUCTION METHOD THEREFOR

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2024-12-19

CARBONIC ANHYDRASE IX-TARGETING RADIOACTIVE DIAGNOSTIC AND THERAPEUTIC MEDICAMENT AND METHOD FOR PREPARING SAME

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HMOX1 INDUCERS

#270
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ORGANIC COMPOUNDS

#271
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COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER

#272
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Methods for treating cancer

#273
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2024-12-05

SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME

#274
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COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY

#275
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2024-11-28

Substituted Quinoxalines

#276
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2024-11-28

QUINACRINE AND DERIVATIVES THEREOF FOR TREATMENT OF VIRAL INFECTIONS

#277
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2024-11-28

ISOQUINOLINONES AND QUINOLINONES AS MODULATORS OF POLRMT

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2024-11-28

PHENYL CORE COMPOUNDS AS MGLU5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME

#279
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Compounds for Treating Cannabinoid Toxicity and Acute Cannabinoid Overdose

#280
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2024-11-21

COMPOUNDS AND METHODS FOR MODULATING INTERLEUKIN-2-INDUCIBLE T-CELL KINASE

#281
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2024-11-21

SMARCA DEGRADERS AND USES THEREOF

#282
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2024-11-21

INHIBITORS OF TRANSGLUTAMINASES

#283
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2024-11-21

BIFUNCTIONAL DEGRADERS COMPRISING A TEAD BINDER

#284
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2024-11-21

NOVEL INHIBITOR OF HYPE-MEDIATED AMPYLATION

#285
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PRMT5 INHIBITOR AND THE USE THEREOF

#286
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2024-11-14

MODULATORS OF PrPC AND USES THEREOF

#287
20240376091
2024-11-14

THIADIAZOLEAMIDE DERIVATIVES AND THEIR APPLICATIONS

#288
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2024-11-14

INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS

#289
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2024-11-14

NAMPT INHIBITORS AND USES THEREOF

#290
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2024-11-14

INHIBITORS OF TRANSGLUTAMINASES

#291
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2024-11-07

N-substituted-dioxocyclobutenylamino-3-hydroxy-picolinamides useful as CCR6 inhibitors

#292
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2024-11-07

CERTAIN PLADIENOLIDE COMPOUNDS AND METHODS OF USE

#293
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2024-11-07

SUBSTITUTED TETRAHYDROFURAN-2-CARBOXAMIDES AS MODULATORS OF SODIUM CHANNELS

#294
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2024-11-07

JAK2 INHIBITORS AND METHODS OF USE THEREOF

#295
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2024-11-07

ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS

#296
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2024-11-07

Fused Heterobicyclic Antiviral Agents

#297
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2024-11-07

BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF

#298
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2024-10-31

RAD51 INHIBITORS

#299
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2024-10-31

SMALL MOLECULE UREA DERIVATIVES AS STING ANTAGONISTS

#300
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2024-10-31

HETEROCYCLIC COMPOUNDS AS SEROTONIN (5-HT) 5-HT2A AND 5-HT2C RECEPTOR POSITIVE ALLOSTERIC MODULATORS