95301 ⎘
Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
PANNEXIN-1 MODULATORS AND METHODS OF TREATING DISORDERS IN WHICH PANNEXIN-1 IS IMPLICATED
#2PEPTIDYL NITRILE COMPOUND AND USE THEREOF
#31H-CYCLOPENTA[B]BENZOFURAN DERIVATIVES FOR THE PREVENTION AND TREATMENT OF VIRUS DISEASES
#41-(5-(2-CYANOPYRIDIN-4-YL)OXAZOLE-2-CARBONYL)-4-METHYLHEXAHYDROPYRROLO[3,4-B]PYR ROLE-5(1H)-CARBONITRILE ASUSP30 INHIBITOR FOR USE IN THE TREATMENT OF MITOCHONDRIAL DYSFUNCTION, CANCER AND FIBROSIS
#5WNT SIGNALING PATHWAY INHIBITORS FOR TREATMENTS OF DISEASE
#6QUINAZOLINE DERIVATIVE COMPOUND AND USE THEREOF
#7NOVEL COMPOUNDS
#8NOVEL ENANTIOMERS OF A SERIES OF ANTIVIRAL COMPOUNDS
#9IMIDAZOLE DERIVATIVES
#10INHIBITORS OF RIPK2 AND MEDICAL USES THEREOF
#11COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH STING ACTIVITY
#12HIPK4 Degraders as Non-Hormonal Male Contraceptives
#13HETEROARYL COMPOUNDS AS MULTI-TARGET PROTEIN KINASE INHIBITORS
#14STAPHYLOCOCCUS AUREUS PBP4 INHIBITORS AND METHOD OF USE
#15MODULATORS OF BETA CATENIN AND USES THEREOF
#16COMPOUND FOR ORGANIC ELECTRONIC DEVICE, ORGANIC ELECTRONIC DEVICE USING THE SAME, AND ELECTRONIC DEVICE THEREOF
#17HETEROAROMATIC INDOLESULFONAMIDES
#18THIOPHENE BASED APYRASE INHIBITORS
#19METHOD FOR PREPARING DITHIOCYCLOPENTENONE DERIVATIVE AND APPLICATION THEREOF
#20SIRTUIN MODULATING COMPOUNDS, INCLUDING SIRTUIN ACTIVATING COMPOUNDS, AND APPLICATIONS THEREOF
#212-AMINO IMIDAZOLE DERIVATIVES AS PRMT5 INHIBITORS
#22HETEROCYCLIC COMPOUNDS AND USES THEREOF
#238-HYDROXYQUINOLINE COMPOUND AND USE THEREOF
#24NEGATIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR 2
#25BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF
#26Small molecule inhibitors of the ribosome biogenesis factor NVL2
#27PLASMODIUM FALCIPARUM BLOOD STAGE INHIBITORS
#28COMPOUNDS FOR TARGETED PROTEIN DEGRADATION
#29BCL-XL/BCL-2 DEGRADERS AND USES THEREOF
#30PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE
#31COMPOSITIONS AND METHODS FOR TREATING CANCER
#32A NOVEL CRYSTALLINE FORM OF PRITELIVIR
#33SUBSTITUTED BENZOFURANYL AND BENZOXAZOLYL COMPOUNDS AND USES THEREOF
#34ACSS2 INHIBITORS AND METHODS OF USE THEREOF
#35Piperidinone Derivatives as MDM2 Inhibitors for the Treatment of Cancer
#36TPK AGONIST AND METHOD FOR USING SAME TO TREAT NEURODEGENERATIVE DISEASES
#37A NOVEL CRYSTALLINE FORM OF PRITELIVIR
#38N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-QUINOLINE-4-CARBOXAMIDES
#39HETEROCYCLE DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS
#40TNKS2 INHIBITORS
#41NOVEL DPP1 INHIBITORS AND USES THEREOF
#42INHIBITORS OF KIF18A AND USES THEREOF
#43PEROXIREDOXIN 3 INHIBITORS AND METHODS OF USE FOR TREATING CANCER
#44KCC2 POTENTIATORS AND USES THEREOF
#45Compounds
#46TOLFENPYRAD DERIVATIVES EXHIBIT POTENT FRANCISELLA-SPECIFIC ANTIBACTERIAL ACTIVITY WITHOUT TOXICITY TO MAMMALIAN CELLS IN VITRO
#47AZOLE PESTICIDAL COMPOUNDS
#48CERTAIN (2S)-N-[(1S)-1-CYANO-2-PHENYLETHYL]-1,4-OXAZEPANE-2-CARBOXAMIDES AS DIPEPTIDYL PEPTIDASE 1 INHIBITORS
#49THIADIAZOLYL DERIVATIVES
#50SARS-COV-2 INHIBITORS FOR TREATING CORONAVIRUS INFECTIONS
#51SMALL MOLECULES AS KCNQ2/3 (KV7.2/3) CHANNEL ACTIVATORS AND THEIR MEDICAL USE THEREOF
#52PHENYLUREA DERIVATIVES AND THEIR PHARMACEUTICAL USES
#53KIT INHIBITORS, COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF USE THEREOF
#54PRODRUGS OF RILUZOLE AND THEIR METHOD OF USE
#55INHIBITORS OF MYC AND USES THEREOF
#56THIADIAZOLONE DERIVATIVES, COMPOSITIONS AND USES THEREOF
#57Generative AI-Assisted Identification of Novel PI3K-alpha Inhibitors
#58NOVEL ISOTHIAZOL-3-YL AND ISOXAZOL-3-YL SULFONAMIDE COMPOUNDS
#59COMPOUNDS AND METHODS FOR THE ENHANCED DEGRADATION OF TARGETED PROTEINS
#60N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (1,3-THIAZOLYL)](SUBSTITUTED)CARBOXAMIDE COMPOUNDS, PHARMACEUTICAL COMPOSITIONS, AND METHODS OF PREPARING THE AMIDE COMPOUNDS AND OF THEIR USE
#61STIMULATOR OF INTERFERON GENES AGONISTS
#62BIARYL DERIVATIVES AND RELATED USES
#63ALKOXY HETEROARYL- CARBOXAMIDE OR THIOAMIDE COMPOUNDS
#64INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE, COMPOSITIONS, AND METHODS OF USE
#65LINEAR DIPEPTIDYL PEPTIDASE 1 INHIBITORS AND USES THEREOF
#66NOVEL INHIBITORS
#67BENZISOTHIAZOLE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF
#68TRIAZOLE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR D
#69INHIBITOR COMPOUNDS
#70PYRIDINE CARBOXAMIDE COMPOUNDS FOR INHIBITING NAV1.8
#71SPIROCYCLOHEXANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS ANTI-APOPTOTIC INHIBITORS
#72Compounds, Compositions and Methods
#73TPK AGONIST AND METHOD FOR TREATING NEURODEGENERATIVE DISEASES USING SAME
#74FUSED BICYCLIC EGFR INHIBITORS AND METHODS OF USE THEREOF
#75COMPOUNDS INDUCING PRODUCTION OF PROTEINS BY IMMUNE CELLS
#763-ALKYNYL CARBOXAMIDES AS AEP MODULATORS
#77NITROGEN-CONTAINING COMPOUND AND USE THEREOF
#78BENZOTHIAZOLE ANAOLOGUES AND USE THEREOF AS BOOSTERS OF ANTI TUBERCULOSIS DRUGS
#79METHODS AND COMPOSITIONS FOR SELECTIVELY INHIBITING PATHOGENIC MICROBES
#80METHODS AND COMPOSITIONS FOR SELECTIVELY INHIBITING PATHOGENIC MICROBES
#81ISOXAZOLINE DERIVATIVE COMPOUND AND INSECTICIDAL COMPOSITION COMPRISING SAME
#82INDAZOLE DERIVATIVES FOR TREATING TRPM3-MEDIATED DISORDERS
#8317-Beta-Hydroxysteroid Dehydrogenase Type 13 Inhibitors and Methods of Use Thereof
#84MASP-2 INHIBITORS AND METHODS OF USE
#85SOLID-STATE FORMS OF N-(2-(4-CYANOTHIAZOLIDIN-3-YL)-2-OXOETHYL)-6-MORPHOLINOQUINOLINE-4-CARBOXAMIDE
#86Novel Substituted 6,7-Dihydro-5H-Benzo[7]Annulene Compounds, Processes for their Preparation and Therapeutic Uses Thereof
#87MASP-2 INHIBITORS AND METHODS OF USE
#88IDENTIFICATION OF NOVEL BENZOTHIAZONES AS TAU-SH3 INTERACTION INHIBITORS FOR THE TREATMENT OF ALZHEIMER’S DISEASE
#891,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF
#90CSF-1R INHIBITORS AND USES THEREOF
#91FLAVIVIRUS INHIBITORS
#92BENZENE SULFONAMIDE THIAZOLE COMPOUNDS AND THEIR USE FOR THE TREATMENT OF CANCERS
#93DEGRADER COMPOUNDS OF QSOX1 mRNA
#94IMIDAZOPYRIDINE AND OXAZOLOPYRIDINE DERIVATIVES AND ANALOGS THEREOF, METHODS OF PREPARATION THEREOF, METHODS OF HIF-1/2A PATHWAY INHIBITION, AND INDUCTION OF FERROPTOSIS
#95NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS
#96AZAQUINOLINONE DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF
#97NEW DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS
#98INTRACELLULAR KINASE ASSOCIATED WITH RESISTANCE AGAINST ANTI-TUMOUR IMMUNE RESPONSES, AND USES THEREOF
#99GPR84 ANTAGONISTS AND USES THEREOF
#100SMALL MOLECULE MODULATORS OF GP130 SIGNALING PATHWAYS
#101IRAK DEGRADERS AND USES THEREOF
#102COMPOUNDS AND METHODS FOR INHIBITING FASCIN
#103DEUTERATED COMPOUNDS
#104CERTAIN PLADIENOLIDE COMPOUNDS AND METHODS OF USE
#105PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY
#106RILUZOLE PRODRUGS AND THEIR USE
#107EIF4E INHIBITORS AND USES THEREOF
#108PIPERAZINE DERIVATIVE OR SALT THEREOF, AND PHARMACEUTICAL COMPOSITION
#109CHROMEN-2-ONE MODULATORS OF POLRMT
#110PI4-Kinase Inhibitors and Methods of Using the Same
#111INHIBITORS OF MsbA AS ANTIBIOTICS, PHARMACEUTICAL COMPOSITIONS, AND USES THEREOF
#112SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS
#113HERBICIDAL DERIVATIVES
#114HSD17B13 INHIBITORS AND USES THEREOF
#115SARM1 MODULATORS, PREPARATIONS, AND USES THEREOF
#116SIALIC ACID DERIVATIVES AND METHODS OF USING SAME
#1172-SUBSTITUTED THIAZOLE AND BENZOTHIAZOLE COMPOSITIONS AND METHODS AS DUX4 INHIBITORS
#118PTPN2 INHIBITORS
#119ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF
#120PHARMACEUTICAL COMPOUNDS AND COMPOSITIONS AS c-KIT KINASE INHIBITORS
#1213,4,6,7-TETRAHYDRO-2,7-NAPHTHYRIDINE-2(1H)-CARBOXAMIDE DERIVATIVES AS GPR65 INHIBITORS FOR THE TREATMENT OF CANCER AND AUTOIMMUNE DISEASES
#122BIOLOGICALLY ACTIVE COMPOUNDS AND METHODS THEREOF
#123Fused Heterobicyclic Antiviral Agents
#124A SYNTHESIS SCHEME AND PROCEDURES FOR PREPARING A SIK3 INHIBITOR AND INTERMEDIATES THEREOF
#125HETEROCYCLIC COMPOUNDS AND USES THEREOF
#126SELECTIVE LIGANDS FOR MODULATION OF GIRK CHANNELS
#127FORMULATIONS COMPRISING N-SUBSTITUTED-DIOXOCYCLOBUTENYLAMINO-3-HYDROXY-PICOLINAMIDE COMPOUNDS AND USES THEREOF
#128TREATMENT OR PROPHYLAXIS OF PROLIFERATIVE CONDITIONS
#129Inhibitors of Molluscum Contagiosum Infection and Methods Using the Same
#130HETEROCYCLIC DERIVATIVES AS MITOGEN-ACTIVATED PROTEIN KINASE (MEK) INHIBITORS
#131REVERSIBLE LYSINE COVALENT MODIFIERS OF CDK2 AND USES THEREOF
#132INDOLE DERIVATIVE, METHOD FOR PREPARING SAME, AND USE THEREOF
#133GONADOTROPIN-RELEASING HORMONE RECEPTOR ANTAGONISTS AND METHODS RELATING THERETO
#134OREXIN RECEPTOR AGONISTS
#135COMPOSITIONS FOR TREATING AND/OR PREVENTING CELL OR TISSUE NECROSIS SPECIFICALLY TARGETING CATHEPSIN C AND/OR CELA1 AND/OR CELA3A AND/OR STRUCTURALLY RELATED ENZYMES THERETO
#1364-AMINOPHENYL-THIAZOLE DERIVATIVES AND METHODS OF USE THEREOF
#1374-METHYLSULFONYL-SUBSTITUTED PIPERIDINE UREA COMPOUNDS
#138PYRAZOLE-SUBSTITUTED CYCLOPENTANOL ESTER DERIVATIVE AND USE THEREOF
#139HUMAN PLASMA KALLIKREIN INHIBITORS
#140METHODS OF TREATING NEUROLOGICAL, METABOLIC, AND OTHER DISORDERS USING ENANTIOPURE DEUTERIUM-ENRICHED PIOGLITAZONE
#141Compounds
#142DEUTERATED DERIVATIVES OF LANIFIBRANOR
#143NOVEL DRP-1 INHIBITORS AS THERAPEUTIC AGENTS
#144HUMAN PLASMA KALLIKREIN INHIBITORS
#1451,4-Substituted Piperidine Derivatives
#146BENZOTHIAZOLE-PHENYLSULFONYL-PIPERIDINE ANALOGS AS ACTIVATORS OF NACYLPHOSPHATIDYLETHANOLAMINE HYDROLYZING PHOSPHOLIPASE D
#147METHODS FOR TREATING CANCER
#148AMIDE-SUBSTITUTED HETEROCYCLIC COMPOUNDS USEFUL AS MODULATORS OF IL-12, IL-23 AND/OR IFN ALPHA RESPONSES
#149CRYSTALLINE FORM OF LANIFIBRANOR
#150A METHOD FOR THE PREPARATION OF INDOLE-3-CARBOXYLIC ACID DERIVATIVES
#1512,3-DIHYDROBENZO[B][1,4]DIOXIN-6-YL CONTAINING COMPOUNDS USEFUL AS IMMUNOMODULATORS
#152QUINAZOLINES AS POTASSIUM ION CHANNEL INHIBITORS
#153POTENT ASGPR-BINDING COMPOUNDS FOR THE DEGRADATION OF IMMUNOGLOBULINS AND OTHER PROTEINS
#154CYCLOOLEFIN SUBSTITUTED HETEROAROMATIC COMPOUNDS AND THEIR USE
#155COMPOUNDS AND METHODS FOR THE TARGETED DEGRADATION OF ANDROGEN RECEPTOR
#156SUBSTITUTED BENZAMIDES AS HERBICIDES
#157THIOBENZIMIDAZOLE DERIVATIVE PREPARATION METHOD AND NOVEL INTERMEDIATE THEREFOR
#158P2X3 INHIBITOR COMPOUND, SALT THEREOF, POLYMORPH THEREOF AND USE THEREOF
#159MULTICYCLIC COMPOUNDS
#160SULFONYL AMIDE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH
#1613,4-DIHYDROQUINOXALINE-2-CARBOXIMIDE DERIVATIVE COMPOUND AND PHARMACEUTICAL COMPOSITION COMPRISING SAME FOR PREVENTING OR TREATING CANCER DISEASE
#162THIOBENZIMIDAZOLE DERIVATIVE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, AND USE THEREOF
#163HETEROCYCLIC COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL AND PSYCHOLOGICAL DISORDERS
#164ANTIMICROBIAL AGENTS
#165COMPOUND, POLYMERIZABLE COMPOSITION, POLYMER, HOLOGRAPHIC RECORDING MEDIUM, OPTICAL MATERIAL, AND OPTICAL COMPONENT
#166THIAZOLE DERIVATIVE COMPOUND AND USES THEREOF
#167METHOD FOR FORMING AMINOTHIAZOLE DERIVATIVES WITH SUPER-PARAMAGNETIC NANOPARTICLE CATALYST
#168MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR
#169Transcription Factor Brn2 Inhibitory Compounds for Use as Therapeutics
#170BCL-XL DEGRADERS AND USES THEREOF
#171COMPOUNDS, SALTS THEREOF AND METHODS FOR TREATMENT OF DISEASES
#172NOVEL RAS INHIBITORS
#1732-OXO-DIHYDROQUINOLINE-3-CARBOXAMIDE DERIVATIVES AS GABA TYPE A RECEPTOR MODULATORS
#174THIADIAZOLE COMPOUND, AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING INFLAMMATORY DISEASES, INCLUDING SAME
#175METHOD OF FORMING BOND BY COUPLING REACTION
#176PROPIONIC ACID DERIVATIVE AND MEDICAL USE THEREOF
#177COMPOUNDS FOR TREATMENT OF CANCER
#178NON-AROMATIC CYCLIC-PYRIMIDINE ANALOGS AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS
#179Telomerase Reverse Transcriptase (TERT) Expression Enhancing Compounds and Methods for Using the Same
#180RIP1 MODULATORS, PREPARATIONS, AND USES THEREOF
#181ELECTRON ACCEPTOR, AND REAGENT LAYER AND SENSOR EACH USING SAME
#182NEW ANTIVIRAL TRIAZOLE DERIVATIVES, THEIR SYNTHESIS AND THEIR USE FOR TREATMENT OF MAMMALIAN VIRAL INFECTIONS
#183INHIBITORS OF RNA HELICASE DHX9 AND USES THEREOF
#184PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS
#185METHOD FOR FORMING A SCHIFF BASE WITH CATALYTIC SUPER-PARAMAGNETIC IRON OXIDE NANOPARTICLES
#186PYRROLIDINE COMPOUNDS
#187MRGPRX2 MODULATORS AND RELATED METHODS OF TREATMENT
#188ARYL-OR HETEROARYL-SUBSTITUTED BENZENE COMPOUNDS
#189MODULATORS OF ACKR3 AND USES THEREOF
#190A METHOD FOR TREATING ROSAH SYNDROME
#191SUBSTITUTED 1,2,4-TRIAZOLES AND METHODS OF USE
#192MCL-1 INHIBITORS
#1931,4-DIHYDROQUINAZOLINONE COMPOUNDS AND USES THEREOF
#194PROTEIN DEGRADERS AND USES THEREOF
#195THIAZOLE COMPOUNDS AND METHODS OF USE THEREOF
#196MODULATORS OF THE INTEGRATED STRESS PATHWAY
#197CATHEPSIN K INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF
#198THIOSTREPTON-INSPIRED COMPOUNDS FOR TREATMENT OF CANCER AND PREPARATION THEREOF
#199RAD51 INHIBITORS
#200THIADIAZOLONE DERIVATIVES USEFUL AS AMPK ACTIVATOR
#201SMO MODULATOR COMPOUNDS
#202PYRIDINYL DERIVATIVES AS SODIUM CHANNEL ACTIVATORS
#203SMALL MOLECULE PROTEIN SYNTHESIS MODULATORS
#204MASP-2 INHIBITORS AND METHODS OF USE
#205MYST Inhibitors
#206PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF
#207KAT6 Inhibitors
#208DIARYL COMPOUND AS TUBULIN/SRC DUAL TARGET INHIBITOR
#209SULFOXIMINE GLYCOSIDASE INHIBITORS
#210cGAS ANTAGONIST COMPOUNDS
#211PYRIDAZINE DERIVATIVES AND RELATED USES
#212BICYCLIC-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS
#213COMPOSITIONS AND METHODS FOR TREATING CANCER
#214PEPTIDYL NITRILE COMPOUND AND USE THEREOF
#215NOVEL KALIRIN INHIBITORS FOR REGULATION OF SYNAPTIC PLASTICITY AND NEUROPATHIC PAIN TREATMENT
#216SPIROCYCLIC CAV2.3 ANTAGONISTS
#2172-SUBSTITUTED THIAZOLE HSD17B13 INHIBITORS AND USES THEREOF
#218MERCAPTOPYRIMIDINE COMPOUNDS THAT INHIBIT NONHOMOLOGOUS END JOINING AND METHODS THEREOF
#219MEK INHIBITORS AND METHODS OF THEIR USE
#220COMPOSITIONS AND METHODS FOR TREATING CANCER
#221RIPK3 INHIBITORS AND METHODS OF USE
#222ENHANCERS OF PARTICULATE GUANYLYL CYCLASE RECEPTOR A
#223COMPOUNDS AND METHODS OF ACTIVATING LIPOPROTEIN LIPASE
#224NOVEL DRP-1 INHIBITORS AS THERAPEUTIC AGENTS
#225COMPOSITIONS AND METHODS FOR MAKING AND USING SMALL MOLECULES FOR TUBULIN-TARGETED THERAPY IN THE TREATMENT OF CANCERS AND RELATED CONDITIONS
#226SMALL MOLECULE PROTEIN SYNTHESIS MODULATORS
#227SUBSTITUTED HETEROCYCLES AS HSET INHIBITORS
#228PYRAZOLE-SUBSTITUTED CYCLOPENTANOL ESTER DERIVATIVE AND USE THEREOF
#229PI3K-ALPHA INHIBITORS AND METHODS OF USE THEREOF
#2304-SUBSTITUTED AMINOISOQUINOLINE DERIVATIVES
#231NSD2-TARGETED CHECMICAL DEGRADERTS AND COMPOSITIONS AND METHODS OF USE THEREOF
#232PYRIDAZINONES AS PARP7 INHIBITORS
#233Novel Aminobenzene Derivative Having Cancer Cell Growth Inhibitory Effect, and Preventive or Therapeutic Pharmaceutical Composition Containing Same as Active Ingredient
#234SUBSTITUTED (1,2,3,4-TETRAHYDROCYCLOPENTA[b]INDOL-3-YL)ACETIC ACID DERIVATIVES USEFUL IN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISORDERS
#235SOLID FORMS OF A BENZTHIAZOLE-PIPERAZINYL-OXAZOLE COMPOUND AND METHODS OF USE THEREOF
#236COMPOSITIONS AND METHODS OF USE TO TREAT 12-LIPOXYGENASE (12-LOX) MEDIATED DISEASES
#237BENZOTHIAZOLE, BENZOISOXAZOLE, AND BENZODIOXOLE ANALOGS AS RXFP1 RECEPTOR AGONISTS
#238NOVEL CANNABICHROMENIC ACID DERIVATIVE, PREPARATION METHOD THEREFOR, AND COMPOSITION COMPRISING SAME FOR IMPROVING COGNITIVE FUNCTION
#239HETEROCYCLIC COMPOUNDS AS DYRK1A INHIBITORS
#240DIAMINOPYRIMIDINES AS P2X3 AND P2X2/3 ANTAGONISTS
#241THIADIAZINE DERIVATIVES
#242Anti-inflammatory Compounds, Pharmaceutical Compositions, and Treatment Methods
#243Pharmaceutical Compounds and Compositions as C-Kit Kinase Inhibitors
#244CARDIAC SARCOMERE INHIBITORS
#245TLR MODULATOR AND USE THEREOF
#246MODULATORS OF MYOCYTE LIPID ACCUMULATION AND INSULIN RESISTANCE AND METHODS OF USE THEREOF
#247SMALL MOLECULE INHIBITORS OF PR3 AND HNE AND USES THEREOF
#248THERAPEUTIC COMPOUNDS AND METHODS
#249CRYSTALLINE FORMS OF A DEOXYCYTIDINE KINASE INHIBITOR AND USES THEREOF
#250N-[5-(aminosulfonyl)-4-methyl-1,3-thiazol-2-yl]-N-methyl-2-[4-(2-pyridinyl)-phenyl]-acetamide free base hemihydrate, methods of manufacture and uses thereof
#251PREPARATION OF INDOLONE-3YL-HYDRAZONO-SUBSTITUTED 1,3-THIAZOLIDINONE DERIVATIVES AND APPLICATION THEREOF
#252CHROMOBOX PROTEIN INHIBITORS AND USES THEREOF
#253QUINOLINE DERIVATIVES
#254EGFR INHIBITORS AND METHODS OF USE THEREOF
#255TETRAHYDROQUINAZOLINE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS
#256N-(5-SUBSTITUTED-[(1,3,4-THIADIAZOLYL) OR (THIAZOLYL)])(SUBSTITUTED)CARBOXAMIDE COMPOUNDS AND USE THEREOF FOR INHIBITING HUMAN POLYMERASE THETA
#257ENHANCERS OF PARTICULATE GUANYLYL CYCLASE RECEPTOR A
#258QUINAZOLINONE DIONE COMPOUNDS AND USES THEREOF
#259ARYL OR HETEROARYL DERIVATIVE, AND PHARMACEUTICAL COMPOSITION COMPRISING SAME AS ACTIVE INGREDIENT FOR PREVENTION OR TREATMENT OF KINASE-RELATED DISEASES
#260SELECTIVE PEPTIDOMIMETIC MODULATORS OF CAV2.2 (N-TYPE) VOLTAGE-GATED CALCIUM CHANNELS AND USES THEREOF
#261PEROXIREDOXIN 3 INHIBITORS AND METHODS OF USE FOR TREATING CANCER
#262ARYL HYDROCARBON RECEPTOR (AHR) AGONISTS AND USES THEREOF
#263LONG-CHAIN COMPOUND THAT ACTS ON ACLY, PREPARATION METHOD THEREFOR AND USE THEREOF
#264HETEROCYCLIC COMPOUNDS AND USES THEREOF
#265FUSED BICYCLIC SUBSTITUTED N-(1H-INDOL-7-YL)BENZENESULFONAMIDES AND USES THEREOF
#266NOVEL PYRIDINE DERIVATIVE COMPOUND AS RON INHIBITOR
#267FLUORINE-CONTAINING PYRAZOLE COMPOUND AND PRODUCTION METHOD THEREFOR
#268CARBONIC ANHYDRASE IX-TARGETING RADIOACTIVE DIAGNOSTIC AND THERAPEUTIC MEDICAMENT AND METHOD FOR PREPARING SAME
#269HMOX1 INDUCERS
#270ORGANIC COMPOUNDS
#271COMPOSITIONS AND METHODS FOR THE TREATMENT OF CANCER
#272Methods for treating cancer
#273SULFONYLUREAS AND RELATED COMPOUNDS AND USE OF SAME
#274COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY
#275Substituted Quinoxalines
#276QUINACRINE AND DERIVATIVES THEREOF FOR TREATMENT OF VIRAL INFECTIONS
#277ISOQUINOLINONES AND QUINOLINONES AS MODULATORS OF POLRMT
#278PHENYL CORE COMPOUNDS AS MGLU5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME
#279Compounds for Treating Cannabinoid Toxicity and Acute Cannabinoid Overdose
#280COMPOUNDS AND METHODS FOR MODULATING INTERLEUKIN-2-INDUCIBLE T-CELL KINASE
#281SMARCA DEGRADERS AND USES THEREOF
#282INHIBITORS OF TRANSGLUTAMINASES
#283BIFUNCTIONAL DEGRADERS COMPRISING A TEAD BINDER
#284NOVEL INHIBITOR OF HYPE-MEDIATED AMPYLATION
#285PRMT5 INHIBITOR AND THE USE THEREOF
#286MODULATORS OF PrPC AND USES THEREOF
#287THIADIAZOLEAMIDE DERIVATIVES AND THEIR APPLICATIONS
#288INHIBITORS OF ALPHA-HEMOLYSIN OF STAPHYLOCOCCUS AUREUS
#289NAMPT INHIBITORS AND USES THEREOF
#290INHIBITORS OF TRANSGLUTAMINASES
#291N-substituted-dioxocyclobutenylamino-3-hydroxy-picolinamides useful as CCR6 inhibitors
#292CERTAIN PLADIENOLIDE COMPOUNDS AND METHODS OF USE
#293SUBSTITUTED TETRAHYDROFURAN-2-CARBOXAMIDES AS MODULATORS OF SODIUM CHANNELS
#294JAK2 INHIBITORS AND METHODS OF USE THEREOF
#295ALLOSTERIC MODULATORS OF NICOTINIC ACETYLCHOLINE RECEPTORS
#296Fused Heterobicyclic Antiviral Agents
#297BICYCLIC 1,4-DIAZEPANONES AND THERAPEUTIC USES THEREOF
#298RAD51 INHIBITORS
#299SMALL MOLECULE UREA DERIVATIVES AS STING ANTAGONISTS
#300HETEROCYCLIC COMPOUNDS AS SEROTONIN (5-HT) 5-HT2A AND 5-HT2C RECEPTOR POSITIVE ALLOSTERIC MODULATORS