ClassID:

95363

C07D471/08 - CPC Classification

Classification description:

Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups  -  in which the condensed system contains two hetero rings Bridged systems

Recent Application in this class:
#1
20260138987
2026-05-21

MUSCARINIC ACETYLCHOLINE M1 RECEPTOR ANTAGONISTS

#2
20260132143
2026-05-14

HETEROCYCLIC INHIBITORS OF KRAS G12C MUTANT PROTEINS AND USES THEREOF

#3
20260132139
2026-05-14

HIV INHIBITOR COMPOUNDS

#4
20260132132
2026-05-14

3A,4,5,6-TETRAHYDRO-1 H-PYRAZOLO[3,4-C]PYRIDIN-7(7AH)-ONE DERIVATIVES AS FACTOR XIIA INHIBITORS

#5
20260103456
2026-04-16

COMPOUND, PHARMACEUTICAL COMPOSITION CONTAINING SAME, SYNTHESIS METHOD THEREFOR AND USE THEREOF

#6
20260098038
2026-04-09

NOVEL DERIVATIVES HAVING 2,3-DIHYDRO-1H-INDENE OR 2,3-DIHYDROBENZOFURAN MOIETY OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME

#7
20260098032
2026-04-09

METHODS AND COMPOUNDS FOR RESTORING MUTANT p53 FUNCTION

#8
20260092057
2026-04-02

BCL-XL/BCL-2 DEGRADERS AND USES THEREOF

#9
20260078103
2026-03-19

ISOQUINOLONES AS PI3K INHIBITORS

#10
20260078094
2026-03-19

ANTI-VIRAL COMPOUNDS

#11
20260078092
2026-03-19

SULFONYL CARBOXAMIDE COMPOUND, THEIR DERIVATIVES, AND USES THEREOF

#12
20260055107
2026-02-26

SERIES OF NITROGEN-CONTAINING BRIDGED HETEROCYCLIC COMPOUNDS AND PREPARATION METHOD THEREFOR

#13
20260049063
2026-02-19

ALKYNYL QUINAZOLINE COMPOUNDS

#14
20260042777
2026-02-12

PIPERIDYLUREA COMPOUNDS AND METHODS OF USE THEREOF

#15
20260042759
2026-02-12

INHIBITOR CONTAINING BICYCLIC DERIVATIVE, PREPARATION METHOD THEREFOR AND USE THEREOF

#16
20260042734
2026-02-12

HETEROCYCLIC RING-SUBSTITUTED AROMATIC COMPOUND, PREPARATION METHOD THEREFOR, AND USE THEREOF

#17
20260035362
2026-02-05

GLP-1R AGONISTS AND USES THEREOF

#18
20260034119
2026-02-05

5-METHOXY-N,N-DIMETHYLTRYPTAMINE ANALOGS, THEIR SYNTHESIS, AND METHODS FOR TREATMENT OF NEUROLOGICAL, PSYCHIATRIC, AND SUBSTANCE USE DISORDERS

#19
20260022108
2026-01-22

ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF

#20
20260015344
2026-01-15

PAN-KRAS INHIBITORS

#21
20260008779
2026-01-08

CRYSTALLINE FORMS OF CFTR MODULATORS

#22
20260008768
2026-01-08

UREA DERIVATIVES FOR INHIBITING NLRP3 AND USES THEREOF

#23
20260007684
2026-01-08

AMIDE DERIVATIVES FOR INHIBITING NLRP3 AND USES THEREOF

#24
20260001860
2026-01-01

METHODS AND COMPOSITIONS OF INHIBITING DCN1-UBC12 INTERACTION

#25
20250387403
2025-12-25

SELECTIVE SIGMA-2 RECEPTOR LIGANDS AS MODULATORS OF TMEM97

#26
20250368644
2025-12-04

DURLOBACTAM CRYSTALLINE FORMS

#27
20250368620
2025-12-04

ARNT Degrading Compounds and Uses Thereof

#28
20250361234
2025-11-27

COMPOUNDS, COMPOSITIONS, AND METHODS

#29
20250340529
2025-11-06

Heterocyclic Compounds as Immunomodulators of PD-L1 Interactions

#30
20250326768
2025-10-23

Benzodiazepine Derivatives as RSV Inhibitors

#31
20250325552
2025-10-23

SUBSTITUTED THIADIAZOLYL DERIVATIVES AS DNA POLYMERASE THETA INHIBITORS

#32
20250320203
2025-10-16

4-(3H-PYRAZOLO[4,3-F]QUINOLIN-7-YL)-N-(2-(DIMETHYLAMINO)ETHYL)BENZAMIDE- OR HYDROXAMIC ACID COMPOUNDS, COMPOSITIONS, AND METHODS OF USE

#33
20250320197
2025-10-16

THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF

#34
20250320185
2025-10-16

AMINOHETEROARYL KINASE INHIBITORS

#35
20250313535
2025-10-09

ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF

#36
20250289818
2025-09-18

HETEROCYCLIC DERIVATIVES, PHARMACEUTICAL COMPOSITIONS AND THEIR USE IN THE TREATMENT, AMELIORATION OR PREVENTION OF CANCER

#37
20250289801
2025-09-18

EGFR INHIBITORS

#38
20250288595
2025-09-18

TROPOMYOSIN-RELATED KINASE (TRK) INHIBITORS

#39
20250282766
2025-09-11

PTPN2/PTP1B Degrader and Therapeutic Method Thereof

#40
20250276964
2025-09-04

Benzisoxazole Derivatives and Uses thereof

#41
20250275959
2025-09-04

COMPOUNDS AND METHODS OF THEIR USE

#42
20250270225
2025-08-28

COMPOSITIONS AND METHODS FOR INHIBITION OF RAS

#43
20250270220
2025-08-28

SOS1 INHIBITORS

#44
20250268910
2025-08-28

NICOTINIC ACETYLCHOLINE RECEPTOR LIGANDS

#45
20250263424
2025-08-21

KRAS INHIBITORS

#46
20250263412
2025-08-21

NON-HYDROXAMATE HDAC6 INHIBITORS AND RELATED METHODS OF USE

#47
20250263405
2025-08-21

HISTONE DEACETYLASE 6 INHIBITOR COMPOUNDS AND USES THEREOF

#48
20250263394
2025-08-21

COMPOUNDS, PREPARATION METHODS AND USES THEREOF

#49
20250257192
2025-08-14

UREA-GLYOXAL CROSSLINKING COMPOUNDS FOR PHENOLIC BINDER COMPOSITIONS

#50
20250257059
2025-08-14

PROTEIN TYROSINE PHOSPHATASE INHIBITORS AND USES THEREOF

#51
20250257035
2025-08-14

1,4-Substituted Piperidine Derivatives

#52
20250250230
2025-08-07

HETEROCYCLIC COMPOUND

#53
20250243210
2025-07-31

CRBN E3 LIGASE LIGAND COMPOUND, PROTEIN DEGRADER DEVELOPED BASED THEREON AND THEIR APPLICATIONS

#54
20250243183
2025-07-31

IMIDAZOLYL PYRIMIDINYLAMINE COMPOUNDS AS CDK2 INHIBITORS

#55
20250241915
2025-07-31

COMPOUNDS FOR THE TREATMENT OF BRAF-ASSOCIATED DISEASES AND DISORDERS

#56
20250236614
2025-07-24

BICYCLIC TETRAHYDROAZEPINE DERIVATIVES

#57
20250230127
2025-07-17

MONO- OR DI-SUBSTITUTED INDOLE DERIVATIVES AS DENGUE VIRAL REPLICATION INHIBITORS

#58
20250223292
2025-07-10

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE

#59
20250214970
2025-07-03

PYRIDINYLACETAMIDE DERIVATIVES AS SODIUM CHANNEL ACTIVATORS

#60
20250214965
2025-07-03

COMPOUND AS KIF18A INHIBITOR

#61
20250213698
2025-07-03

BICYCLIC HETEROCYCLES AND THEIR LIGANDS FOR TARGETED DELIVERY OF THERAPEUTIC AGENTS

#62
20250213555
2025-07-03

SUBSTITUTED TETRAHYDROFURAN ANALOGS AS MODULATORS OF SODIUM CHANNELS

#63
20250206760
2025-06-26

NITROGEN-CONTAINING HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATION THEREOF

#64
20250206752
2025-06-26

PI3K INHIBITORS

#65
20250206724
2025-06-26

SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS

#66
20250206717
2025-06-26

COMPOUND HAVING ANTI-TUMOR ACTIVITY AND USE THEREOF

#67
20250197395
2025-06-19

IBOGAINE AND NORIBOGAINE ANALOGS AND USES THEREOF

#68
20250179065
2025-06-05

HDAC6 INHIBITORS AND USES THEREOF

#69
20250179032
2025-06-05

HETEROCYCLIC INHIBITORS OF GLUT9 FOR TREATMENT OF DISEASE

#70
20250171462
2025-05-29

COMPOUNDS, COMPOSITIONS, AND METHODS

#71
20250171453
2025-05-29

HETEROCYCLIC COMPOUNDS AND USES THEREOF

#72
20250171432
2025-05-29

COMPOUNDS AND METHODS OF USE

#73
20250171431
2025-05-29

HETEROCYCLIC INHIBITORS OF IGF-1R FOR TREATMENT OF DISEASE

#74
20250160204
2025-05-15

MATERIALS FOR ELECTRONIC DEVICES

#75
20250154141
2025-05-15

BCL-XL/BCL-2 DUAL DEGRADERS FOR TREATMENT OF CANCERS

#76
20250154114
2025-05-15

MATERIAL FOR METAL PATTERNING, HETEROCYCLIC COMPOUND, THIN FILM FOR METAL PATTERNING, ORGANIC ELECTROLUMINESCENT DEVICE, ELECTRONIC DEVICE, AND METHOD FOR FORMING METAL PATTERN

#77
20250145617
2025-05-08

SIGMA-2 RECEPTOR LIGAND DRUG CONJUGATES AS ANTITUMOR COMPOUNDS, METHODS OF SYNTHESIS AND USES THEREOF

#78
20250145589
2025-05-08

PYRIDINE DERIVATIVE AND USE THEREOF

#79
20250129058
2025-04-24

PTPN2/PTP1B degrader and therapeutic method thereof

#80
20250129044
2025-04-24

PYRIDINYL DERIVATIVES AS SODIUM CHANNEL ACTIVATORS

#81
20250129027
2025-04-24

FATTY ACID AMIDE HYDROLASE MODULATORS, COMPOSITIONS COMPRISING THE SAME AND USES THEREOF

#82
20250122185
2025-04-17

COMPOSITIONS AND METHODS COMPRISING SUBSTITUTED N-(2-CHLORO-6-METHYLPHENYL)-2-((6-(6-MEMBERED HETEROCYCLOALKYL)-2-METHYLPYRIMIDIN-4-YL)AMINO)THIAZOLE-5-CARBOXAMIDE ANALOGUES

#83
20250115608
2025-04-10

HORMONE RECEPTOR MODULATORS FOR TREATING METABOLIC CONDITIONS AND DISORDERS

#84
20250115591
2025-04-10

NOVEL SULFONAMIDE CARBOXAMIDE COMPOUNDS

#85
20250115586
2025-04-10

BENZAMIDES OF PYRAZOLYLAMINO- PYRIMIDINYL DERIVATIVES, AND COMPOSITIONS AND METHODS THEREOF

#86
20250115579
2025-04-10

QUINOLINE cGAS ANTAGONIST COMPOUNDS

#87
20250115574
2025-04-10

2-PYRAZOLE ANILINES AND RELATED ANALOGS FOR INHIBITING YAP/TAZ-TEAD

#88
20250109122
2025-04-03

CYCLOALKYL PYRIMIDINES AS FERROPORTIN INHIBITORS

#89
20250092057
2025-03-20

HETEROCYCLIC RIP1 INHIBITORY COMPOUNDS

#90
20250092031
2025-03-20

RIPK3 INHIBITORS AND METHODS OF USE

#91
20250084082
2025-03-13

HUPERZINE B CRYSTAL AND PREPARATION AND APPLICATION THEREOF

#92
20250084064
2025-03-13

2-AMINO-N-HETEROARYL-NICOTINAMIDES AS NAV1.8 INHIBITORS

#93
20250082609
2025-03-13

HETEROCYCLIC SULFONAMIDE DERIVATIVES AND PHARMACEUTICAL USES THEREOF

#94
20250066398
2025-02-27

RECEPTOR INHIBITOR, PHARMACEUTICAL COMPOSITION COMPRISING SAME, AND USE THEREOF

#95
20250064993
2025-02-27

NOVEL BISPIDINE-BASED METAL CHELATING LIGANDS DISPLAYING GOOD RELAXIVITY

#96
20250059191
2025-02-20

CRYSTALLINE FORMS OF DIAZABICYCLOOCTANE DERIVATIVE AND PRODUCTION PROCESS THEREOF

#97
20250059179
2025-02-20

Heterocyclic Compounds and Methods of Use

#98
20250059141
2025-02-20

TLR MODULATOR AND USE THEREOF

#99
20250057817
2025-02-20

KRAS G12C INHIBITORS AND METHODS OF USING THE SAME

#100
20250051344
2025-02-13

BIFUNCTIONAL SELECTIVE DEGRADERS OF SMARCA2 AND THERAPEUTIC USES THEREOF

#101
20250051326
2025-02-13

Crystalline forms of CFTR modulators

#102
20250042910
2025-02-06

HIV INHIBITOR COMPOUNDS

#103
20250034116
2025-01-30

1,4-DIHETEROCYCLIC SUBSTITUTED AROMATIC RING OR AROMATIC HETEROCYCLIC COMPOUND AND USE THEREOF

#104
20250034110
2025-01-30

LPAR1 ANTAGONISTS AND USES THEREOF

#105
20250032454
2025-01-30

KDM1A INHIBITORS FOR THE TREATMENT OF DISEASE

#106
20250026749
2025-01-23

GLUCOSYLCERAMIDE SYNTHASE INHIBITORS

#107
20250026722
2025-01-23

SUBSTITUTED QUINOLINES AS IMPROVED NF-KB-INDUCING KINASE (NIK) INHIBITORS

#108
20250025443
2025-01-23

COMPOUNDS AND METHODS FOR TREATING CORONA VIRUSES

#109
20250019376
2025-01-16

CHROMANE AMIDINE MONOBACTAM ANTIBIOTICS

#110
20250002471
2025-01-02

6-SUBSTITUTED INDOLE COMPOUNDS

#111
20240425490
2024-12-26

SULFAMIDE RIBONUCLEOTIDE REDUCTASE (RNR) INHIBITORS AND USES THEREOF

#112
20240417388
2024-12-19

BENZIMIDAZOLONE DERIVED INHIBITORS OF BCL6

#113
20240415847
2024-12-19

BETA-LACTAMASE INHIBITORS AND USES THEREOF

#114
20240400591
2024-12-05

COMPOUNDS TARGETING MUTANT OF P53

#115
20240400584
2024-12-05

COMPOUNDS AND METHODS FOR MODULATING SPLICING

#116
20240398959
2024-12-05

C3-CARBON LINKED GLUTARIMIDE DEGRONIMERS FOR TARGET PROTEIN DEGRADATION

#117
20240398828
2024-12-05

HETERO-ATOM CONTAINING COMPOUNDS AND USES THEREOF

#118
20240391920
2024-11-28

RING-MODIFIED PROLINE SHORT PEPTIDE COMPOUND AND USE THEREOF

#119
20240391919
2024-11-28

DIAZABICYCLOOCTANONES AS INHIBITORS OF SERINE BETA-LACTAMASES

#120
20240391882
2024-11-28

Substituted Quinoxalines

#121
20240390383
2024-11-28

DIOXAZINES AND THEIR USE IN TREATMENT OF GBA-RELATED DISEASES

#122
20240383897
2024-11-21

THERAPEUTIC COMPOUNDS

#123
20240383884
2024-11-21

COMPOUNDS AND METHODS FOR MODULATING INTERLEUKIN-2-INDUCIBLE T-CELL KINASE

#124
20240383876
2024-11-21

TLR7/8 ANTAGONISTS AND USES THEREOF

#125
20240382494
2024-11-21

THERAPEUTIC COMPOUNDS

#126
20240376055
2024-11-14

INHIBITORS OF TRANSGLUTAMINASES

#127
20240368205
2024-11-07

CHELATE COMPOUNDS

#128
20240368163
2024-11-07

COMPOUNDS AND METHODS FOR MODULATING SPLICING

#129
20240368136
2024-11-07

BENZOLACTAM COMPOUNDS AS PROTEIN KINASE INHIBITORS

#130
20240368129
2024-11-07

SULPHONYL UREA DERIVATIVES AS NLRP3 INFLAMMASOME MODULATORS

#131
20240368119
2024-11-07

RIP1 INHIBITORY COMPOUNDS AND METHODS FOR MAKING AND USING THE SAME

#132
20240368079
2024-11-07

PROCESS FOR THE PREPARATION OF OPTICALLY PURE ENANTIOMERS OF CYCLIC IMINIUM SALTS AND THEIR USE AS CATALYSTS

#133
20240366802
2024-11-07

GADOLINIUM BEARING PCTA-BASED CONTRAST AGENTS

#134
20240360165
2024-10-31

INHIBITORS OF CYCLIN DEPENDENT KINASE 7 (CDK7)

#135
20240360155
2024-10-31

Benzodiazepine derivatives as RSV inhibitors

#136
20240360146
2024-10-31

BRUTON'S TYROSINE KINASE AND MUTANT DEGRADER, COMPOSITION AND APPLICATION THEREOF

#137
20240336611
2024-10-10

ANALOGS FOR THE TREATMENT OF DISEASE

#138
20240336596
2024-10-10

PARP7 INHIBITOR AND USE THEREOF

#139
20240327392
2024-10-03

HETEROCYCLOALKYL-SUBSTITUTED POLYHETEROAZOLE DERIVATIVES AS MEDICAMENTS FOR TREATING AND/OR PREVENTING RS VIRUS INFECTIONS

#140
20240327380
2024-10-03

BTK INHIBITORS

#141
20240327378
2024-10-03

INHIBITORS OF (ALPHA-V)(BETA-6) INTEGRIN

#142
20240327354
2024-10-03

GRAM-NEGATIVE BACTERIA EFFLUX PUMP INHIBITORS

#143
20240317769
2024-09-26

KRAS G12D INHIBITORS

#144
20240300964
2024-09-12

COMPOSITIONS AND METHODS FOR INHIBITION OF RAS

#145
20240300940
2024-09-12

Phenothiazinyl Compounds and Uses

#146
20240294499
2024-09-05

TARGETED PROTEIN DEGRADATION USING BIFUNCTIONAL COMPOUNDS THAT BIND UBIQUITIN LIGASE AND TARGET MCL-1 PROTEIN

#147
20240287108
2024-08-29

nSMASE2 INHIBITOR PRODRUGS WITH ENHANCED ORAL AND BRAIN EXPOSURES

#148
20240287020
2024-08-29

SUBSTITUTED BENZODIAZOLES AND USE THEREOF IN THERAPY

#149
20240285817
2024-08-29

BISPIDINE DERIVATIVES AND THE USE THEREOF

#150
20240285808
2024-08-29

MOLECULAR PROBES FOR IN VIVO DETECTION OF ALDEHYDES

#151
20240285614
2024-08-29

PHENOL RIBONUCLEOTIDE REDUCTASE (RNR) INHIBITORS AND USES THEREOF

#152
20240270700
2024-08-15

COMPOSITIONS AND USES THEREOF

#153
20240254126
2024-08-01

NOVEL BISPIDONE LIGANDS AND TRANSITION METAL COMPLEXES THEREOF

#154
20240246973
2024-07-25

Cathinone Derivatives, Pharmaceutical Formulations, and Methods

#155
20240246909
2024-07-25

EBNA1 Inhibitors and Methods Using Same

#156
20240239788
2024-07-18

SMALL MOLECULE INHIBITORS OF KRAS G12D MUTANT

#157
20240228506
2024-07-11

RIPK1 INHIBITORS AND METHODS OF USE

#158
20240217964
2024-07-04

QUINUCLIDINONE ANALOGUES AS ANTICANCER AGENTS

#159
20240217953
2024-07-04

BICYCLIC SUBSTITUTED AROMATIC CARBOXYLIC ACID COMPOUNDS

#160
20240208993
2024-06-27

Five- and six-membered compound, and preparation method therefor and pharmaceutical composition and use thereof

#161
20240190846
2024-06-13

Thyroid hormone receptor agonists and use thereof

#162
20240190842
2024-06-13

SUBSTITUTED QUINOLINONE-8-CARBONITRILE DERIVATIVES HAVING ANDROGEN DEGRADATION ACTIVITY AND USES THEREOF

#163
20240189322
2024-06-13

Tropomyosin-related kinase (trk) inhibitors

#164
20240182684
2024-06-06

UREA-GLYOXAL CROSSLINKING COMPOUNDS FOR PHENOLIC BINDER COMPOSITIONS

#165
20240182471
2024-06-06

METHODS AND COMPOSITIONS FOR SUBSTITUTED ARYLCYCLOHEPTANE ANALOGS

#166
20240182414
2024-06-06

Mono- or di-substituted indole derivatives as dengue viral replication inhibitors

#167
20240174642
2024-05-30

HETEROCYCLIC COMPOUNDS CAPABLE OF ACTIVATING STING

#168
20240174641
2024-05-30

HETEROCYCLIC COMPOUNDS CAPABLE OF ACTIVATING STING

#169
20240173307
2024-05-30

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#170
20240150285
2024-05-09

Modulators of complex I

#171
20240140957
2024-05-02

BRIDGED COMPOUNDS AS KRAS G12D INHIBITOR AND DEGRADER AND THE USE THEREOF

#172
20240140932
2024-05-02

Cycloalkyl pyrimidines as ferroportin inhibitors

#173
20240132499
2024-04-25

FUSED PYRROLINES WHICH ACT AS UBIQUITIN-SPECIFIC PROTEASE 30 (USP30) INHIBITORS

#174
20240132497
2024-04-25

Azabicyclo and diazepine derivatives

#175
20240132496
2024-04-25

IONIC COMPOUND, ABSORBENT AND ABSORPTION DEVICE

#176
20240124422
2024-04-18

MUTANT PI3K-ALPHA INHIBITORS AND THEIR USE AS PHARMACEUTICALS

#177
20240117407
2024-04-11

Morphinan compounds

#178
20240114782
2024-04-04

INDOLO[3.2.1-JK]CARBAZOLE-6-CARBONITRILE DERIVATIVES AS BLUE FLUORESCENT EMITTERS FOR USE IN OLEDS

#179
20240109890
2024-04-04

BRIDGED HETEROCYCLYL-SUBSTITUTED PYRIMIDINE COMPOUNDS, PREPARATION METHOD AND MEDICAL USE THEREOF

#180
20240109868
2024-04-04

EP300/CBP MODULATOR, PREPARATION METHOD THEREFOR AND USE THEREOF

#181
20240101552
2024-03-28

CARBONYL HETEROCYCLIC COMPOUND AND APPLICATION THEREOF

#182
20240101535
2024-03-28

DIHYDROISOQUINOLINONE DERIVATIVE AND APPLICATION THEREOF

#183
20240093265
2024-03-21

MORPHINAN COMPOUNDS

#184
20240092760
2024-03-21

Quinoline cGAS antagonist compounds

#185
20240083881
2024-03-14

Benzamides of pyrazolyl-amino-pyrimidinyl derivatives, and compositions and methods thereof

#186
20240083872
2024-03-14

CYCLIC AMINE DERIVATIVES HAVING SEROTONIN RECEPTOR BINDING ACTIVITY

#187
20240076291
2024-03-07

MODIFIED ISOINDOLINONES AS GLUCOSYLCERAMIDE SYNTHASE INHIBITORS

#188
20240059691
2024-02-22

ENZYME INHIBITORS

#189
20240051959
2024-02-15

Small molecule inhibitors targeting sporulation

#190
20240051940
2024-02-15

SULFONAMIDES WITH EGFR INHIBITION ACTIVITIES AND THEIR USE THEREOF

#191
20240034733
2024-02-01

KRAS G12D INHIBITORS

#192
20240025882
2024-01-25

Benzamides of pyrazolylamino-pyrimidinyl derivatives, and compositions and methods thereof

#193
20240018143
2024-01-18

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ARYL DERIVATIVES FOR TREATING TRPM3 MEDIATED DISORDERS

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1,4-substituted piperidine derivatives

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MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR

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PYRIDAZINE DERIVATIVES FOR MODULATING NUCLEIC ACID SPLICING

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Aryl, heteroaryl, and heterocyclic pharmaceutical compounds for treatment of medical disorders

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CXCR6 SULFONAMIDE COMPOUNDS

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COMPOUNDS FOR TREATING HUNTINGTON'S DISEASE

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RIP1 Inhibitory Compounds and Methods for Making and Using the Same

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2-OXO-IMIDAZOLIDINE-4-CARBOXAMIDES AS NAV1.8 INHIBITORS

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QUINOLINE COMPOUNDS

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NLRP3 MODULATORS

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ANTAGONIST COMPOUNDS

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Isoquinolin-3-yl carboxamides and preparation and use thereof

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Morphinan derivatives and use thereof

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2-pyrazole anilines and related analogs for inhibiting YAP/TAZ-TEAD

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Compounds useful as inhibitors of ATR kinase

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Pan-tropic entry inhibitors

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GLP-1R MODULATING COMPOUNDS

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CHEMICAL COMPOUNDS

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MORPHINAN DERIVATIVE

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COMPOUNDS AND METHODS FOR MODULATING SPLICING

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FACTOR XI ACTIVATION INHIBITORS

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Sulphonyl urea derivatives as NLRP3 inflammasome modulators

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TARGETED NITROXIDE AGENTS

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HETEROCYCLIC RIP1 INHIBITORY COMPOUNDS

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PYRIDAZINE DERIVATIVES FOR MODULATING NUCLEIC ACID SPLICING

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Hormone receptor modulators for treating metabolic conditions and disorders

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SOS1 inhibitors

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NAMPT MODULATORS

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Fused pyrrolines which act as ubiquitin-specific protease 30 (USP30) inhibitors

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GPR84 ANTAGONISTS AND USES THEREOF

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RIP1 INHIBITORY COMPOUNDS AND METHODS FOR MAKING AND USING THE SAME

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Therapeutic compounds

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COMPOUNDS AND COMPOSITIONS FOR TREATING CNS DISORDERS

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Receptor inhibitor, pharmaceutical composition comprising same, and use thereof

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sGC STIMULATORS

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TRNA SYNTHETASE INHIBITORS

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COMPOUND USED AS KINASE INHIBITOR AND USE THEREOF

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AZEPANE DERIVATIVE

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Quinoline cGAS antagonist compounds

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Tropomyosin-related kinase (Trk) inhibitors

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Substituted indoles and methods of use thereof

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Antimicrobial Compounds and Methods

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COMPOUNDS

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HETEROCYCLIC RIP1 KINASE INHIBITORS

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Phenoxy-pyridyl-pyrimidine compounds and methods of use

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EGFR inhibitors

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1,3-THIAZOL-2-YL SUBSTITUTED BENZAMIDES

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New compounds for treatment of diseases related to DUX4 expression

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SMALL MOLECULE RPN13 INHIBITORS WITH ANTITUMOR PROPERTIES

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MATRIPTASE 2 INHIBITORS AND USES THEREOF

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Sulfonamide carboxamide compounds

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METHODS AND COMPOSITIONS FOR MODULATING SPLICING

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HIV inhibitor compounds

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EGFR inhibitors

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Imidazolyl pyrimidinylamine compounds as CDK2 inhibitors

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BICYCLIC COMPOUND AND USE THEREOF

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METHODS AND COMPOSITIONS FOR MODULATING SPLICING

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Benzolactam compounds as protein kinase inhibitors

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1-AMINOSULFONYL-2-CARBOXYPYRROLE DERIVATIVES AS METALLO-BETA-LACTAMASE INHIBITORS

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HETEROCYCLIC TRPML1 AGONISTS

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Pyrrolo[2,3-d]pyrimidinyl, pyrrolo[2,3-b]pyrazinyl and pyrrolo[2,3-d]pyridinyl acrylamides

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METHODS AND COMPOSITIONS FOR MODULATING SPLICING

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Small molecule inhibitors targeting sporulation

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2023-01-05

NOVEL COMPOUNDS HAVING INHIBITORY ACTIVITY AGAINST GLUCOSYLCERAMIDE SYNTHASE OR PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, PROCESSES FOR PREPARING THE SAME, AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME

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