ClassID:

20409

A61K31/4965 - CPC Classification

Classification description:

Medicinal preparations containing organic active ingredients; Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two nitrogen atoms as the only ring heteroatoms, e.g. piperazine Non-condensed pyrazines

Sub-classes:
Recent Application in this class:
#1
20260152565
2026-06-04

BCMA VH-ONLY CARS

#2
20260151389
2026-06-04

Use of Tetramethylpyrazine Nitrone Derivatives In The Treatment of Ischemic Stroke

#3
20260139035
2026-05-21

HUMAN ANTIBODY AGAINST CORONAVIRUS VARIANTS OR ANTIGEN-BINDING FRAGMENT THEREOF

#4
20260138956
2026-05-21

NOVEL COMPOUNDS AND USES THEREOF

#5
20260137766
2026-05-21

LIPOSOME FORMULATIONS FOR TREATMENT OF ACTIVE TUBERCULOSIS

#6
20260125359
2026-05-07

HETEROARYL COMPOUNDS AS MULTI-TARGET PROTEIN KINASE INHIBITORS

#7
20260124197
2026-05-07

NOVEL HETEROBICYCLIC COMPOUND FOR INHIBITING YAP-TEAD INTERACTION AND PHARMACEUTICAL COMPOSITION COMPRISING SAME

#8
20260097007
2026-04-09

CYSTEAMINE FOR THE TREATMENT, MITIGATION AND PREVENTION OF CORONAVIRAL, E.G., SARS-CoV-2, INFECTIONS

#9
20260085083
2026-03-26

NOVEL COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF

#10
20260085030
2026-03-26

ARTEMISINIC ACID DERIVATIVE, AND PREPARATION METHOD THEREFOR AND APPLICATION THEREOF

#11
20260076961
2026-03-19

COMBINATION TREATMENTS

#12
20260041683
2026-02-12

Compounds with Anti-Acinetobacter Baumannii Activity

#13
20260021109
2026-01-22

PROSTANOID RECEPTOR AGONISTS AS NON-TUBERCULOUS ANTI-MYCOBACTERIAL AGENTS

#14
20260021048
2026-01-22

CONTROLLED RELEASE PHARMACEUTICAL COMPOSITION OF SELEXIPAG OR IT'S ACTIVE METABOLITE

#15
20260007659
2026-01-08

METHOD FOR DETECTING OR TREATING TRIPLE NEGATIVE BREAST CANCER

#16
20260007603
2026-01-08

ALPHA-KETOGLUTARATE (AKG)-BASED POLYMERIC MICROPARTICLES AND METHODS OF USE

#17
20250388542
2025-12-25

ANALOGUES OF PENTAMIDINE AND USES THEREFOR

#18
20250382283
2025-12-18

COMPOUNDS AND THEIR USES AS CD38 INHIBITORS

#19
20250378918
2025-12-11

Phenotype-Based Chemical Screens

#20
20250375443
2025-12-11

IDENTIFICATION AND USE OF SHP2 CONFORMATIONAL DISRUPTORS FOR CANCER TREATMENT

#21
20250368595
2025-12-04

NOVEL MOLECULES

#22
20250333396
2025-10-30

INHIBITING ATAXIA TELANGIECTASIA AND RAD3-RELATED PROTEIN (ATR)

#23
20250332162
2025-10-30

INHIBITING PURINE BIOSYNTHESIS TO INCREASE FAVIPIRAVIR POTENCY AGAINST RNA VIRUS INFECTIONS

#24
20250332161
2025-10-30

PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY

#25
20250332151
2025-10-30

METHODS OF TREATMENT FOR CYSTIC FIBROSIS

#26
20250313535
2025-10-09

ALPHA 4 BETA 7 INTEGRIN MODULATORS AND USES THEREOF

#27
20250312335
2025-10-09

FLT COMBINATION THERAPY FOR CANCER AND COMPOSITIONS THEREFOR

#28
20250304537
2025-10-02

HETEROARENES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND METHODS OF USING THE SAME

#29
20250302775
2025-10-02

METHODS FOR THE TREATMENT OF DEPRESSION

#30
20250296909
2025-09-25

NOVEL BENZENE DERIVATIVE AND IMMUNOSUPPRESSION-RELATED USE THEREOF

#31
20250289826
2025-09-18

PLPRO PROTEIN INHIBITOR, AND PREPARATION METHOD AND APPLICATION THEREOF

#32
20250281482
2025-09-11

BILE ACID RECYCLING INHIBITORS FOR TREATMENT OF PEDIATRIC CHOLESTATIC LIVER DISEASES

#33
20250270173
2025-08-28

PYRIDINE DERIVATIVES FOR TREATING PSYCHIATRIC DISORDERS

#34
20250262273
2025-08-21

MODIFIED CAVEOLIN-1 PEPTIDES FOR THE TREATMENT OF CHRONIC KIDNEY DISEASE

#35
20250241928
2025-07-31

CALMODULIN INHIBITORS FOR THE TREATMENT OF RIBOSOMAL DISORDERS AND RIBOSOMOPATHIES

#36
20250230129
2025-07-17

POLYAMIDE COMPOUNDS, METHOD FOR PREPARING SAME, AND MEDICAL USE THEREOF

#37
20250214942
2025-07-03

INHIBITORS OF RECEPTOR INTERACTING PROTEIN KINASE I FOR THE TREATMENT OF DISEASE

#38
20250214930
2025-07-03

TETRALIN AND TETRAHYDROQUINOLINE COMPOUNDS AS INHIBITORS OF HIF-2ALPHA

#39
20250205518
2025-06-26

PULMONARY HYPERTENSION TREATMENT

#40
20250205260
2025-06-26

ADJUNCTIVE TREATMENT OF MYCOBACTERIAL DISEASES

#41
20250186374
2025-06-12

ALLOSTERIC INHIBITORS OF THE MAIN PROTEASE OF SARS-COV-2

#42
20250170126
2025-05-29

NOVEL B0AT1 INHIBITOR

#43
20250152583
2025-05-15

AMILORIDE FOR USE IN THE TOPICAL TREATMENT OF SOMATOSENSORY IMPAIRMENTS

#44
20250145564
2025-05-08

SULFONYLUREA COMPOUND, PREPARATION METHOD THEREFOR, AND APPLICATION THEREOF

#45
20250144040
2025-05-08

COMPOSITE PARTICLE FORMULATIONS AND APPLICATIONS THEREOF

#46
20250136558
2025-05-01

PYRAZINE COMPOUNDS AS IRREVERSIBLE INHIBITORS OF FLT3

#47
20250134850
2025-05-01

PLANT-DERIVED SMALL MOLECULES AS MARBURG VIRUS INHIBITORS

#48
20250127781
2025-04-24

USE OF INHIBITORS OF BRUTON'S TYROSINE KINASE (BTK)

#49
20250127778
2025-04-24

CANCER IMMUNOTHERAPY COMPOSITION CONTAINING INTERACTION INHIBITOR OF STING AND TRIM29 AS ACTIVE INGREDIENT

#50
20250120969
2025-04-17

METHODS AND COMPOSITIONS FOR TREATING INFLAMMATION INJURY IN THE LUNGS

#51
20250115569
2025-04-10

SULFONAMIDE COMPOUNDS FOR THE TREATMENT OF NEUROLOGICAL CONDITIONS

#52
20250115561
2025-04-10

BIPHENYL-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS

#53
20250109110
2025-04-03

BICYCLIC-SUBSTITUTED EPITHELIAL SODIUM CHANNEL BLOCKING COMPOUNDS

#54
20250099458
2025-03-27

USE OF ANTI-IDIOPATHIC PULMONARY FIBROSIS DRUG NINTEDANIB IN TREATMENT OF TUBERCULOSIS

#55
20250082584
2025-03-13

TRANSDERMAL THERAPEUTIC SYSTEM FOR THE TRANSDERMAL ADMINISTRATION OF SELEXIPAG

#56
20250074938
2025-03-06

CELL-PERMEANT INHIBITORS OF VIRAL CYSTEINE PROTEASES

#57
20250064844
2025-02-27

N4-HYDROXYCYTIDINE AND DERIVATIVES AND ANTI-VIRAL USES RELATED THERETO

#58
20250064789
2025-02-27

KETOAMIDE DERIVATIVES AND PHARMACEUTICAL USES THEREOF

#59
20250051263
2025-02-13

NOVEL IONIZABLE LIPIDS AND LIPID NANOPARTICLES AND METHODS OF USING THE SAME

#60
20250041374
2025-02-06

WILLOW EXTRACT AND ITS USE IN TREATING A VIRAL INFECTION, ALLERGIC REACTION, AND OTHER MEDICAL CONDITIONS

#61
20250034139
2025-01-30

AMINE COMPOUNDS HAVING ANTI-INFLAMMATORY, ANTIFUNGAL, ANTIPARASITIC, AND ANTICANCER ACTIVITY

#62
20250025484
2025-01-23

POLYMERSOME NANOPARTICLES EXHAUSTING INTRACELLUAR AMINO ACID FOR CANCER THERAPY AND METHODS THEREOF

#63
20250025445
2025-01-23

METHOD OF CARDIOPROTECTION

#64
20250017920
2025-01-16

Magnetic nano-drug with double targeting VEGF-VEGFR, and preparation method and application thereof

#65
20250017870
2025-01-16

ADHESIVE PATCH CONTAINING SELEXIPAG AS ACTIVE INGREDIENT

#66
20250011288
2025-01-09

RXFP1 AGONISTS

#67
20250009739
2025-01-09

METHOD OF TREATING A SKIN DISORDER

#68
20250009693
2025-01-09

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#69
20250002463
2025-01-02

NEW SALT FORMS OF AMILORIDE AND ITS DERIVATIVES FOR PHARMACEUTICAL USE

#70
20240425464
2024-12-26

Substituted Monohydrazides as Potent Antifungal Agents

#71
20240425463
2024-12-26

PROCESS FOR MANUFACTURING A DIPHENYLPHRAZINE DERIVATIVE

#72
20240400586
2024-12-05

HETEROARYL DERIVATIVE PARP INHIBITOR AND USE THEREOF

#73
20240400518
2024-12-05

SOS1 INHIBITOR AND USE THEREOF

#74
20240390457
2024-11-28

COMPOSITION AND METHOD OF TREATING BRAIN CANCER

#75
20240374585
2024-11-14

EPITHELIAL SODIUM CHANNEL (ENAC) INHIBITOR CONJUGATES AND METHODS FOR USE THEREOF

#76
20240366592
2024-11-07

ANTICOAGULANT REVERSAL AGENTS

#77
20240360203
2024-10-31

Antigen Binding Molecules Targeting SARS-CoV-2

#78
20240336577
2024-10-10

PYRAZINE COMPOUND, AND METHOD OF PREPARATION AND USE THEREOF

#79
20240327334
2024-10-03

Covalent Inhibitors As Antiviral Agents

#80
20240325387
2024-10-03

COMBINATION THERAPY

#81
20240325386
2024-10-03

THERAPEUTIC AGENT FOR COVID-19

#82
20240325321
2024-10-03

COMPOSITIONS AND METHODS FOR INHIBITING PLpro PROTEASE ACTIVITY AND FOR PREVENTING AND TREATING SARS-CoV-2 INFECTION

#83
20240308992
2024-09-19

DRAK2 INHIBITOR, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#84
20240307382
2024-09-19

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#85
20240307293
2024-09-19

METHODS AND DEVICES FOR MODULATING ELECTROLYTE EXCRETION

#86
20240277701
2024-08-22

PYRUVATE KINASE ACTIVATORS FOR USE IN THERAPY

#87
20240254113
2024-08-01

COMPOUNDS AND THEIR USES AS CD38 INHIBITORS

#88
20240254079
2024-08-01

Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2alpha

#89
20240254075
2024-08-01

FATTY ACID AMIDE HYDROLASE (FAAH) CLEAVABLE PRODRUGS OF THYROMIMETICS AND COMBINATION WITH PERIPHERALLY RESTRICTED FAAH INHIBITORS

#90
20240245679
2024-07-25

AGENT FOR TREATING INFECTIOUS DISEASES AGAINST MUTANT VIRUSES OF NOVEL CORONAVIRUS

#91
20240238274
2024-07-18

INHIBITORS OF UBIQUITIN SPECIFIC PEPTIDASE 22 (USP22) AND USES THEREOF FOR TREATING DISEASE AND DISORDERS

#92
20240216365
2024-07-04

METHODS AND USES OF PROTEIN DISULFIDE ISOMERASE INHIBITORY COMPOUNDS

#93
20240199564
2024-06-20

TRPM8 AGONISTS AS COOLING AGENTS AND FOR THE TREATMENT OF DISEASE

#94
20240199554
2024-06-20

Inhibitors of receptor interacting protein kinase I for the treatment of disease

#95
20240197724
2024-06-20

THERAPEUTIC AGENT FOR GAIT DISTURBANCE

#96
20240189305
2024-06-13

THERAPEUTIC AGENT FOR CORONAVIRUS INFECTION

#97
20240182419
2024-06-06

ANTI-CANCER COMPOUNDS

#98
20240180955
2024-06-06

FIBER SUPPLEMENTATION PROTECTS FROM ANTIBIOTIC-INDUCED GUT MICROBIOME DYSBIOSIS BY MODULATING REDOX METABOLISM

#99
20240180895
2024-06-06

USE OF KAPPA OPIOID RECEPTOR AGONISTS TO TREAT CARDIOVASCULAR DISEASE

#100
20240180880
2024-06-06

METHODS OF USING EHMT2 INHIBITORS IN TREATING OR PREVENTING BLOOD DISORDERS

#101
20240173307
2024-05-30

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#102
20240173277
2024-05-30

ANTI-MYCOBACTERIAL DRUGS

#103
20240148723
2024-05-09

MYCOBACTERIUM TUBERCULOSIS COMPOSITIONS AND METHODS

#104
20240139207
2024-05-02

METHODS FOR TREATING PULMONARY HYPERTENSION

#105
20240131024
2024-04-25

PHARMACEUTICAL COMPOSITIONS COMPRISING SORBITAN ESTERS

#106
20240130984
2024-04-25

AMINONAPHTHOQUINONE COMPOUNDS FOR TREATMENT AND/OR PREVENTION OF FIBROSIS DISEASES

#107
20240115664
2024-04-11

Diketopiperazine Salts for Drug Delivery and Related Methods

#108
20240108617
2024-04-04

AN INHALABLE DRY POWDER COMPOSITION FOR PULMONARY DISEASES

#109
20240091238
2024-03-21

Calmodulin inhibitors for the treatment of ribosomal disorders and ribosomopathies

#110
20240075049
2024-03-07

DRUGS, THERAPEUTIC COMBINATIONS AND METHODS FOR PREVENTING VIRAL AND MICROBIAL INFECTIONS AND THEIR SEQUELAE

#111
20240058327
2024-02-22

Pharmaceutical Compositions Comprising Sorbitan Esters

#112
20240058315
2024-02-22

Pyridine and Pyrazine derivative for the Treatment of CF, COPD, and Bronchiectasis

#113
20240041868
2024-02-08

Methods, Compositions, and Uses of Novel FYN Kinase Inhibitors

#114
20240041867
2024-02-08

PHARMACEUTICAL COMPOSITION

#115
20240041866
2024-02-08

PHARMACEUTICAL COMPOSITION

#116
20240024311
2024-01-25

A CONTROLLED RELEASE PHARMACEUTICAL COMPOSITION OF SELEXIPAG OR IT'S ACTIVE METABOLITE

#117
20240000789
2024-01-04

THERAPEUTIC COMBINATIONS COMPRISING A CRAF INHIBITOR

#118
20240000777
2024-01-04

USE OF AN ERK INHIBITOR FOR THE TREATMENT OF MYELOFIBROSIS

#119
20240000732
2024-01-04

Anti-mycobacterial drugs

#120
20230416236
2023-12-28

INHIBITING ATAXIA TELANGIECTASIA AND RAD3-RELATED PROTEIN (ATR)

#121
20230414625
2023-12-28

Combination Antibacterial Composition and Short-Course Antibacterial Regimen

#122
20230414608
2023-12-28

USE OF ATR AND CHK1 INHIBITOR COMPOUNDS

#123
20230404954
2023-12-21

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#124
20230404921
2023-12-21

LYOTROPIC LIQUID CRYSTALLINE PHASE PARTICLE

#125
20230398112
2023-12-14

SPRAY-DRIED METAL-ORGANIC FRAMEWORKS FOR TREATMENT AND/OR DIAGNOSIS OF PULMONARY DISEASE

#126
20230372534
2023-11-23

CONJUGATES OF ACTIVE PHARMACEUTICAL INGREDIENTS

#127
20230372458
2023-11-23

ANTIVIRAL AGENT FOR COMBINED THERAPY OF COVID-19 (SARS-COV-2)

#128
20230372381
2023-11-23

COMPOSITIONS AND METHODS UTILIZING PROTEIN INHIBITORS FOR SYNERGISTIC INHIBITION AND TREATMENT OF SARS-CoV-2

#129
20230372334
2023-11-23

USE OF AN ERK INHIBITOR FOR THE TREATMENT OF MYELOFIBROSIS

#130
20230365550
2023-11-16

Lithium oxyhalide electrochemical cell design for high-rate discharge

#131
20230357367
2023-11-09

Antigen Binding Molecules Targeting SARS-CoV-2

#132
20230357366
2023-11-09

Antigen binding molecules targeting SARS-CoV-2

#133
20230355517
2023-11-09

USE OF ACTIVE SUBSTANCES WITH ANTIVIRAL, ANTI MALARIAL, AND/OR MUCOLYTIC PROPERTIES IN THE TREATMENT OF VIRAL LUNG DISEASES INCLUDING COVID-19 BY SOFT MIST INHALER OR VIBRATION MESH TECHNOLOGY NEBULIZER THROUGH INHALATION ROUTE

#134
20230338369
2023-10-26

COMBINATION OF A PROTEASOME INHIBITOR AND A HDAC INHIBITOR AND ITS USE FOR THE TREATMENT OF GENETIC DISEASES LINKED TO A PROTEIN CONFORMATIONAL DISORDER

#135
20230321008
2023-10-12

INHIBITORS OF ACID SPHINGOMYELINASE FOR PREVENTING AND TREATING THE COVID-19 DISEASE

#136
20230310544
2023-10-05

ANTI-RNA VIRAL PHARMACEUTICAL COMBINATION THERAPY WITH APROTININ + anti-RNA DRUG

#137
20230310421
2023-10-05

MOLECULES FOR USE IN THE TREATMENT OF VIRAL INFECTIONS

#138
20230285435
2023-09-14

COMPOSITIONS AND METHODS FOR TREATING VIRAL INFECTIONS

#139
20230277629
2023-09-07

FORMULATIONS AND METHODS FOR TREATMENT OF FIBROMYALGIA AND RELATED MYOFASCIAL PAIN DISORDERS

#140
20230277528
2023-09-07

COMPOSITIONS AND METHODS FOR HAIR FOLLICLE REGENERATION

#141
20230272449
2023-08-31

Identification of inhibitors of TcpC and TIR NADase activity

#142
20230271931
2023-08-31

Carboxylic acid aromatic amides as antagonists of bradykinin B1 receptor

#143
20230263827
2023-08-24

EXPANDED MEMORY SUBSETS OF GAMMA DELTA T CELLS FOR IMMUNOTHERAPY

#144
20230248721
2023-08-10

METHOD FOR DETECTING OR TREATING TRIPLE NEGATIVE BREAST CANCER

#145
20230241095
2023-08-03

PARTIALLY DESULFATED HEPARIN FOR TREATING CORONAVIRAL INFECTIONS

#146
20230241026
2023-08-03

NOVEL DRUG-CONTROLLED SYSTEMS AND USES THEREOF

#147
20230240984
2023-08-03

DIMETHYL SULFOXIDE (DMSO) AND METHYLSULFONYLMETHANE (MSM) FORMULATIONS TO TREAT OSTEOARTHRITIS

#148
20230234984
2023-07-27

Cysteine protease inhibitors and methods of use thereof

#149
20230233576
2023-07-27

ECLITASERTIB FOR USE IN TREATING CONDITIONS INVOLVING SYSTEMIC HYPERINFLAMMATORY RESPONSE

#150
20230226149
2023-07-20

MODIFIED CAVEOLIN-1 PEPTIDES FOR THE TREATMENT OF PATHOGEN-INDUCED LUNG INJURY

#151
20230218542
2023-07-13

MEDICAMENT FOR TREATING HYPERTENSION

#152
20230213515
2023-07-06

DRUG AND DIAGNOSTIC COMBINATION SYSTEM TO IDENTIFY AND TREAT SINGLE-STRANDED RNA VIRUSES INCLUDING CORONAVIRUSES AND MONKEYPOX

#153
20230210848
2023-07-06

CORONAVIRUS INFECTION THERAPEUTIC AGENT FORMED THROUGH COMBINATION OF PYRAZINE DERIVATIVE AND ANOTHER CORONAVIRUS INFECTION THERAPEUTIC DRUG

#154
20230201238
2023-06-29

THERAPEUTIC AGENT FOR AN RNA VIRUS INFECTION COMPRISING A COMBINATION OF A PYRAZINE DERIVATIVE AND A THIOPURINE DERIVATIVE

#155
20230158021
2023-05-25

SARS-CoV-2 Antiviral Pharmaceutical Composition and Application Thereof

#156
20230158020
2023-05-25

Method for treating RNA viral infections, including COVID-19 (SARS-CoV-2)

#157
20230143612
2023-05-11

SUBSTITUTED 1,1'-BIPHENYL COMPOUNDS AND METHODS USING SAME

#158
20230143415
2023-05-11

Treatment of aneurysms

#159
20230137585
2023-05-04

6-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING DISEASES AND CONDITIONS MEDIATED BY DEFICIENT CFTR ACTIVITY

#160
20230130925
2023-04-27

METHODS TO PREVENT, AMELIORATE AND TREAT COMPLICATIONS FROM VIRAL INFECTIONS

#161
20230128176
2023-04-27

Anti-RNA virus, including anti-SARS-CoV-2 virus, pharmaceutical composition Avifavir

#162
20230127703
2023-04-27

THERAPEUTIC AGENT FOR CORONAVIRUS INFECTION

#163
20230121825
2023-04-20

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#164
20230119141
2023-04-20

USES OF TAXIFOLIN FOR RESPIRATORY HEALTH

#165
20230117606
2023-04-20

COMPOSITIONS AND METHODS FOR THE TREATMENT OF INTRACELLULAR BACTERIAL INFECTIONS

#166
20230114153
2023-04-13

IMIDAZOLYL THIOPEHENE SULFONYL CARBAMATES FOR USE IN THE TREATMENT OF DISEASES ASSOCIATED WITH ANGIOTENSIN II

#167
20230113077
2023-04-13

CONTROLLED RELEASE SELEXIPAG COMPOSITION

#168
20230107186
2023-04-06

COBICISTAT FOR PREVENTION AND/OR TREATMENT OF CORONAVIRUS INFECTIONS

#169
20230106864
2023-04-06

COMPOSITIONS AND METHODS FOR THE TREATMENT OF INTRACELLULAR BACTERIAL INFECTIONS

#170
20230106592
2023-04-06

METHOD FOR TREATING CANCER USING A COMBINATION OF DNA DAMAGING AGENTS AND ATR INHIBITORS

#171
20230090389
2023-03-23

A TRIPLE PHARMACEUTICAL COMBINATION COMPRISING DABRAFENIB, AN ERK INHIBITOR AND A SHP2 INHIBITOR

#172
20230076066
2023-03-09

Use of sodium dichloroisocyanurate (NaDCC) and a pharmaceutical formulation prepared therefrom

#173
20230073428
2023-03-09

METHODS OF TREATING AND ASSESSING PULMONARY ARTERIAL HYPERTENSION WITH SELEXIPAG

#174
20230073008
2023-03-09

ANTISENSE NUCLEIC ACID THAT INDUCES SKIPPING OF EXON 50

#175
20230043209
2023-02-09

Carboxylic acid aromatic amides

#176
20230032813
2023-02-02

METHODS OF TREATING PULMONARY ARTERIAL HYPERTENSION

#177
20230028660
2023-01-26

Anti-cancer compounds

#178
20230027929
2023-01-26

MrgprX2 Antagonists and Uses Thereof

#179
20230021476
2023-01-26

Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2alpha

#180
20230020241
2023-01-19

Pharmaceutical Composition For The Treatment Of Pulmonary Arterial Hypertension

#181
20230000816
2023-01-05

SODIUM-GLUCOSE LINKED TRANSPORTER INHIBITORS FOR THE MANAGEMENT OF CHRONIC KIDNEY DISEASE, HYPERTENSION, AND HEART FAILURE IN COMPANION ANIMALS

#182
20220409694
2022-12-29

POLYPEPTIDE, AND PREPARATION METHOD THEREFOR AND USE THEREOF

#183
20220409542
2022-12-29

Inhalable antimicrobial particles and methods of making the same

#184
20220401554
2022-12-22

USE OF MEMBRANE INHIBITORS TO ENHANCE VACCINE DEVELOPMENT AGAINST ENVELOPED VIRUSES

#185
20220401441
2022-12-22

PHARMACEUTICAL COMPOSITION COMPRISING SELEXIPAG

#186
20220388955
2022-12-08

EP2 ANTAGONIST

#187
20220370444
2022-11-24

Compositions of Clofazimine, Combinations Comprising Them, Processes for Their Preparation, Uses and Methods of Treatment Comprising Them

#188
20220347449
2022-11-03

THREE-DIMENSIONAL MICROFLUIDICS DEVICES FOR THE DELIVERY OF ACTIVES

#189
20220347172
2022-11-03

COMBINATION TREATMENTS

#190
20220333112
2022-10-20

Antisense nucleic acid that induces skipping of exon 50

#191
20220331346
2022-10-20

Substituted bicyclic compounds

#192
20220331313
2022-10-20

METHODS FOR TREATING SARCOIDOSIS-ASSOCIATED PULMONARY HYPERTENSION

#193
20220326255
2022-10-13

METHODS OF MONITORING MUCOSAL HEALING

#194
20220323531
2022-10-13

Willow extract and its use in treating a viral infection, allergic reaction, and other medical conditions

#195
20220323437
2022-10-13

METHODS FOR TREATING PULMONARY ARTERIAL HYPERTENSION

#196
20220305092
2022-09-29

MEDICAMENT AND FOOD FOR PREVENTING OR TREATING NOVEL CORONAVIRUS PNEUMONIA COVID-19 AND USE THEREOF

#197
20220304957
2022-09-29

ANTI-CANCER COMPOSITIONS AND METHODS OF USE

#198
20220273689
2022-09-01

POTENTIATION OF ANTIVIRAL NUCLEOBASES AS RNA VIRUS THERAPY

#199
20220265649
2022-08-25

BILE ACID RECYCLING INHIBITORS FOR TREATMENT OF PEDIATRIC CHOLESTATIC LIVER DISEASES

#200
20220257594
2022-08-18

TRANSITIONING PATIENTS TREATED FOR PULMONARY ARTERIAL HYPERTENSION TO SELEXIPAG

#201
20220249489
2022-08-11

METHOD FOR TREATING CANCER USING A COMBINATION OF CHK1 AND ATR INHIBITORS

#202
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2022-08-04

Pulmonary hypertension treatment

#203
20220233521
2022-07-28

COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE AND COMBINATION THERAPIES THEREOF

#204
20220226336
2022-07-21

COMBINATION THERAPY FOR TREATING CANCER

#205
20220218801
2022-07-14

COMBINATION GMCI AND ATRI CANCER TREATMENT

#206
20220214332
2022-07-07

Methods for Detecting A Mycobacterium Tuberculosis Infection

#207
20220202812
2022-06-30

Use of ligustrazine nitrone derivatives in treatment and prevention of diabetic complication diseases

#208
20220175769
2022-06-09

METHOD OF TREATMENT OF ACTINIC KERATOSES

#209
20220169685
2022-06-02

Treatment of ischemia

#210
20220168299
2022-06-02

PHARMACEUTICAL COMPOSITION COMPRISING TBN, OR SALT OR HYDRATE THEREOF, AND PREPARATION METHOD THEREOF

#211
20220168268
2022-06-02

SMALL-MOLECULE INHIBITOR OF PD-1/PD-L1, PHARMACEUTICAL COMPOSITION THEREOF WITH PD-L1 ANTIBODY, AND APPLICATION OF SAME

#212
20220152228
2022-05-19

COMPOSITIONS AND METHODS FOR RADIOTHERAPY USING CHELATED RADIOTHERAPEUTIC AGENTS AND NON-TARGET TISSUE BLOCKADE

#213
20220152041
2022-05-19

Calmodulin inhibitors for the treatment of ribosomal disorders and ribosomapathies

#214
20220127237
2022-04-28

FLUORESCENT PYRAZINE DERIVATIVES AND METHODS OF USING THE SAME IN ASSESSING RENAL FUNCTION

#215
20220117968
2022-04-21

THIENO[2,3-D)PYRIMIDINES AND BENZOFURO(3,2-D)PYRIMIDINES AS ANTIMICROBIAL AGENTS

#216
20220096476
2022-03-31

Pharmaceutical composition for the treatment of pulmonary arterial hypertension

#217
20220096468
2022-03-31

Therapeutic agent for RNA viral infection comprising a combination of pyrazine derivative and compound which increases amount of pyrazine derivative ribose triphosphate in cell

#218
20220088012
2022-03-24

PZA and cytochrome Bc1 inhibitor combination treatment

#219
20220081390
2022-03-17

FARNESOID X RECEPTOR AGONISTS AND USES THEREOF

#220
20220079920
2022-03-17

PHARMACEUTICAL COMPOSITION CONTAINING AMLODIPINE, CHLORTHALIDONE, AND AMILORIDE AND APPLICATION THEREOF

#221
20220062379
2022-03-03

METHODS AND COMPOSITIONS FOR MODULATING IMMUNE DYSREGULATION

#222
20220062234
2022-03-03

Drug-controlled systems and uses thereof

#223
20220047686
2022-02-17

METHODS FOR TREATING INFECTIOUS DISEASES

#224
20220047586
2022-02-17

Composition and methods for preventing or reducing the incidence of transient ischemic attacks

#225
20220031668
2022-02-03

METHODS OF INHIBITING PROCOLLAGEN-LYSINE, 2-OXOGLUTARATE 5-DIOXYGENASE 2

#226
20220023296
2022-01-27

Bile acid recycling inhibitors for treatment of pediatric cholestatic liver diseases

#227
20220017482
2022-01-20

Synthetic Antibacterial Compounds and Uses Thereof

#228
20220008426
2022-01-13

Therapeutic combinations comprising a c-RAF inhibitor

#229
20220000808
2022-01-06

Cysteamine for the Treatment, Mitigation and Prevention of Coronaviral, e.g., SARS-CoV-2, Infections

#230
20210401802
2021-12-30

PKC-Delta-I inhibitor formulations and uses thereof

#231
20210393600
2021-12-23

[1.1.1] bicyclo compounds as indoleamine 2,3-dioxygenase inhibitors

#232
20210393599
2021-12-23

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#233
20210386752
2021-12-16

Uses of Electron Transport Chain Complex I or Complex II Inhibitors in Treating Cancer, Combination Therapies, and Diagnostic Methods Related Thereto

#234
20210386709
2021-12-16

COMPOSITIONS AND METHODS FOR SUPPRESSING MSUT2

#235
20210369680
2021-12-02

METHODS OF TREATING DISEASES AND DISORDERS RESULTING FROM BETA CORONAVIRUS INFECTION

#236
20210361657
2021-11-25

USE OF INHIBITORS OF BRUTONS TYROSINE KINASE (BTK)

#237
20210353620
2021-11-18

Method of treating severe acute respiratory syndrome (SARS) virus infection by administering a protein disulfide isomerase (PDI) inhibitor

#238
20210346376
2021-11-11

Use of Favipiravir in treatment of coronavirus infection

#239
20210330809
2021-10-28

LIPID-COATED PARTICLES FOR TREATING VIRAL INFECTIONS

#240
20210322407
2021-10-21

Use of Trimetazidine in Preparation of Drugs for Preventing and Treating Liver Diseases

#241
20210317079
2021-10-14

Tetralin and tetrahydroquinoline compounds as inhibitors of HIF-2α

#242
20210300905
2021-09-30

Inhibiting ataxia telangiectasia and RAD3-related protein (ATR)

#243
20210290651
2021-09-23

METHODS OF TREATING VIRAL INFECTIONS USING INHIBITORS OF NUCLEOTIDE SYNTHESIS PATHWAYS

#244
20210290629
2021-09-23

ACC INHIBITORS FOR USE IN TREATING MYCOBACTERIAL DISEASES

#245
20210290617
2021-09-23

Ophthalmic formulations of cetirizine and methods of use

#246
20210290531
2021-09-23

Method for treatment of a viral-mediated infectious disease

#247
20210277007
2021-09-09

Hetero-halo inhibitors of histone deacetylase

#248
20210275616
2021-09-09

Composition for ameliorating peripheral sensory neuropathy

#249
20210269399
2021-09-02

MODULATORS OF THE INTEGRATED STRESS PATHWAY

#250
20210267953
2021-09-02

Substituted oxazolidinones for the treatment of mammalian infections

#251
20210260055
2021-08-26

TOPICAL FORMULATIONS OF DGAT1 INHIBITORS AND THEIR METHODS OF USE

#252
20210260040
2021-08-26

METHODS OF USING EHMT2 INHIBITORS IN TREATING OR PREVENTING BLOOD DISORDERS

#253
20210252033
2021-08-19

N4-HYDROXYCYTIDINE AND DERIVATIVES AND ANTI-VIRAL USES RELATED THERETO

#254
20210228554
2021-07-29

Pyridine and pyrazine derivative for the treatment of chronic bronchitis

#255
20210223233
2021-07-22

Mitochondrial Conductance Inhibitors and Methods of Use Thereof

#256
20210220354
2021-07-22

Composition for reducing nervous system injury and method of making and use thereof

#257
20210220353
2021-07-22

USE OF FAVIPIRAVIR IN TREATMENT OF CORONAVIRUS INFECTION

#258
20210220351
2021-07-22

Pyruvate kinase activators for use in therapy

#259
20210214323
2021-07-15

NOVEL COMPOUNDS AND COMPOSITIONS FOR INHIBITION OF FASN

#260
20210212993
2021-07-15

Use of prostacyclin antagonists for treating ocular surface nociception

#261
20210196734
2021-07-01

Substituted 6-membered aryl or heteroaryl allosteric modulators of nicotinic acetylcholine receptors

#262
20210196715
2021-07-01

Pharmaceutical composition for the treatment of pulmonary arterial hypertension

#263
20210186969
2021-06-24

AZA-PYRIDONE COMPOUNDS AND USES THEREOF

#264
20210186960
2021-06-24

MODULATORS OF INDOLEAMINE 2,3-DIOXYGENASE

#265
20210179566
2021-06-17

Compositions and methods for delivering pharmaceutical agents

#266
20210171466
2021-06-10

THIOACETATE COMPOUNDS, COMPOSITIONS AND METHODS OF USE

#267
20210169874
2021-06-10

ANTICOAGULANT REVERSAL AGENTS

#268
20210163476
2021-06-03

Imidazoquinolyl compounds having anti-inflammatory, antifungal, antiparasitic, and anticancer activity

#269
20210161840
2021-06-03

COMPOSITIONS AND METHODS FOR TREATMENT OF IRON OVERLOAD

#270
20210154191
2021-05-27

Methods of treatment of cancer

#271
20210154190
2021-05-27

SHP2 INHIBITOR COMPOSITIONS AND METHODS FOR TREATING CANCER

#272
20210138084
2021-05-13

Conjugates of active pharmaceutical ingredients

#273
20210138041
2021-05-13

Diketopiperazine salts for drug delivery and related methods

#274
20210121527
2021-04-29

METHODS OF TREATING MINIMAL RESIDUAL CANCER

#275
20210113495
2021-04-22

METHOD OF TREATING EPILEPSY OR EPILEPTIC ENCEPHALOPATHY WITH FENFLURAMINE IN PATIENTS WITHOUT PULMONARY HYPERTENSION

#276
20210100844
2021-04-08

RAR selective agonists in combination with immune modulators for cancer immunotherapy

#277
20210094921
2021-04-01

Inhibitors of receptor interacting protein kinase I for the treatment of disease

#278
20210093640
2021-04-01

Polycyclic carbamoylpyridone derivatives, pharmaceutical compositions and use thereof

#279
20210077511
2021-03-18

Substituted 6-membered aryl or heteroaryl allosteric modulators of nicotinic acetylcholine receptors

#280
20210069187
2021-03-11

Stable pharmaceutical composition of Selexipag

#281
20210059947
2021-03-04

Method for producing freeze-dried formulation

#282
20210032236
2021-02-04

NOVEL GLUTAMINASE INHIBITORS

#283
20210032195
2021-02-04

Farnesoid X receptor agonists and uses thereof

#284
20210030753
2021-02-04

Methods, compositions, and uses of novel FYN kinase inhibitors

#285
20210024471
2021-01-28

3,5-diamino-6-chloro-N-(N-(4-(4-(2-(hexyl(2,3,4,5,6-pentahydroxyhexyl)amino)ethoxy)phenyl)butyl)carbamimidoyl)pyrazine-2-carboxamide

#286
20210013550
2021-01-14

Lithium oxyhalide electrochemical cell design for high-rate discharge

#287
20210009682
2021-01-14

REDUCING CUTANEOUS SCAR FORMATION AND TREATING SKIN CONDITIONS

#288
20210008072
2021-01-14

FORMULATIONS OF AZAINDOLE COMPOUNDS

#289
20200405711
2020-12-31

Ophthalmic formulations of cetirizine and methods of use

#290
20200399247
2020-12-24

Inhibiting ataxia telangiectasia and Rad3-related protein (ATR)

#291
20200397700
2020-12-24

GRANULAR COMPOSITION, PRODUCTION METHOD FOR GRANULAR COMPOSITION, AND DISSOLUTION PROPERTY IMPROVEMENT METHOD FOR GRANULAR COMPOSITION

#292
20200390761
2020-12-17

TREATING CANCER WITH ATR INHIBITORS

#293
20200383960
2020-12-10

Pyridine and Pyrazine derivative for the Treatment of CF, COPD, and Bronchiectasis

#294
20200375930
2020-12-03

MODULATORS OF THE PROSTACYCLIN (PGI2) RECEPTOR USEFUL FOR THE TREATMENT OF DISORDERS RELATED THERETO

#295
20200368244
2020-11-26

Pulmonary hypertension treatment

#296
20200368243
2020-11-26

THERAPIES FOR HEMATOLOGIC MALIGNANCIES

#297
20200361876
2020-11-19

Process for the preparation of diphenylpyrazine derivatives

#298
20200360373
2020-11-19

Controlled-release preparation

#299
20200354415
2020-11-12

Treatment of ischemia

#300
20200347025
2020-11-05

Compounds and compositions for inhibition of FASN