ClassID:

20412

A61K31/4985 - page 3 - CPC Classification

Classification description:

Medicinal preparations containing organic active ingredients; Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two nitrogen atoms as the only ring heteroatoms, e.g. piperazine Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems

Recent Application in this class:
#601
20240165122
2024-05-23

COMBINATION THERAPY FOR PI3K-ASSOCIATED DISEASE OR DISORDER

#602
20240165111
2024-05-23

ORGANIC COMPOUNDS

#603
20240165110
2024-05-23

SELECTIVE AND NON-SELECTIVE OPIOID RECEPTOR FUNCTIONAL ANTAGONISTS AND METHODS RELATED THERETO FOR TREATMENT OF ADDICTION, OPIOD DEPENDENCE, AND NEUROPATHIC PAIN

#604
20240156831
2024-05-16

HETEROCYCLIC COMPOUNDS AS PAD INHIBITORS

#605
20240156827
2024-05-16

PDE5 INHIBITOR POWDER FORMULATIONS AND METHODS RELATING THERETO

#606
20240148745
2024-05-09

COMPOUNDS FOR USE IN PROGRESSIVE MULTIPLE SCLEROSIS

#607
20240148744
2024-05-09

SULFONAMIDES AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES

#608
20240139182
2024-05-02

Certain Triazolopyridines and Triazolopyrazines, Compositions Thereof and Methods of Use Therefor

#609
20240139164
2024-05-02

RAPAMYCIN ANALOGS AND USES THEREOF

#610
20240132470
2024-04-25

Antibacterial Compounds

#611
20240131026
2024-04-25

BROMOCRIPTINE FORMULATIONS

#612
20240131012
2024-04-25

RAPAMYCIN ANALOGS AND USES THEREOF

#613
20240131007
2024-04-25

METHODS AND COMPOSITIONS FOR PICORNAVIRUS ANTI-VIRAL AGENTS

#614
20240130964
2024-04-25

SOFT CHEWABLE FORMULATIONS WITH ACTIVE INGREDIENTS

#615
20240122925
2024-04-18

SHP2 PHOSPHATASE INHIBITORS AND METHODS OF MAKING AND USING THE SAME

#616
20240122924
2024-04-18

NOVEL METHODS

#617
20240122923
2024-04-18

METHODS OF TREATING HIDRADENITIS SUPPURATIVA

#618
20240122855
2024-04-18

Methods for the preparation of biologically active compounds in nanoparticulate form

#619
20240115577
2024-04-11

SMALL MOLECULE REGULATORS OF ALVEOLAR TYPE 2 CELL PROLIFERATION FOR THE TREATMENT OF PULMONARY DISEASES

#620
20240115565
2024-04-11

Amorphous solid dispersions

#621
20240108633
2024-04-04

METHOD FOR PREVENTING OR TREATING DISEASE OR CONDITION ASSOCIATED WITH ANTITUMOR AGENT

#622
20240108627
2024-04-04

Phosphodiesterase Inhibitor Treatment

#623
20240108621
2024-04-04

NOVEL USES

#624
20240108620
2024-04-04

Treatment Regimen

#625
20240108619
2024-04-04

INTRANASAL DHE FOR THE TREATMENT OF HEADACHE

#626
20240108618
2024-04-04

KRAS G12C INHIBITOR DOSING REGIMENS

#627
20240100048
2024-03-28

DIPEPTIDYLPEPTIDASE 4 INHIBITION ENHANCES LYMPHOCYTE TRAFFICKING, IMPROVING BOTH NATURALLY OCCURRING TUMOR IMMUNITY AND IMMUNOTHERAPY

#628
20240100047
2024-03-28

COMPOSITION AND METHOD FOR TREATING COVID-19

#629
20240091224
2024-03-21

Pharmaceutical capsule compositions comprising lumateperone mono-tosylate

#630
20240083910
2024-03-14

AMIDO-SUBSTITUTED PYRIDYL COMPOUNDS AND METHODS OF USE THEREOF FOR THE TREATMENT OF HERPESVIRUSES

#631
20240082245
2024-03-14

Methods for Treating HCV

#632
20240082223
2024-03-14

DIHYDROFUROPYRIDINE DERIVATIVES AS RHO- KINASE INHIBITORS

#633
20240082221
2024-03-14

COMPOSITIONS AND METHODS FOR THE IDENTIFICATION OF COMPOUNDS THAT PROTECT AGAINST LIPOFUSCIN CYTOTOXICITY

#634
20240075028
2024-03-07

PHARMACEUTICAL COMPOSITION COMPRISING TADALAFIL OR PHARMACEUTICALLLY ACCEPTABLE SALT THEREOF AND DUTASTERIDE OR PHARMACEUTICALLLY ACCEPTABLE SALT THEREOF EXHIBITING NOVEL DISSOLUTION RATE

#635
20240075026
2024-03-07

Solid Pharmaceutical Compositions for Treating HCV

#636
20240066030
2024-02-29

Methods

#637
20240066029
2024-02-29

Substituted pyrazolo[1,5-a]pyridine compounds as RET kinase inhibitors

#638
20240066020
2024-02-29

COMPOSITIONS AND METHODS TO TREAT NON-ALCOHOLIC FATTY LIVER DISEASES (NAFLD)

#639
20240058450
2024-02-22

BCL-XL Inhibitory Compounds Having Low Cell Permeability and Antibody Drug Conjugates Including the Same

#640
20240058342
2024-02-22

TREATMENT OF CONGENITAL ADRENAL HYPERPLASIA

#641
20240058334
2024-02-22

METHODS FOR TREATING SMALL CELL LUNG CANCER AND OTHER NEUROENDOCRINE CANCERS

#642
20240050430
2024-02-15

KRAS G12C INHIBITORS AND METHODS OF USING THE SAME

#643
20240044916
2024-02-08

METHODS OF MONITORING INFLAMMATORY BOWEL DISEASES

#644
20240043393
2024-02-08

cGAS antagonist compounds

#645
20240041871
2024-02-08

METHODS AND COMPOSITIONS FOR SLEEP DISORDERS AND OTHER DISORDERS

#646
20240041870
2024-02-08

METHODS OF TREATING SYSTEMIC LUPUS ERYTHEMATOSUS

#647
20240041868
2024-02-08

Methods, Compositions, and Uses of Novel FYN Kinase Inhibitors

#648
20240041798
2024-02-08

OVARIAN CANCER VACCINES

#649
20240034740
2024-02-01

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#650
20240033330
2024-02-01

TYPE I DIABETES THERAPY

#651
20240033262
2024-02-01

NOVEL METHODS

#652
20240033258
2024-02-01

COMPOSITIONS AND METHODS FOR THE TREATMENT OF ADDICTION AND OTHER NEUROPSYCHIATRIC DISORDERS

#653
20240025891
2024-01-25

HETEROCYCLIC COMPOUNDS AND THEIR USE FOR TREATMENT OF HELMINTHIC INFECTIONS AND DISEASES

#654
20240024334
2024-01-25

NOVEL METHODS

#655
20240024312
2024-01-25

PHARMACEUTICAL COMPOSITIONS OF SITAGLIPTIN

#656
20240016840
2024-01-18

METHODS AND COMPOSITIONS FOR USE OF THERAPEUTIC T CELLS IN COMBINATION WITH KINASE INHIBITORS

#657
20240016802
2024-01-18

TRANSMUCOSAL METHODS FOR TREATING PSYCHIATRIC AND NEUROLOGICAL CONDITIONS

#658
20240010656
2024-01-11

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#659
20240009188
2024-01-11

PHARMACEUTICAL COMPOSITIONS OF NILOTINIB

#660
20240009130
2024-01-11

RAPIDLY INFUSING COMPOSITIONS FOR ORAL MUCOSAL DELIVERY AND METHODS

#661
20240000798
2024-01-04

Modulation of solubility, stability, absorption, metabolism, and pharmacokinetic profile of lipophilic drugs by sterols

#662
20240000781
2024-01-04

AMORPHOUS SOLID DISPERSIONS

#663
20240000780
2024-01-04

PED5 INHIBITOR SEMI-SOLID COMPOSITIONS AND METHODS OF MAKING AND USING THEREOF

#664
20230414699
2023-12-28

TREATMENT OF DERMATOLOGICAL CONDITIONS

#665
20230414628
2023-12-28

METHODS FOR TREATING DISEASES MEDIATED BY GLUTATHIONE PEROXIDASE 4

#666
20230414610
2023-12-28

THERAPIES FOR CANCER USING SMALL MOLECULES THAT BIND TO AND INHIBIT RAIL INTERACTING PROTEINS

#667
20230414582
2023-12-28

METHODS OF TREATING DISEASES AND DISORDERS

#668
20230405095
2023-12-21

DOSING REGIMEN

#669
20230404941
2023-12-21

Use of cannabidiol in treatment of pulmonary hypertension

#670
20230399333
2023-12-14

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#671
20230398126
2023-12-14

RIFT VALLEY FEVER SMALL MOLECULE TREATMENT

#672
20230390318
2023-12-07

Antiviral Prodrugs and Pharmaceutical Compositions Thereof

#673
20230390221
2023-12-07

PHARMACEUTICAL COMPOSITIONS WITH LOW AMOUNTS OF NITROSAMINE IMPURITIES AND METHODS FOR PRODUCING THE SAME

#674
20230381187
2023-11-30

Liquid oral formulations for sildenafil

#675
20230381175
2023-11-30

Therapeutic agent composition and method of use, for treatment of mild congnitive impairment, depression, and psychological disorders

#676
20230381174
2023-11-30

THIONOESTER-DERIVATIVE OF RABEXIMOD FOR THE TREATMENT OF INFLAMMATORY AND AUTOIMMUNE DISORDERS

#677
20230381173
2023-11-30

METHODS AND PHARMACEUTICAL COMPOSITION FOR TREATING DISEASES

#678
20230381158
2023-11-30

COMPOSITIONS FOR THE TREATMENT OF NON-ALCOHOLIC FATTY LIVER DISEASE AND NON-ALCOHOLIC STEATOHEPATITIS

#679
20230374027
2023-11-23

PROCESSES FOR THE PREPARATION OF (3S,4R)-3-ETHYL-4-(3H-IMIDAZO[1,2-a]PYRROLO[2,3-e]-PYRAZIN-8-YL)-N-(2,2,2-TRIFLUOROETHYL)PYRROLIDINE-1-CARBOXAMIDE AND SOLID STATE FORMS THEREOF

#680
20230372351
2023-11-23

Treatment of erectile dysfunction and other indications

#681
20230372345
2023-11-23

Inhaled PDE-V Inhibitor Drugs

#682
20230372336
2023-11-23

NOVEL METHODS

#683
20230372335
2023-11-23

TREATMENT OF COGNITIVE IMPAIRMENT WITH A CNS-PENETRANT sGC STIMULATOR

#684
20230372249
2023-11-23

PALATABLE FORMULATIONS

#685
20230365610
2023-11-16

Aryl Glucoside Derivative

#686
20230364081
2023-11-16

METHOD AND FORMULATION FOR TREATING MALE PREMATURE EJACULATION

#687
20230364080
2023-11-16

TREATING SPONDYLOARTHRITIC AND PSORIATIC CONDITIONS WITH UPADACITINIB

#688
20230364079
2023-11-16

COMPOUND AS BRAIN-PERMEABLE BTK OR HER2 INHIBITOR, PREPARATION METHOD THEREFOR, AND USE THEREOF

#689
20230364078
2023-11-16

METHOD OF PREPARING NANOPARTICLES COMPRISING POORLY WATER SOLUBLE DRUGS FOR TREATING HEPATITIS

#690
20230355636
2023-11-09

COMBINATIONS OF 15-PGDH INHIBITORS WITH CORTICOSTEROIDS AND/OR TNF INHIBITORS AND USES THEREOF

#691
20230355630
2023-11-09

SOLID PHARMACEUTICAL COMPOSITIONS COMPRISING BIOPTERIN DERIVATIVES AND USES OF SUCH COMPOSITIONS

#692
20230355626
2023-11-09

INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

#693
20230355616
2023-11-09

METHODS AND COMPOSITIONS FOR SLEEP DISORDERS AND OTHER DISORDERS

#694
20230355593
2023-11-09

N-methyl-D-aspartic Acid Receptor Modulators

#695
20230348481
2023-11-02

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#696
20230346787
2023-11-02

Organic compounds

#697
20230346781
2023-11-02

Small molecule inhibitors of cancer stem cells and mesenchymal cancer types

#698
20230346779
2023-11-02

DOSAGE FORM COMPOSITIONS COMPRISING AN INHIBITOR OF BTK AND MUTANTS THEREOF

#699
20230346748
2023-11-02

PHARMACEUTICAL COMBINATION, COMPOSITION AND COMPOUND PREPARATION CONTAINING GLUCOKINASE ACTIVATOR AND K-ATP CHANNEL BLOCKER, PREPARATION METHOD THEREFOR AND USE THEREOF

#700
20230339968
2023-10-26

KRAS Gl2C INHIBITORS

#701
20230339957
2023-10-26

DOSAGE FORM COMPOSITIONS COMPRISING AN INHIBITOR OF BRUTON'S TYROSINE KINASE

#702
20230339951
2023-10-26

Pharmaceutical compositions comprising 4-((6bR, 10aS)-3-methyl-2,3,6b,9,10,10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)butan-1-one for treating central nervous system disorders

#703
20230338449
2023-10-26

PLANT EXTRACTS WITH ANTI-DIABETIC AND OTHER USEFUL ACTIVITIES

#704
20230338370
2023-10-26

Treatment of Cancer with TOR Kinase Inhibitors

#705
20230338366
2023-10-26

PARENTERAL UNIT DOSAGE FORM OF DIHYDROERGOTAMINE

#706
20230338304
2023-10-26

USE OF CANNABINOIDS IN TREATING ANTI-DEPRESSANT-INDUCED FEMALE SEXUAL DYSFUNCTION

#707
20230331735
2023-10-19

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#708
20230331732
2023-10-19

HETEROCYCLIC GLP-1 AGONISTS

#709
20230331729
2023-10-19

4-IMIDAZOPYRIDAZIN-1-YL-BENZAMIDES AS BTK INHIBITORS

#710
20230330099
2023-10-19

Substituted indole Mcl-1 inhibitors

#711
20230330086
2023-10-19

Antiproliferative compounds and second active agents for combined use

#712
20230322794
2023-10-12

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#713
20230322747
2023-10-12

OXADIAZOLE HDAC6 INHIBITORS AND USES THEREOF

#714
20230321090
2023-10-12

Bromocriptine formulations

#715
20230321089
2023-10-12

COMBINATION OF CABOTEGRAVIR AND LEVONORGESTREL

#716
20230321086
2023-10-12

METHODS AND MATERIALS FOR INHIBITING NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE ACTIVITY

#717
20230312595
2023-10-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#718
20230312594
2023-10-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#719
20230312593
2023-10-05

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1- carboxamide and solid state forms thereof

#720
20230310444
2023-10-05

COMPOSITIONS AND METHODS FOR TREATING DISEASES AND DISORDERS

#721
20230310424
2023-10-05

METHODS AND MATERIALS FOR INCREASING NICOTINAMIDE PHOSPHORIBOSYL TRANSFERASE ACTIVITY

#722
20230303582
2023-09-28

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#723
20230301995
2023-09-28

Transmucosal methods for treating psychiatric and neurological conditions

#724
20230301994
2023-09-28

BICYCLIC COMPOUNDS AND METHODS FOR THEIR USE IN TREATING PITT HOPKINS SYNDROME

#725
20230293517
2023-09-21

ANTAGONIST COMPOUNDS

#726
20230286974
2023-09-14

Composition and Method for Treating Metabolic Disorders

#727
20230285691
2023-09-14

Heating unit for use in a drug delivery device

#728
20230285435
2023-09-14

COMPOSITIONS AND METHODS FOR TREATING VIRAL INFECTIONS

#729
20230285398
2023-09-14

Liquid oral formulations for tadalafil

#730
20230285345
2023-09-14

Combination methods and compositions including sleep therapeutics for treating mood

#731
20230285283
2023-09-14

PHARMACEUTICAL FORMULATIONS COMPRISING TADALAFIL

#732
20230279012
2023-09-07

HETEROARYL PYRIDONE AND AZA-PYRIDONE COMPOUNDS

#733
20230277629
2023-09-07

FORMULATIONS AND METHODS FOR TREATMENT OF FIBROMYALGIA AND RELATED MYOFASCIAL PAIN DISORDERS

#734
20230277465
2023-09-07

ANTIDIABETIC PHARMACEUTICAL COMPOSITIONS

#735
20230277448
2023-09-07

CHEWABLE FORMULATIONS

#736
20230271974
2023-08-31

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-α]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms therof

#737
20230271962
2023-08-31

Pharmaceutical compositions comprising 4-((6bR, 10aS)-3-methyl-2,3,6b,9,10, 10a-hexahydro-1H,7H-pyrido[3′,4′:4,5]pyrrolo[1,2,3-de]quinoxalin-8-yl)-1-(4-fluorophenyl)butan-1-ol for treating central nervous system disorders

#738
20230270677
2023-08-31

LONG-ACTING THERAPEUTIC AGENT COMBINATIONS AND METHODS THEREOF

#739
20230260595
2023-08-17

DETERMINATION OF NFKB PATHWAY ACTIVITY USING UNIQUE COMBINATION OF TARGET GENES

#740
20230255963
2023-08-17

SUBSTITUTED BENZALDEHYDE COMPOUNDS AND METHODS FOR THEIR USE IN INCREASING TISSUE OXYGENATION

#741
20230255962
2023-08-17

COMBINATION OF A BTK INHIBITOR AND AN INHIBITOR OF CDK9 TO TREAT CANCER

#742
20230255890
2023-08-17

COMPOSITE FORMULATION COMPRISING SITAGLIPTIN AND DAPAGLIFLOZIN AND PREPARATION METHOD THEREFOR

#743
20230248724
2023-08-10

Method of Injecting Dihydroergotamine Into The Body

#744
20230248723
2023-08-10

PYRROLO[2,3-B]PYRAZINE COMPOUNDS AS CCCDNA INHIBITORS FOR THE TREATMENT OF HEPATITIS B VIRUS (HBV) INFECTION

#745
20230241059
2023-08-03

ANTI-NEOPLASTIC COMBINATIONS AND DOSING REGIMENS USING CDK4/6 INHIBITOR COMPOUNDS TO TREAT RB-POSITIVE TUMORS

#746
20230234967
2023-07-27

Fused Azole Heterocycles as AHR Antagonists

#747
20230233555
2023-07-27

METHOD OF ADMINISTERING UPADACITINIB TO AVOID ADVERSE DRUG INTERACTIONS AND EFFECTS

#748
20230233554
2023-07-27

USE OF PHOSPHODIESTERASE 5 INHIBITOR IN PREPARATION OF MEDICAMENT FOR RESISTING FIBROTIC DISEASES

#749
20230228740
2023-07-20

METHOD OF USING HUMAN SPHEROIDS FOR DRUG DISCOVERY

#750
20230227463
2023-07-20

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#751
20230227455
2023-07-20

METHOD FOR PREPARING A CRYSTALLINE FORM OF RABEXIMOD

#752
20230226062
2023-07-20

HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS

#753
20230226054
2023-07-20

Compositions and use of varenicline for treating dry eye

#754
20230226053
2023-07-20

Compositions and use of varenicline for treating dry eye

#755
20230226052
2023-07-20

Compositions and use of varenicline for treating dry eye

#756
20230226050
2023-07-20

METHOD OF ACHIEVING HIV VIRAL REMISSION USING LONG-ACTING ANTIRETROVIRAL AGENTS

#757
20230226049
2023-07-20

ACALABRUTINIB MALEATE DOSAGE FORMS

#758
20230226048
2023-07-20

NEW USE OF RABEXIMOD

#759
20230219968
2023-07-13

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#760
20230219967
2023-07-13

Pyrazole derivatives useful as 5-lipoxygenase activating protein (FLAP) inhibitors

#761
20230218597
2023-07-13

SUBSTITUTED PYRIDINES AND METHODS OF USE

#762
20230210850
2023-07-06

Process for preparing substituted pyrazolo[1,5-a]pyrazines

#763
20230203051
2023-06-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1- carboxamide and solid state forms thereof

#764
20230203050
2023-06-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#765
20230203049
2023-06-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#766
20230203037
2023-06-29

Organic compounds

#767
20230201194
2023-06-29

COMBINATION COMPOSITIONS FOR IMMUNOTHERAPY

#768
20230192758
2023-06-22

COMPOUNDS WITH HIV MATURATION INHIBITORY ACTIVITY

#769
20230190741
2023-06-22

LONG-LASTING REABSORBABLE SUBCUTANEOUS IMPLANT WITH SUSTAINED RELEASE OF PRE-CONCENTRATED PHARMACOLOGICALLY ACTIVE SUBSTANCE IN POLYMER FOR THE TREATMENT OF ERECTILE DYSFUNCTION AND BENIGN PROSTATIC HYPERPLASIA

#770
20230190740
2023-06-22

AN NK-1 RECEPTOR ANTAGONIST FOR TREATING A DISEASE SELECTING FROM SEPSIS, SEPTIC SHOCK, ACUTE RESPIRATORY DISTRESS SYNDROME (ARDS) OR MULTIPLE ORGAN DYSFUNCTION SYNDROME (MODS)

#771
20230190690
2023-06-22

THERAPEUTIC AND/OR PREVENTIVE AGENT FOR CORONAVIRUS DISEASE 2019 (COVID-19)

#772
20230183257
2023-06-15

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]- pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#773
20230183225
2023-06-15

USE OF SELECTIVE GABA A ALPHA 5 NEGATIVE ALLOSTERIC MODULATORS FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM CONDITIONS

#774
20230181577
2023-06-15

STABLE COMPOSITIONS OF VARENICLINE

#775
20230181576
2023-06-15

Organic compounds

#776
20230181556
2023-06-15

USE OF PSYCHOTROPIC DRUGS FOR THE TREATMENT OF CORONAVIRUS INFECTIONS

#777
20230181527
2023-06-15

APICAL SODIUM-DEPENDENT TRANSPORTER INHIBITOR COMPOSITIONS

#778
20230181463
2023-06-15

OLEOGEL AND OLEOPASTE COMPOSITIONS AND USES THEREOF

#779
20230174562
2023-06-08

RADIO-AND CHEMO-PROTECTIVE COMPOUNDS

#780
20230172902
2023-06-08

Methods for the prophylaxis and treatment of COVID and COVID-19

#781
20230165855
2023-06-01

USE OF CYCLO-HISPRO (CHP) FOR LOWERING BLOOD PRESSURE

#782
20230165854
2023-06-01

Compounds and compositions for treating conditions associated with APJ receptor activity

#783
20230158023
2023-05-25

Crystalline succinate salt of 6-(6-aminopyrazin-2-yl)-n-(4-(4-(oxetan-3-yl)piperazin-1-yl)phenyl)imidazo[1,2-a]pyrazin-8-amine as a Syk inhibitor

#784
20230158022
2023-05-25

METHODS OF USING MYT1 INHIBITORS

#785
20230150999
2023-05-18

Composition and Method for Treating Metabolic Disorders

#786
20230149395
2023-05-18

METHODS OF TREATING RELAPSING MULTIPLE SCLEROSIS USING AN INHIBITOR OF BRUTON'S TYROSINE KINASE

#787
20230149314
2023-05-18

ORAL COMPLEX TABLET COMPRISING SITAGLIPTIN, DAPAGLIFLOZIN, AND METFORMIN

#788
20230148226
2023-05-11

COMPOSITIONS OF STABLE FORMULATIONS OF VARENICLINE SALT OR BASE FORM WITH CONTROL ON NITROSO IMPURITIES

#789
20230146514
2023-05-11

Oral compositions and the preparation methods thereof

#790
20230143119
2023-05-11

PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF DIABETES AND METABOLIC DISEASES ASSOCIATED THEREWITH

#791
20230136702
2023-05-04

Inhibitors of Human Herpesviruses

#792
20230133176
2023-05-04

COMPOSITION AND METHOD FOR TREATMENT OF DIABETES

#793
20230132378
2023-04-27

COMPOSITIONS AND METHODS FOR TREATING HEMORRHAGIC STROKE

#794
20230127304
2023-04-27

NEW INHIBITORS FOR THE KEAP1-NRF2 PROTEIN-PROTEIN INTERACTION

#795
20230125427
2023-04-27

Methods of measuring signaling pathway activity for selection of therapeutic agents

#796
20230121337
2023-04-20

CDK2 inhibitors and methods of using the same

#797
20230120910
2023-04-20

REGIMENS FOR TREATING HIV INFECTIONS AND AIDS

#798
20230119894
2023-04-20

THERAPEUTIC OR PROPHYLACTIC METHOD FOR DIABETES USING COMBINATION MEDICINE

#799
20230117286
2023-04-20

PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF NONALCOHOLIC STEATOHEPATITIS

#800
20230114946
2023-04-13

MESOSCALE NANOPARTICLES FOR SELECTIVE TARGETING TO THE KIDNEY AND METHODS OF THEIR THERAPEUTIC USE

#801
20230113598
2023-04-13

HETEROCYCLIC COMPOUNDS USEFUL AS PDK1 INHIBITORS

#802
20230112832
2023-04-13

Chemokine CXCR4 Receptor Modulators and Uses Related Thereto

#803
20230110784
2023-04-13

TREATMENT OF ADDICTION AND IMPULSE-CONTROL DISORDERS USING PDE7 INHIBITORS

#804
20230109858
2023-04-13

Heterocyclic inhibitors of PTPN11

#805
20230109839
2023-04-13

THERAPEUTIC AGENT FOR TAUOPATHIES

#806
20230109662
2023-04-06

INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

#807
20230107195
2023-04-06

TREATMENT OF CANCER WITH SMG1-INHIBITORS

#808
20230107039
2023-04-06

SOFT CHEWABLE FORMED BODY FOR THE ADMINISTRATION TO ANIMALS

#809
20230106238
2023-04-06

PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING NK/T-CELLLYMPHOMA OR NK-CELL LEUKEMIA, COMPRISING PHOSPHODIESTERASE TYPE 5 INHIBITOR

#810
20230100102
2023-03-30

CXCR7 INHIBITORS FOR THE TREATMENT OF CANCER

#811
20230097057
2023-03-30

Compositions for Inhibition of Herpesviruses

#812
20230095530
2023-03-30

COMPOUND USED AS RET KINASE INHIBITOR AND APPLICATION THEREOF

#813
20230095075
2023-03-30

COMPOSITIONS AND METHODS TO PROTECT MAMMALIAN TISSUE AGAINST COLD AND OTHER METABOLIC STRESSES

#814
20230095043
2023-03-30

POLYCYCLIC COMPOUND ACTING AS KINASE INHIBITOR

#815
20230094463
2023-03-30

ANTIBODIES THAT DISRUPT THE INTERACTION OF GAL3 AND INSULIN RECEPTOR OR INTEGRINS AND METHODS OF USE THEREOF

#816
20230090520
2023-03-23

SUBSTITUTED PYRAZOLO[1,5-A]PYRIDINE COMPOUNDS AS RET KINASE INHIBITORS

#817
20230089368
2023-03-23

POLYAROMATIC UREA DERIVATIVES AND THEIR USE IN THE TREATMENT OF MUSCLE DISEASES

#818
20230087744
2023-03-23

POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE

#819
20230087118
2023-03-23

IMIDAZO[1,2-a]PYRIDINYL DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE

#820
20230084803
2023-03-16

COMPOSITIONS AND METHODS FOR TREATING METABOLIC DISEASES

#821
20230081911
2023-03-16

NOVEL PROCESS FOR THE PREPARATION OF ACALABRUTINIB AND ITS INTERMEDIATES

#822
20230079407
2023-03-16

ANTI-MSR1 ANTIBODIES AND METHODS OF USE THEREOF

#823
20230074330
2023-03-09

PDE5 compositions and methods for immunotherapy

#824
20230074252
2023-03-09

DOSAGES AND METHODS FOR TREATING PULMONARY ARTERIAL HYPERTENSION WITH RODATRISTAT

#825
20230064417
2023-03-02

COMPOUNDS

#826
20230062486
2023-03-02

KRAS G12C INHIBITOR AND PHARMACEUTICAL USE THEREOF

#827
20230058001
2023-02-23

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#828
20230057844
2023-02-23

MOLECULAR TARGETS FOR ADDICTION

#829
20230057084
2023-02-23

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#830
20230052586
2023-02-16

DISUBSTITUTED ALKYNE DERIVATIVES

#831
20230049719
2023-02-16

PYRAZOLO[3,4-B]PYRAZINE SHP2 PHOSPHATASE INHIBITORS

#832
20230049113
2023-02-16

METHODS OF TREATING WHSC1-OVEREXPRESSING CANCERS BY INHIBITING SETD2

#833
20230047314
2023-02-16

Oral film formulation for modulating absorption profile

#834
20230046317
2023-02-16

Inhibitors of Glutathione S-Transferases (GSTS) and NAD(P)H:Quinone Oxidoreductase 1 (NQO1), Pharmaceutical Compositions, and Uses in Managing Cancer

#835
20230045509
2023-02-09

PHARMACEUTICAL COMPOSITIONS COMPRISING CABOTEGRAVIR

#836
20230045252
2023-02-09

Pyrazolo[1,5-a]pyrazin-4-yl derivatives

#837
20230044941
2023-02-09

TRIARYL COMPOUNDS FOR TREATMENT OF PD-L1 DISEASES

#838
20230043030
2023-02-09

Substituted pyridines, pyridazines, pyrimidines, and 1,2,3-triazines as bruton's tyrosine kinase inhibitors

#839
20230041761
2023-02-09

SMALL MOLECULE MODULATORS OF SIGMA-1 AND SIGMA-2 RECEPTORS AND USES THEREOF

#840
20230039319
2023-02-09

DEUTERIUM-ENRICHED SUBSTITUTED PHENOXYPHENYL ACETIC ACIDS AND ACYLSULFONAMIDES

#841
20230039309
2023-02-09

Substituted indole Mcl-1 inhibitors

#842
20230039022
2023-02-09

NK-3 RECEPTOR ANTAGONISTS FOR THERAPEUTIC OR COSMETIC TREATMENT OF EXCESS BODY FAT

#843
20230033410
2023-02-02

COMPLEX FORMULATION COMPRISING SITAGLIPTIN AND DAPAGLIFLOZIN, AND PREPARATION METHOD THEREFOR

#844
20230032813
2023-02-02

METHODS OF TREATING PULMONARY ARTERIAL HYPERTENSION

#845
20230029372
2023-01-26

THERAPEUTIC COMPOSITIONS AND METHODS FOR PREVENTION AND TREATMENT OF DIASTOLIC DYSFUNCTION

#846
20230021705
2023-01-26

GLP-1R MODULATING COMPOUNDS

#847
20230020241
2023-01-19

Pharmaceutical Composition For The Treatment Of Pulmonary Arterial Hypertension

#848
20230019094
2023-01-19

NOVEL COMPOUND AND PHARMACEUTICAL COMPOSITION FOR PREVENTION OR TREATMENT OF CANCER COMPRISING SAME

#849
20230017155
2023-01-19

Sleep improving agent

#850
20230014578
2023-01-19

GRANULES AND PREPARATION USING SAME

#851
20230014173
2023-01-19

Antibacterial compounds

#852
20230012449
2023-01-12

COMPOUNDS FOR THE TREATMENT OF HIV

#853
20230010803
2023-01-12

TREATMENTS FOR DIFFUSE LARGE B-CELL LYMPHOMA

#854
20230008047
2023-01-12

Imidazopiperazine inhibitors of transcription activating proteins

#855
20230000860
2023-01-05

INTRANASAL DHE FOR THE TREATMENT OF HEADACHE

#856
20230000842
2023-01-05

METHODS OF TREATING CARTILAGE DISORDERS THROUGH INHIBITION OF CLK AND DYRK

#857
20220409621
2022-12-29

Liquid oral formulations for sildenafil

#858
20220409619
2022-12-29

INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

#859
20220409615
2022-12-29

HTT modulators for treating Huntington's disease

#860
20220409589
2022-12-29

CHEMOKINE RECEPTOR BINDING HETEROCYCLIC COMPOUNDS WITH ENHANCED EFFICACY

#861
20220406428
2022-12-22

METHODS FOR TREATING ERECTILE DYSFUNCTION WITH A CGMP-SPECIFIC PHOSPHODIESTERASE 5 INHIBITOR PHARMACEUTICAL COMPOSITION

#862
20220403001
2022-12-22

PDE5 DERIVED REGULATORY CONSTRUCTS AND METHODS OF USE IN IMMUNOTHERAPY

#863
20220401442
2022-12-22

THERAPEUTIC COMBINATIONS OF ACALABRUTINIB AND CAPIVASERTIB TO TREAT B-CELL MALIGNANCIES

#864
20220401381
2022-12-22

PERIPHERALLY ACTING CANNABIDIOL (CBD)-CONTAINING COMPOUNDS AND USES THEREOF FOR ENHANCING FEMALE SEXUAL FUNCTION OR TREATING FEMALE SEXUAL DISORDERS

#865
20220395504
2022-12-15

KRAS G12C inhibitors and methods of using the same

#866
20220390454
2022-12-08

BIOMARKER PANEL TARGETED TO DISEASES DUE TO MULTIFACTORIAL ONTOLOGY OF GLYCOCALYX DISRUPTION

#867
20220387427
2022-12-08

Oral gliptin compositions and method for preparation thereof

#868
20220387426
2022-12-08

BICYCLIC COMPOUNDS AND METHODS FOR THEIR USE IN TREATING PITT HOPKINS SYNDROME

#869
20220387395
2022-12-08

UREA, AMIDE, AND SUBSTITUTED HETEROARYL COMPOUNDS FOR CBL-B INHIBITION

#870
20220378795
2022-12-01

Fused heterotricyclic organic compounds, pharmaceutical compositions, and medical uses thereof

#871
20220370451
2022-11-24

INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

#872
20220370420
2022-11-24

Spirocyclic 2,3-dihydro-7-azaindole compounds and uses thereof

#873
20220370395
2022-11-24

ENHANCER OF PHOTODYNAMIC EFFECT IN ALA-PDT OR ALA-PDD

#874
20220363675
2022-11-17

Novel Ferroportin Inhibitors

#875
20220362357
2022-11-17

Synergistic Combinations of Amino Acid Depletion Agent Sensitizers (AADAS) and Amino Acid Depletion Agents (AADA), and Therapeutic Methods of Use Thereof

#876
20220362251
2022-11-17

TREATMENT OF TACHYCARDIA

#877
20220362241
2022-11-17

NOVEL METHODS

#878
20220362238
2022-11-17

BILE ACID RECYCLING INHIBITORS AND SATIOGENS FOR TREATMENT OF DIABETES, OBESITY, AND INFLAMMATORY GASTROINTESTINAL CONDITIONS

#879
20220356182
2022-11-10

INHIBITORS OF HEPATITIS C VIRUS REPLICATION

#880
20220356158
2022-11-10

CGAS antagonist compounds

#881
20220354859
2022-11-10

SUBSTITUTED IMIDAZOQUINOXALINE COMPOUNDS AND USES THEREOF

#882
20220348582
2022-11-03

Crystal forms of (s)-4-(8-amino-3-(1-(but-2-ynoyl)pyrrolidin-2-yl)imidazo[1,5-a]pyrazin-1-yl)-n-(pyridin-2-yl)benzamide

#883
20220347174
2022-11-03

Method for treating HIV with Cabotegravir and Rilpivirine

#884
20220340575
2022-10-27

Use of a DPP-4 inhibitor in SIRS and/or sepsis

#885
20220339109
2022-10-27

Drug delivery system

#886
20220332751
2022-10-20

ANTIVIRAL PRODRUGS AND PHARMACEUTICAL COMPOSITIONS THEREOF

#887
20220331314
2022-10-20

COMPOSITIONS COMPRISING TIGOLANER FOR CONTROLLING PARASITES

#888
20220324835
2022-10-13

INHIBITORS OF CBL-B AND METHODS OF USE THEREOF

#889
20220323457
2022-10-13

Modulators of BCL6 proteolysis and associated methods of use

#890
20220323446
2022-10-13

SOTORASIB DOSING REGIMEN

#891
20220323434
2022-10-13

TREATMENT FOR DIABETES IN PATIENTS INAPPROPRIATE FOR METFORMIN THERAPY

#892
20220323358
2022-10-13

POWDER FOR ORAL SUSPENSION CONTAINING TADALAFIL

#893
20220315597
2022-10-06

TRICYCLIC COMPOUNDS AND THEIR USE

#894
20220313692
2022-10-06

Amorphous solid dispersions

#895
20220313641
2022-10-06

SPREADABLE NUTRITIONAL SUPPLEMENT AND SPREADABLE MEDICINE

#896
20220307034
2022-09-29

INHIBITING APE2 EXPRESSION IN A SUBJECT TREATED WITH A DRUG AGENT THAT CAUSES INCREASED APE2 EXPRESSION

#897
20220306643
2022-09-29

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]-pyrazin-8-yl)-N-(2,2,2-trifluoroethyl)pyrrolidine-1-carboxamide and solid state forms thereof

#898
20220305009
2022-09-29

IRAK4 KINASE INHIBITOR AND PREPARATION METHOD THEREFOR

#899
20220304893
2022-09-29

PROTECTION OF OXYGEN SENSITIVE COMPOUNDS

#900
20220298166
2022-09-22

Processes for the preparation of (3S,4R)-3-ethyl-4-(3H-imidazo[1,2-a]pyrrolo[2,3-e]-pyrazin-8-yl)-n-(2,2,2-trifluoroethyl)pyrrolidine-1 carboxamide and solid state forms thereof