94770 ⎘
Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
Compositions and methods of treating retinal disease
#302Guanidine compound
#303HETEROARYLS AND USES THEREOF
#304Carboxamide or sulfonamide substituted thiazoles and related derivatives as modulators for the orphan nuclear receptor ROR[γ]
#305Cyclic protein tyrosine kinase inhibitors
#306Inhibitors of the activity of complex (III) of the mitochondrial electron transport chain and use thereof
#307PREPARATION OF FEBUXOSTAT
#308Bicyclic thiazole compounds
#309Tertiary amines for use in the treatment of cardiac disorders
#310NEPRILYSIN INHIBITORS
#311Dual-acting thiophene, pyrrole, thiazole and furan antihypertensive agents
#312Novel halogen-substituted compounds
#313Piperidine/piperazine derivatives
#314Substituted biphenyl amides as P2Xand P2Xantagonists
#315Heteroaryl compounds with cyclic bridging unit
#316Bicyclo[3.2.1]octyl amide derivatives and uses of same
#317Heteroaryl compounds with A-cyclic bridging unit
#318Processes for preparing tubulysin derivatives and conjugates thereof
#319Inhibition of MCL-1 and/or BFL-1/A1
#320Aromatic 5-membered heterocyclic derivative having TRPV4-Inhibiting activity
#321Heteroarylcarboxylic acid ester derivative
#322COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES
#3235-membered heterocyclic amides and related compounds
#324Guanidinobenzoic acid compound
#325TRPM8 antagonists
#326METHOD FOR REDUCING BLOOD PRESSURE USING INHIBITORS OF PLASMA KALLIKREIN
#327Haloalkyl heteroaryl benzamide compounds
#328GLP-1 receptor stabilizers and modulators
#329METHODS FOR TREATING HYPERTENSION
#330Substituted arylcyclopentenes as therapeutic agents
#331Acylamino-substituted fused cyclopentanecarboxylic acid derivatives and their use as pharmaceuticals
#332Metalloenzyme inhibitor compounds
#333Modulators of C3a receptors
#334PROCESS FOR THE PREPARATION OF FEBUXOSTAT POLYMORPHS
#335THIAZOLE COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATMENT OF DEGENERATIVE DISEASES AND DISORDERS
#336Compositions, formulations and methods for treating ocular diseases
#337Substituted hydroxamic acids and uses thereof
#338Heteroaromatic compounds as BTK inhibitors
#339Molecules that induce disease resistance and improve growth in plants
#340Stem cell cultures
#341Macrocyclic inhibitors of hepatitis C virus
#342THERAPEUTIC AGENT AND PREVENTIVE AGENT FOR DEMYELINATING DISEASE
#343VINYL-PHENYL DERIVATIVES FOR INFLAMMATION AND IMMUNE-RELATED USES
#344Compounds that modulate intracellular calcium
#345Substituted hydroxamic acids and uses thereof
#346Compounds for treatment of cancer
#347Benzylamine derivatives as inhibitors of plasma kallikrein
#348Amide derivatives, process for preparation thereof and use thereof as insecticide
#349Cyclic protein tyrosine kinase inhibitors
#350Fungicide N-cycloalkyl-N-biphenylmethyl-carboxamide derivatives
#351Compound having detrusor muscle-contracting activity and urethral sphincter muscle-relaxing activity
#352Synthesis of tetracyclines and analogues thereof
#353Amidine compound or salt thereof
#354Biaryl derivatives as nAChR modulators
#355Thiazole compounds, methods for preparation and use thereof
#356Specific carboxamides as KCNQ2/3 modulators
#357Thiazole derivatives
#358Dual-acting thiophene, pyrrole, thiazole and furan antihypertensive agents
#359Heterocyclic inhibitors of necroptosis
#360Isoxazoline derivatives as pesticides
#361PROCESS FOR FEBUXOSTAT
#362Amide derivative, pest control agent containing the amide derivative, and pest controlling method
#363COMPOUNDS FOR INFLAMMATION AND IMMUNE-RELATED USES
#364Guanidine compound
#3652-(3-aminoaryl) amino-4-aryl-thiazoles and their use as c-kit inhibitors
#366Phenicol antibacterial agents
#367O-cyclopropylcyclohexyl-carboxanilides and their use as fungicides
#368Heteroarylcarboxylic acid ester derivative
#369Method for producing aminothiazole derivative and production intermediate
#370Method for producing aminothiazole derivative and production intermediate
#371BIARYL DERIVATIVES AS SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 2 INHIBITORS
#372Neprilysin inhibitors
#373HETEROAROMATIC COMPOUNDS AS BTK INHIBITORS
#374Neprilysin inhibitors
#375Aminoindanes amides having a high fungicidal activity and their phytosanitary compositions
#376Neprilysin inhibitors
#377NOVEL BICYCLIC THIAZOLE COMPOUNDS
#378PROCESS FOR THE PREPARATION OF 2-ARYLTHIAZOLE DERIVATIVES
#379Inhibitors of matrix metalloproteinases
#380THIAZOLE AND OXAZOLE-SUBSTITUTED ARYLAMIDES AS P2X3 AND P2X2/3 ANTAGONISTS
#381Fungicidal N-(2-phenoxyethyl)carboxamide derivatives and their aza, thia and sila analogues
#382Process for the preparation of febuxostat
#383Crystalline forms of febuxostat
#384POLYMORPHS OF FEBUXOSTAT
#385Cyclic amide derivative
#386ACYLSULFONAMIDES AND PROCESSES FOR PRODUCING THE SAME
#387Compounds for treatment of cancer
#388SUBSTANTIALLY PURE SALTS OF FEBUXOSTAT AND PROCESSES FOR PREPARATION THEREOF
#389PROCESS FOR PREPARING THE CRYSTALLINE FORM II OF FEBUXOSTAT
#390Compound having detrusor muscle-contracting activity and urethral sphincter muscle-relaxing activity
#391Crystalline forms of Febuxostat
#392PROCESS TO PREPARE ETHYL 4-METHYL-2-(4-(2-METHYLPROPYLOXY)-3-CYANOPHENYL)-5-THIAZOLECARBOXYLATE
#3932-alkyl-cycloalk(en)yl-carboxamides
#394Cysteine protease inhibitors
#395Preparation of febuxostat
#396Pyridinyl amides as P2X3 and P2X2/3 inhibitors
#397Method for producing phenyl-substituted heterocyclic derivative by means of coupling method using palladium compound
#398Process for preparing the crystalline form A of (2-[3-cyano-4-(2-I-butoxy)phenyl]-4-methyl-5-thiazole-carboxylic acid (febuxostat)
#399Guanidine compound
#400Polymorphs of an active pharmaceutical ingredient
#401LIGANDS FOR ANTIBODY AND Fc-FUSION PROTEIN PURIFICATION BY AFFINITY CHROMATOGRAPHY
#402Compounds and methods of treating brain disorders
#403C7-fluoro substituted tetracycline compounds
#404Thiazoles, imidazoles, and pyrazoles useful as inhibitors of protein kinases
#405Carboxylation catalysts
#4062′,2-bisthiazole non-nucleoside compounds, preparation methods, pharmaceutical compositions and uses as hepatitis virus inhibitors thereof
#4073-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals
#408DESAZADESFERROTHIOCIN AND DESAZADESFERROTHIOCIN POLYETHER ANALOGUES AS METAL CHELATION AGENTS
#409Benzamide derivatives
#410FUSED BICYCLIC HETEROARYL DERIVATIVE
#411Acylamino-substituted fused cyclopentanecarboxylic acid derivatives and their use as pharmaceuticals
#412Convenient Synthesis of Azolines to Azoles
#413NOVEL INHIBITORS OF STEAROYL-CoA-DESATURASE-1 AND THEIR USES
#414THERAPEUTIC COMPOUNDS
#415Anilinopiperazine derivatives and methods of use thereof
#416Electrochromic device
#417Heterocyclic inhibitors of necroptosis
#418Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
#419C7-fluoro substituted tetracycline compounds
#420INSECTICIDAL COMPOUNDS
#421Hematopoietic growth factor mimetic small molecule compounds and their uses
#422CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS
#423Heteroarylcarboxylic acid ester derivative
#424IRE-1α inhibitors
#425Arginine Derivatives with NP-I Antagonistic Activity
#426Amide derivatives, process for preparation thereof and use thereof as insecticide
#427Carboxy oxazole or thiazole compounds as DGAT-1 inhibitors useful for the treatment of obesity
#4283H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents
#429Compounds, pharmaceutical compositions and uses thereof
#430Method for carrying out chemical reactions with the aid of an inductively heated heating medium
#431Bicyclo[3.2.1]octyl amide derivatives and uses of same
#432Substituted amide compound
#433NOVEL GLUCOKINASE ACTIVATORS AND PROCESSES FOR THE PREPARATION THEREOF
#434Heteroaryls and uses thereof
#435Heteroaryls and uses thereof
#436Macrocylic inhibitors of hepatitis C virus
#437Neprilysin inhibitors
#438Neprilysin inhibitors
#439Arginine derivatives with NP-1 antagonistic activity
#440Process for producing crystals of polymorphic 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-5-thiazolecaboxylic acid by poor-solvent addition method
#441Compositions including 6-aminohexanoic acid derivatives as HDAC inhibitors
#442Compound having detrusor muscle-contracting activity and urethral sphincter muscle-relaxing activity
#443LPA RECEPTOR ANTAGONIST
#444Compounds for treatment of cancer
#445Sulfonylhydrazide compounds for treating proliferative disorders
#446Hydroxamates as therapeutic agents
#447Herbicidally active ketosultams and diketopyridines
#4482-(3-aminoaryl) amino-4-aryl-thiazoles and their use as c-kit inhibitors
#449DIACYLETHYLENEDIAMINE COMPOUND
#450Cycloalkylidene and heterocycloalkylidene inhibitor compounds
#451SUBSTITUTED ACYLGUANIDINE DERIVATIVES (AS AMENDED)
#452Substituted thiazol-2-ylamine derivatives, pharmaceutical compositions, and methods of use as 11-beta HSD1 modulators
#453Kinase Knockdown Via Electrophilically Enhanced Inhibitors
#454Herbicides
#455NOVEL HETEROCYCLIC NF-kB INHIBITORS
#456Thiazole and oxazole-substituted arylamides as P2Xand P2Xantagonists
#4571-(4-ureidobenzoyl)piperazine derivatives
#458METHOD FOR REDUCING BLOOD PRESSURE USING INHIBITORS OF PLASMA KALLIKREIN
#459Process for producing phenyl-substituted heterocyclic derivative through coupling using transition metal catalyst
#460Cysteine protease inhibitors
#461Halogen-substituted compounds
#462ARYL CARBONYL DERIVATIVES AS THERAPEUTIC AGENTS
#463Macrocyclic inhibitors of hepatitis C virus
#464Stem cell cultures
#465HIGH-PURITY FEBUXOSTAT AND THE METHOD FOR PREPARATION
#466Treatment of a stomach or small intestine ulcer with 2-(3-cyano-4-isobutyloxyphenyl)-4-methyl-1,3-thiazole-5-carboxylic acid
#467Desazadesferrothiocin and desazadesferrothiocin polyether analogues as metal chelation agents
#468Heteroaryl diamide compounds useful as MMP-13 inhibitors
#469Fungicidal carboxamides
#470High penetration compositions and their applications
#471Therapeutic compounds
#472Tubulysin D Analogues
#473Compositions and methods of treating retinal disease
#474Bradykinin B1-antagonists
#475Compounds
#476Agent for overcoming resistance to anti-cancer agent
#477Compounds for treatment of cancer
#478Novel amido derivatives and their use as positive allosteric modulators of metabotropic glutamate receptors
#4792-alkyl-cycloalk(en)yl-carboxamides
#480Isoxazoline derivatives as pesticides
#481Stem cell cultures
#482Inhibitors of STAT3
#483Substituted hydroxamic acids and uses thereof
#484SUBSTITUTED HYDROXAMIC ACIDS AND USES THEREOF
#485Fused-ring derivative and medical application of same
#4862-(3-aminoaryl) amino-4-aryl-thiazoles and their use as c-kit inhibitors
#487Sulfonamide compounds or salts thereof
#488Diacylglycerol acyltransferase inhibitors
#489Anti-Heparin Compounds
#490Dual-acting thiophene, pyrrole, thiazole and furan antihypertensive agents
#491N-hydroxyamidinoheterocycles as modulators of indoleamine 2,3-dioxygenase
#492BIARYL AMINO ACIDS AND THEIR USE IN DNA BINDING OLIGOMERS
#493Compounds, isomer thereof, or pharmaceutically acceptable salts thereof as vanilloid receptor antagonist and pharmaceutical compositions containing the same
#494Compounds that Inhibit HIV Particle Formation
#495Acylamino-substituted fused cyclopentanecarboxylic acid derivatives and their use as pharmaceuticals
#496Therapeutic compounds
#497Thiazoles and oxazoles useful as modulators of ATP-binding cassette transporters
#4982-oxothiazole compounds and method of using same for chronic inflammatory disorders
#499Amide derivative, pest control agent containing the amide derivative, and pest controlling method
#500N-2-(hetero)arylethylcarboxamide derivative, and pest-controlling agent comprising the same
#501NOVEL CARBOXYLIC ACID ANALOGS AS GLYCOGEN SYNTHASE ACTIVATORS
#502Acylsulfonamides and processes for producing the same
#503Biphenyl carboxylic acids and bioisosteres as glycogen synthase activators
#5042-substituted-ethynylthiazole derivatives and uses of same
#5057-And 9-Carbamate, Urea, Thiourea, Thiocarbamate, And Heteroaryl-Amino Substituted Tetracycline Compounds
#506Compounds which modulate the CB2 receptor
#507Therapeutic substituted cyclopentanes
#508Heteroaryl-ureas and their use as glucokinase activators
#509Therapeutic compounds
#510Therapeutic compounds
#511Agent for regeneration and/or protection of nerves
#512Potent immunosuppressive agents, derivatives and uses
#513NPY Y5 ANTAGONIST
#514Luminescent substrate for liciferase
#515Tubulysin D analogues
#516Bis-(Sulfonylamino) Derivatives in Therapy 066
#517Hydroxamates as therapeutic agents
#518Blood flow promoters for cauda equina tissues
#519Tetrahydropyridine, tetrahydroazepine, and dihydropyrrole derivatives for inflammation and immune-related uses
#520Synthesis of tetracyclines and analogues thereof
#521THIAZOLECARBOXANILIDES
#522Glucokinase activators and methods of using same
#523Biphenyl amides as P2Xand P2Xantagonists
#524Crystalline form of febuxostat
#525Heterocyclic inhibitors of necroptosis
#526Compounds as adenosine Areceptor antagonists
#527AMIDE COMPOUNDS AND USE THEREOF FOR PLANT DISEASE CONTROL
#528Thiazol-Guanidine Derivatives Useful As A (Beta)-Related Pathologies
#529NPY Y5 antagonist
#530Haloalkyl heteroaryl benzamide compounds
#5315-Membered Heterocyclic Amides And Related Compounds
#532Fungicide N-cycloalkyl-benzyl-amide derivatives
#533Substituted pyrazine compounds
#534Novel Heterocyclic NF-kB Inhibitors
#535EP2 Receptor Agonists
#536Fungicidal composition containing acid amide derivative
#537FUNGICIDAL COMPOSITION CONTAINING ACID AMIDE DERIVATIVE
#538Method for Carrying Out Chemical Reactions with the Aid of an Inductively Heated Heating Medium
#539LPA receptor antagonist
#540Azolecarboxamide compound or salt thereof
#541AGENT FOR OVERCOMING RESISTANCE TO ANTI-CANCER AGENT
#5424-ARYL-BUTANE-1,3-DIAMIDES
#543Compounds and methods for the treatment of viruses and cancer
#544BIPHENYLCARBOXAMIDES
#545TNIK INHIBITOR AND THE USE
#546Piperidine/piperazine derivatives
#547Heterocyclic amide derivatives useful as microbiocides
#548Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
#549Heteroaryl-ureas and their use as glucokinase activators
#550Heterocyclic a amide derivatives useful as microbiocides
#551Viral polymerase inhibitors
#5521,3-dihydroxy substituted phenylamide glucokinase activators
#553Modified malonate derivatives
#554ESTER COMPOUND AND MEDICAL USE THEREOF
#555Organic Compounds
#556Aminothiazole derivatives as human stearoyl-CoA desaturase inhibitors
#5572,4-disubstituted-5-aminocarbonyl-1,3-thiazole derivatives for therapeutic agent of antiinflammatory disease, method thereof for preparation, therapeutic agent for antiinflammatory disease induced by SPC activity containing the same
#558Regulation of protein synthesis
#559Compounds, compositions and methods comprising heteroaromatic derivatives
#560TNIK INHIBITOR AND THE USE
#561Substituted arylcyclopentenes as therapeutic agents
#562NOVEL AMIDO DERIVATIVES AND THEIR USE AS POSITIVE ALLOSTERIC MODULATORS OF METABOTROPIC GLUTAMATE RECEPTORS
#563Sphingosine Kinase Inhibitors and Methods of Their Use
#564Biaryl Sulfonamides and Methods for Using Same
#565Cytoskeletal active compounds, composition and use
#5662-aminothiazole-4-carboxylic amides as protein kinase inhibitors
#567Thiazolidine derivatives as orexin receptor antagonists
#568INHIBITORS OF 11-BETA-HYDROXY STERIOD DEHYDROGENASE TYPE 1
#569OXAZOLE AND THIAZOLE COMBINATORIAL LIBRARIES
#570C7-fluoro substituted tetracycline compounds
#571Compounds, Compositions and Methods Comprising Thiazole Derivatives
#572Hydrazone derivative
#573Thiazole compounds and their use for inhibiting phosphodiesterase 4, TNF-α, and IL-4
#574AMIDE AND UREA DERIVATIVES FOR THE TREATMENT OF METABOLIC DISEASES
#575Heteroaryl compounds as P2Yreceptor inhibitors
#576Fungicide N-(3-phenylpropyl) carboxamide derivatives
#577Insecticidal compounds
#578Certain Chemical Entities, Compositions, and Methods
#579Heterocyclic non-nucleoside compounds, their preparation, pharmaceutical composition and their use as antiviral agents
#5802-aminothiazole-4-carboxylic amides as protein kinase inhibitors
#581Therapeutic compounds
#582NOVEL HETEROCYCLIC NF-kB INHIBITORS
#583FUSED BICYCLIC HETEROARYL DERIVATIVE
#584Thiazolyl biphenyl amides
#585N-hydroxyamide derivatives possessing antibacterial activity
#586Microbiocides
#587Cycloalkylidene and heterocycloalkylidene inhibitor compounds
#588Arginine derivatives with NP-I antagonistic activity
#5894-(3,3-DIHALO-ALLYLOXY)PHENOL DERIVATIVES HAVING PESTICIDAL PROPERTIES
#590Heterocyclocarboxamide derivatives
#591P-38 INHIBITORS
#592Novel Heterocyclic NF-kB Inhibitors
#593Compounds for treatment of cancer
#594TYROSINE DERIVATIVE
#595Ethenyl carboxamide derivatives useful as microbiocides
#596Compounds, Compositions and Methods Comprising Heteroaromatic Derivatives
#597ANTI-VIRAL INHIBITORS AND METHODS OF USE
#598Imidazopyridinyl benzamide mitotic kinesin inhibitors
#599Thiazoles, imidazoles, and pyrazoles useful as inhibitors of protein kinases
#600Imidazopyridinyl benzamide mitotic kinesin inhibitors