ClassID:

95252

C07D403/12 - page 18 - CPC Classification

Classification description:

Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links

Recent Application in this class:
#5101
20120178764
2012-07-12

Novel Compounds

#5102
20120178758
2012-07-12

STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS

#5103
20120178741
2012-07-12

Sulfonylamino-derivatives as novel inhibitors of histone deacetylase

#5104
20120178735
2012-07-12

2H-CHROMENE COMPOUND AND DERIVATIVE THEREOF

#5105
20120178678
2012-07-12

Derivatives of 2H pyridazin-3-ones, their preparation and their use as SCD-1 inhibitors

#5106
20120178622
2012-07-12

Aminoquinazoline compounds for combating invertebrate pests

#5107
20120175598
2012-07-12

Carbazole derivative and organic electroluminescent devices utilizing the same and fabrication method thereof

#5108
20120172591
2012-07-05

Inhibitors of human phosphatidylinositol 3-kinase delta

#5109
20120172385
2012-07-05

ORTHO SUBSTITUTED PYRIMIDINE COMPOUNDS AS JAK INHIBITORS

#5110
20120172384
2012-07-05

HETEROCYCLYLAMINOPYRIMIDINES AS KINASE INHIBITORS

#5111
20120172378
2012-07-05

Compounds

#5112
20120172364
2012-07-05

Rate-controlled particles

#5113
20120172361
2012-07-05

TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS

#5114
20120168741
2012-07-05

Stilbene derivatives, light-emitting element, display device, and electronic device

#5115
20120165520
2012-06-28

PROCESS FOR THE SYNTHESIS OF PRODRUGS OF OPIOIDS

#5116
20120165519
2012-06-28

Fused bicyclic derivatives of 2,4-diaminopyrimidine as ALK and c-MET inhibitors

#5117
20120165352
2012-06-28

6-amino quinazoline or 3-cyano quinoline derivatives, preparation methods and pharmaceutical uses thereof

#5118
20120165351
2012-06-28

QUINAZOLINE DERIVATIVES

#5119
20120165347
2012-06-28

Compounds and their use as BACE inhibitors

#5120
20120165343
2012-06-28

Glucagon receptor modulators

#5121
20120165332
2012-06-28

SULFONAMIDES AND SULFAMIDES AS ZAP-70 INHIBITORS

#5122
20120165330
2012-06-28

QUINAZOLINONE AND RELATED ANALOGS AS SIRTUIN MODULATORS

#5123
20120165319
2012-06-28

INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME

#5124
20120165318
2012-06-28

Heterocyclic compounds for the inhibition of PASK

#5125
20120165305
2012-06-28

Substituted imidazopyridazines and benzimidazoles as inhibitors of FGFR3

#5126
20120164288
2012-06-28

Dyes with changeable solubilities, and methods for their use

#5127
20120157484
2012-06-21

Tryptophan hydroxylase inhibitors

#5128
20120157437
2012-06-21

VLA-4 INHIBITORY DRUG

#5129
20120157429
2012-06-21

Compounds useful as inhibitors of Janus kinases

#5130
20120157427
2012-06-21

Pyrazole aminopyrimidine derivatives as LRRK2 modulators

#5131
20120157426
2012-06-21

Mutant-selective EGFR inhibitors and uses thereof

#5132
20120157412
2012-06-21

Substituted pyrimidinyl oxime kinase inhibitors

#5133
20120157306
2012-06-21

Substituted fused pyrimidinones and dihydropyrimidinones

#5134
20120156279
2012-06-21

High penetration prodrug compositions of peptides and peptide-related compounds

#5135
20120156219
2012-06-21

NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF

#5136
20120149696
2012-06-14

Ethylene diamine modulators of fatty acid hydrolase

#5137
20120149677
2012-06-14

Ether benzotriazole derivatives

#5138
20120149676
2012-06-14

Compounds

#5139
20120149573
2012-06-14

Herbicidal pyrimidone derivatives

#5140
20120148534
2012-06-14

Methods and compositions of treating a family viral infection

#5141
20120148531
2012-06-14

Fused heterocyclic derivatives and methods of use

#5142
20120148514
2012-06-14

N-ALKYL LACTAM ETHERS, AND COMPOSITIONS AND USES THEREOF

#5143
20120142921
2012-06-07

Substituted hydrazide compounds and use thereof

#5144
20120142717
2012-06-07

Pyrimidinone compounds for use in the treatment of diseases or conditions mediated by Lp-PLA

#5145
20120142716
2012-06-07

4-pyrimidinesulfamide derivative

#5146
20120142711
2012-06-07

Acid-labile trigger units

#5147
20120142705
2012-06-07

ISATIN AND OXINDOLE COMPOUNDS

#5148
20120142689
2012-06-07

Serotonin reuptake inhibitors

#5149
20120142686
2012-06-07

Viral polymerase inhibitors

#5150
20120142677
2012-06-07

Pyrrolidine compounds which modulate the CB2 receptor

#5151
20120142668
2012-06-07

CATHEPSIN C INHIBITORS

#5152
20120142660
2012-06-07

AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS

#5153
20120142647
2012-06-07

Compounds as respiratory stimulants for treatment of breathing control disorders or diseases

#5154
20120141392
2012-06-07

METHODS OF MODULATING THE ACTIVITY OF THE MC1 RECEPTOR AND TREATMENT OF CONDITIONS RELATED TO THIS RECEPTOR

#5155
20120136016
2012-05-31

4, 5, 6-trisubstituted pyrimidine derivatives as factor IXa inhibitors

#5156
20120136001
2012-05-31

SUBSTITUTED OXINDOLE DERIVATIVES, MEDICAMENTS CONTAINING THE LATTER AND USE THEREOF

#5157
20120135997
2012-05-31

PHARMACEUTICAL COMPOSITION COMPRISING A LACTAM OR BENZENESULFONAMIDE COMPOUND

#5158
20120135994
2012-05-31

Inhibitors of human phosphatidylinositol 3-kinase delta

#5159
20120135987
2012-05-31

Phenylimidazole derivatives as PDE10A enzyme inhibitors

#5160
20120135977
2012-05-31

Ether benzotriazole derivatives

#5161
20120134963
2012-05-31

Compositions and methods for enhancing virus efficacy

#5162
20120134930
2012-05-31

Pyrazine derivatives for bioconjugation

#5163
20120130087
2012-05-24

Stereomerically pure fused bicyclic proline compounds useful for preparing hepatitis C protease inhibitors

#5164
20120130073
2012-05-24

Inhibitors of SYK and JAK protein kinases

#5165
20120130069
2012-05-24

Indazole derivatives or pharmaceutically acceptable salts thereof as protein kinase inhibitors for proliferative diseases treatment, and a pharmaceutical composition containing the same as an active ingredient

#5166
20120129867
2012-05-24

Inhibitors of protein kinases

#5167
20120129862
2012-05-24

Prokineticin 1 receptor antagonists

#5168
20120129844
2012-05-24

N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl]-4-(3,4-dimethylpiperazin-1-yl)benzamide and salts thereof

#5169
20120129830
2012-05-24

7-aza-spiro[3.5]nonane-7-carboxylate derivatives, preparation thereof and therapeutic use thereof

#5170
20120129829
2012-05-24

Indole modulators of S1P receptors

#5171
20120129765
2012-05-24

Specific HCV NS3 protease inhibitors

#5172
20120122930
2012-05-17

1H-benzimidazole-5-carboxamides as anti-inflammatory agents

#5173
20120122904
2012-05-17

Solid forms of (S)-2-amino-3-(4-(2-amino-6-((R)-1-(4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl)-2,2,2-trifluoroethoxy)pyrimidin-4-yl)phenyl)propanoic acid

#5174
20120122889
2012-05-17

SMALL MOLECULE INHIBITORS OF NECROPTOSIS

#5175
20120122868
2012-05-17

Apaf-1 inhibitor compounds

#5176
20120122857
2012-05-17

HETEROBICYCLIC CARBOXAMIDES AS INHIBITORS FOR KINASES

#5177
20120122854
2012-05-17

Carbocyclic Fused Cyclic Amines

#5178
20120122842
2012-05-17

NAMPT and rock inhibitors

#5179
20120122837
2012-05-17

Substituted quinoxalines as inhibitors of fatty acid binding protein

#5180
20120121502
2012-05-17

Pyrimidine hydroxy amide compounds as protein deacetylase inhibitors and methods of use thereof

#5181
20120115918
2012-05-10

Anti-Viral Compounds

#5182
20120115903
2012-05-10

Substituted Heteroaromatic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands

#5183
20120115902
2012-05-10

3H-imidazo [4, 5-B] pyridine-6-carboxamides as anti-inflammatory agents

#5184
20120115893
2012-05-10

Substituted Bicyclic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands

#5185
20120115869
2012-05-10

TETRAZOLE DERIVATIVES

#5186
20120115868
2012-05-10

Triazole compounds II

#5187
20120115844
2012-05-10

Triazole compounds I

#5188
20120115825
2012-05-10

Cyclohexyloxy-substituted heterocyclics, medicines containing these compounds and method for the production thereof

#5189
20120114696
2012-05-10

Small-molecule botulinum toxin inhibitors

#5190
20120114535
2012-05-10

Compound for inhibiting activity of ribonuclease, and container for storing nucleic acid containing the same

#5191
20120110704
2012-05-03

Pyridazine compounds for controlling invertebrate pests

#5192
20120108639
2012-05-03

Nitrogen-containing aromatic heterocyclyl compound

#5193
20120108631
2012-05-03

Sulfonamides for the modulation of PKM2

#5194
20120108603
2012-05-03

AMINOCARBONYL-DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE

#5195
20120108565
2012-05-03

PYRROLE CARBOXYLIC ACID DERIVATIVES AS ANTIBACTERIAL AGENTS

#5196
20120107273
2012-05-03

NEW PIPERAZINE COMPOUND AND USE THEREOF AS A HCV POLYMERASE INHIBITOR

#5197
20120101275
2012-04-26

Inhibitors of syk and JAK protein kinases

#5198
20120101081
2012-04-26

Amino-pyrrolidine-azetidine diamides as monoacylglycerol lipase inhibitors

#5199
20120101078
2012-04-26

AMIDE DERIVATIVES AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS

#5200
20120101072
2012-04-26

Triazole compounds that modulate Hsp90 activity

#5201
20120097925
2012-04-26

Organic light-emitting device

#5202
20120095211
2012-04-19

SUBSTITUTED PROLINE INHIBITORS OF HEPATITIS C VIRUS REPLICATION

#5203
20120095068
2012-04-19

Imidazolidine-2,4-dione derivatives and use thereof as a medicament

#5204
20120095040
2012-04-19

Cyclopenta[C]pyrrole-2-carboxylate derivatives, preparation thereof and therapeutic use thereof

#5205
20120095036
2012-04-19

Substituted indazole and aza-indazole derivatives as gamma secretase modulators

#5206
20120095015
2012-04-19

TRIAZOLE COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR

#5207
20120094997
2012-04-19

Substituted hydroxamic acids and uses thereof

#5208
20120094993
2012-04-19

-pyridin-3-yl or -pyrazin-2-yl carboxamides

#5209
20120094976
2012-04-19

Chemical compounds

#5210
20120094974
2012-04-19

SMOOTHENED RECEPTOR MODULATORS

#5211
20120094968
2012-04-19

Sulfonic amide and sulfoximine-substituted diaryl-dihydropyrimidinones and usage thereof

#5212
20120088919
2012-04-12

Dual-acting antihypertensive agents

#5213
20120088911
2012-04-12

Carboxylic acid derivatives, their preparation and use

#5214
20120088797
2012-04-12

1-heterocyclylsulfonyl, 3-aminomethyl, 5- (hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors

#5215
20120088779
2012-04-12

Heterocyclic sulfonamides

#5216
20120088778
2012-04-12

AZOLE DERIVATIVES AND FUSED BICYCLIC AZOLE DERIVATIVES AS THERAPEUTIC AGENTS

#5217
20120088772
2012-04-12

NOVEL PHARMACEUTICAL COMPOSITION FOR PREVENTION AND/OR TREATMENT OF ATTENTION DEFICIT/HYPERACTIVITY DISORDER

#5218
20120088768
2012-04-12

Pinane-substituted pyrimidinediamine derivatives useful as Axl inhibitors

#5219
20120088758
2012-04-12

Five-membered heterocycles useful as serine protease inhibitors

#5220
20120088754
2012-04-12

Sulfonyl-derivatives as novel inhibitors of histone deacetylase

#5221
20120088752
2012-04-12

Hedgehog pathway antagonists and therapeutic applications thereof

#5222
20120088740
2012-04-12

Co-crystals and pharmaceutical compositions comprising the same

#5223
20120083500
2012-04-05

Oxazolone and pyrrolidinone-substituted biphenyls as P2Xand P2Xantagonists

#5224
20120083488
2012-04-05

Tetracyclic compound

#5225
20120083483
2012-04-05

Inhibitors of hepatitis C virus replication

#5226
20120083475
2012-04-05

Indole amide derivatives and related compounds for use in the treatment of neurodegenerative diseases

#5227
20120083474
2012-04-05

Heterocyclic amides as modulators of TRPA1

#5228
20120077991
2012-03-29

Insecticides

#5229
20120077811
2012-03-29

Prodrug forms of kinase inhibitors and their use in therapy

#5230
20120077809
2012-03-29

Pyrimidopyridazine derivatives useful as P38 MAPK inhibitors

#5231
20120077796
2012-03-29

Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy

#5232
20120076835
2012-03-29

HIV INHIBITING PYRIMIDINES DERIVATIVES

#5233
20120071657
2012-03-22

Triazole compounds useful as protein kinase inhibitors

#5234
20120071479
2012-03-22

Pyrazine derivatives as enac blockers

#5235
20120071472
2012-03-22

Riminophenazines with 2-(heteroaryl)amino substituents and their anti-microbial activity

#5236
20120071466
2012-03-22

Inhibitor compounds of 11-beta-hydroxysteroid dehydrogenase type 1

#5237
20120071447
2012-03-22

Antiviral drugs for treatment of arenavirus infection

#5238
20120070413
2012-03-22

Method of treating cancer with substituted amide derivatives

#5239
20120065234
2012-03-15

Substituted N-phenyl-bipyrrolidine carboxamides and therapeutic use thereof

#5240
20120065216
2012-03-15

Quinazolinedione derivatives as PARP inhibitors

#5241
20120065214
2012-03-15

Compounds and their uses 708

#5242
20120065196
2012-03-15

AMIDE COMPOUNDS

#5243
20120065162
2012-03-15

N, N-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitors

#5244
20120059014
2012-03-08

Compounds for the Treatment of Metabolic Disorders

#5245
20120059002
2012-03-08

Anti-inflammatory agents

#5246
20120058996
2012-03-08

Carbazole carboxamide compounds useful as kinase inhibitors

#5247
20120058990
2012-03-08

-4-[[(5)-5-[[[3,5-bis(trifluoromethyl)phenyl]methyl] (2-methyl-2-tetrazol-5-yl)amino]-2,3,4,5-tetrahydro-7,9-dimethyl-1-1-benzazepin-1-yl]methyl]-cyclohexanecarboxylic acid

#5248
20120058988
2012-03-08

Carbazole and carboline kinase inhibitors

#5249
20120058892
2012-03-08

N-(tetrazol-5-yl)- and N-(triazol-5-yl)arylcarboxamides and their use as herbicides

#5250
20120053345
2012-03-01

Indazole Compounds

#5251
20120053195
2012-03-01

Hydrobromide salts of a pyrazolylaminoquinazoline

#5252
20120053194
2012-03-01

Optically active pyrazolylaminoquinazoline, and pharmaceutical compositions and methods of use thereof

#5253
20120053193
2012-03-01

Optically active pyrazolylaminoquinazoline, and pharmaceutical compositions and methods of use thereof

#5254
20120053183
2012-03-01

Piperazinylpyrimidine analogues as protein kinase inhibitors

#5255
20120053181
2012-03-01

Pyrrolidine-derived beta 3 adrenergic receptor agonists

#5256
20120053180
2012-03-01

CYCLOHEXANE ANALOGUES AS GPR119 AGONISTS

#5257
20120053179
2012-03-01

Rho-Kinase Inhibitors

#5258
20120053176
2012-03-01

ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF

#5259
20120053165
2012-03-01

Novel Phenyl Imidazoles and Phenyl Triazoles As Gamma-Secretase Modulators

#5260
20120046327
2012-02-23

METHOD FOR INHIBITING THE INDUCTION AND FORMATION OF OSTEOCLASTS

#5261
20120046308
2012-02-23

NOVEL ALPHA-PHENOXYBENZENEACETIC ACID DERIVATIVE AND PHARMACEUTICAL PREPARATION COMPRISING SAME

#5262
20120046287
2012-02-23

Dihydroindolone compounds, a process for their preparation and pharmaceutical compositions containing them

#5263
20120046275
2012-02-23

Cytoskeletal active rho kinase inhibitor compounds, composition and use

#5264
20120046269
2012-02-23

Amino azaheterocyclic carboxamides

#5265
20120046250
2012-02-23

Methods and compositions useful in treating cancer and reducing Wnt mediated effects in a cell

#5266
20120046245
2012-02-23

Compositions and methods for inhibition of the JAK pathway

#5267
20120045851
2012-02-23

LABELS, THEIR PRODUCTION PROCESS AND THEIR USES

#5268
20120045454
2012-02-23

2,4-pyrimidinediamine compounds and their uses

#5269
20120041008
2012-02-16

4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use

#5270
20120041001
2012-02-16

Carbonylamino-derivatives as novel inhibitors of histone deacetylase

#5271
20120040990
2012-02-16

INDOL-3-Y-CARBONYL-PIPERIDIN AND PIPERAZIN-DERIVATIVES

#5272
20120040977
2012-02-16

INHIBITORS OF HCV NS5A

#5273
20120040968
2012-02-16

Diamino heterocyclic carboxamide compound

#5274
20120040967
2012-02-16

Pyrazin-2-yl-pyridin-2-yl-amine and pyrazin-2-yl-pyrimidin-4-yl-amine compounds and their use

#5275
20120040955
2012-02-16

FLUORO SUBSTITUTED PYRIMIDINE COMPOUNDS AS JAK3 INHIBITORS

#5276
20120040954
2012-02-16

Anti-inflammatory agents

#5277
20120040948
2012-02-16

Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy

#5278
20120040935
2012-02-16

COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED ION CHANNELS

#5279
20120035407
2012-02-09

Compounds useful as inhibitors of ATR kinase

#5280
20120035239
2012-02-09

2-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses

#5281
20120035195
2012-02-09

1,4,5,6-tetrahydro-pyrimidin-2-ylamine compounds

#5282
20120035194
2012-02-09

SUBSTITUTED 2-AMINO-FUSED HETEROCYCLIC COMPOUNDS

#5283
20120035168
2012-02-09

N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides

#5284
20120035155
2012-02-09

INDOLE-2-CARBOXAMIDE DEIVATIVE

#5285
20120035154
2012-02-09

Modulators of Cellular Adhesion

#5286
20120029192
2012-02-02

Pyrazole Derivatives

#5287
20120029188
2012-02-02

Substituted aniline derivatives

#5288
20120029011
2012-02-02

Nitrogen-containing heteroaryl compounds and methods of use thereof

#5289
20120028997
2012-02-02

Prokineticin 1 receptor antagonists

#5290
20120028994
2012-02-02

Compounds for the reduction of beta-amyloid production

#5291
20120028963
2012-02-02

Hydroxamate derivative, a production method for the same, and a pharmaceutical composition comprising the same

#5292
20120028961
2012-02-02

6 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HTreceptor agonist

#5293
20120022254
2012-01-26

Sirtuin modulating compounds

#5294
20120022253
2012-01-26

Indazole, benzisoxazole, and benzisothiazole kinase inhibitors

#5295
20120022118
2012-01-26

Compounds for the treatment of proliferative disorders

#5296
20120022096
2012-01-26

Pro-neurogenic compounds

#5297
20120022090
2012-01-26

Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators

#5298
20120022066
2012-01-26

Insecticidal triazines and pyrimidines

#5299
20120022065
2012-01-26

C-met modulators and method of use

#5300
20120022057
2012-01-26

BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYGLYCEROL ACYLTRANSFERASE

#5301
20120021976
2012-01-26

Bicyclic piperidine and piperazine derivatives as GPCR modulators for the treatment of obesity, diabetes and other metabolic disorders

#5302
20120020915
2012-01-26

Substituted imidazole derivatives and methods of use thereof for treating cancer

#5303
20120016131
2012-01-19

Compositions and methods for inhibition of the JAK pathway

#5304
20120016122
2012-01-19

Compositions and methods for inhibition of the JAK pathway

#5305
20120015966
2012-01-19

PPAR ACTIVE COMPOUNDS

#5306
20120015959
2012-01-19

Heterocyclic compounds as autotaxin inhibitors

#5307
20120015954
2012-01-19

Therapeutic agents useful for treating pain

#5308
20120015951
2012-01-19

Polymorphs of brimonidine pamoate

#5309
20120015938
2012-01-19

1,4-BENZODIAZEPIN-2-ON DERIVATIVES

#5310
20120015927
2012-01-19

Crystalline forms of N-[2-[[(2,3-difluorophenyl)methyl]THIO]-6-{[(1R,2S)-2,3-dihydroxy-1-methylpropyl]oxy}-4-pyrimidinyl]-1-azetidinesulfonamide

#5311
20120015905
2012-01-19

Compounds for the prevention and treatment of cardiovascular diseases

#5312
20120014914
2012-01-19

Inhibitors of serine proteases, particularly HCV NS3-NS4A proteases

#5313
20120010407
2012-01-12

Compositions and methods for inhibition of the JAK pathway

#5314
20120010406
2012-01-12

Compositions and methods for inhibition of the JAK pathway

#5315
20120010235
2012-01-12

N-SUBSTITUTED PYRROLIDINES

#5316
20120010204
2012-01-12

Phthalazinone derivatives

#5317
20120010182
2012-01-12

Chemical compounds

#5318
20120009151
2012-01-12

Triazines And Related Compounds Having Antiviral Activity, Compositions And Methods Thereof

#5319
20120009124
2012-01-12

USE OF BUFFERS FOR RADIONUCLIDE COMPLEXATION

#5320
20120004422
2012-01-05

Intermediates useful in the preparation of maleimide functionalized polymers

#5321
20120004217
2012-01-05

Therapeutic agents useful for treating pain

#5322
20120004206
2012-01-05

Inhibitors of the 11-beta-hydroxysteroid dehydrogenase type 1 enzyme

#5323
20120003229
2012-01-05

MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN ALPHAVBETA3 RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY

#5324
20110319468
2011-12-29

Cyclic amine compounds

#5325
20110319447
2011-12-29

Triazole compounds that modulate HSP90 activity

#5326
20110319436
2011-12-29

Methods and compositions for modulating IRE1, SRC, and ABL activity

#5327
20110319430
2011-12-29

Fungicidal pyrazoles

#5328
20110319429
2011-12-29

Substituted 1,1,3,1-tetraoxidobenzo[D][1,3,2]dithiazoles as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction

#5329
20110319414
2011-12-29

Triazine derivative and pharmaceutical composition comprising the same

#5330
20110319413
2011-12-29

Piperazine compound capable of inhibiting prostaglandin D synthase

#5331
20110319412
2011-12-29

Piperidine and pyrrolidine derivatives having NPY Y5 receptor antagonism

#5332
20110319411
2011-12-29

ISOINDOLINONE AND RELATED ANALOGS AS SIRTUIN MODULATORS

#5333
20110319410
2011-12-29

PYRAZINE DERIVATIVES AND USE AS PI3K INHIBITORS

#5334
20110319403
2011-12-29

Bicyclic compounds as inhibitors of diacylglycerol acyltransferase

#5335
20110319396
2011-12-29

BENZODIAZEPIN-2-ON DERIVATIVES

#5336
20110319379
2011-12-29

Substituted Indazole Amides And Their Use As Glucokinase Activators

#5337
20110319362
2011-12-29

STAT3 LIGANDS AND THERAPEUTIC USES THEREOF

#5338
20110318393
2011-12-29

Substituted Pyrazole Compounds

#5339
20110313167
2011-12-22

Substituted Heterocycles as Therapeutic agents for treating cancer

#5340
20110312996
2011-12-22

NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION

#5341
20110312964
2011-12-22

Cysteine protease inhibitors

#5342
20110312963
2011-12-22

P38 MAP kinase inhibitors

#5343
20110312960
2011-12-22

Pyrazine derivatives and use as PI3K inhibitors

#5344
20110312955
2011-12-22

Triazine compounds as PI3 kinase and mTOR inhibitors

#5345
20110312949
2011-12-22

PHARMACEUTICAL USE OF SUBSTITUTED AMIDES

#5346
20110312945
2011-12-22

CRTH2 MODULATORS

#5347
20110312936
2011-12-22

Cyclohexyl-azetidinyl antagonists of CCR2

#5348
20110312935
2011-12-22

1H-benz imidazole-5-carboxamides as anti-inflammatory agents

#5349
20110312921
2011-12-22

N-myristoyl transferase inhibitors

#5350
20110312908
2011-12-22

Small molecule myristate inhibitors of BCR-ABL and methods of use

#5351
20110311648
2011-12-22

Methods for the treatment of cancer

#5352
20110311482
2011-12-22

Hepatitis C virus inhibitors

#5353
20110306628
2011-12-15

Non-peptidyl, potent, and selective mu opioid receptor antagonists

#5354
20110306611
2011-12-15

Transcription factor modulating compounds and methods of use thereof

#5355
20110306602
2011-12-15

4, 6-disubstituted aminopyrimidine derivatives as inhibitors of protein kinases

#5356
20110306592
2011-12-15

Cyclohexyl-azetidinyl antagonists of CCR2

#5357
20110306589
2011-12-15

Nitrogen containing heteroaryl compounds

#5358
20110301349
2011-12-08

Methods of preparing 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds

#5359
20110301193
2011-12-08

Methods and compositions of targeted drug development

#5360
20110301192
2011-12-08

Inhibitors of Cyclin Kinase Inhibitor p21

#5361
20110301175
2011-12-08

5-(4-(haloalkoxy)phenyl) pyrimidine-2-amine compounds and compositions as kinase inhibitors

#5362
20110301174
2011-12-08

1-heterocyclylsulfonyl, 3-aminomethyl, 5- (hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors

#5363
20110301173
2011-12-08

1-heterocyclylsulfonyl, 3-aminomethyl, 5-(hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors

#5364
20110301162
2011-12-08

AURORA KINASE MODULATORS AND METHODS OF USE

#5365
20110301161
2011-12-08

Benzimidazole inhibitors of leukotriene production

#5366
20110301157
2011-12-08

BICYCLIC AMIDES AS KINASE INHIBITORS

#5367
20110301155
2011-12-08

INDAZOLE COMPOUNDS FOR ACTIVATING GLUCOKINASE

#5368
20110301146
2011-12-08

GLYCOGEN SYNTHASE KINASE-3 BETA INHIBITORS CONTAINING 7-HYDROXY-BENZOIMIDAZOLE-4-YL-METHANONE DERIVATIVES

#5369
20110301145
2011-12-08

Pyridazinones, method of making, and method of use thereof

#5370
20110301128
2011-12-08

Pyrrole derivatives as pharmaceutical agents

#5371
20110301113
2011-12-08

PYRIDINEAMINE DERIVATIVES

#5372
20110301109
2011-12-08

Phenylpyrimidone compounds, the pharmaceutical compositions, preparation methods and uses thereof

#5373
20110295004
2011-12-01

Quinazoline based EGFR inhibitors

#5374
20110294850
2011-12-01

Indoline derivatives

#5375
20110294812
2011-12-01

P38 MAP kinase inhibitors

#5376
20110294798
2011-12-01

IL-12 Modulatory compounds

#5377
20110294796
2011-12-01

Benzotriazine inhibitors of kinases

#5378
20110294749
2011-12-01

DIAMINOPYRIMIDINECARBOXAMIDE DERIVATIVE

#5379
20110288227
2011-11-24

Polymerizable ionic liquid compositions

#5380
20110288139
2011-11-24

Substituted amino-benzimidazoles, medicaments comprimising said compound, their use and their method of manufacture

#5381
20110288109
2011-11-24

NEW COMPOUNDS

#5382
20110288083
2011-11-24

Method of treating cancer by inhibition of protein kinase-like endoplasmic reticulum protein kinase

#5383
20110288076
2011-11-24

Acetanilide sphingosine-1-phosphate receptor antagonists

#5384
20110288075
2011-11-24

Methods of treating disorders mediated by histamine Hreceptors using pyridazinone derivatives

#5385
20110288071
2011-11-24

Substituted pyrimidines for the treatment of diseases such as cancer

#5386
20110288065
2011-11-24

Aminopyrazine derivative and medicine

#5387
20110281913
2011-11-17

Melanocortin receptor antagonist compounds, process for preparing them and use thereof in human medicine and cosmetics

#5388
20110281881
2011-11-17

Substituted bicyclic heterocyclic compounds as gamma secretase modulators

#5389
20110281875
2011-11-17

Inhibitors of IAP

#5390
20110281846
2011-11-17

Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as Axl inhibitors

#5391
20110281843
2011-11-17

Substituted indazole derivatives active as kinase inhibitors

#5392
20110281840
2011-11-17

N-substituted saturated heterocyclic sulfone compounds with CB2 receptor agonistic activity

#5393
20110281356
2011-11-17

COMPOUNDS FOR STEM CELL DIFFERENTIATION

#5394
20110275819
2011-11-10

Organic compounds and their uses

#5395
20110275800
2011-11-10

2-sulfonylamino-4-heteroaryl butyramide antagonists of CCR10

#5396
20110275762
2011-11-10

Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes

#5397
20110275673
2011-11-10

INHIBITORS OF SPHINGOSINE KINASE 1

#5398
20110275657
2011-11-10

Melanocortin receptor modulators, process for preparing them and use there in human medicine and cosmetics

#5399
20110275656
2011-11-10

3H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents

#5400
20110275633
2011-11-10

2,4-diaminopyrimidine derivates as PTK2-inhibitors for the treatment of abnormal cell growth