95252 ⎘
Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group containing two hetero rings linked by a chain containing hetero atoms as chain links
Novel Compounds
#5102STYRYL-TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS
#5103Sulfonylamino-derivatives as novel inhibitors of histone deacetylase
#51042H-CHROMENE COMPOUND AND DERIVATIVE THEREOF
#5105Derivatives of 2H pyridazin-3-ones, their preparation and their use as SCD-1 inhibitors
#5106Aminoquinazoline compounds for combating invertebrate pests
#5107Carbazole derivative and organic electroluminescent devices utilizing the same and fabrication method thereof
#5108Inhibitors of human phosphatidylinositol 3-kinase delta
#5109ORTHO SUBSTITUTED PYRIMIDINE COMPOUNDS AS JAK INHIBITORS
#5110HETEROCYCLYLAMINOPYRIMIDINES AS KINASE INHIBITORS
#5111Compounds
#5112Rate-controlled particles
#5113TRIAZINE DERIVATIVES AND THEIR THERAPEUTICAL APPLICATIONS
#5114Stilbene derivatives, light-emitting element, display device, and electronic device
#5115PROCESS FOR THE SYNTHESIS OF PRODRUGS OF OPIOIDS
#5116Fused bicyclic derivatives of 2,4-diaminopyrimidine as ALK and c-MET inhibitors
#51176-amino quinazoline or 3-cyano quinoline derivatives, preparation methods and pharmaceutical uses thereof
#5118QUINAZOLINE DERIVATIVES
#5119Compounds and their use as BACE inhibitors
#5120Glucagon receptor modulators
#5121SULFONAMIDES AND SULFAMIDES AS ZAP-70 INHIBITORS
#5122QUINAZOLINONE AND RELATED ANALOGS AS SIRTUIN MODULATORS
#5123INHIBITORS OF INTERLEUKIN-1 BETA CONVERTING ENZYME
#5124Heterocyclic compounds for the inhibition of PASK
#5125Substituted imidazopyridazines and benzimidazoles as inhibitors of FGFR3
#5126Dyes with changeable solubilities, and methods for their use
#5127Tryptophan hydroxylase inhibitors
#5128VLA-4 INHIBITORY DRUG
#5129Compounds useful as inhibitors of Janus kinases
#5130Pyrazole aminopyrimidine derivatives as LRRK2 modulators
#5131Mutant-selective EGFR inhibitors and uses thereof
#5132Substituted pyrimidinyl oxime kinase inhibitors
#5133Substituted fused pyrimidinones and dihydropyrimidinones
#5134High penetration prodrug compositions of peptides and peptide-related compounds
#5135NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS AND MEDICINAL USE THEREOF
#5136Ethylene diamine modulators of fatty acid hydrolase
#5137Ether benzotriazole derivatives
#5138Compounds
#5139Herbicidal pyrimidone derivatives
#5140Methods and compositions of treating a family viral infection
#5141Fused heterocyclic derivatives and methods of use
#5142N-ALKYL LACTAM ETHERS, AND COMPOSITIONS AND USES THEREOF
#5143Substituted hydrazide compounds and use thereof
#5144Pyrimidinone compounds for use in the treatment of diseases or conditions mediated by Lp-PLA
#51454-pyrimidinesulfamide derivative
#5146Acid-labile trigger units
#5147ISATIN AND OXINDOLE COMPOUNDS
#5148Serotonin reuptake inhibitors
#5149Viral polymerase inhibitors
#5150Pyrrolidine compounds which modulate the CB2 receptor
#5151CATHEPSIN C INHIBITORS
#5152AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS
#5153Compounds as respiratory stimulants for treatment of breathing control disorders or diseases
#5154METHODS OF MODULATING THE ACTIVITY OF THE MC1 RECEPTOR AND TREATMENT OF CONDITIONS RELATED TO THIS RECEPTOR
#51554, 5, 6-trisubstituted pyrimidine derivatives as factor IXa inhibitors
#5156SUBSTITUTED OXINDOLE DERIVATIVES, MEDICAMENTS CONTAINING THE LATTER AND USE THEREOF
#5157PHARMACEUTICAL COMPOSITION COMPRISING A LACTAM OR BENZENESULFONAMIDE COMPOUND
#5158Inhibitors of human phosphatidylinositol 3-kinase delta
#5159Phenylimidazole derivatives as PDE10A enzyme inhibitors
#5160Ether benzotriazole derivatives
#5161Compositions and methods for enhancing virus efficacy
#5162Pyrazine derivatives for bioconjugation
#5163Stereomerically pure fused bicyclic proline compounds useful for preparing hepatitis C protease inhibitors
#5164Inhibitors of SYK and JAK protein kinases
#5165Indazole derivatives or pharmaceutically acceptable salts thereof as protein kinase inhibitors for proliferative diseases treatment, and a pharmaceutical composition containing the same as an active ingredient
#5166Inhibitors of protein kinases
#5167Prokineticin 1 receptor antagonists
#5168N-[5-[2-(3,5-dimethoxyphenyl)ethyl]-1h-pyrazol-3-yl]-4-(3,4-dimethylpiperazin-1-yl)benzamide and salts thereof
#51697-aza-spiro[3.5]nonane-7-carboxylate derivatives, preparation thereof and therapeutic use thereof
#5170Indole modulators of S1P receptors
#5171Specific HCV NS3 protease inhibitors
#51721H-benzimidazole-5-carboxamides as anti-inflammatory agents
#5173Solid forms of (S)-2-amino-3-(4-(2-amino-6-((R)-1-(4-chloro-2-(3-methyl-1H-pyrazol-1-yl)phenyl)-2,2,2-trifluoroethoxy)pyrimidin-4-yl)phenyl)propanoic acid
#5174SMALL MOLECULE INHIBITORS OF NECROPTOSIS
#5175Apaf-1 inhibitor compounds
#5176HETEROBICYCLIC CARBOXAMIDES AS INHIBITORS FOR KINASES
#5177Carbocyclic Fused Cyclic Amines
#5178NAMPT and rock inhibitors
#5179Substituted quinoxalines as inhibitors of fatty acid binding protein
#5180Pyrimidine hydroxy amide compounds as protein deacetylase inhibitors and methods of use thereof
#5181Anti-Viral Compounds
#5182Substituted Heteroaromatic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands
#51833H-imidazo [4, 5-B] pyridine-6-carboxamides as anti-inflammatory agents
#5184Substituted Bicyclic Carboxamide and Urea Compounds as Vanilloid Receptor Ligands
#5185TETRAZOLE DERIVATIVES
#5186Triazole compounds II
#5187Triazole compounds I
#5188Cyclohexyloxy-substituted heterocyclics, medicines containing these compounds and method for the production thereof
#5189Small-molecule botulinum toxin inhibitors
#5190Compound for inhibiting activity of ribonuclease, and container for storing nucleic acid containing the same
#5191Pyridazine compounds for controlling invertebrate pests
#5192Nitrogen-containing aromatic heterocyclyl compound
#5193Sulfonamides for the modulation of PKM2
#5194AMINOCARBONYL-DERIVATIVES AS NOVEL INHIBITORS OF HISTONE DEACETYLASE
#5195PYRROLE CARBOXYLIC ACID DERIVATIVES AS ANTIBACTERIAL AGENTS
#5196NEW PIPERAZINE COMPOUND AND USE THEREOF AS A HCV POLYMERASE INHIBITOR
#5197Inhibitors of syk and JAK protein kinases
#5198Amino-pyrrolidine-azetidine diamides as monoacylglycerol lipase inhibitors
#5199AMIDE DERIVATIVES AS NEUROPEPTIDE Y5 RECEPTOR LIGANDS
#5200Triazole compounds that modulate Hsp90 activity
#5201Organic light-emitting device
#5202SUBSTITUTED PROLINE INHIBITORS OF HEPATITIS C VIRUS REPLICATION
#5203Imidazolidine-2,4-dione derivatives and use thereof as a medicament
#5204Cyclopenta[C]pyrrole-2-carboxylate derivatives, preparation thereof and therapeutic use thereof
#5205Substituted indazole and aza-indazole derivatives as gamma secretase modulators
#5206TRIAZOLE COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE DOPAMINE D3 RECEPTOR
#5207Substituted hydroxamic acids and uses thereof
#5208-pyridin-3-yl or -pyrazin-2-yl carboxamides
#5209Chemical compounds
#5210SMOOTHENED RECEPTOR MODULATORS
#5211Sulfonic amide and sulfoximine-substituted diaryl-dihydropyrimidinones and usage thereof
#5212Dual-acting antihypertensive agents
#5213Carboxylic acid derivatives, their preparation and use
#52141-heterocyclylsulfonyl, 3-aminomethyl, 5- (hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors
#5215Heterocyclic sulfonamides
#5216AZOLE DERIVATIVES AND FUSED BICYCLIC AZOLE DERIVATIVES AS THERAPEUTIC AGENTS
#5217NOVEL PHARMACEUTICAL COMPOSITION FOR PREVENTION AND/OR TREATMENT OF ATTENTION DEFICIT/HYPERACTIVITY DISORDER
#5218Pinane-substituted pyrimidinediamine derivatives useful as Axl inhibitors
#5219Five-membered heterocycles useful as serine protease inhibitors
#5220Sulfonyl-derivatives as novel inhibitors of histone deacetylase
#5221Hedgehog pathway antagonists and therapeutic applications thereof
#5222Co-crystals and pharmaceutical compositions comprising the same
#5223Oxazolone and pyrrolidinone-substituted biphenyls as P2Xand P2Xantagonists
#5224Tetracyclic compound
#5225Inhibitors of hepatitis C virus replication
#5226Indole amide derivatives and related compounds for use in the treatment of neurodegenerative diseases
#5227Heterocyclic amides as modulators of TRPA1
#5228Insecticides
#5229Prodrug forms of kinase inhibitors and their use in therapy
#5230Pyrimidopyridazine derivatives useful as P38 MAPK inhibitors
#5231Phenalkylamine derivatives, pharmaceutical compositions containing them, and their use in therapy
#5232HIV INHIBITING PYRIMIDINES DERIVATIVES
#5233Triazole compounds useful as protein kinase inhibitors
#5234Pyrazine derivatives as enac blockers
#5235Riminophenazines with 2-(heteroaryl)amino substituents and their anti-microbial activity
#5236Inhibitor compounds of 11-beta-hydroxysteroid dehydrogenase type 1
#5237Antiviral drugs for treatment of arenavirus infection
#5238Method of treating cancer with substituted amide derivatives
#5239Substituted N-phenyl-bipyrrolidine carboxamides and therapeutic use thereof
#5240Quinazolinedione derivatives as PARP inhibitors
#5241Compounds and their uses 708
#5242AMIDE COMPOUNDS
#5243N, N-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitors
#5244Compounds for the Treatment of Metabolic Disorders
#5245Anti-inflammatory agents
#5246Carbazole carboxamide compounds useful as kinase inhibitors
#5247-4-[[(5)-5-[[[3,5-bis(trifluoromethyl)phenyl]methyl] (2-methyl-2-tetrazol-5-yl)amino]-2,3,4,5-tetrahydro-7,9-dimethyl-1-1-benzazepin-1-yl]methyl]-cyclohexanecarboxylic acid
#5248Carbazole and carboline kinase inhibitors
#5249N-(tetrazol-5-yl)- and N-(triazol-5-yl)arylcarboxamides and their use as herbicides
#5250Indazole Compounds
#5251Hydrobromide salts of a pyrazolylaminoquinazoline
#5252Optically active pyrazolylaminoquinazoline, and pharmaceutical compositions and methods of use thereof
#5253Optically active pyrazolylaminoquinazoline, and pharmaceutical compositions and methods of use thereof
#5254Piperazinylpyrimidine analogues as protein kinase inhibitors
#5255Pyrrolidine-derived beta 3 adrenergic receptor agonists
#5256CYCLOHEXANE ANALOGUES AS GPR119 AGONISTS
#5257Rho-Kinase Inhibitors
#5258ADENOSINE A3 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF
#5259Novel Phenyl Imidazoles and Phenyl Triazoles As Gamma-Secretase Modulators
#5260METHOD FOR INHIBITING THE INDUCTION AND FORMATION OF OSTEOCLASTS
#5261NOVEL ALPHA-PHENOXYBENZENEACETIC ACID DERIVATIVE AND PHARMACEUTICAL PREPARATION COMPRISING SAME
#5262Dihydroindolone compounds, a process for their preparation and pharmaceutical compositions containing them
#5263Cytoskeletal active rho kinase inhibitor compounds, composition and use
#5264Amino azaheterocyclic carboxamides
#5265Methods and compositions useful in treating cancer and reducing Wnt mediated effects in a cell
#5266Compositions and methods for inhibition of the JAK pathway
#5267LABELS, THEIR PRODUCTION PROCESS AND THEIR USES
#52682,4-pyrimidinediamine compounds and their uses
#52694-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds and methods of their use
#5270Carbonylamino-derivatives as novel inhibitors of histone deacetylase
#5271INDOL-3-Y-CARBONYL-PIPERIDIN AND PIPERAZIN-DERIVATIVES
#5272INHIBITORS OF HCV NS5A
#5273Diamino heterocyclic carboxamide compound
#5274Pyrazin-2-yl-pyridin-2-yl-amine and pyrazin-2-yl-pyrimidin-4-yl-amine compounds and their use
#5275FLUORO SUBSTITUTED PYRIMIDINE COMPOUNDS AS JAK3 INHIBITORS
#5276Anti-inflammatory agents
#5277Aminoindane derivatives, pharmaceutical compositions containing them, and their use in therapy
#5278COMPOSITIONS USEFUL AS INHIBITORS OF VOLTAGE-GATED ION CHANNELS
#5279Compounds useful as inhibitors of ATR kinase
#52802-oxo-1-pyrrolidine derivatives, processes for preparing them and their uses
#52811,4,5,6-tetrahydro-pyrimidin-2-ylamine compounds
#5282SUBSTITUTED 2-AMINO-FUSED HETEROCYCLIC COMPOUNDS
#5283N-((6-amino-pyridin-3-yl)methyl)-heteroaryl-carboxamides
#5284INDOLE-2-CARBOXAMIDE DEIVATIVE
#5285Modulators of Cellular Adhesion
#5286Pyrazole Derivatives
#5287Substituted aniline derivatives
#5288Nitrogen-containing heteroaryl compounds and methods of use thereof
#5289Prokineticin 1 receptor antagonists
#5290Compounds for the reduction of beta-amyloid production
#5291Hydroxamate derivative, a production method for the same, and a pharmaceutical composition comprising the same
#52926 substituted 2, 3,4,5 tetrahydro-1H-benzo[d]azepines as 5-HTreceptor agonist
#5293Sirtuin modulating compounds
#5294Indazole, benzisoxazole, and benzisothiazole kinase inhibitors
#5295Compounds for the treatment of proliferative disorders
#5296Pro-neurogenic compounds
#5297Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazopyridine derivatives as gamma secretase modulators
#5298Insecticidal triazines and pyrimidines
#5299C-met modulators and method of use
#5300BICYCLIC COMPOUNDS AS INHIBITORS OF DIACYGLYCEROL ACYLTRANSFERASE
#5301Bicyclic piperidine and piperazine derivatives as GPCR modulators for the treatment of obesity, diabetes and other metabolic disorders
#5302Substituted imidazole derivatives and methods of use thereof for treating cancer
#5303Compositions and methods for inhibition of the JAK pathway
#5304Compositions and methods for inhibition of the JAK pathway
#5305PPAR ACTIVE COMPOUNDS
#5306Heterocyclic compounds as autotaxin inhibitors
#5307Therapeutic agents useful for treating pain
#5308Polymorphs of brimonidine pamoate
#53091,4-BENZODIAZEPIN-2-ON DERIVATIVES
#5310Crystalline forms of N-[2-[[(2,3-difluorophenyl)methyl]THIO]-6-{[(1R,2S)-2,3-dihydroxy-1-methylpropyl]oxy}-4-pyrimidinyl]-1-azetidinesulfonamide
#5311Compounds for the prevention and treatment of cardiovascular diseases
#5312Inhibitors of serine proteases, particularly HCV NS3-NS4A proteases
#5313Compositions and methods for inhibition of the JAK pathway
#5314Compositions and methods for inhibition of the JAK pathway
#5315N-SUBSTITUTED PYRROLIDINES
#5316Phthalazinone derivatives
#5317Chemical compounds
#5318Triazines And Related Compounds Having Antiviral Activity, Compositions And Methods Thereof
#5319USE OF BUFFERS FOR RADIONUCLIDE COMPLEXATION
#5320Intermediates useful in the preparation of maleimide functionalized polymers
#5321Therapeutic agents useful for treating pain
#5322Inhibitors of the 11-beta-hydroxysteroid dehydrogenase type 1 enzyme
#5323MODULATORS OF CYTOKINE MEDIATED SIGNALLING PATHWAYS AND INTEGRIN ALPHAVBETA3 RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
#5324Cyclic amine compounds
#5325Triazole compounds that modulate HSP90 activity
#5326Methods and compositions for modulating IRE1, SRC, and ABL activity
#5327Fungicidal pyrazoles
#5328Substituted 1,1,3,1-tetraoxidobenzo[D][1,3,2]dithiazoles as MGLUR4 allosteric potentiators, compositions, and methods of treating neurological dysfunction
#5329Triazine derivative and pharmaceutical composition comprising the same
#5330Piperazine compound capable of inhibiting prostaglandin D synthase
#5331Piperidine and pyrrolidine derivatives having NPY Y5 receptor antagonism
#5332ISOINDOLINONE AND RELATED ANALOGS AS SIRTUIN MODULATORS
#5333PYRAZINE DERIVATIVES AND USE AS PI3K INHIBITORS
#5334Bicyclic compounds as inhibitors of diacylglycerol acyltransferase
#5335BENZODIAZEPIN-2-ON DERIVATIVES
#5336Substituted Indazole Amides And Their Use As Glucokinase Activators
#5337STAT3 LIGANDS AND THERAPEUTIC USES THEREOF
#5338Substituted Pyrazole Compounds
#5339Substituted Heterocycles as Therapeutic agents for treating cancer
#5340NOVEL INHIBITORS OF HEPATITIS C VIRUS REPLICATION
#5341Cysteine protease inhibitors
#5342P38 MAP kinase inhibitors
#5343Pyrazine derivatives and use as PI3K inhibitors
#5344Triazine compounds as PI3 kinase and mTOR inhibitors
#5345PHARMACEUTICAL USE OF SUBSTITUTED AMIDES
#5346CRTH2 MODULATORS
#5347Cyclohexyl-azetidinyl antagonists of CCR2
#53481H-benz imidazole-5-carboxamides as anti-inflammatory agents
#5349N-myristoyl transferase inhibitors
#5350Small molecule myristate inhibitors of BCR-ABL and methods of use
#5351Methods for the treatment of cancer
#5352Hepatitis C virus inhibitors
#5353Non-peptidyl, potent, and selective mu opioid receptor antagonists
#5354Transcription factor modulating compounds and methods of use thereof
#53554, 6-disubstituted aminopyrimidine derivatives as inhibitors of protein kinases
#5356Cyclohexyl-azetidinyl antagonists of CCR2
#5357Nitrogen containing heteroaryl compounds
#5358Methods of preparing 4-phenyl-6-(2,2,2-trifluoro-1-phenylethoxy)pyrimidine-based compounds
#5359Methods and compositions of targeted drug development
#5360Inhibitors of Cyclin Kinase Inhibitor p21
#53615-(4-(haloalkoxy)phenyl) pyrimidine-2-amine compounds and compositions as kinase inhibitors
#53621-heterocyclylsulfonyl, 3-aminomethyl, 5- (hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors
#53631-heterocyclylsulfonyl, 3-aminomethyl, 5-(hetero-) aryl substituted 1-H-pyrrole derivatives as acid secretion inhibitors
#5364AURORA KINASE MODULATORS AND METHODS OF USE
#5365Benzimidazole inhibitors of leukotriene production
#5366BICYCLIC AMIDES AS KINASE INHIBITORS
#5367INDAZOLE COMPOUNDS FOR ACTIVATING GLUCOKINASE
#5368GLYCOGEN SYNTHASE KINASE-3 BETA INHIBITORS CONTAINING 7-HYDROXY-BENZOIMIDAZOLE-4-YL-METHANONE DERIVATIVES
#5369Pyridazinones, method of making, and method of use thereof
#5370Pyrrole derivatives as pharmaceutical agents
#5371PYRIDINEAMINE DERIVATIVES
#5372Phenylpyrimidone compounds, the pharmaceutical compositions, preparation methods and uses thereof
#5373Quinazoline based EGFR inhibitors
#5374Indoline derivatives
#5375P38 MAP kinase inhibitors
#5376IL-12 Modulatory compounds
#5377Benzotriazine inhibitors of kinases
#5378DIAMINOPYRIMIDINECARBOXAMIDE DERIVATIVE
#5379Polymerizable ionic liquid compositions
#5380Substituted amino-benzimidazoles, medicaments comprimising said compound, their use and their method of manufacture
#5381NEW COMPOUNDS
#5382Method of treating cancer by inhibition of protein kinase-like endoplasmic reticulum protein kinase
#5383Acetanilide sphingosine-1-phosphate receptor antagonists
#5384Methods of treating disorders mediated by histamine Hreceptors using pyridazinone derivatives
#5385Substituted pyrimidines for the treatment of diseases such as cancer
#5386Aminopyrazine derivative and medicine
#5387Melanocortin receptor antagonist compounds, process for preparing them and use thereof in human medicine and cosmetics
#5388Substituted bicyclic heterocyclic compounds as gamma secretase modulators
#5389Inhibitors of IAP
#5390Bridged bicyclic aryl and bridged bicyclic heteroaryl substituted triazoles useful as Axl inhibitors
#5391Substituted indazole derivatives active as kinase inhibitors
#5392N-substituted saturated heterocyclic sulfone compounds with CB2 receptor agonistic activity
#5393COMPOUNDS FOR STEM CELL DIFFERENTIATION
#5394Organic compounds and their uses
#53952-sulfonylamino-4-heteroaryl butyramide antagonists of CCR10
#5396Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes
#5397INHIBITORS OF SPHINGOSINE KINASE 1
#5398Melanocortin receptor modulators, process for preparing them and use there in human medicine and cosmetics
#53993H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents
#54002,4-diaminopyrimidine derivates as PTK2-inhibitors for the treatment of abnormal cell growth